中文名称 |
英文名称 |
CAS号 |
化学式 |
结构式图片 |
—— |
2-methyl-1-[(3R)-3-[(5S,7R)-2-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]propan-1-one |
—— |
C17H25F3N4O |
|
—— |
(4S)-1-methyl-4-[(3S)-3-[(5S,7R)-2-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidine-1-carbonyl]pyrrolidin-2-one |
—— |
C19H26F3N5O2 |
|
—— |
[(3R)-3-[(5S,7R)-7-(difluoromethyl)-2-methyl-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-[(1R,2S)-2-methylcyclopropyl]methanone |
—— |
C18H26F2N4O |
|
—— |
[(3R)-3-[(5S,7R)-2-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-(1,3-thiazol-4-yl)methanone |
—— |
C17H20F3N5OS |
|
—— |
[(1R,3S)-3-methoxycyclohexyl]-[(3R)-3-[(5S,7R)-2-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]methanone |
—— |
C21H31F3N4O2 |
|
—— |
(2S)-1-[(3R)-3-[(5S,7R)-7-(difluoromethyl)-2-methyl-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-2-(2-fluorophenoxy)propan-1-one |
—— |
C22H27F3N4O2 |
|
—— |
3-(3-methoxy-1,2-oxazol-5-yl)-1-[(3R)-3-[(5S,7R)-2-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]propan-1-one |
—— |
C20H26F3N5O3 |
|
—— |
2-[(1R)-cyclopent-2-en-1-yl]-1-[(3R)-3-[(5S,7R)-7-(difluoromethyl)-2-methyl-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]ethanone |
—— |
C20H28F2N4O |
|
—— |
(4R)-5,5-dimethyl-4-[(3R)-3-[(5S,7R)-2-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidine-1-carbonyl]oxolan-2-one |
—— |
C20H27F3N4O3 |
|
—— |
[(3S)-3-[(5S,7R)-7-(difluoromethyl)-2-methyl-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-[(2R)-oxolan-2-yl]methanone |
—— |
C18H26F2N4O2 |
|
—— |
(2S)-2-methyl-1-[(3R)-3-[(5S,7R)-2-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-3-thiophen-2-ylpropan-1-one |
—— |
C21H27F3N4OS |
|
—— |
(2S)-1-[(3R)-3-[(5S,7R)-7-(difluoromethyl)-2-methyl-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-2-(3-fluorophenoxy)propan-1-one |
—— |
C22H27F3N4O2 |
|
—— |
3-cyclopentyl-1-[(3R)-3-[(5S,7R)-2-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]propan-1-one |
—— |
C21H31F3N4O |
|
—— |
(2S)-1-[(3R)-3-[(5S,7R)-7-(difluoromethyl)-2-methyl-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-2-(4-fluorophenoxy)propan-1-one |
—— |
C22H27F3N4O2 |
|
—— |
1-[(3S)-3-[(5S,7R)-2-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-3-[(2S)-oxolan-2-yl]propan-1-one |
—— |
C20H29F3N4O2 |
|
—— |
(4R)-1-methyl-4-[(3S)-3-[(5S,7R)-2-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidine-1-carbonyl]pyrrolidin-2-one |
—— |
C19H26F3N5O2 |
|
—— |
(2S)-1-[(3S)-3-[(5S,7R)-7-(difluoromethyl)-2-methyl-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-2-(3-fluorophenoxy)propan-1-one |
—— |
C22H27F3N4O2 |
|
—— |
(2R)-1-[(3R)-3-[(5S,7R)-7-(difluoromethyl)-2-methyl-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-2-(3-fluorophenoxy)propan-1-one |
—— |
C22H27F3N4O2 |
|
—— |
1-[(3S)-3-[(5S,7R)-7-(difluoromethyl)-2-methyl-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-4-pyridin-4-ylbutan-1-one |
—— |
C22H29F2N5O |
|
—— |
(4R)-1-methyl-4-[(3R)-3-[(5S,7R)-2-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidine-1-carbonyl]pyrrolidin-2-one |
—— |
C19H26F3N5O2 |
|
—— |
[(3S)-3-[(5S,7R)-7-(difluoromethyl)-2-methyl-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-(2-methoxypyridin-4-yl)methanone |
—— |
C20H25F2N5O2 |
|
—— |
1-[(3R)-3-[(5S,7R)-7-(difluoromethyl)-2-methyl-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-2-[[(2R)-oxan-2-yl]methoxy]ethanone |
—— |
C21H32F2N4O3 |
|
—— |
1-[(3S)-3-[(5S,7R)-7-(difluoromethyl)-2-methyl-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-3-(2-fluorophenyl)propan-1-one |
—— |
C22H27F3N4O |
|
—— |
(4S)-5,5-dimethyl-4-[(3R)-3-[(5S,7R)-2-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidine-1-carbonyl]oxolan-2-one |
—— |
C20H27F3N4O3 |
|
—— |
(4R)-4-[(3S)-3-[(5S,7R)-7-(difluoromethyl)-2-methyl-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidine-1-carbonyl]-1-methylpyrrolidin-2-one |
—— |
C19H27F2N5O2 |
|
—— |
[(3R)-3-[(5S,7R)-7-(difluoromethyl)-2-methyl-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-[(2S)-oxolan-2-yl]methanone |
—— |
C18H26F2N4O2 |
|
—— |
1-[4-[(3R)-3-[(5S,7R)-7-(difluoromethyl)-2-methyl-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-4-oxobutyl]pyrrolidin-2-one |
—— |
C21H31F2N5O2 |
|
—— |
[(3R)-3-[(5S,7R)-2-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-[(2R)-oxolan-2-yl]methanone |
—— |
C18H25F3N4O2 |
|
—— |
1-[(3S)-3-[(5S,7R)-7-(difluoromethyl)-2-methyl-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-3-pyridin-3-ylpropan-1-one |
—— |
C21H27F2N5O |
|
—— |
(4S)-5,5-dimethyl-4-[(3S)-3-[(5S,7R)-2-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidine-1-carbonyl]oxolan-2-one |
—— |
C20H27F3N4O3 |
|
—— |
(2S)-1-[(3S)-3-[(5S,7R)-7-(difluoromethyl)-2-methyl-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-2-(2-methoxyphenoxy)propan-1-one |
—— |
C23H30F2N4O3 |
|
—— |
[(1S,3S)-3-methoxycyclohexyl]-[(3R)-3-[(5S,7R)-2-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]methanone |
—— |
C21H31F3N4O2 |
|
—— |
(2R)-2-methyl-1-[(3S)-3-[(5S,7R)-2-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-3-thiophen-2-ylpropan-1-one |
—— |
C21H27F3N4OS |
|
—— |
1-[(3R)-3-[(5S,7R)-2-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-3-[(2S)-oxolan-2-yl]propan-1-one |
—— |
C20H29F3N4O2 |
|
—— |
2-cyclopentyl-1-[(3R)-3-[(5S,7R)-2-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]ethanone |
—— |
C20H29F3N4O |
|
—— |
(2S)-1-[(3R)-3-[(5S,7R)-7-(difluoromethyl)-2-methyl-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-2-(2-methoxyphenoxy)propan-1-one |
—— |
C23H30F2N4O3 |
|
—— |
(2R)-1-[(3S)-3-[(5S,7R)-7-(difluoromethyl)-2-methyl-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-2-(3-methoxyphenoxy)propan-1-one |
—— |
C23H30F2N4O3 |
|
—— |
(4R)-4-[(3R)-3-[(5S,7R)-7-(difluoromethyl)-2-methyl-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidine-1-carbonyl]-1-prop-2-enylpyrrolidin-2-one |
—— |
C21H29F2N5O2 |
|
—— |
[(3R)-3-[(5S,7R)-2-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-[(2S)-oxolan-2-yl]methanone |
—— |
C18H25F3N4O2 |
|
—— |
(2S)-1-[(3S)-3-[(5S,7R)-7-(difluoromethyl)-2-methyl-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-2-(4-fluorophenoxy)propan-1-one |
—— |
C22H27F3N4O2 |
|
—— |
1-[(3S)-3-[(5S,7R)-2-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-3-[(2R)-oxolan-2-yl]propan-1-one |
—— |
C20H29F3N4O2 |
|
—— |
cyclohexyl-[(3R)-3-[(5S,7R)-7-(difluoromethyl)-2-methyl-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]methanone |
—— |
C20H30F2N4O |
|
—— |
1-[(3S)-3-[(5S,7R)-2-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-2-[(2S)-oxolan-2-yl]ethanone |
—— |
C19H27F3N4O2 |
|
—— |
(4-methoxycyclohexyl)-[(3R)-3-[(5S,7R)-2-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]methanone |
—— |
C21H31F3N4O2 |
|
—— |
cyclopropyl-[(3R)-3-[(5S,7R)-7-(difluoromethyl)-2-methyl-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]methanone |
—— |
C17H24F2N4O |
|
—— |
[(3S)-3-[(5S,7R)-7-(difluoromethyl)-2-methyl-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-[(2S)-oxolan-2-yl]methanone |
—— |
C18H26F2N4O2 |
|
—— |
(2R)-1-[(3S)-3-[(5S,7R)-7-(difluoromethyl)-2-methyl-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-2-(2-fluorophenoxy)propan-1-one |
—— |
C22H27F3N4O2 |
|
—— |
(2R)-1-[(3S)-3-[(5S,7R)-7-(difluoromethyl)-2-methyl-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-2-(4-fluorophenoxy)propan-1-one |
—— |
C22H27F3N4O2 |
|
—— |
1-[(3R)-3-[(5S,7R)-7-(difluoromethyl)-2-methyl-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-3-pyridin-3-ylpropan-1-one |
—— |
C21H27F2N5O |
|
—— |
(4S)-4-[(3S)-3-[(5S,7R)-7-(difluoromethyl)-2-methyl-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidine-1-carbonyl]-1-prop-2-enylpyrrolidin-2-one |
—— |
C21H29F2N5O2 |
|