中文名称 |
英文名称 |
CAS号 |
化学式 |
结构式图片 |
—— |
1-[(2R)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]-2-methoxyethanone |
—— |
C16H23F3N4O2 |
|
—— |
[(3S)-3-[(5S,7R)-5-propan-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]-pyrimidin-5-ylmethanone |
—— |
C19H23F3N6O |
|
—— |
1-[(2S)-2-[(5S,7R)-5-tert-butyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-2-pyrazol-1-ylethanone |
—— |
C21H29F3N6O |
|
—— |
2-(2-fluorophenoxy)-1-[4-[(5S,7R)-2-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]ethanone |
—— |
C21H24F4N4O2 |
|
—— |
[(3R)-3-[(5S,7R)-2-tert-butyl-7-(difluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-pyridin-4-ylmethanone |
—— |
C22H29F2N5O |
|
—— |
[(3S)-3-[(5S,7R)-2-tert-butyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-pyridin-4-ylmethanone |
—— |
C22H28F3N5O |
|
—— |
1-[(3S)-3-[(5S,7R)-2-tert-butyl-7-(difluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-3-(1,2-oxazol-5-yl)propan-1-one |
—— |
C22H31F2N5O2 |
|
—— |
[(3R)-3-[(5S,7R)-2-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-pyridin-3-ylmethanone |
—— |
C19H22F3N5O |
|
—— |
[(3S)-3-[(5S,7R)-7-(difluoromethyl)-2-methyl-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-[(3R)-1,1-dioxothiolan-3-yl]methanone |
—— |
C18H26F2N4O3S |
|
—— |
5-[4-[(5S,7R)-2-tert-butyl-7-(difluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidine-1-carbonyl]-1-methylpyridin-2-one |
—— |
C23H31F2N5O2 |
|
—— |
2-[(2S)-oxolan-2-yl]-1-[(2R)-2-[(5S,7R)-5-propan-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]ethanone |
—— |
C20H29F3N4O2 |
|
—— |
[(3R)-3-[(5S,7R)-5-tert-butyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]-(2-methylpyrazol-3-yl)methanone |
—— |
C20H27F3N6O |
|
—— |
(4,5-dimethylthiophen-2-yl)-[4-[(5S,7R)-2-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]methanone |
—— |
C20H25F3N4OS |
|
—— |
[(2S)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]-(3-methyl-1,2-oxazol-5-yl)methanone |
—— |
C18H22F3N5O2 |
|
—— |
cyclopropyl-[(2R)-2-[(5R,7R)-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]methanone |
—— |
C16H21F3N4O |
|
—— |
[(3R)-1,1-dioxothiolan-3-yl]-[(2R)-2-[(5S,7R)-5-propan-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]methanone |
—— |
C19H27F3N4O3S |
|
—— |
[(2S)-2-[(5R,7R)-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-pyridin-4-ylmethanone |
—— |
C19H22F3N5O |
|
—— |
cyclopropyl-[(2S)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]methanone |
—— |
C17H23F3N4O |
|
—— |
(2-methoxypyridin-4-yl)-[(2S)-2-[(5S,7R)-5-propan-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]methanone |
—— |
C21H26F3N5O2 |
|
—— |
(1,3-dimethylpyrazol-4-yl)-[(2R)-2-[(5S,7R)-5-propan-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]methanone |
—— |
C20H27F3N6O |
|
—— |
cyclohexyl-[(3R)-3-[(5S,7R)-2-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]methanone |
—— |
C20H29F3N4O |
|
—— |
(4-methyl-1,3-thiazol-5-yl)-[(2R)-2-[(5S,7R)-5-propan-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]methanone |
—— |
C19H24F3N5OS |
|
—— |
(5-ethyl-3-methyl-1,2-oxazol-4-yl)-[(2S)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]methanone |
—— |
C20H26F3N5O2 |
|
—— |
[(3R)-3-[(5S,7R)-2-tert-butyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-cyclopropylmethanone |
—— |
C20H29F3N4O |
|
—— |
[4-[(5S,7R)-2-tert-butyl-7-(difluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-(6-methylpyridin-3-yl)methanone |
—— |
C23H31F2N5O |
|
—— |
(3-ethyl-1,2-oxazol-5-yl)-[(3S)-3-[(5S,7R)-2-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]methanone |
—— |
C19H24F3N5O2 |
|
—— |
(2,4-dimethyl-1,3-oxazol-5-yl)-[4-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]methanone |
—— |
C20H26F3N5O2 |
|
—— |
3-[(2R)-oxolan-2-yl]-1-[(2S)-2-[(5S,7R)-5-propan-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]propan-1-one |
—— |
C21H31F3N4O2 |
|
—— |
[(3S)-3-[(5S,7R)-2-tert-butyl-7-(difluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-pyridin-4-ylmethanone |
—— |
C22H29F2N5O |
|
—— |
3-cyclopentyl-1-[4-[(5S,7R)-7-(difluoromethyl)-2-methyl-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]propan-1-one |
—— |
C21H32F2N4O |
|
—— |
1-[(2S)-2-[(5S,7R)-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]butan-1-one |
—— |
C19H23F3N4OS |
|
—— |
3-[(2S)-oxolan-2-yl]-1-[(2R)-2-[(5S,7R)-5-propan-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]propan-1-one |
—— |
C21H31F3N4O2 |
|
—— |
ethyl (5R,7S)-5-[(3S)-1-(3,6-dihydro-2H-pyran-5-ylmethyl)piperidin-3-yl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxylate |
—— |
C21H29F3N4O3 |
|
—— |
5-[(2S)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidine-1-carbonyl]-1-methylpyridin-2-one |
—— |
C20H24F3N5O2 |
|
—— |
(4-methyl-1,3-thiazol-5-yl)-[(2S)-2-[(5S,7R)-5-propan-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]methanone |
—— |
C19H24F3N5OS |
|
—— |
(4R)-4-[4-[(5S,7R)-2-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidine-1-carbonyl]-1-prop-2-enylpyrrolidin-2-one |
—— |
C21H28F3N5O2 |
|
—— |
[(2S)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]-(4-methyl-1,3-thiazol-5-yl)methanone |
—— |
C18H22F3N5OS |
|
—— |
4-[(3R)-3-[(5S,7R)-2-tert-butyl-7-(difluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidine-1-carbonyl]-1-methylpyridin-2-one |
—— |
C23H31F2N5O2 |
|
—— |
1-[4-[4-[(5S,7R)-2-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-4-oxobutyl]pyrrolidin-2-one |
—— |
C21H30F3N5O2 |
|
—— |
(2-methoxypyridin-4-yl)-[(2R)-2-[(5S,7R)-5-propan-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]methanone |
—— |
C21H26F3N5O2 |
|
—— |
1-[4-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]butan-1-one |
—— |
C18H27F3N4O |
|
—— |
(1,3-dimethylpyrazol-4-yl)-[(2S)-2-[(5S,7R)-5-propan-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]methanone |
—— |
C20H27F3N6O |
|
—— |
1-[4-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-2,2-dimethylpropan-1-one |
—— |
C19H29F3N4O |
|
—— |
3-[(2S)-oxolan-2-yl]-1-[(2S)-2-[(5S,7R)-5-propan-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]propan-1-one |
—— |
C21H31F3N4O2 |
|
—— |
(5R,7R)-5-ethyl-2-(1-prop-2-enylsulfonylpiperidin-4-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine |
—— |
C17H25F3N4O2S |
|
—— |
ethyl (5R,7S)-5-[(3R)-1-(3,6-dihydro-2H-pyran-5-ylmethyl)piperidin-3-yl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxylate |
—— |
C21H29F3N4O3 |
|
—— |
2-(4-methyl-1,2,5-oxadiazol-3-yl)-1-[(2S)-2-[(5S,7R)-5-propan-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]ethanone |
—— |
C19H25F3N6O2 |
|
—— |
2-[(2S)-oxolan-2-yl]-1-[(2S)-2-[(5S,7R)-5-propan-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]ethanone |
—— |
C20H29F3N4O2 |
|
—— |
(1-methylpyrazol-3-yl)-[(2R)-2-[(5S,7R)-5-propan-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]methanone |
—— |
C19H25F3N6O |
|
—— |
[(2S)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]-(2-methylpyrazol-3-yl)methanone |
—— |
C18H23F3N6O |
|