中文名称 |
英文名称 |
CAS号 |
化学式 |
结构式图片 |
—— |
3-methyl-5-pyridin-2-yl-2-thiophen-2-yl-1H-pyrazolo[1,5-a]pyrimidin-7-one |
—— |
C16H12N4OS |
|
—— |
3-methyl-5-pyridin-4-yl-2-thiophen-2-yl-1H-pyrazolo[1,5-a]pyrimidin-7-one |
—— |
C16H12N4OS |
|
—— |
7-[(3R)-1-benzylpyrrolidin-3-yl]-3-methyl-2-thiophen-2-ylpyrazolo[1,5-a]pyrimidine |
—— |
C22H22N4S |
|
—— |
7-[(3S)-1-benzylpyrrolidin-3-yl]-3-methyl-2-thiophen-2-ylpyrazolo[1,5-a]pyrimidine |
—— |
C22H22N4S |
|
—— |
1-[(2R)-2-(2-tert-butylpyrazolo[1,5-a]pyrimidin-7-yl)piperidin-1-yl]-2-(3,4,5-trimethylpyrazol-1-yl)ethanone |
—— |
C23H32N6O |
|
—— |
(2S)-1-[[2-(furan-2-yl)-5,6-dimethylpyrazolo[1,5-a]pyrimidin-7-yl]amino]-3-morpholin-4-ylpropan-2-ol |
—— |
C19H25N5O3 |
|
—— |
5,6-Dimethyl-2-(oxan-4-yl)-7-prop-2-enoxypyrazolo[1,5-a]pyrimidine |
—— |
C16H21N3O2 |
|
—— |
(2R)-1-[[2-(furan-2-yl)-5,6-dimethylpyrazolo[1,5-a]pyrimidin-7-yl]amino]-3-morpholin-4-ylpropan-2-ol |
—— |
C19H25N5O3 |
|
—— |
2-tert-butyl-7-[(2S)-1-(1,5-dimethylpyrazol-4-yl)sulfonylpyrrolidin-2-yl]pyrazolo[1,5-a]pyrimidine |
—— |
C19H26N6O2S |
|
—— |
(1,5-dimethylpyrazol-4-yl)-[(2R)-2-[(5R,7R)-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]methanone |
—— |
C18H23F3N6O |
|
—— |
(1,5-dimethylpyrazol-4-yl)-[(2R)-2-[5-propan-2-yl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]methanone |
—— |
C20H23F3N6O |
|
—— |
(1,5-dimethylpyrazol-4-yl)-[(2R)-2-[(5S,7R)-5-propan-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]methanone |
—— |
C20H27F3N6O |
|
—— |
(1,5-dimethylpyrazol-4-yl)-[(3S)-3-[(5S,7R)-5-propan-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]methanone |
—— |
C20H27F3N6O |
|
—— |
(1,5-dimethylpyrazol-4-yl)-[(2S)-2-[5-propan-2-yl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]methanone |
—— |
C20H23F3N6O |
|
—— |
2-tert-butyl-7-[(2S)-1-[1-(difluoromethyl)-5-methylpyrazol-4-yl]sulfonylpyrrolidin-2-yl]pyrazolo[1,5-a]pyrimidine |
—— |
C19H24F2N6O2S |
|
—— |
2-tert-butyl-7-[(2R)-1-[1-(difluoromethyl)-5-methylpyrazol-4-yl]sulfonylpyrrolidin-2-yl]pyrazolo[1,5-a]pyrimidine |
—— |
C19H24F2N6O2S |
|
—— |
(1,5-dimethylpyrazol-4-yl)-[(3R)-3-[(5S,7R)-5-propan-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]methanone |
—— |
C20H27F3N6O |
|
—— |
(2,4-dimethylpyrimidin-5-yl)-[(2R)-2-[(5S,7R)-5-propan-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]methanone |
—— |
C21H27F3N6O |
|
—— |
(2,4-dimethylpyrimidin-5-yl)-[(2S)-2-[(5S,7R)-5-propan-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]methanone |
—— |
C21H27F3N6O |
|
—— |
(2,4-dimethylpyrimidin-5-yl)-[(2S)-2-[5-propan-2-yl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]methanone |
—— |
C21H23F3N6O |
|
—— |
2-[(2R)-1-[(4-ethoxy-3-methoxyphenyl)methyl]pyrrolidin-2-yl]-5-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine |
—— |
C22H25F3N4O2 |
|
—— |
1-[4-[(5S,7R)-7-(difluoromethyl)-2-methyl-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-3-(4-ethoxyphenyl)propan-1-one |
—— |
C24H32F2N4O2 |
|
—— |
2-[(3R)-1-[(4-ethoxy-3-methoxyphenyl)methyl]pyrrolidin-3-yl]-5-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine |
—— |
C22H25F3N4O2 |
|
—— |
(5R,7R)-2-[(2R)-1-[(4-ethoxy-3-methoxyphenyl)methyl]pyrrolidin-2-yl]-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine |
—— |
C22H29F3N4O2 |
|
—— |
2-[(3S)-1-[(4-ethoxy-3-methoxyphenyl)methyl]pyrrolidin-3-yl]-5-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine |
—— |
C22H25F3N4O2 |
|
—— |
2-[(2S)-1-[(4-ethoxy-3-methoxyphenyl)methyl]pyrrolidin-2-yl]-5-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine |
—— |
C22H25F3N4O2 |
|
—— |
3-(3-ethoxy-1,2-oxazol-5-yl)-1-[(2R)-2-(2-methylpyrazolo[1,5-a]pyrimidin-7-yl)piperidin-1-yl]propan-1-one |
—— |
C20H25N5O3 |
|
—— |
(2-Tert-butyl-7-ethylpyrazolo[1,5-a]pyrimidin-6-yl)-(1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl)methanone |
—— |
C23H34N4O |
|
—— |
1-[(3S)-3-[(5S,7R)-7-(difluoromethyl)-2-methyl-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-3-(3-ethoxy-1,2-oxazol-5-yl)propan-1-one |
—— |
C21H29F2N5O3 |
|
—— |
1-[(3R)-3-[(5S,7R)-7-(difluoromethyl)-2-methyl-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-3-(3-ethoxy-1,2-oxazol-5-yl)propan-1-one |
—— |
C21H29F2N5O3 |
|
—— |
3-(3-ethoxy-1,2-oxazol-5-yl)-1-[(2S)-2-(2-methylpyrazolo[1,5-a]pyrimidin-7-yl)piperidin-1-yl]propan-1-one |
—— |
C20H25N5O3 |
|
—— |
1-[4-[(5S,7R)-7-(difluoromethyl)-2-methyl-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]-3-(3-ethoxy-1,2-oxazol-5-yl)propan-1-one |
—— |
C21H29F2N5O3 |
|
—— |
2-[(2R)-1-[(3-ethoxy-4-methoxyphenyl)methyl]pyrrolidin-2-yl]-5-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine |
—— |
C22H25F3N4O2 |
|
—— |
2-[(2S)-1-[(3-ethoxy-4-methoxyphenyl)methyl]pyrrolidin-2-yl]-5-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine |
—— |
C22H25F3N4O2 |
|
—— |
(5R,7R)-2-[(2S)-1-[(3-ethoxy-4-methoxyphenyl)methyl]pyrrolidin-2-yl]-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine |
—— |
C22H29F3N4O2 |
|
—— |
(5R,7R)-2-[(2R)-1-[(3-ethoxy-4-methoxyphenyl)methyl]pyrrolidin-2-yl]-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine |
—— |
C22H29F3N4O2 |
|
—— |
(2-ethoxypyridin-3-yl)-[(3S)-3-[(5S,7S)-2-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]methanone |
—— |
C21H26F3N5O2 |
|
—— |
ethyl (5S,7R)-5-[1-[(2R)-oxolane-2-carbonyl]piperidin-4-yl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxylate |
—— |
C20H27F3N4O4 |
|
—— |
ethyl (5S,7R)-5-[(3R)-1-[(3R)-oxolane-3-carbonyl]piperidin-3-yl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxylate |
—— |
C20H27F3N4O4 |
|
—— |
(2-ethoxypyridin-3-yl)-[(3S)-3-[(5R,7S)-2-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]methanone |
—— |
C21H26F3N5O2 |
|
—— |
(2-ethoxypyridin-3-yl)-[(3S)-3-[(5S,7R)-2-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]methanone |
—— |
C21H26F3N5O2 |
|
—— |
ethyl (5S,7R)-5-[(3S)-1-(3-methoxypropanoyl)piperidin-3-yl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxylate |
—— |
C19H27F3N4O4 |
|
—— |
ethyl (5S,7R)-5-[(3S)-1-(2,2-dimethylpropanoyl)piperidin-3-yl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxylate |
—— |
C20H29F3N4O3 |
|
—— |
ethyl (5S,7R)-5-[(3R)-1-(cyclopentanecarbonyl)piperidin-3-yl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxylate |
—— |
C21H29F3N4O3 |
|
—— |
ethyl (5S,7R)-5-[1-[(2S)-oxolane-2-carbonyl]piperidin-4-yl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxylate |
—— |
C20H27F3N4O4 |
|
—— |
ethyl (5S,7R)-5-[1-[(1S,2R)-2-methylcyclopropanecarbonyl]piperidin-4-yl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxylate |
—— |
C20H27F3N4O3 |
|
—— |
ethyl (5S,7R)-5-[1-(2-methylpropanoyl)piperidin-4-yl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxylate |
—— |
C19H27F3N4O3 |
|
—— |
ethyl (5S,7R)-5-[1-[(1S,2S)-2-methylcyclopropanecarbonyl]piperidin-4-yl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxylate |
—— |
C20H27F3N4O3 |
|
—— |
ethyl (5S,7R)-5-[1-[(3R)-oxolane-3-carbonyl]piperidin-4-yl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxylate |
—— |
C20H27F3N4O4 |
|
—— |
ethyl (5S,7R)-5-[(3S)-1-[(1S,2S)-2-methylcyclopropanecarbonyl]piperidin-3-yl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxylate |
—— |
C20H27F3N4O3 |
|