中文名称 |
英文名称 |
CAS号 |
化学式 |
结构式图片 |
—— |
[(3R)-3-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-pyridin-2-ylmethanone |
—— |
C20H24F3N5O |
|
—— |
1-[2-[(2R)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]-2-oxoethyl]pyrimidine-2,4-dione |
—— |
C19H23F3N6O3 |
|
—— |
4-[(3S)-3-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidine-1-carbonyl]-1-methylpyridin-2-one |
—— |
C21H26F3N5O2 |
|
—— |
1-[(2R)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]-2-pyridin-2-ylethanone |
—— |
C20H24F3N5O |
|
—— |
(5R,7R)-5-ethyl-2-[(2R)-1-pyrrolidin-1-ylsulfonylpiperidin-2-yl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine |
—— |
C18H28F3N5O2S |
|
—— |
[(2S)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-(3-methylpyridin-4-yl)methanone |
—— |
C21H26F3N5O |
|
—— |
[(2R)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]-(1H-pyrazol-5-yl)methanone |
—— |
C17H21F3N6O |
|
—— |
[(2R)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-(5-propan-2-yl-1,2-oxazol-3-yl)methanone |
—— |
C21H28F3N5O2 |
|
—— |
(4S)-4-[(2R)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidine-1-carbonyl]-1-methylpyrrolidin-2-one |
—— |
C20H28F3N5O2 |
|
—— |
4-[(2S)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidine-1-carbonyl]-1-methylpyridin-2-one |
—— |
C21H26F3N5O2 |
|
—— |
[(2R)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-(3-propan-2-yl-1,2-oxazol-5-yl)methanone |
—— |
C21H28F3N5O2 |
|
—— |
[(2R)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]-(1-methylpyrazol-3-yl)methanone |
—— |
C18H23F3N6O |
|
—— |
1-[2-[(2S)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]-2-oxoethyl]pyrimidine-2,4-dione |
—— |
C19H23F3N6O3 |
|
—— |
[(2S)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]-(1-methylpyrazol-3-yl)methanone |
—— |
C18H23F3N6O |
|
—— |
[(3R)-1,1-dioxothiolan-3-yl]-[(2S)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]methanone |
—— |
C18H25F3N4O3S |
|
—— |
4-[(2S)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidine-1-carbonyl]-1-methylpyridin-2-one |
—— |
C20H24F3N5O2 |
|
—— |
[(2R)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-(5-methoxythiophen-2-yl)methanone |
—— |
C20H25F3N4O2S |
|
—— |
(4S)-4-[(2R)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidine-1-carbonyl]-1-methylpyrrolidin-2-one |
—— |
C19H26F3N5O2 |
|
—— |
5-[(3S)-3-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidine-1-carbonyl]-1H-pyridin-2-one |
—— |
C20H24F3N5O2 |
|
—— |
(5R,7R)-5-ethyl-2-[(3S)-1-[(2-methylpyrimidin-5-yl)methyl]piperidin-3-yl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine |
—— |
C20H27F3N6 |
|
—— |
(4R)-4-[(2R)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidine-1-carbonyl]-1-methylpyrrolidin-2-one |
—— |
C20H28F3N5O2 |
|
—— |
[(2S)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-(1-methylpyrazol-3-yl)methanone |
—— |
C19H25F3N6O |
|
—— |
[(2R)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-(1-methylpyrazol-4-yl)methanone |
—— |
C19H25F3N6O |
|
—— |
[(2S)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-(3-propan-2-yl-1,2-oxazol-5-yl)methanone |
—— |
C21H28F3N5O2 |
|
—— |
[(2R)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-(2-methoxypyridin-4-yl)methanone |
—— |
C21H26F3N5O2 |
|
—— |
(4R)-4-[(2S)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidine-1-carbonyl]-1-methylpyrrolidin-2-one |
—— |
C19H26F3N5O2 |
|
—— |
[(2S)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-(2-methoxypyridin-4-yl)methanone |
—— |
C21H26F3N5O2 |
|
—— |
(2R)-1-[(2R)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]-2-(5-methylpyrazol-1-yl)propan-1-one |
—— |
C20H27F3N6O |
|
—— |
cyclohexyl-[(3R)-3-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]methanone |
—— |
C21H31F3N4O |
|
—— |
4-[(2R)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidine-1-carbonyl]-1-methylpyridin-2-one |
—— |
C21H26F3N5O2 |
|
—— |
[(2S)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-(1,3-thiazol-4-yl)methanone |
—— |
C18H22F3N5OS |
|
—— |
(5R,7R)-5-ethyl-2-[(2S)-1-pyrrolidin-1-ylsulfonylpiperidin-2-yl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine |
—— |
C18H28F3N5O2S |
|
—— |
[(2S)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-(5-propan-2-yl-1H-pyrazol-3-yl)methanone |
—— |
C21H29F3N6O |
|
—— |
[(2R)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-(5-methylpyrazin-2-yl)methanone |
—— |
C20H25F3N6O |
|
—— |
[(2S)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-(5-methoxythiophen-2-yl)methanone |
—— |
C20H25F3N4O2S |
|
—— |
[(2S)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-(5-propan-2-yl-1,2-oxazol-3-yl)methanone |
—— |
C21H28F3N5O2 |
|
—— |
[(2S)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-[(2R)-oxolan-2-yl]methanone |
—— |
C19H27F3N4O2 |
|
—— |
1-[(2S)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-2-methoxyethanone |
—— |
C17H25F3N4O2 |
|
—— |
[(2S)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-(4-methylthiadiazol-5-yl)methanone |
—— |
C18H23F3N6OS |
|
—— |
[(2R)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-(4-methylthiadiazol-5-yl)methanone |
—— |
C18H23F3N6OS |
|
—— |
[(2R)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-[(2S)-oxolan-2-yl]methanone |
—— |
C19H27F3N4O2 |
|
—— |
[(2S)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-(4-methyl-1,2,5-oxadiazol-3-yl)methanone |
—— |
C18H23F3N6O2 |
|
—— |
(2,4-dimethyl-1,3-thiazol-5-yl)-[(2S)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]methanone |
—— |
C20H26F3N5OS |
|
—— |
(2,4-dimethyl-1,3-thiazol-5-yl)-[(2R)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]methanone |
—— |
C20H26F3N5OS |
|
—— |
1-[(2R)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-2-methoxyethanone |
—— |
C17H25F3N4O2 |
|
—— |
[(2S)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-[(2S)-oxolan-2-yl]methanone |
—— |
C19H27F3N4O2 |
|
—— |
(4S)-4-[(2S)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidine-1-carbonyl]-1-methylpyrrolidin-2-one |
—— |
C20H28F3N5O2 |
|
—— |
(5S,7R)-2-[(2R)-1-ethylsulfonylpiperidin-2-yl]-5-propan-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine |
—— |
C17H27F3N4O2S |
|
—— |
(5R,7R)-2-(1-ethylsulfonylpiperidin-4-yl)-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine |
—— |
C15H23F3N4O2S |
|
—— |
(5S,7R)-5-tert-butyl-2-[(2S)-1-ethylsulfonylpiperidin-2-yl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine |
—— |
C18H29F3N4O2S |
|