中文名称 |
英文名称 |
CAS号 |
化学式 |
结构式图片 |
—— |
1-[(3R)-3-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-2-pyrazol-1-ylethanone |
—— |
C19H25F3N6O |
|
—— |
[(3R)-3-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-(2-methoxypyridin-4-yl)methanone |
—— |
C21H26F3N5O2 |
|
—— |
(4,5-dimethylthiophen-2-yl)-[(3S)-3-[(5R,7R)-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]methanone |
—— |
C20H25F3N4OS |
|
—— |
(3R)-1-(4-ethyl-11,13-dimethyl-3,7,8,10-tetrazatricyclo[7.4.0.02,7]trideca-1,3,5,8,10,12-hexaen-6-yl)piperidine-3-carboxamide |
—— |
C19H24N6O |
|
—— |
(3S)-1-(4-ethyl-11,13-dimethyl-3,7,8,10-tetrazatricyclo[7.4.0.02,7]trideca-1,3,5,8,10,12-hexaen-6-yl)piperidine-3-carboxamide |
—— |
C19H24N6O |
|
—— |
[(3S)-3-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-pyridin-3-ylmethanone |
—— |
C20H24F3N5O |
|
—— |
cyclohexyl-[(3R)-3-[(5R,7R)-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]methanone |
—— |
C20H29F3N4O |
|
—— |
[(3S)-3-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-(3-methylpyridin-4-yl)methanone |
—— |
C21H26F3N5O |
|
—— |
(4,5-dimethylthiophen-2-yl)-[(3R)-3-[(5R,7R)-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]methanone |
—— |
C20H25F3N4OS |
|
—— |
(2,4-dimethyl-1,3-thiazol-5-yl)-[(3S)-3-[(5R,7R)-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]methanone |
—— |
C19H24F3N5OS |
|
—— |
[(3S)-3-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-(1-methylpyrazol-4-yl)methanone |
—— |
C19H25F3N6O |
|
—— |
2,2-dimethyl-1-[(3S)-3-[(5S,7R)-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]propan-1-one |
—— |
C21H27F3N4OS |
|
—— |
[(3R)-3-[(5S,7R)-5-tert-butyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-pyridin-4-ylmethanone |
—— |
C22H28F3N5O |
|
—— |
cyclohexyl-[(3S)-3-[(5R,7R)-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]methanone |
—— |
C20H29F3N4O |
|
—— |
1-[(3S)-3-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-2-pyrazol-1-ylethanone |
—— |
C19H25F3N6O |
|
—— |
[(3R)-3-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-(1-methylpyrazol-4-yl)methanone |
—— |
C19H25F3N6O |
|
—— |
[(3R)-3-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-pyridin-3-ylmethanone |
—— |
C20H24F3N5O |
|
—— |
[(3S)-3-[(5S,7R)-5-tert-butyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-pyridin-3-ylmethanone |
—— |
C22H28F3N5O |
|
—— |
[(3R)-3-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-(2-methoxypyrimidin-5-yl)methanone |
—— |
C20H25F3N6O2 |
|
—— |
2-(3,5-dimethylpyrazol-1-yl)-1-[(3S)-3-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]ethanone |
—— |
C21H29F3N6O |
|
—— |
2-(3,5-dimethylpyrazol-1-yl)-1-[(3R)-3-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]ethanone |
—— |
C21H29F3N6O |
|
—— |
1-[(3S)-3-[(5S,7R)-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]butan-1-one |
—— |
C20H25F3N4OS |
|
—— |
[(3R)-3-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-(3-methylpyridin-4-yl)methanone |
—— |
C21H26F3N5O |
|
—— |
(2,4-dimethyl-1,3-thiazol-5-yl)-[(3R)-3-[(5R,7R)-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]methanone |
—— |
C19H24F3N5OS |
|
—— |
1-[(3S)-3-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-2,2-dimethylpropan-1-one |
—— |
C19H29F3N4O |
|
—— |
2-methoxy-1-[(3R)-3-[(5S,7R)-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]ethanone |
—— |
C19H23F3N4O2S |
|
—— |
[(3S)-3-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-(2-methoxypyridin-4-yl)methanone |
—— |
C21H26F3N5O2 |
|
—— |
(1,5-dimethylpyrazol-4-yl)-[4-[(5S,7R)-5-propan-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]methanone |
—— |
C21H29F3N6O |
|
—— |
1-[(3R)-3-[(5S,7R)-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]butan-1-one |
—— |
C20H25F3N4OS |
|
—— |
(5S,7R)-5-propan-2-yl-2-(1-pyrrolidin-1-ylsulfonylpiperidin-4-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine |
—— |
C19H30F3N5O2S |
|
—— |
3-methoxy-1-[(3S)-3-[(5S,7R)-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]propan-1-one |
—— |
C20H25F3N4O2S |
|
—— |
2-methoxy-1-[(3S)-3-[(5S,7R)-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]ethanone |
—— |
C19H23F3N4O2S |
|
—— |
[(3S)-3-[(5S,7R)-5-tert-butyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-pyridin-4-ylmethanone |
—— |
C22H28F3N5O |
|
—— |
(2,4-dimethyl-1,3-thiazol-5-yl)-[(3S)-3-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]methanone |
—— |
C20H26F3N5OS |
|
—— |
(2-methoxypyrimidin-5-yl)-[4-[(5R,7R)-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]methanone |
—— |
C19H23F3N6O2 |
|
—— |
[4-[(5S,7R)-5-tert-butyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-(2-methylpyrazol-3-yl)methanone |
—— |
C21H29F3N6O |
|
—— |
(2,4-dimethyl-1,3-thiazol-5-yl)-[(3R)-3-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]methanone |
—— |
C20H26F3N5OS |
|
—— |
[(1R,2S)-2-methylcyclopropyl]-[4-[(5S,7R)-5-propan-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]methanone |
—— |
C20H29F3N4O |
|
—— |
[(3R)-3-[(5S,7R)-5-tert-butyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-pyridin-3-ylmethanone |
—— |
C22H28F3N5O |
|
—— |
[(2R)-2-[(5S,7R)-5-tert-butyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-(1-methylpyrazol-3-yl)methanone |
—— |
C21H29F3N6O |
|
—— |
[(3R)-3-[(5S,7R)-5-tert-butyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]-(3-methyl-1,2-oxazol-5-yl)methanone |
—— |
C20H26F3N5O2 |
|
—— |
[(3S)-3-[(5S,7R)-5-tert-butyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]-(2-methylpyrazol-3-yl)methanone |
—— |
C20H27F3N6O |
|
—— |
(5S,7R)-2-(1-ethylsulfonylpiperidin-4-yl)-5-propan-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine |
—— |
C17H27F3N4O2S |
|
—— |
[4-[(5S,7R)-5-propan-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-pyridin-4-ylmethanone |
—— |
C21H26F3N5O |
|
—— |
(2-methylpyridin-3-yl)-[4-[(5S,7R)-5-propan-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]methanone |
—— |
C22H28F3N5O |
|
—— |
[(3R)-3-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]-pyridin-4-ylmethanone |
—— |
C19H22F3N5O |
|
—— |
1-[(3R)-3-[(5S,7R)-2-tert-butyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-2-methylpropan-1-one |
—— |
C20H31F3N4O |
|
—— |
[(1S,2S)-2-methylcyclopropyl]-[4-[(5S,7R)-5-propan-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]methanone |
—— |
C20H29F3N4O |
|
—— |
(2,4-dimethyl-1,3-oxazol-5-yl)-[4-[(5R,7R)-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]methanone |
—— |
C19H24F3N5O2 |
|
—— |
(1,3-dimethylpyrazol-4-yl)-[4-[(5S,7R)-5-propan-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]methanone |
—— |
C21H29F3N6O |
|