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吡唑并嘧啶类

中文名称 英文名称 CAS号 化学式 结构式图片
—— (7S)-7-(2-methoxyphenyl)-5-methyl-3-N-(3-methylphenyl)-6-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide —— C29H27N5O3
(7S)-7-(2-methoxyphenyl)-5-methyl-3-N-(3-methylphenyl)-6-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide
—— (7S)-6-N-(2-methoxyphenyl)-5-methyl-7-(3-methylphenyl)-3-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide —— C29H27N5O3
(7S)-6-N-(2-methoxyphenyl)-5-methyl-7-(3-methylphenyl)-3-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide
—— 2-tert-butyl-N-[5-(diethylamino)pentan-2-yl]-7-ethylpyrazolo[1,5-a]pyrimidine-6-carboxamide —— C22H37N5O
2-tert-butyl-N-[5-(diethylamino)pentan-2-yl]-7-ethylpyrazolo[1,5-a]pyrimidine-6-carboxamide
—— N-[(1R,2R,3S)-2,3-dimethylcyclohexyl]-4-[(5-oxo-6,7-dihydropyrazolo[1,5-a]pyrimidin-4-yl)methyl]benzamide —— C22H28N4O2
N-[(1R,2R,3S)-2,3-dimethylcyclohexyl]-4-[(5-oxo-6,7-dihydropyrazolo[1,5-a]pyrimidin-4-yl)methyl]benzamide
—— 4-[(5-oxo-6,7-dihydropyrazolo[1,5-a]pyrimidin-4-yl)methyl]-N-[(2S)-4-phenylbutan-2-yl]benzamide —— C24H26N4O2
4-[(5-oxo-6,7-dihydropyrazolo[1,5-a]pyrimidin-4-yl)methyl]-N-[(2S)-4-phenylbutan-2-yl]benzamide
—— N-[(1R,2S)-2-methylcyclohexyl]-4-[(5-oxo-6,7-dihydropyrazolo[1,5-a]pyrimidin-4-yl)methyl]benzamide —— C21H26N4O2
N-[(1R,2S)-2-methylcyclohexyl]-4-[(5-oxo-6,7-dihydropyrazolo[1,5-a]pyrimidin-4-yl)methyl]benzamide
—— 4-[(5-oxo-6,7-dihydropyrazolo[1,5-a]pyrimidin-4-yl)methyl]-N-[(2R)-4-phenylbutan-2-yl]benzamide —— C24H26N4O2
4-[(5-oxo-6,7-dihydropyrazolo[1,5-a]pyrimidin-4-yl)methyl]-N-[(2R)-4-phenylbutan-2-yl]benzamide
—— N-[3-[(2R)-2-methylpiperidin-1-yl]propyl]-4-[(5-oxo-6,7-dihydropyrazolo[1,5-a]pyrimidin-4-yl)methyl]benzamide —— C23H31N5O2
N-[3-[(2R)-2-methylpiperidin-1-yl]propyl]-4-[(5-oxo-6,7-dihydropyrazolo[1,5-a]pyrimidin-4-yl)methyl]benzamide
—— N-[3-[(3R)-3-methylpiperidin-1-yl]propyl]-4-[(5-oxo-6,7-dihydropyrazolo[1,5-a]pyrimidin-4-yl)methyl]benzamide —— C23H31N5O2
N-[3-[(3R)-3-methylpiperidin-1-yl]propyl]-4-[(5-oxo-6,7-dihydropyrazolo[1,5-a]pyrimidin-4-yl)methyl]benzamide
—— 4-[(2-methyl-5-oxo-6,7-dihydropyrazolo[1,5-a]pyrimidin-4-yl)methyl]-N-[(2R)-4-phenylbutan-2-yl]benzamide —— C25H28N4O2
4-[(2-methyl-5-oxo-6,7-dihydropyrazolo[1,5-a]pyrimidin-4-yl)methyl]-N-[(2R)-4-phenylbutan-2-yl]benzamide
—— N-[(1S,2R,3S)-2,3-dimethylcyclohexyl]-2,3,7-triazatricyclo[7.6.0.02,6]pentadeca-1(9),3,5,7-tetraene-5-carboxamide —— C21H30N4O
N-[(1S,2R,3S)-2,3-dimethylcyclohexyl]-2,3,7-triazatricyclo[7.6.0.02,6]pentadeca-1(9),3,5,7-tetraene-5-carboxamide
—— N-[3-[(2S)-2-methylpiperidin-1-yl]propyl]-4-[(5-oxo-6,7-dihydropyrazolo[1,5-a]pyrimidin-4-yl)methyl]benzamide —— C23H31N5O2
N-[3-[(2S)-2-methylpiperidin-1-yl]propyl]-4-[(5-oxo-6,7-dihydropyrazolo[1,5-a]pyrimidin-4-yl)methyl]benzamide
—— N-[3-[(3S)-3-methylpiperidin-1-yl]propyl]-4-[(5-oxo-6,7-dihydropyrazolo[1,5-a]pyrimidin-4-yl)methyl]benzamide —— C23H31N5O2
N-[3-[(3S)-3-methylpiperidin-1-yl]propyl]-4-[(5-oxo-6,7-dihydropyrazolo[1,5-a]pyrimidin-4-yl)methyl]benzamide
—— N-[3-[(2R)-2-ethylpiperidin-1-yl]propyl]-4-[(5-oxo-6,7-dihydropyrazolo[1,5-a]pyrimidin-4-yl)methyl]benzamide —— C24H33N5O2
N-[3-[(2R)-2-ethylpiperidin-1-yl]propyl]-4-[(5-oxo-6,7-dihydropyrazolo[1,5-a]pyrimidin-4-yl)methyl]benzamide
—— N-[(2R)-butan-2-yl]-4-[(5-oxo-6,7-dihydropyrazolo[1,5-a]pyrimidin-4-yl)methyl]benzamide —— C18H22N4O2
N-[(2R)-butan-2-yl]-4-[(5-oxo-6,7-dihydropyrazolo[1,5-a]pyrimidin-4-yl)methyl]benzamide
—— N-[(2S)-butan-2-yl]-4-[(5-oxo-6,7-dihydropyrazolo[1,5-a]pyrimidin-4-yl)methyl]benzamide —— C18H22N4O2
N-[(2S)-butan-2-yl]-4-[(5-oxo-6,7-dihydropyrazolo[1,5-a]pyrimidin-4-yl)methyl]benzamide
—— N-[[(2R)-1-ethylpyrrolidin-2-yl]methyl]-4-[(5-oxo-6,7-dihydropyrazolo[1,5-a]pyrimidin-4-yl)methyl]benzamide —— C21H27N5O2
N-[[(2R)-1-ethylpyrrolidin-2-yl]methyl]-4-[(5-oxo-6,7-dihydropyrazolo[1,5-a]pyrimidin-4-yl)methyl]benzamide
—— 4-[(5-oxo-6,7-dihydropyrazolo[1,5-a]pyrimidin-4-yl)methyl]-N-[(2S)-2-phenylpropyl]benzamide —— C23H24N4O2
4-[(5-oxo-6,7-dihydropyrazolo[1,5-a]pyrimidin-4-yl)methyl]-N-[(2S)-2-phenylpropyl]benzamide
—— N-[(1R,2R)-2-methylcyclohexyl]-4-[(5-oxo-6,7-dihydropyrazolo[1,5-a]pyrimidin-4-yl)methyl]benzamide —— C21H26N4O2
N-[(1R,2R)-2-methylcyclohexyl]-4-[(5-oxo-6,7-dihydropyrazolo[1,5-a]pyrimidin-4-yl)methyl]benzamide
—— N-[(1S,2R,3S)-2,3-dimethylcyclohexyl]-4-[(5-oxo-6,7-dihydropyrazolo[1,5-a]pyrimidin-4-yl)methyl]benzamide —— C22H28N4O2
N-[(1S,2R,3S)-2,3-dimethylcyclohexyl]-4-[(5-oxo-6,7-dihydropyrazolo[1,5-a]pyrimidin-4-yl)methyl]benzamide
—— N-[(1R,2R,3R)-2,3-dimethylcyclohexyl]-4-[(5-oxo-6,7-dihydropyrazolo[1,5-a]pyrimidin-4-yl)methyl]benzamide —— C22H28N4O2
N-[(1R,2R,3R)-2,3-dimethylcyclohexyl]-4-[(5-oxo-6,7-dihydropyrazolo[1,5-a]pyrimidin-4-yl)methyl]benzamide
—— N-[(2S)-4-phenylbutan-2-yl]-2,3,7-triazatricyclo[7.6.0.02,6]pentadeca-1(9),3,5,7-tetraene-5-carboxamide —— C23H28N4O
N-[(2S)-4-phenylbutan-2-yl]-2,3,7-triazatricyclo[7.6.0.02,6]pentadeca-1(9),3,5,7-tetraene-5-carboxamide
—— 4-[(5-oxo-6,7-dihydropyrazolo[1,5-a]pyrimidin-4-yl)methyl]-N-[(2R)-2-phenylpropyl]benzamide —— C23H24N4O2
4-[(5-oxo-6,7-dihydropyrazolo[1,5-a]pyrimidin-4-yl)methyl]-N-[(2R)-2-phenylpropyl]benzamide
—— N-[(1S,2S)-2-methylcyclohexyl]-4-[(5-oxo-6,7-dihydropyrazolo[1,5-a]pyrimidin-4-yl)methyl]benzamide —— C21H26N4O2
N-[(1S,2S)-2-methylcyclohexyl]-4-[(5-oxo-6,7-dihydropyrazolo[1,5-a]pyrimidin-4-yl)methyl]benzamide
—— N-[(1R,2R)-2-methylcyclohexyl]-2,3,7-triazatricyclo[7.5.0.02,6]tetradeca-1(9),3,5,7-tetraene-5-carboxamide —— C19H26N4O
N-[(1R,2R)-2-methylcyclohexyl]-2,3,7-triazatricyclo[7.5.0.02,6]tetradeca-1(9),3,5,7-tetraene-5-carboxamide
—— N-[[(2R)-1-ethylpyrrolidin-2-yl]methyl]-2,3,7-triazatricyclo[7.6.0.02,6]pentadeca-1(9),3,5,7-tetraene-5-carboxamide —— C20H29N5O
N-[[(2R)-1-ethylpyrrolidin-2-yl]methyl]-2,3,7-triazatricyclo[7.6.0.02,6]pentadeca-1(9),3,5,7-tetraene-5-carboxamide
—— N-[(1R,2S)-2-methylcyclohexyl]-2,3,7-triazatricyclo[7.6.0.02,6]pentadeca-1(9),3,5,7-tetraene-5-carboxamide —— C20H28N4O
N-[(1R,2S)-2-methylcyclohexyl]-2,3,7-triazatricyclo[7.6.0.02,6]pentadeca-1(9),3,5,7-tetraene-5-carboxamide
—— N-[(2R)-2-phenylpropyl]-2,3,7-triazatricyclo[7.6.0.02,6]pentadeca-1(9),3,5,7-tetraene-5-carboxamide —— C22H26N4O
N-[(2R)-2-phenylpropyl]-2,3,7-triazatricyclo[7.6.0.02,6]pentadeca-1(9),3,5,7-tetraene-5-carboxamide
—— N-[(1S)-1-phenylethyl]-2,3,7-triazatricyclo[7.6.0.02,6]pentadeca-1(9),3,5,7-tetraene-5-carboxamide —— C21H24N4O
N-[(1S)-1-phenylethyl]-2,3,7-triazatricyclo[7.6.0.02,6]pentadeca-1(9),3,5,7-tetraene-5-carboxamide
—— N-[(1S,2R)-2-methylcyclohexyl]-2,3,7-triazatricyclo[7.6.0.02,6]pentadeca-1(9),3,5,7-tetraene-5-carboxamide —— C20H28N4O
N-[(1S,2R)-2-methylcyclohexyl]-2,3,7-triazatricyclo[7.6.0.02,6]pentadeca-1(9),3,5,7-tetraene-5-carboxamide
—— N-[(2R)-butan-2-yl]-2,3,7-triazatricyclo[7.6.0.02,6]pentadeca-1(9),3,5,7-tetraene-5-carboxamide —— C17H24N4O
N-[(2R)-butan-2-yl]-2,3,7-triazatricyclo[7.6.0.02,6]pentadeca-1(9),3,5,7-tetraene-5-carboxamide
—— N-[[(2S)-oxolan-2-yl]methyl]-2,3,7-triazatricyclo[7.6.0.02,6]pentadeca-1(9),3,5,7-tetraene-5-carboxamide —— C18H24N4O2
N-[[(2S)-oxolan-2-yl]methyl]-2,3,7-triazatricyclo[7.6.0.02,6]pentadeca-1(9),3,5,7-tetraene-5-carboxamide
—— N-[(1S,2S)-2-methylcyclohexyl]-2,3,7-triazatricyclo[7.5.0.02,6]tetradeca-1(9),3,5,7-tetraene-5-carboxamide —— C19H26N4O
N-[(1S,2S)-2-methylcyclohexyl]-2,3,7-triazatricyclo[7.5.0.02,6]tetradeca-1(9),3,5,7-tetraene-5-carboxamide
—— [(3R,5S)-3,5-dimethylpiperidin-1-yl]-(2,3,7-triazatricyclo[7.6.0.02,6]pentadeca-1(9),3,5,7-tetraen-5-yl)methanone —— C20H28N4O
[(3R,5S)-3,5-dimethylpiperidin-1-yl]-(2,3,7-triazatricyclo[7.6.0.02,6]pentadeca-1(9),3,5,7-tetraen-5-yl)methanone
—— N-[(1R,2R,3S)-2,3-dimethylcyclohexyl]-2,3,7-triazatricyclo[7.6.0.02,6]pentadeca-1(9),3,5,7-tetraene-5-carboxamide —— C21H30N4O
N-[(1R,2R,3S)-2,3-dimethylcyclohexyl]-2,3,7-triazatricyclo[7.6.0.02,6]pentadeca-1(9),3,5,7-tetraene-5-carboxamide
—— N-[(2S)-butan-2-yl]-2,3,7-triazatricyclo[7.6.0.02,6]pentadeca-1(9),3,5,7-tetraene-5-carboxamide —— C17H24N4O
N-[(2S)-butan-2-yl]-2,3,7-triazatricyclo[7.6.0.02,6]pentadeca-1(9),3,5,7-tetraene-5-carboxamide
—— N-[(1R,2S)-2-methylcyclohexyl]-2,3,7-triazatricyclo[7.5.0.02,6]tetradeca-1(9),3,5,7-tetraene-5-carboxamide —— C19H26N4O
N-[(1R,2S)-2-methylcyclohexyl]-2,3,7-triazatricyclo[7.5.0.02,6]tetradeca-1(9),3,5,7-tetraene-5-carboxamide
—— N-[[(2R)-oxolan-2-yl]methyl]-2,3,7-triazatricyclo[7.6.0.02,6]pentadeca-1(9),3,5,7-tetraene-5-carboxamide —— C18H24N4O2
N-[[(2R)-oxolan-2-yl]methyl]-2,3,7-triazatricyclo[7.6.0.02,6]pentadeca-1(9),3,5,7-tetraene-5-carboxamide
—— N-[(2R)-4-phenylbutan-2-yl]-2,3,7-triazatricyclo[7.6.0.02,6]pentadeca-1(9),3,5,7-tetraene-5-carboxamide —— C23H28N4O
N-[(2R)-4-phenylbutan-2-yl]-2,3,7-triazatricyclo[7.6.0.02,6]pentadeca-1(9),3,5,7-tetraene-5-carboxamide
—— N-[(1S)-1-phenylethyl]-2,3,7-triazatricyclo[7.5.0.02,6]tetradeca-1(9),3,5,7-tetraene-5-carboxamide —— C20H22N4O
N-[(1S)-1-phenylethyl]-2,3,7-triazatricyclo[7.5.0.02,6]tetradeca-1(9),3,5,7-tetraene-5-carboxamide
—— N-[(1R,2R,3R)-2,3-dimethylcyclohexyl]-2,3,7-triazatricyclo[7.6.0.02,6]pentadeca-1(9),3,5,7-tetraene-5-carboxamide —— C21H30N4O
N-[(1R,2R,3R)-2,3-dimethylcyclohexyl]-2,3,7-triazatricyclo[7.6.0.02,6]pentadeca-1(9),3,5,7-tetraene-5-carboxamide
—— N-[(1S,2R)-2-methylcyclohexyl]-2,3,7-triazatricyclo[7.5.0.02,6]tetradeca-1(9),3,5,7-tetraene-5-carboxamide —— C19H26N4O
N-[(1S,2R)-2-methylcyclohexyl]-2,3,7-triazatricyclo[7.5.0.02,6]tetradeca-1(9),3,5,7-tetraene-5-carboxamide
—— N-[(1S,2R,3R)-2,3-dimethylcyclohexyl]-2,3,7-triazatricyclo[7.6.0.02,6]pentadeca-1(9),3,5,7-tetraene-5-carboxamide —— C21H30N4O
N-[(1S,2R,3R)-2,3-dimethylcyclohexyl]-2,3,7-triazatricyclo[7.6.0.02,6]pentadeca-1(9),3,5,7-tetraene-5-carboxamide
—— N-[(1S,2S)-2-methylcyclohexyl]-2,3,7-triazatricyclo[7.6.0.02,6]pentadeca-1(9),3,5,7-tetraene-5-carboxamide —— C20H28N4O
N-[(1S,2S)-2-methylcyclohexyl]-2,3,7-triazatricyclo[7.6.0.02,6]pentadeca-1(9),3,5,7-tetraene-5-carboxamide
—— N-[(2S)-2-phenylpropyl]-2,3,7-triazatricyclo[7.6.0.02,6]pentadeca-1(9),3,5,7-tetraene-5-carboxamide —— C22H26N4O
N-[(2S)-2-phenylpropyl]-2,3,7-triazatricyclo[7.6.0.02,6]pentadeca-1(9),3,5,7-tetraene-5-carboxamide
—— N-[(2R)-2-phenylpropyl]-2,3,7-triazatricyclo[7.5.0.02,6]tetradeca-1(9),3,5,7-tetraene-5-carboxamide —— C21H24N4O
N-[(2R)-2-phenylpropyl]-2,3,7-triazatricyclo[7.5.0.02,6]tetradeca-1(9),3,5,7-tetraene-5-carboxamide
—— N-[(2S)-2-phenylpropyl]-2,3,7-triazatricyclo[7.5.0.02,6]tetradeca-1(9),3,5,7-tetraene-5-carboxamide —— C21H24N4O
N-[(2S)-2-phenylpropyl]-2,3,7-triazatricyclo[7.5.0.02,6]tetradeca-1(9),3,5,7-tetraene-5-carboxamide
—— 4-[(5-oxo-6,7-dihydropyrazolo[1,5-a]pyrimidin-4-yl)methyl]-N-[[(2R)-oxolan-2-yl]methyl]benzamide —— C19H22N4O3
4-[(5-oxo-6,7-dihydropyrazolo[1,5-a]pyrimidin-4-yl)methyl]-N-[[(2R)-oxolan-2-yl]methyl]benzamide
—— N-[(1R)-1-phenylethyl]-2,3,7-triazatricyclo[7.5.0.02,6]tetradeca-1(9),3,5,7-tetraene-5-carboxamide —— C20H22N4O
N-[(1R)-1-phenylethyl]-2,3,7-triazatricyclo[7.5.0.02,6]tetradeca-1(9),3,5,7-tetraene-5-carboxamide
—— [(3S,5S)-3,5-dimethylpiperidin-1-yl]-(2,3,7-triazatricyclo[7.6.0.02,6]pentadeca-1(9),3,5,7-tetraen-5-yl)methanone —— C20H28N4O
[(3S,5S)-3,5-dimethylpiperidin-1-yl]-(2,3,7-triazatricyclo[7.6.0.02,6]pentadeca-1(9),3,5,7-tetraen-5-yl)methanone