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—— 5-nitro-N-[(1R)-1-(2-oxo-1,3-dihydroindol-5-yl)ethyl]thiophene-2-carboxamide —— C15H13N3O4S
5-nitro-N-[(1R)-1-(2-oxo-1,3-dihydroindol-5-yl)ethyl]thiophene-2-carboxamide
—— (5Z)-5-(4-tert-butylbenzylidene)-3-(4-fluorophenyl)-2-thioxo-1,3-thiazolidin-4-one —— C20H18FNOS2
(5Z)-5-(4-tert-butylbenzylidene)-3-(4-fluorophenyl)-2-thioxo-1,3-thiazolidin-4-one
—— 5-(4-acetylphenyl)-N-[(1R)-1-(3-hydroxyphenyl)ethyl]-N-methylfuran-2-carboxamide —— C22H21NO4
5-(4-acetylphenyl)-N-[(1R)-1-(3-hydroxyphenyl)ethyl]-N-methylfuran-2-carboxamide
—— 5-[(3aS,4S,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[(1R)-1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]pentanamide —— C20H27N3O4S
5-[(3aS,4S,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[(1R)-1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]pentanamide
—— 5-[(3aS,4S,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[(1R)-1-(2,4-dichloro-5-fluorophenyl)ethyl]pentanamide —— C18H22Cl2FN3O2S
5-[(3aS,4S,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[(1R)-1-(2,4-dichloro-5-fluorophenyl)ethyl]pentanamide
—— 5-[[(1R)-1-(3,4-difluorophenyl)ethyl]sulfanylmethyl]-3-(methylsulfonylmethyl)-1,2,4-oxadiazole —— C13H14F2N2O3S2
5-[[(1R)-1-(3,4-difluorophenyl)ethyl]sulfanylmethyl]-3-(methylsulfonylmethyl)-1,2,4-oxadiazole
—— 5-cyclopropyl-N-[(1R)-1-(2,4-dimethoxyphenyl)ethyl]-1-phenyltriazole-4-carboxamide —— C22H24N4O3
5-cyclopropyl-N-[(1R)-1-(2,4-dimethoxyphenyl)ethyl]-1-phenyltriazole-4-carboxamide
—— 5-[1-[(1S)-1-(2,4-difluorophenyl)ethyl]piperidin-4-yl]-3-pyridin-2-yl-1,2,4-oxadiazole —— C20H20F2N4O
5-[1-[(1S)-1-(2,4-difluorophenyl)ethyl]piperidin-4-yl]-3-pyridin-2-yl-1,2,4-oxadiazole
—— 5-[1-[(1R)-1-(2,4-difluorophenyl)ethyl]piperidin-4-yl]-3-pyridin-2-yl-1,2,4-oxadiazole —— C20H20F2N4O
5-[1-[(1R)-1-(2,4-difluorophenyl)ethyl]piperidin-4-yl]-3-pyridin-2-yl-1,2,4-oxadiazole
—— (5E)-5-[[3-[4-[(4-chlorophenyl)methoxy]phenyl]-1-phenylpyrazol-4-yl]methylidene]-3-[(4-methylphenyl)methyl]-2-sulfanylidene-1,3-thiazolidin-4-one —— C34H26ClN3O2S2
(5E)-5-[[3-[4-[(4-chlorophenyl)methoxy]phenyl]-1-phenylpyrazol-4-yl]methylidene]-3-[(4-methylphenyl)methyl]-2-sulfanylidene-1,3-thiazolidin-4-one
—— 5-[[(1S)-1-(3,4-difluorophenyl)ethyl]sulfanylmethyl]-3-(methylsulfonylmethyl)-1,2,4-oxadiazole —— C13H14F2N2O3S2
5-[[(1S)-1-(3,4-difluorophenyl)ethyl]sulfanylmethyl]-3-(methylsulfonylmethyl)-1,2,4-oxadiazole
—— 5-[(3aS,4S,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[(1S)-1-(2,4-dichloro-5-fluorophenyl)ethyl]pentanamide —— C18H22Cl2FN3O2S
5-[(3aS,4S,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[(1S)-1-(2,4-dichloro-5-fluorophenyl)ethyl]pentanamide
—— (5E)-3-ethyl-5-{[3-(4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methylene}-2-thioxo-1,3-thiazolidin-4-one —— C22H19N3O2S2
(5E)-3-ethyl-5-{[3-(4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methylene}-2-thioxo-1,3-thiazolidin-4-one
—— (5E)-5-{[2,5-dimethyl-1-(pyridin-4-yl)-1H-pyrrol-3-yl]methylidene}-2-thioxoimidazolidin-4-one —— C15H14N4OS
(5E)-5-{[2,5-dimethyl-1-(pyridin-4-yl)-1H-pyrrol-3-yl]methylidene}-2-thioxoimidazolidin-4-one
—— (5E)-3-(3-ethoxypropyl)-5-[[9-methyl-4-oxo-2-(2-phenylethylamino)pyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C26H28N4O3S2
(5E)-3-(3-ethoxypropyl)-5-[[9-methyl-4-oxo-2-(2-phenylethylamino)pyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5E)-5-[(3,5-dimethylpiperidin-1-yl)methylidene]-3-ethyl-2-sulfanylidene-1,3-thiazolidin-4-one —— C13H20N2OS2
(5E)-5-[(3,5-dimethylpiperidin-1-yl)methylidene]-3-ethyl-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5Z)-5-[(E)-3-(furan-2-yl)prop-2-enylidene]-3-prop-2-enyl-2-sulfanylidene-1,3-thiazolidin-4-one —— C13H11NO2S2
(5Z)-5-[(E)-3-(furan-2-yl)prop-2-enylidene]-3-prop-2-enyl-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5E)-5-[(4-propoxyphenyl)methylidene]-3-propyl-2-sulfanylidene-1,3-thiazolidin-4-one —— C16H19NO2S2
(5E)-5-[(4-propoxyphenyl)methylidene]-3-propyl-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5S)-3-(5-chlorothiophen-2-yl)-N-[(2R)-1-(2,4-difluorophenoxy)propan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C17H15ClF2N2O3S
(5S)-3-(5-chlorothiophen-2-yl)-N-[(2R)-1-(2,4-difluorophenoxy)propan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— 5-[(3aS,4S,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-benzyl-N-[(2S)-1-(2-methoxyphenyl)propan-2-yl]pentanamide —— C27H35N3O3S
5-[(3aS,4S,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-benzyl-N-[(2S)-1-(2-methoxyphenyl)propan-2-yl]pentanamide
—— 5-[(3aS,4S,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-benzyl-N-[(2R)-1-(2-methoxyphenyl)propan-2-yl]pentanamide —— C27H35N3O3S
5-[(3aS,4S,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-benzyl-N-[(2R)-1-(2-methoxyphenyl)propan-2-yl]pentanamide
—— (5E)-3-benzyl-5-[(3,5-dibromo-4-hydroxyphenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C17H11Br2NO2S2
(5E)-3-benzyl-5-[(3,5-dibromo-4-hydroxyphenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5S)-3-(2,5-difluorophenyl)-N-[(2S,3S)-4-hydroxy-3-methylbutan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C15H18F2N2O3
(5S)-3-(2,5-difluorophenyl)-N-[(2S,3S)-4-hydroxy-3-methylbutan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5E)-5-[[3-(4-chlorophenyl)-1-phenylpyrazol-4-yl]methylidene]-2-(4-hydroxy-N-methylanilino)-1,3-thiazol-4-one —— C26H19ClN4O2S
(5E)-5-[[3-(4-chlorophenyl)-1-phenylpyrazol-4-yl]methylidene]-2-(4-hydroxy-N-methylanilino)-1,3-thiazol-4-one
—— 5-bromo-N-[(2R)-1-methoxypropan-2-yl]pyridin-3-amine —— C9H13BrN2O
5-bromo-N-[(2R)-1-methoxypropan-2-yl]pyridin-3-amine
—— (5R)-3-(5-chlorothiophen-2-yl)-N-[(2S)-1-(2,4-difluorophenoxy)propan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C17H15ClF2N2O3S
(5R)-3-(5-chlorothiophen-2-yl)-N-[(2S)-1-(2,4-difluorophenoxy)propan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— [5-[[(2R)-2-hydroxypropyl]amino]-2-nitrophenyl]-pyrrolidin-1-ylmethanone —— C14H19N3O4
[5-[[(2R)-2-hydroxypropyl]amino]-2-nitrophenyl]-pyrrolidin-1-ylmethanone
—— (5E)-3-ethyl-2-sulfanylidene-5-[(1,2,4-triazol-4-ylamino)methylidene]-1,3-thiazolidin-4-one —— C8H9N5OS2
(5E)-3-ethyl-2-sulfanylidene-5-[(1,2,4-triazol-4-ylamino)methylidene]-1,3-thiazolidin-4-one
—— (5E,5'Z)-3,3'-ethane-1,2-diylbis{2-(4-methoxyphenyl)-5-[4-(propan-2-yloxy)benzylidene]-3,5-dihydro-4H-imidazol-4-one} —— C42H42N4O6
(5E,5'Z)-3,3'-ethane-1,2-diylbis{2-(4-methoxyphenyl)-5-[4-(propan-2-yloxy)benzylidene]-3,5-dihydro-4H-imidazol-4-one}
—— 5-(3-chlorophenyl)-N-[(2R)-2-morpholin-4-ylpropyl]-1H-pyrazole-4-carboxamide —— C17H21ClN4O2
5-(3-chlorophenyl)-N-[(2R)-2-morpholin-4-ylpropyl]-1H-pyrazole-4-carboxamide
—— (5S)-3-(5-chlorothiophen-2-yl)-N-[(2S)-1-(2,4-difluorophenoxy)propan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C17H15ClF2N2O3S
(5S)-3-(5-chlorothiophen-2-yl)-N-[(2S)-1-(2,4-difluorophenoxy)propan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5E)-5-[(1-methylpyrrol-2-yl)methylidene]-2-sulfanylideneimidazolidin-4-one —— C9H9N3OS
(5E)-5-[(1-methylpyrrol-2-yl)methylidene]-2-sulfanylideneimidazolidin-4-one
—— (5E)-5-[[1-[(4-chlorophenyl)methyl]indol-3-yl]methylidene]-3-prop-2-enyl-2-sulfanylidene-1,3-thiazolidin-4-one —— C22H17ClN2OS2
(5E)-5-[[1-[(4-chlorophenyl)methyl]indol-3-yl]methylidene]-3-prop-2-enyl-2-sulfanylidene-1,3-thiazolidin-4-one
—— 5-(4-methoxyphenyl)-1,3-dimethyl-10-[(E)-2-phenylethenyl]-1,7,8,10-tetrahydro-2H-pyrimido[4',5':3,4]pyrrolo[2,1-c][1,4]oxazine-2,4(3H)-dione —— C26H25N3O4
5-(4-methoxyphenyl)-1,3-dimethyl-10-[(E)-2-phenylethenyl]-1,7,8,10-tetrahydro-2H-pyrimido[4',5':3,4]pyrrolo[2,1-c][1,4]oxazine-2,4(3H)-dione
—— 5-bromo-N-[(2S)-1-methoxypropan-2-yl]pyridin-3-amine —— C9H13BrN2O
5-bromo-N-[(2S)-1-methoxypropan-2-yl]pyridin-3-amine
—— (5E)-5-benzylidene-3-{1-[2-(2-hydroxyethyl)piperidin-1-yl]-1-oxopropan-2-yl}-2-thioxo-1,3-thiazolidin-4-one —— C20H24N2O3S2
(5E)-5-benzylidene-3-{1-[2-(2-hydroxyethyl)piperidin-1-yl]-1-oxopropan-2-yl}-2-thioxo-1,3-thiazolidin-4-one
—— (5Z)-2-[2-(1-adamantyl)-2-oxoethyl]sulfanyl-3-(4-methylphenyl)-5-[(4-propan-2-ylphenyl)methylidene]imidazol-4-one —— C32H36N2O2S
(5Z)-2-[2-(1-adamantyl)-2-oxoethyl]sulfanyl-3-(4-methylphenyl)-5-[(4-propan-2-ylphenyl)methylidene]imidazol-4-one
—— (5E)-5-[(1,3-dimethyl-1H-pyrazol-4-yl)methylidene]-3-(4-fluorophenyl)-2-thioxoimidazolidin-4-one —— C15H13FN4OS
(5E)-5-[(1,3-dimethyl-1H-pyrazol-4-yl)methylidene]-3-(4-fluorophenyl)-2-thioxoimidazolidin-4-one
—— (5E)-5-[(1-methyl-1H-pyrazol-4-yl)methylidene]-3-(propan-2-yl)-2-thioxo-1,3-thiazolidin-4-one —— C11H13N3OS2
(5E)-5-[(1-methyl-1H-pyrazol-4-yl)methylidene]-3-(propan-2-yl)-2-thioxo-1,3-thiazolidin-4-one
—— (5E)-3-[4-(2-ethylpiperidin-1-yl)-4-oxobutyl]-5-[(4-methylphenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C22H28N2O2S2
(5E)-3-[4-(2-ethylpiperidin-1-yl)-4-oxobutyl]-5-[(4-methylphenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5E)-5-[[4-(dimethylamino)phenyl]methylidene]-3-ethyl-1,3-thiazolidine-2,4-dione —— C14H16N2O2S
(5E)-5-[[4-(dimethylamino)phenyl]methylidene]-3-ethyl-1,3-thiazolidine-2,4-dione
—— (5E)-5-[(1,3-diphenyl-1H-pyrazol-4-yl)methylidene]-3-(4-fluorophenyl)-2-thioxoimidazolidin-4-one —— C25H17FN4OS
(5E)-5-[(1,3-diphenyl-1H-pyrazol-4-yl)methylidene]-3-(4-fluorophenyl)-2-thioxoimidazolidin-4-one
—— (5E)-5-[(2E)-2-methyl-3-phenylprop-2-en-1-ylidene]-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-2-thioxo-1,3-thiazolidin-4-one —— C20H23N3O2S2
(5E)-5-[(2E)-2-methyl-3-phenylprop-2-en-1-ylidene]-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-2-thioxo-1,3-thiazolidin-4-one
—— (5Z)-3-[3-(4-benzylpiperidin-1-yl)-3-oxopropyl]-5-[(E)-3-phenylprop-2-enylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C27H28N2O2S2
(5Z)-3-[3-(4-benzylpiperidin-1-yl)-3-oxopropyl]-5-[(E)-3-phenylprop-2-enylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5E)-3-(1-phenylethyl)-5-(1H-pyrrol-2-ylmethylidene)-2-sulfanylidene-1,3-thiazolidin-4-one —— C16H14N2OS2
(5E)-3-(1-phenylethyl)-5-(1H-pyrrol-2-ylmethylidene)-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5Z)-3-[3-(4-methylpiperazin-1-yl)-3-oxopropyl]-5-[(E)-3-phenylprop-2-enylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C20H23N3O2S2
(5Z)-3-[3-(4-methylpiperazin-1-yl)-3-oxopropyl]-5-[(E)-3-phenylprop-2-enylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5S)-3-(2,5-difluorophenyl)-N-[(2R,3S)-4-hydroxy-3-methylbutan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C15H18F2N2O3
(5S)-3-(2,5-difluorophenyl)-N-[(2R,3S)-4-hydroxy-3-methylbutan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5E)-3-butyl-5-[[4-(dimethylamino)phenyl]methylidene]-1,3-thiazolidine-2,4-dione —— C16H20N2O2S
(5E)-3-butyl-5-[[4-(dimethylamino)phenyl]methylidene]-1,3-thiazolidine-2,4-dione
—— (5S)-3-(2,5-difluorophenyl)-N-[(2R,3R)-4-hydroxy-3-methylbutan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C15H18F2N2O3
(5S)-3-(2,5-difluorophenyl)-N-[(2R,3R)-4-hydroxy-3-methylbutan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— [5-[[(2S)-2-hydroxypropyl]amino]-2-nitrophenyl]-pyrrolidin-1-ylmethanone —— C14H19N3O4
[5-[[(2S)-2-hydroxypropyl]amino]-2-nitrophenyl]-pyrrolidin-1-ylmethanone