中文名称 |
英文名称 |
CAS号 |
化学式 |
结构式图片 |
—— |
[(3R)-3-[(5S,7R)-2-tert-butyl-7-(difluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-(1,3-thiazol-4-yl)methanone |
—— |
C20H27F2N5OS |
|
—— |
3-(1,3-benzothiazol-2-yl)-1-[(2R)-2-(2-tert-butylpyrazolo[1,5-a]pyrimidin-7-yl)pyrrolidin-1-yl]propan-1-one |
—— |
C24H27N5OS |
|
—— |
1-[(2R)-2-(2-tert-butylpyrazolo[1,5-a]pyrimidin-7-yl)pyrrolidin-1-yl]-2,2-dimethylpropan-1-one |
—— |
C19H28N4O |
|
—— |
(2-Aminopyridin-3-yl)-[4-[5-tert-butyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]methanone |
—— |
C22H25F3N6O |
|
—— |
1-[(2S)-2-(2-tert-butylpyrazolo[1,5-a]pyrimidin-7-yl)pyrrolidin-1-yl]-2,2-dimethylpropan-1-one |
—— |
C19H28N4O |
|
—— |
1-[4-[(5S,7R)-2-tert-butyl-7-(difluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-2-[(2S)-oxolan-2-yl]ethanone |
—— |
C22H34F2N4O2 |
|
—— |
1-[(3R)-3-[(5S,7R)-2-tert-butyl-7-(difluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-2-pyridin-2-ylethanone |
—— |
C23H31F2N5O |
|
—— |
4-[4-[(5S,7R)-2-tert-butyl-7-(difluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidine-1-carbonyl]-1-methylpyridin-2-one |
—— |
C23H31F2N5O2 |
|
—— |
[(3S)-3-[(5S,7R)-2-tert-butyl-7-(difluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-pyridin-3-ylmethanone |
—— |
C22H29F2N5O |
|
—— |
[(3R)-3-[(5S,7R)-2-tert-butyl-7-(difluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-cyclohexylmethanone |
—— |
C23H36F2N4O |
|
—— |
1-[(3S)-3-[(5S,7R)-2-tert-butyl-7-(difluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-2-[(1S)-cyclopent-2-en-1-yl]ethanone |
—— |
C23H34F2N4O |
|
—— |
1-[4-[(5S,7R)-2-tert-butyl-7-(difluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-2-pyridin-2-ylethanone |
—— |
C23H31F2N5O |
|
—— |
[(2S)-2-[(5S,7R)-5-tert-butyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-cyclopropylmethanone |
—— |
C20H29F3N4O |
|
—— |
(5S,7R)-5-tert-butyl-2-[1-[[(3S)-oxolan-3-yl]methyl]piperidin-4-yl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine |
—— |
C21H33F3N4O |
|
—— |
(5S,7R)-5-tert-butyl-2-[(2R)-1-(pyridin-3-ylmethyl)piperidin-2-yl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine |
—— |
C22H30F3N5 |
|
—— |
[(2R)-2-[(5S,7R)-5-tert-butyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-pyridin-3-ylmethanone |
—— |
C22H28F3N5O |
|
—— |
(5R,7S)-2-tert-butyl-7-(difluoromethyl)-5-[(3S)-1-(3,6-dihydro-2H-pyran-5-ylmethyl)piperidin-3-yl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine |
—— |
C22H34F2N4O |
|
—— |
1-[(3S)-3-[(5S,7R)-5-tert-butyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-2-[(2S)-oxolan-2-yl]ethanone |
—— |
C22H33F3N4O2 |
|
—— |
[(3R)-3-[(5S,7R)-2-tert-butyl-7-(difluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-cyclopentylmethanone |
—— |
C22H34F2N4O |
|
—— |
[(2S)-2-[5-tert-butyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-pyridin-3-ylmethanone |
—— |
C22H24F3N5O |
|
—— |
[4-[5-Tert-butyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-(1-methylpyrazol-4-yl)methanone |
—— |
C21H25F3N6O |
|
—— |
[(3S)-3-[(5S,7R)-2-tert-butyl-7-(difluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-(1,3-thiazol-4-yl)methanone |
—— |
C20H27F2N5OS |
|
—— |
(5S,7R)-5-tert-butyl-2-[(2S)-1-[(1-methylpyrazol-4-yl)methyl]piperidin-2-yl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine |
—— |
C21H31F3N6 |
|
—— |
1-[(3R)-3-[(5S,7R)-2-tert-butyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-2-[(1S)-cyclopent-2-en-1-yl]ethanone |
—— |
C23H33F3N4O |
|
—— |
(5R,7S)-2-tert-butyl-7-(difluoromethyl)-5-[(3S)-1-(pyridin-2-ylmethyl)piperidin-3-yl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine |
—— |
C22H31F2N5 |
|
—— |
(5S,7R)-5-tert-butyl-2-[(3S)-1-prop-2-enylsulfonylpyrrolidin-3-yl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine |
—— |
C18H27F3N4O2S |
|
—— |
[(3R)-3-[(5S,7R)-2-tert-butyl-7-(difluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-[(1R)-cyclohex-3-en-1-yl]methanone |
—— |
C23H34F2N4O |
|
—— |
[4-[(5S,7R)-5-tert-butyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-(1-methylpyrazol-3-yl)methanone |
—— |
C21H29F3N6O |
|
—— |
1-[(3S)-3-[(5S,7R)-5-tert-butyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-2-[(2R)-oxolan-2-yl]ethanone |
—— |
C22H33F3N4O2 |
|
—— |
(5S,7R)-5-tert-butyl-2-[1-[[(3R)-oxolan-3-yl]methyl]piperidin-4-yl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine |
—— |
C21H33F3N4O |
|
—— |
1-[(2S)-2-[5-tert-butyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-2-pyridin-2-ylethanone |
—— |
C23H26F3N5O |
|
—— |
[(2R)-2-[(5S,7R)-5-tert-butyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-pyridin-2-ylmethanone |
—— |
C22H28F3N5O |
|
—— |
(5S,7R)-5-tert-butyl-2-[(3S)-1-pyrrolidin-1-ylsulfonylpyrrolidin-3-yl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine |
—— |
C19H30F3N5O2S |
|
—— |
[(3S)-3-[(5S,7R)-2-tert-butyl-7-(difluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-cyclopropylmethanone |
—— |
C20H30F2N4O |
|
—— |
1-[(2R)-2-[(5S,7R)-5-tert-butyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-2-pyridin-2-ylethanone |
—— |
C23H30F3N5O |
|
—— |
1-[4-[(5S,7R)-5-tert-butyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-2-methoxyethanone |
—— |
C19H29F3N4O2 |
|
—— |
(5R,7S)-2-tert-butyl-7-(difluoromethyl)-5-[(3R)-1-(3,6-dihydro-2H-pyran-5-ylmethyl)piperidin-3-yl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine |
—— |
C22H34F2N4O |
|
—— |
1-[(3S)-3-[(5S,7R)-5-tert-butyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-2,2-dimethylpropan-1-one |
—— |
C21H33F3N4O |
|
—— |
[(2S)-2-[(5S,7R)-5-tert-butyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-(1-methylpyrazol-4-yl)methanone |
—— |
C21H29F3N6O |
|
—— |
(5-Aminopyridin-3-yl)-[4-[5-tert-butyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]methanone |
—— |
C22H25F3N6O |
|
—— |
[(2S)-2-[(5S,7R)-5-tert-butyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-[(2S)-oxolan-2-yl]methanone |
—— |
C21H31F3N4O2 |
|
—— |
1-[4-[(5S,7R)-5-tert-butyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-2-hydroxyethanone |
—— |
C18H27F3N4O2 |
|
—— |
3-[(3S)-3-[(5R,7S)-2-tert-butyl-7-(difluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-N,N,2,2-tetramethylpropan-1-amine |
—— |
C23H41F2N5 |
|
—— |
1-[(3S)-3-[(5S,7R)-5-tert-butyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]-3-[(2S)-oxolan-2-yl]propan-1-one |
—— |
C22H33F3N4O2 |
|
—— |
1-[(3R)-3-[(5S,7R)-2-tert-butyl-7-(difluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-3-methoxypropan-1-one |
—— |
C20H32F2N4O2 |
|
—— |
[(3S)-3-[(5S,7R)-2-tert-butyl-7-(difluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-cyclohexylmethanone |
—— |
C23H36F2N4O |
|
—— |
(5S,7R)-5-tert-butyl-2-[(2R)-1-[(1-methylpyrazol-4-yl)methyl]piperidin-2-yl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine |
—— |
C21H31F3N6 |
|
—— |
(5R,7S)-2-tert-butyl-5-[(3S)-1-(pyridin-2-ylmethyl)piperidin-3-yl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine |
—— |
C22H30F3N5 |
|
—— |
[(3S)-3-[(5S,7R)-2-tert-butyl-7-(difluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-[(2R)-oxolan-2-yl]methanone |
—— |
C21H32F2N4O2 |
|
—— |
1-[(3S)-3-[(5S,7R)-2-tert-butyl-7-(difluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-2-[(1R)-cyclopent-2-en-1-yl]ethanone |
—— |
C23H34F2N4O |
|