中文名称 |
英文名称 |
CAS号 |
化学式 |
结构式图片 |
—— |
[(2R)-2-[5-propan-2-yl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]-pyridin-4-ylmethanone |
—— |
C20H20F3N5O |
|
—— |
cyclopropyl-[(3R)-3-[5-propan-2-yl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]methanone |
—— |
C19H23F3N4O |
|
—— |
(2-methyl-5-propan-2-ylpyrazol-3-yl)-[(3S)-3-[5-propan-2-yl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]methanone |
—— |
C22H27F3N6O |
|
—— |
2-tert-butyl-5-[(3S)-1-[3-[(2S)-oxolan-2-yl]propanoyl]pyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one |
—— |
C21H30N4O3 |
|
—— |
2,2-dimethyl-1-[(3R)-3-[5-thiophen-2-yl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]propan-1-one |
—— |
C21H23F3N4OS |
|
—— |
2-tert-butyl-5-[(3S)-1-(4-imidazol-1-ylbutanoyl)pyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one |
—— |
C21H28N6O2 |
|
—— |
1-[(3R)-3-[2-tert-butyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-2-methoxyethanone |
—— |
C19H25F3N4O2 |
|
—— |
2-tert-butyl-5-[(3S)-1-[3-[(2R)-oxolan-2-yl]propanoyl]pyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one |
—— |
C21H30N4O3 |
|
—— |
2-tert-butyl-5-[(3R)-1-[3-[(2S)-oxolan-2-yl]propanoyl]pyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one |
—— |
C21H30N4O3 |
|
—— |
1-methylsulfonyl-N-[2-(5-thiophen-2-ylpyrazolo[1,5-a]pyrimidin-2-yl)ethyl]piperidine-4-carboxamide |
—— |
C19H23N5O3S2 |
|
—— |
2-benzofuran-1-yl-[(3S)-3-[2-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]methanone |
—— |
C22H19F3N4O2 |
|
—— |
3-(3-chloro-1,2-oxazol-5-yl)-N-[2-(5-pyridin-4-ylpyrazolo[1,5-a]pyrimidin-2-yl)ethyl]propanamide |
—— |
C19H17ClN6O2 |
|
—— |
1-methyl-4-[(2S)-2-[(5R,7R)-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidine-1-carbonyl]pyridin-2-one |
—— |
C20H24F3N5O2 |
|
—— |
[(3S)-1,1-dioxothiolan-3-yl]-[(2R)-2-[(5S,7R)-5-propan-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]methanone |
—— |
C19H27F3N4O3S |
|
—— |
1-methyl-5-[4-[(5S,7R)-2-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidine-1-carbonyl]pyridin-2-one |
—— |
C20H24F3N5O2 |
|
—— |
[4-[(5S,7R)-5-tert-butyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-pyridin-4-ylmethanone |
—— |
C22H28F3N5O |
|
—— |
(4-methylthiadiazol-5-yl)-[4-[(5S,7R)-5-propan-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]methanone |
—— |
C19H25F3N6OS |
|
—— |
1-[(3S)-3-[(5S,7R)-2-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-3-phenylpropan-1-one |
—— |
C22H27F3N4O |
|
—— |
[4-[(5S,7R)-5-tert-butyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-pyridin-2-ylmethanone |
—— |
C22H28F3N5O |
|
—— |
1-[4-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-2-methylpropan-1-one |
—— |
C18H27F3N4O |
|
—— |
[(2R)-2-[(5S,7R)-5-propan-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-pyridin-2-ylmethanone |
—— |
C21H26F3N5O |
|
—— |
(4-methyl-1,3-thiazol-5-yl)-[4-[(5S,7R)-2-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]methanone |
—— |
C18H22F3N5OS |
|
—— |
[(3S)-1,1-dioxothiolan-3-yl]-[(2S)-2-[(5S,7R)-5-propan-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]methanone |
—— |
C19H27F3N4O3S |
|
—— |
[(1R,2S)-2-methylcyclopropyl]-[(2R)-2-[(5S,7R)-5-propan-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]methanone |
—— |
C20H29F3N4O |
|
—— |
(4-ethylthiadiazol-5-yl)-[(2S)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]methanone |
—— |
C18H23F3N6OS |
|
—— |
1-[(3R)-3-[(5S,7R)-7-(difluoromethyl)-2-methyl-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-3-(4-ethoxyphenyl)propan-1-one |
—— |
C24H32F2N4O2 |
|
—— |
(5R,7R)-5-ethyl-2-(1-pyrrolidin-1-ylsulfonylpiperidin-4-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine |
—— |
C18H28F3N5O2S |
|
—— |
[4-[(5S,7R)-5-tert-butyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-pyridin-3-ylmethanone |
—— |
C22H28F3N5O |
|
—— |
1-[(2R)-2-[(5S,7R)-5-tert-butyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-2-pyrazol-1-ylethanone |
—— |
C21H29F3N6O |
|
—— |
[(2R)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]-(3-methyl-1,2-oxazol-5-yl)methanone |
—— |
C18H22F3N5O2 |
|
—— |
1-[(3R)-3-[(5S,7R)-2-tert-butyl-7-(difluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-2-methylpropan-1-one |
—— |
C20H32F2N4O |
|
—— |
(3,5-dimethyl-1,2-oxazol-4-yl)-[(2R)-2-[(5R,7R)-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]methanone |
—— |
C18H22F3N5O2 |
|
—— |
(3R)-1-(4-ethyl-11,13-dimethyl-3,7,8,10-tetrazatricyclo[7.4.0.02,7]trideca-1,3,5,8,10,12-hexaen-6-yl)piperidin-3-ol |
—— |
C18H23N5O |
|
—— |
[(3S)-3-[(5S,7R)-2-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-pyridin-4-ylmethanone |
—— |
C19H22F3N5O |
|
—— |
[(1S,2S)-2-methylcyclopropyl]-[(2R)-2-[(5S,7R)-5-propan-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]methanone |
—— |
C20H29F3N4O |
|
—— |
[7-(difluoromethyl)-5-methylpyrazolo[1,5-a]pyrimidin-3-yl]-[(3R)-3-(5-fluorobenzotriazol-1-yl)piperidin-1-yl]methanone |
—— |
C20H18F3N7O |
|
—— |
3-methoxy-1-[(3R)-3-[(5S,7R)-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]propan-1-one |
—— |
C20H25F3N4O2S |
|
—— |
(2R)-1-[(3R)-3-[(5S,7R)-7-(difluoromethyl)-2-methyl-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-2-(3,5-dimethylphenoxy)propan-1-one |
—— |
C24H32F2N4O2 |
|
—— |
1-[(2R)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]-3-(3-methylpyrazol-1-yl)propan-1-one |
—— |
C20H27F3N6O |
|
—— |
5-[(3R)-1-[(2S)-3-(1,3-benzodioxol-5-yl)-2-methylpropyl]piperidin-3-yl]-2-methylpyrazolo[1,5-a]pyrimidin-7-amine |
—— |
C23H29N5O2 |
|
—— |
1-[4-[(5S,7R)-5-tert-butyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-2-[(2S)-oxolan-2-yl]ethanone |
—— |
C22H33F3N4O2 |
|
—— |
4-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]-N,N-dimethylpiperidine-1-sulfonamide |
—— |
C16H26F3N5O2S |
|
—— |
1-[4-[(5S,7R)-2-tert-butyl-7-(difluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-3-phenylpropan-1-one |
—— |
C25H34F2N4O |
|
—— |
(5S,7R)-2-(1-methylsulfonylpiperidin-4-yl)-5-propan-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine |
—— |
C16H25F3N4O2S |
|
—— |
1-[(3R)-3-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-2,2-dimethylpropan-1-one |
—— |
C19H29F3N4O |
|
—— |
[(3S)-3-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]-pyridin-4-ylmethanone |
—— |
C19H22F3N5O |
|
—— |
[(3S)-3-[(5S,7R)-5-tert-butyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]-pyrimidin-5-ylmethanone |
—— |
C20H25F3N6O |
|
—— |
2,2-dimethyl-1-[(3R)-3-[(5S,7R)-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]propan-1-one |
—— |
C21H27F3N4OS |
|
—— |
(5R,7R)-5-ethyl-2-(1-methylsulfonylpiperidin-4-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine |
—— |
C15H23F3N4O2S |
|
—— |
[4-[(5S,7R)-5-tert-butyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-(2-methylpyridin-3-yl)methanone |
—— |
C23H30F3N5O |
|