中文名称 |
英文名称 |
CAS号 |
化学式 |
结构式图片 |
—— |
3-(3,5-dimethylpyrazol-1-yl)-1-[(2R)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]propan-1-one |
—— |
C21H29F3N6O |
|
—— |
(5R,7R)-5-ethyl-2-(1-propan-2-ylsulfonylpiperidin-4-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine |
—— |
C17H27F3N4O2S |
|
—— |
[(2R)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-(4-methyl-1,2,5-oxadiazol-3-yl)methanone |
—— |
C18H23F3N6O2 |
|
—— |
(1,3-dimethylpyrazol-4-yl)-[4-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]methanone |
—— |
C20H27F3N6O |
|
—— |
(2S)-1-[(2S)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]-2-(5-methylpyrazol-1-yl)propan-1-one |
—— |
C20H27F3N6O |
|
—— |
(3,5-dimethyl-1,2-oxazol-4-yl)-[(2S)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]methanone |
—— |
C19H24F3N5O2 |
|
—— |
[(2R)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-(1H-pyrazol-5-yl)methanone |
—— |
C18H23F3N6O |
|
—— |
(2R)-1-[(2S)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]-2-(5-methylpyrazol-1-yl)propan-1-one |
—— |
C20H27F3N6O |
|
—— |
(4R)-4-[(2S)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidine-1-carbonyl]-1-methylpyrrolidin-2-one |
—— |
C20H28F3N5O2 |
|
—— |
(4R)-4-[(2R)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidine-1-carbonyl]-1-methylpyrrolidin-2-one |
—— |
C19H26F3N5O2 |
|
—— |
[(3S)-3-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-pyridin-2-ylmethanone |
—— |
C20H24F3N5O |
|
—— |
2-[2-[(2R)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]-2-oxoethyl]-6-methylpyridazin-3-one |
—— |
C20H25F3N6O2 |
|
—— |
1-[(2R)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]-3-(4-methylpyrazol-1-yl)propan-1-one |
—— |
C20H27F3N6O |
|
—— |
3-(3,5-dimethylpyrazol-1-yl)-1-[(2S)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]propan-1-one |
—— |
C21H29F3N6O |
|
—— |
1-[(2S)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]-3-pyridin-3-ylpropan-1-one |
—— |
C21H26F3N5O |
|
—— |
2-ethyl-1-[4-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]butan-1-one |
—— |
C20H31F3N4O |
|
—— |
[(2R)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-[(2R)-oxolan-2-yl]methanone |
—— |
C19H27F3N4O2 |
|
—— |
[(3S)-1,1-dioxothiolan-3-yl]-[(2R)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]methanone |
—— |
C18H25F3N4O3S |
|
—— |
1-[(2S)-2-[(5R,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]-3-(4-methylpyrazol-1-yl)propan-1-one |
—— |
C20H27F3N6O |
|
—— |
1-[(3R)-3-[(5R,7R)-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]butan-1-one |
—— |
C16H23F3N4O |
|
—— |
5-ethyl-2-[(2S)-1-(1-propylpiperidin-4-yl)pyrrolidin-2-yl]-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine |
—— |
C21H30F3N5 |
|
—— |
1-[(2R)-2-[(5R,7R)-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]butan-1-one |
—— |
C16H23F3N4O |
|
—— |
ethyl (5S,7R)-5-[(3R)-1-butanoylpiperidin-3-yl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxylate |
—— |
C19H27F3N4O3 |
|
—— |
(5S,7S)-5-ethyl-2-[(3R)-1-[(3-methylpyridin-4-yl)methyl]piperidin-3-yl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine |
—— |
C21H28F3N5 |
|
—— |
(2S)-2-[(5S,7R)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]-N,N-dimethylpyrrolidine-1-sulfonamide |
—— |
C15H24F3N5O2S |
|
—— |
(2S)-2-[(5R,7S)-5-ethyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]-N,N-dimethylpyrrolidine-1-sulfonamide |
—— |
C15H24F3N5O2S |
|
—— |
(5R,7S)-5-ethyl-2-[(2S)-1-(1-ethylpyrazol-4-yl)sulfonylpyrrolidin-2-yl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine |
—— |
C18H25F3N6O2S |
|
—— |
1-[(2S)-2-[(5R,7R)-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]butan-1-one |
—— |
C16H23F3N4O |
|
—— |
1-[4-[(5S,7R)-2-tert-butyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]butan-1-one |
—— |
C20H31F3N4O |
|
—— |
1-[4-[(5S,7R)-2-tert-butyl-7-(difluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]butan-1-one |
—— |
C20H32F2N4O |
|
—— |
1-[(2R)-2-(2-tert-butylpyrazolo[1,5-a]pyrimidin-7-yl)piperidin-1-yl]propan-1-one |
—— |
C18H26N4O |
|
—— |
[(1R,2R)-2-methylcyclopropyl]-[(2R)-2-[5-thiophen-2-yl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]methanone |
—— |
C21H21F3N4OS |
|
—— |
[(1R,2S)-2-methylcyclopropyl]-[(2R)-2-[5-thiophen-2-yl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]methanone |
—— |
C21H21F3N4OS |
|
—— |
5-propan-2-yl-2-[(2R)-1-[(3R)-thiolan-3-yl]pyrrolidin-2-yl]-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine |
—— |
C18H23F3N4S |
|
—— |
5-propan-2-yl-2-[(2S)-1-(pyridin-4-ylmethyl)pyrrolidin-2-yl]-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine |
—— |
C20H22F3N5 |
|
—— |
1-[(2S)-2-[5-propan-2-yl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]-2-pyridin-2-ylethanone |
—— |
C21H22F3N5O |
|
—— |
(5S,7R)-5-propan-2-yl-2-[(2S)-1-pyrrolidin-1-ylsulfonylpiperidin-2-yl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine |
—— |
C19H30F3N5O2S |
|
—— |
(1-methylpyrazol-4-yl)-[(2S)-2-[(5S,7R)-5-propan-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]methanone |
—— |
C19H25F3N6O |
|
—— |
[(2S)-oxolan-2-yl]-[(2S)-2-[(5S,7R)-5-propan-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]methanone |
—— |
C20H29F3N4O2 |
|
—— |
cyclopropyl-[(2S)-2-[(5S,7R)-5-propan-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]methanone |
—— |
C18H25F3N4O |
|
—— |
[(3S)-1,1-dioxothiolan-3-yl]-[(3S)-3-[(5S,7R)-5-propan-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]methanone |
—— |
C19H27F3N4O3S |
|
—— |
[(2S)-2-[(5S,7R)-5-propan-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]-(1,3-thiazol-4-yl)methanone |
—— |
C18H22F3N5OS |
|
—— |
(1-methylpyrazol-4-yl)-[(2R)-2-[(5S,7R)-5-propan-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]methanone |
—— |
C19H25F3N6O |
|
—— |
(5S,7R)-5-propan-2-yl-2-[(3R)-1-prop-2-enylsulfonylpyrrolidin-3-yl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine |
—— |
C17H25F3N4O2S |
|
—— |
(1-methylpyrazol-4-yl)-[4-[(5S,7R)-5-propan-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]methanone |
—— |
C20H27F3N6O |
|
—— |
1-[(2R)-2-[(5S,7R)-5-propan-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-2-pyridin-2-ylethanone |
—— |
C22H28F3N5O |
|
—— |
[4-[(5S,7R)-5-propan-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-(1H-pyrazol-5-yl)methanone |
—— |
C19H25F3N6O |
|
—— |
[(2R)-2-[(5S,7R)-5-propan-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-pyrimidin-5-ylmethanone |
—— |
C20H25F3N6O |
|
—— |
(5S,7R)-5-propan-2-yl-2-[(2R)-1-(pyridin-2-ylmethyl)pyrrolidin-2-yl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine |
—— |
C20H26F3N5 |
|
—— |
[(3R)-3-[(5R,7S)-5-propan-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]piperidin-1-yl]-pyridin-4-ylmethanone |
—— |
C21H26F3N5O |
|