中文名称 |
英文名称 |
CAS号 |
化学式 |
结构式图片 |
—— |
1-[(2S)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]-3-(3-methylpyrazol-1-yl)propan-1-one |
—— |
C20H27F3N6O |
|
—— |
(4-methyl-1,3-thiazol-5-yl)-[(2R)-2-[(5R,7R)-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]methanone |
—— |
C17H20F3N5OS |
|
—— |
[(3R)-3-[(5S,7R)-2-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-pyridin-4-ylmethanone |
—— |
C19H22F3N5O |
|
—— |
1-[(3S)-3-[(5S,7R)-2-tert-butyl-7-(difluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-2-methylpropan-1-one |
—— |
C20H32F2N4O |
|
—— |
[(3R)-3-[(5S,7R)-2-tert-butyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-pyridin-4-ylmethanone |
—— |
C22H28F3N5O |
|
—— |
1-[(2R)-2-[(5S,7R)-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]butan-1-one |
—— |
C19H23F3N4OS |
|
—— |
[(3R)-3-[(5S,7R)-7-(difluoromethyl)-2-methyl-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-[(3R)-1,1-dioxothiolan-3-yl]methanone |
—— |
C18H26F2N4O3S |
|
—— |
cyclopropyl-[(3R)-3-[(5S,7R)-2-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]methanone |
—— |
C17H23F3N4O |
|
—— |
(3-ethyl-1,2-oxazol-5-yl)-[(3R)-3-[(5S,7R)-2-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]methanone |
—— |
C19H24F3N5O2 |
|
—— |
1-[4-[(3S)-3-[(5S,7R)-2-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-4-oxobutyl]pyrrolidin-2-one |
—— |
C21H30F3N5O2 |
|
—— |
1-methyl-5-[(3S)-3-[(5S,7R)-2-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidine-1-carbonyl]pyridin-2-one |
—— |
C20H24F3N5O2 |
|
—— |
(4S)-4-[(3R)-3-[(5S,7R)-2-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidine-1-carbonyl]-1-propan-2-ylpyrrolidin-2-one |
—— |
C21H30F3N5O2 |
|
—— |
[(3R)-3-[(5S,7R)-2-tert-butyl-7-(difluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-(2-methoxypyridin-4-yl)methanone |
—— |
C23H31F2N5O2 |
|
—— |
(3-ethyl-1,2-oxazol-5-yl)-[4-[(5S,7R)-2-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]methanone |
—— |
C19H24F3N5O2 |
|
—— |
(2,4-dimethylpyrimidin-5-yl)-[(2R)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]methanone |
—— |
C20H25F3N6O |
|
—— |
3-[(2R)-oxolan-2-yl]-1-[(2R)-2-[(5S,7R)-5-propan-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]propan-1-one |
—— |
C21H31F3N4O2 |
|
—— |
1-[(3R)-3-[(5S,7R)-2-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-3-phenylpropan-1-one |
—— |
C22H27F3N4O |
|
—— |
(4R)-4-[(3S)-3-[(5S,7R)-2-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidine-1-carbonyl]-1-propan-2-ylpyrrolidin-2-one |
—— |
C21H30F3N5O2 |
|
—— |
[(3S)-3-[(5S,7R)-7-(difluoromethyl)-2-methyl-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-(5-methylthiophen-3-yl)methanone |
—— |
C19H24F2N4OS |
|
—— |
1-[4-[(5S,7R)-2-tert-butyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-2-methylpropan-1-one |
—— |
C20H31F3N4O |
|
—— |
1-methyl-5-[(3R)-3-[(5S,7R)-2-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidine-1-carbonyl]pyridin-2-one |
—— |
C20H24F3N5O2 |
|
—— |
(5-ethyl-2,4-dimethylpyrazol-3-yl)-[(3R)-3-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]methanone |
—— |
C21H29F3N6O |
|
—— |
(4S)-4-[(3S)-3-[(5S,7R)-2-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidine-1-carbonyl]-1-propan-2-ylpyrrolidin-2-one |
—— |
C21H30F3N5O2 |
|
—— |
[(3S)-3-[(5S,7R)-2-tert-butyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-cyclopropylmethanone |
—— |
C20H29F3N4O |
|
—— |
(5S,7R)-5-propan-2-yl-2-[(2S)-1-pyrrolidin-1-ylsulfonylpyrrolidin-2-yl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine |
—— |
C18H28F3N5O2S |
|
—— |
[(3R)-3-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]-[(2R)-oxolan-2-yl]methanone |
—— |
C18H25F3N4O2 |
|
—— |
1-[(2R)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]-2-(4-methylpyrazol-1-yl)ethanone |
—— |
C19H25F3N6O |
|
—— |
[(3R)-3-[(5S,7R)-2-tert-butyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-cyclopentylmethanone |
—— |
C22H33F3N4O |
|
—— |
[(3S)-3-[(5S,7R)-7-(difluoromethyl)-2-methyl-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-[(3S)-1,1-dioxothiolan-3-yl]methanone |
—— |
C18H26F2N4O3S |
|
—— |
1-[(3S)-3-[(5S,7R)-7-(difluoromethyl)-2-methyl-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-2-(2-fluorophenoxy)ethanone |
—— |
C21H25F3N4O2 |
|
—— |
[(3S)-3-[(5S,7R)-2-tert-butyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-(1,3-thiazol-4-yl)methanone |
—— |
C20H26F3N5OS |
|
—— |
(3-methyl-1,2-oxazol-5-yl)-[(3S)-3-[(5S,7R)-2-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]methanone |
—— |
C18H22F3N5O2 |
|
—— |
1-[(2R)-2-[(5S,7R)-5-propan-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-3-pyrazol-1-ylpropan-1-one |
—— |
C21H29F3N6O |
|
—— |
cyclopropyl-[(3S)-3-[(5S,7R)-2-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]methanone |
—— |
C17H23F3N4O |
|
—— |
1-[(3S)-3-[(5S,7R)-7-(difluoromethyl)-2-methyl-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-3-(4-ethoxyphenyl)propan-1-one |
—— |
C24H32F2N4O2 |
|
—— |
[(3R)-1,1-dioxothiolan-3-yl]-[(2S)-2-[(5S,7R)-5-propan-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]methanone |
—— |
C19H27F3N4O3S |
|
—— |
1-[4-[(5S,7R)-5-tert-butyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]butan-1-one |
—— |
C20H31F3N4O |
|
—— |
1-[4-[(5S,7R)-5-tert-butyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-2-pyrazol-1-ylethanone |
—— |
C21H29F3N6O |
|
—— |
1-[4-[(3R)-3-[(5S,7R)-2-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-4-oxobutyl]pyrrolidin-2-one |
—— |
C21H30F3N5O2 |
|
—— |
2-[(2R)-oxolan-2-yl]-1-[(2R)-2-[(5S,7R)-5-propan-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]ethanone |
—— |
C20H29F3N4O2 |
|
—— |
1-[(3R)-3-[(5S,7R)-7-(difluoromethyl)-2-methyl-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-2-(2-fluorophenoxy)ethanone |
—— |
C21H25F3N4O2 |
|
—— |
(2R)-1-[(3S)-3-[(5S,7R)-7-(difluoromethyl)-2-methyl-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-2-(3,5-dimethylphenoxy)propan-1-one |
—— |
C24H32F2N4O2 |
|
—— |
(4,5-dimethylthiophen-3-yl)-[(3R)-3-[(5S,7R)-2-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]methanone |
—— |
C20H25F3N4OS |
|
—— |
1-methyl-4-[(3S)-3-[(5S,7R)-2-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidine-1-carbonyl]pyridin-2-one |
—— |
C20H24F3N5O2 |
|
—— |
1-methyl-4-[(3R)-3-[(5S,7R)-2-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidine-1-carbonyl]pyridin-2-one |
—— |
C20H24F3N5O2 |
|
—— |
(3,5-dimethyl-1,2-oxazol-4-yl)-[(2S)-2-[(5R,7R)-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]methanone |
—— |
C18H22F3N5O2 |
|
—— |
[(2R)-2-[(5R,7R)-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-pyridin-4-ylmethanone |
—— |
C19H22F3N5O |
|
—— |
[(3R)-3-[(5S,7R)-7-(difluoromethyl)-2-methyl-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-[(3S)-1,1-dioxothiolan-3-yl]methanone |
—— |
C18H26F2N4O3S |
|
—— |
[(2R)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]-(4-methylthiadiazol-5-yl)methanone |
—— |
C17H21F3N6OS |
|
—— |
(4-methylthiadiazol-5-yl)-[(2R)-2-[(5R,7R)-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]methanone |
—— |
C16H19F3N6OS |
|