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吡唑并嘧啶类

中文名称 英文名称 CAS号 化学式 结构式图片
—— (7R)-5-(4-bromophenyl)-7-(2-fluorophenyl)-N-(4-fluorophenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C25H17BrF2N4O
(7R)-5-(4-bromophenyl)-7-(2-fluorophenyl)-N-(4-fluorophenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (7R)-7-(2-chlorophenyl)-N-(4-fluorophenyl)-5-(3-methoxyphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C26H20ClFN4O2
(7R)-7-(2-chlorophenyl)-N-(4-fluorophenyl)-5-(3-methoxyphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (7S)-5-(4-ethylphenyl)-7-(3-methoxyphenyl)-N-(4-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C29H28N4O2
(7S)-5-(4-ethylphenyl)-7-(3-methoxyphenyl)-N-(4-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (7R)-7-(4-chlorophenyl)-5-(3-methoxyphenyl)-N-(4-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C27H23ClN4O2
(7R)-7-(4-chlorophenyl)-5-(3-methoxyphenyl)-N-(4-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (7R)-7-(2-chlorophenyl)-N,5-bis(4-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C27H23ClN4O
(7R)-7-(2-chlorophenyl)-N,5-bis(4-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (7S)-7-(2-chlorophenyl)-N,5-bis(4-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C27H23ClN4O
(7S)-7-(2-chlorophenyl)-N,5-bis(4-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (7S)-7-(4-chlorophenyl)-5-(3-methoxyphenyl)-N-(4-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C27H23ClN4O2
(7S)-7-(4-chlorophenyl)-5-(3-methoxyphenyl)-N-(4-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (7R)-5-(3-methoxyphenyl)-7-(4-methoxyphenyl)-N-(4-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C28H26N4O3
(7R)-5-(3-methoxyphenyl)-7-(4-methoxyphenyl)-N-(4-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (7S)-5-(4-ethylphenyl)-N-(4-fluorophenyl)-7-(3-methoxyphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C28H25FN4O2
(7S)-5-(4-ethylphenyl)-N-(4-fluorophenyl)-7-(3-methoxyphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (7S)-7-(2-chlorophenyl)-N-(4-fluorophenyl)-5-(3-methoxyphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C26H20ClFN4O2
(7S)-7-(2-chlorophenyl)-N-(4-fluorophenyl)-5-(3-methoxyphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (7S)-5-(4-chlorophenyl)-7-(2-fluorophenyl)-N-(4-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C26H20ClFN4O
(7S)-5-(4-chlorophenyl)-7-(2-fluorophenyl)-N-(4-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (2S)-N-(4-bromo-2-fluorophenyl)-2-(4-methyl-2-oxopyrimido[1,2-b]indazol-6-yl)butanamide —— C21H18BrFN4O2
(2S)-N-(4-bromo-2-fluorophenyl)-2-(4-methyl-2-oxopyrimido[1,2-b]indazol-6-yl)butanamide
—— (2S)-2-(4-methyl-2-oxopyrimido[1,2-b]indazol-6-yl)-N-(2,3,5,6-tetrafluorophenyl)propanamide —— C20H14F4N4O2
(2S)-2-(4-methyl-2-oxopyrimido[1,2-b]indazol-6-yl)-N-(2,3,5,6-tetrafluorophenyl)propanamide
—— (2R)-N-[4-(diethylamino)-2-methylphenyl]-2-(4-methyl-2-oxopyrimido[1,2-b]indazol-6-yl)butanamide —— C26H31N5O2
(2R)-N-[4-(diethylamino)-2-methylphenyl]-2-(4-methyl-2-oxopyrimido[1,2-b]indazol-6-yl)butanamide
—— (2S)-N-[4-(diethylamino)-2-methylphenyl]-2-(4-methyl-2-oxopyrimido[1,2-b]indazol-6-yl)butanamide —— C26H31N5O2
(2S)-N-[4-(diethylamino)-2-methylphenyl]-2-(4-methyl-2-oxopyrimido[1,2-b]indazol-6-yl)butanamide
—— (7R)-7-(4-bromophenyl)-N-(4-fluorophenyl)-5-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C25H18BrFN4O
(7R)-7-(4-bromophenyl)-N-(4-fluorophenyl)-5-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (7R)-7-(2-fluorophenyl)-N,5-bis(4-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C27H23FN4O
(7R)-7-(2-fluorophenyl)-N,5-bis(4-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (2R)-N-[2-(N-ethylanilino)ethyl]-2-(4-methyl-2-oxopyrimido[1,2-b]indazol-6-yl)butanamide —— C25H29N5O2
(2R)-N-[2-(N-ethylanilino)ethyl]-2-(4-methyl-2-oxopyrimido[1,2-b]indazol-6-yl)butanamide
—— (2R)-N-[3-(3-chlorophenyl)-1,2-oxazol-5-yl]-2-(4-methyl-2-oxopyrimido[1,2-b]indazol-6-yl)butanamide —— C24H20ClN5O3
(2R)-N-[3-(3-chlorophenyl)-1,2-oxazol-5-yl]-2-(4-methyl-2-oxopyrimido[1,2-b]indazol-6-yl)butanamide
—— (2R)-2-(4-methyl-2-oxopyrimido[1,2-b]indazol-6-yl)-N-(2,3,4,5,6-pentafluorophenyl)butanamide —— C21H15F5N4O2
(2R)-2-(4-methyl-2-oxopyrimido[1,2-b]indazol-6-yl)-N-(2,3,4,5,6-pentafluorophenyl)butanamide
—— (2S)-N-[2-(N-ethylanilino)ethyl]-2-(4-methyl-2-oxopyrimido[1,2-b]indazol-6-yl)butanamide —— C25H29N5O2
(2S)-N-[2-(N-ethylanilino)ethyl]-2-(4-methyl-2-oxopyrimido[1,2-b]indazol-6-yl)butanamide
—— (2S)-N-[(2-bromophenyl)methyl]-2-(4-methyl-2-oxopyrimido[1,2-b]indazol-6-yl)butanamide —— C22H21BrN4O2
(2S)-N-[(2-bromophenyl)methyl]-2-(4-methyl-2-oxopyrimido[1,2-b]indazol-6-yl)butanamide
—— (2S)-N-[3-(3-chlorophenyl)-1,2-oxazol-5-yl]-2-(4-methyl-2-oxopyrimido[1,2-b]indazol-6-yl)butanamide —— C24H20ClN5O3
(2S)-N-[3-(3-chlorophenyl)-1,2-oxazol-5-yl]-2-(4-methyl-2-oxopyrimido[1,2-b]indazol-6-yl)butanamide
—— (2R)-N-(4-bromo-3-methylphenyl)-2-(4-methyl-2-oxopyrimido[1,2-b]indazol-6-yl)butanamide —— C22H21BrN4O2
(2R)-N-(4-bromo-3-methylphenyl)-2-(4-methyl-2-oxopyrimido[1,2-b]indazol-6-yl)butanamide
—— (2R)-N-(4-bromo-2-fluorophenyl)-2-(4-methyl-2-oxopyrimido[1,2-b]indazol-6-yl)butanamide —— C21H18BrFN4O2
(2R)-N-(4-bromo-2-fluorophenyl)-2-(4-methyl-2-oxopyrimido[1,2-b]indazol-6-yl)butanamide
—— (2S)-N-(2-bromophenyl)-2-(4-methyl-2-oxopyrimido[1,2-b]indazol-6-yl)butanamide —— C21H19BrN4O2
(2S)-N-(2-bromophenyl)-2-(4-methyl-2-oxopyrimido[1,2-b]indazol-6-yl)butanamide
—— (2S)-N-(2-bromo-4,6-difluorophenyl)-2-(4-methyl-2-oxopyrimido[1,2-b]indazol-6-yl)butanamide —— C21H17BrF2N4O2
(2S)-N-(2-bromo-4,6-difluorophenyl)-2-(4-methyl-2-oxopyrimido[1,2-b]indazol-6-yl)butanamide
—— (2S)-N-[(3-bromophenyl)methyl]-2-(4-methyl-2-oxopyrimido[1,2-b]indazol-6-yl)propanamide —— C21H19BrN4O2
(2S)-N-[(3-bromophenyl)methyl]-2-(4-methyl-2-oxopyrimido[1,2-b]indazol-6-yl)propanamide
—— (2S)-N-(4-bromo-3-methylphenyl)-2-(4-methyl-2-oxopyrimido[1,2-b]indazol-6-yl)butanamide —— C22H21BrN4O2
(2S)-N-(4-bromo-3-methylphenyl)-2-(4-methyl-2-oxopyrimido[1,2-b]indazol-6-yl)butanamide
—— (2R)-N-[(2-bromophenyl)methyl]-2-(4-methyl-2-oxopyrimido[1,2-b]indazol-6-yl)propanamide —— C21H19BrN4O2
(2R)-N-[(2-bromophenyl)methyl]-2-(4-methyl-2-oxopyrimido[1,2-b]indazol-6-yl)propanamide
—— (2S)-N-(5-chloro-2-methoxyphenyl)-2-(4-methyl-2-oxopyrimido[1,2-b]indazol-6-yl)butanamide —— C22H21ClN4O3
(2S)-N-(5-chloro-2-methoxyphenyl)-2-(4-methyl-2-oxopyrimido[1,2-b]indazol-6-yl)butanamide
—— (2R)-N-[(3-bromophenyl)methyl]-2-(4-methyl-2-oxopyrimido[1,2-b]indazol-6-yl)butanamide —— C22H21BrN4O2
(2R)-N-[(3-bromophenyl)methyl]-2-(4-methyl-2-oxopyrimido[1,2-b]indazol-6-yl)butanamide
—— (7S)-7-(2-fluorophenyl)-N,5-bis(4-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C27H23FN4O
(7S)-7-(2-fluorophenyl)-N,5-bis(4-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (2R)-N-[2-[[(2R)-butan-2-yl]-cyclohexylamino]ethyl]-2-(4-methyl-2-oxopyrimido[1,2-b]indazol-6-yl)butanamide —— C27H39N5O2
(2R)-N-[2-[[(2R)-butan-2-yl]-cyclohexylamino]ethyl]-2-(4-methyl-2-oxopyrimido[1,2-b]indazol-6-yl)butanamide
—— (7R)-7-(2-chlorophenyl)-N-(4-fluorophenyl)-5-(4-methoxyphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C26H20ClFN4O2
(7R)-7-(2-chlorophenyl)-N-(4-fluorophenyl)-5-(4-methoxyphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (2R)-N-[(2-bromophenyl)methyl]-2-(4-methyl-2-oxopyrimido[1,2-b]indazol-6-yl)butanamide —— C22H21BrN4O2
(2R)-N-[(2-bromophenyl)methyl]-2-(4-methyl-2-oxopyrimido[1,2-b]indazol-6-yl)butanamide
—— (2R)-N-[(3-bromophenyl)methyl]-2-(4-methyl-2-oxopyrimido[1,2-b]indazol-6-yl)propanamide —— C21H19BrN4O2
(2R)-N-[(3-bromophenyl)methyl]-2-(4-methyl-2-oxopyrimido[1,2-b]indazol-6-yl)propanamide
—— (2S)-N-[(2-bromophenyl)methyl]-2-(4-methyl-2-oxopyrimido[1,2-b]indazol-6-yl)propanamide —— C21H19BrN4O2
(2S)-N-[(2-bromophenyl)methyl]-2-(4-methyl-2-oxopyrimido[1,2-b]indazol-6-yl)propanamide
—— (2S)-N-[(5-bromo-2-methoxyphenyl)methyl]-2-(4-methyl-2-oxopyrimido[1,2-b]indazol-6-yl)propanamide —— C22H21BrN4O3
(2S)-N-[(5-bromo-2-methoxyphenyl)methyl]-2-(4-methyl-2-oxopyrimido[1,2-b]indazol-6-yl)propanamide
—— (2R)-N-[(5-bromo-2-methoxyphenyl)methyl]-2-(4-methyl-2-oxopyrimido[1,2-b]indazol-6-yl)propanamide —— C22H21BrN4O3
(2R)-N-[(5-bromo-2-methoxyphenyl)methyl]-2-(4-methyl-2-oxopyrimido[1,2-b]indazol-6-yl)propanamide
—— (7R)-6-N-(2-methoxyphenyl)-5-methyl-3-N-(3-methylphenyl)-7-(4-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide —— C30H29N5O3
(7R)-6-N-(2-methoxyphenyl)-5-methyl-3-N-(3-methylphenyl)-7-(4-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide
—— (7R)-6-N-(2,4-dimethylphenyl)-5-methyl-3-N-(3-methylphenyl)-7-(4-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide —— C31H31N5O2
(7R)-6-N-(2,4-dimethylphenyl)-5-methyl-3-N-(3-methylphenyl)-7-(4-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide
—— (7S)-6-N-(4-methoxyphenyl)-5-methyl-3-N,7-bis(3-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide —— C30H29N5O3
(7S)-6-N-(4-methoxyphenyl)-5-methyl-3-N,7-bis(3-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide
—— (7S)-3-N-(4-fluorophenyl)-7-(2-methoxyphenyl)-5-methyl-6-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide —— C28H24FN5O3
(7S)-3-N-(4-fluorophenyl)-7-(2-methoxyphenyl)-5-methyl-6-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide
—— (7S)-7-(3-chlorophenyl)-6-N-(2,4-dimethylphenyl)-5-methyl-3-N-(4-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide —— C30H28ClN5O2
(7S)-7-(3-chlorophenyl)-6-N-(2,4-dimethylphenyl)-5-methyl-3-N-(4-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide
—— (7R)-6-N-(4-methoxyphenyl)-5-methyl-3-N,7-bis(4-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide —— C30H29N5O3
(7R)-6-N-(4-methoxyphenyl)-5-methyl-3-N,7-bis(4-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide
—— (7R)-6-N-(2,4-dimethylphenyl)-7-(4-fluorophenyl)-5-methyl-3-N-(3-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide —— C30H28FN5O2
(7R)-6-N-(2,4-dimethylphenyl)-7-(4-fluorophenyl)-5-methyl-3-N-(3-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide
—— (7S)-7-(4-chlorophenyl)-5-methyl-3-N-(4-methylphenyl)-6-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide —— C28H24ClN5O2
(7S)-7-(4-chlorophenyl)-5-methyl-3-N-(4-methylphenyl)-6-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide
—— (7R)-6-N-(2-methoxyphenyl)-7-(4-methoxyphenyl)-5-methyl-3-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide —— C29H27N5O4
(7R)-6-N-(2-methoxyphenyl)-7-(4-methoxyphenyl)-5-methyl-3-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide
—— (7S)-5-methyl-3-N-(3-methylphenyl)-7-(4-methylphenyl)-6-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide —— C29H27N5O2
(7S)-5-methyl-3-N-(3-methylphenyl)-7-(4-methylphenyl)-6-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide