中文名称 |
英文名称 |
CAS号 |
化学式 |
结构式图片 |
—— |
[(3S)-3-[(5S,7R)-2-tert-butyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-(2-methylpyridin-3-yl)methanone |
—— |
C23H30F3N5O |
|
—— |
2-(2-methylfuran-3-yl)-5-[(3S)-1-(pyridin-4-ylmethyl)piperidin-3-yl]pyrazolo[1,5-a]pyrimidin-7-amine |
—— |
C22H24N6O |
|
—— |
[4-[(5S,7R)-2-tert-butyl-7-(difluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-(2-methylpyridin-3-yl)methanone |
—— |
C23H31F2N5O |
|
—— |
12-[[2-(Methylamino)pyridin-3-yl]methyl]-5-(2-methylfuran-3-yl)-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one |
—— |
C21H22N6O2 |
|
—— |
(1,3-dimethylpyrazol-4-yl)-[(3R)-3-[(5S,7R)-5-propan-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]methanone |
—— |
C20H27F3N6O |
|
—— |
N-(3-imidazol-1-ylpropyl)-11-methyl-10-thiophen-2-yl-1,8,12-triazatricyclo[7.3.0.03,7]dodeca-2,7,9,11-tetraen-2-amine |
—— |
C20H22N6S |
|
—— |
(3,5-dimethyl-1,2-oxazol-4-yl)-[(2R)-2-[5-propan-2-yl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]methanone |
—— |
C20H22F3N5O2 |
|
—— |
2-{8,9-Dimethoxy-4-methyl-2-oxo-2H,6H-pyrimido[1,2-B]indazol-6-YL}-N-[(4-ethoxyphenyl)methyl]acetamide |
—— |
C24H26N4O5 |
|
—— |
(3,5-dimethyl-1,2-oxazol-4-yl)-[(2S)-2-[5-propan-2-yl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]methanone |
—— |
C20H22F3N5O2 |
|
—— |
2-[(3S)-1-[(3-ethylimidazol-4-yl)methyl]piperidin-3-yl]-5-propan-2-yl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine |
—— |
C21H27F3N6 |
|
—— |
6-Benzyl-5-methyl-2-(oxan-4-yl)-7-prop-2-ynoxypyrazolo[1,5-a]pyrimidine |
—— |
C22H23N3O2 |
|
—— |
2-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[(3R)-3-[(5S,7R)-5-propan-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]ethanone |
—— |
C21H29F3N6O |
|
—— |
2-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[(3S)-3-[(5S,7R)-5-propan-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]ethanone |
—— |
C21H29F3N6O |
|
—— |
2-[(3R)-1-[(3-ethylimidazol-4-yl)methyl]piperidin-3-yl]-5-propan-2-yl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine |
—— |
C21H27F3N6 |
|
—— |
(5S,7R)-2-[(2R)-1-[(5-methyl-1H-imidazol-4-yl)methyl]piperidin-2-yl]-5-propan-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine |
—— |
C20H29F3N6 |
|
—— |
(5S,7R)-2-[(2S)-1-[(5-methyl-1H-imidazol-4-yl)methyl]piperidin-2-yl]-5-propan-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine |
—— |
C20H29F3N6 |
|
—— |
cyclopropyl-[4-[(5R,7R)-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]methanone |
—— |
C17H23F3N4O |
|
—— |
1-[(2S)-2-[(5R,7R)-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]-2-pyridin-3-yloxyethanone |
—— |
C19H22F3N5O2 |
|
—— |
[2-methoxy-5-[[(2S)-2-[(5R,7R)-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]methyl]phenyl]methanol |
—— |
C21H27F3N4O2 |
|
—— |
2-methyl-1-[(2R)-2-[(5R,7R)-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]propan-1-one |
—— |
C16H23F3N4O |
|
—— |
1-[(3S)-3-[(5R,7R)-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]-4-pyridin-4-ylbutan-1-one |
—— |
C21H26F3N5O |
|
—— |
(3S)-1-[(2S)-2-[(5R,7R)-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]-3-pyrazol-1-ylbutan-1-one |
—— |
C19H25F3N6O |
|
—— |
(2-methyl-5-propan-2-ylpyrazol-3-yl)-[(3S)-3-[(5R,7R)-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]methanone |
—— |
C21H29F3N6O |
|
—— |
(5R,7R)-5-methyl-2-[(3R)-1-propan-2-ylsulfonylpyrrolidin-3-yl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine |
—— |
C15H23F3N4O2S |
|
—— |
[(2R)-2-[(5R,7R)-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]-[(2R)-oxolan-2-yl]methanone |
—— |
C17H23F3N4O2 |
|
—— |
(2-methyl-5-propan-2-ylpyrazol-3-yl)-[(3S)-3-[(5R,7R)-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]methanone |
—— |
C20H27F3N6O |
|
—— |
(5R,7R)-2-[(2R)-1-[[4-(2-methoxyethoxy)phenyl]methyl]pyrrolidin-2-yl]-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine |
—— |
C22H29F3N4O2 |
|
—— |
2-[(1S)-cyclopent-2-en-1-yl]-1-[(2R)-2-[(5R,7R)-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]ethanone |
—— |
C19H25F3N4O |
|
—— |
[(2S)-2-[(5R,7R)-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]-pyridin-4-ylmethanone |
—— |
C18H20F3N5O |
|
—— |
[(3R)-3-[(5R,7R)-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-pyridin-3-ylmethanone |
—— |
C19H22F3N5O |
|
—— |
(5R,7R)-2-[(2R)-1-[(4-methoxyphenyl)methyl]pyrrolidin-2-yl]-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine |
—— |
C20H25F3N4O |
|
—— |
(5R,7R)-2-[(2S)-1-[[4-(2-methoxyethoxy)phenyl]methyl]pyrrolidin-2-yl]-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine |
—— |
C22H29F3N4O2 |
|
—— |
1-[(2R)-2-[(5R,7R)-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]-3-[(2R)-oxolan-2-yl]propan-1-one |
—— |
C19H27F3N4O2 |
|
—— |
(5R,7R)-5-methyl-2-[(2R)-1-[[(3S)-oxolan-3-yl]methyl]pyrrolidin-2-yl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine |
—— |
C17H25F3N4O |
|
—— |
2,2-dimethyl-1-[4-[(5R,7R)-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]propan-1-one |
—— |
C18H27F3N4O |
|
—— |
(5R,7R)-5-methyl-2-(1-propan-2-ylsulfonylpiperidin-4-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine |
—— |
C16H25F3N4O2S |
|
—— |
(1-methylpyrazol-3-yl)-[(2R)-2-[(5R,7R)-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]methanone |
—— |
C17H21F3N6O |
|
—— |
[(2R)-2-[(5R,7R)-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]-(5-propan-2-yl-1H-pyrazol-3-yl)methanone |
—— |
C19H25F3N6O |
|
—— |
(5R,7R)-5-methyl-2-[(3R)-1-pyrrolidin-1-ylsulfonylpyrrolidin-3-yl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine |
—— |
C16H24F3N5O2S |
|
—— |
3-methoxy-1-[(2R)-2-[(5R,7R)-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]propan-1-one |
—— |
C16H23F3N4O2 |
|
—— |
2-methyl-1-[(2S)-2-[(5R,7R)-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]propan-1-one |
—— |
C16H23F3N4O |
|
—— |
(5-tert-butyl-2-methylpyrazol-3-yl)-[(3R)-3-[(5R,7R)-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]methanone |
—— |
C21H29F3N6O |
|
—— |
[(2R)-2-[(5R,7R)-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]-(1-propan-2-ylpyrazol-4-yl)methanone |
—— |
C19H25F3N6O |
|
—— |
(1-methylpyrazol-4-yl)-[(2S)-2-[(5R,7R)-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]methanone |
—— |
C17H21F3N6O |
|
—— |
[(2S)-2-[(5R,7R)-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]-[(2R)-oxolan-2-yl]methanone |
—— |
C17H23F3N4O2 |
|
—— |
(5R,7R)-5-methyl-2-[(3R)-1-prop-2-enylsulfonylpyrrolidin-3-yl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine |
—— |
C15H21F3N4O2S |
|
—— |
[(3S)-3-[(5R,7R)-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-pyridin-3-ylmethanone |
—— |
C19H22F3N5O |
|
—— |
1-[(2S)-2-[(5R,7R)-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]-2-pyridin-2-ylethanone |
—— |
C19H22F3N5O |
|
—— |
(2-methylpyrazol-3-yl)-[(2R)-2-[(5R,7R)-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]methanone |
—— |
C17H21F3N6O |
|
—— |
1-[(3R)-3-[(5R,7R)-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-2-pyridin-3-yloxyethanone |
—— |
C20H24F3N5O2 |
|