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—— ethyl (2Z,5S)-5-(4-methoxyphenyl)-7-methyl-3-oxo-2-[[3-(2-phenoxyethoxy)phenyl]methylidene]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C32H30N2O6S
ethyl (2Z,5S)-5-(4-methoxyphenyl)-7-methyl-3-oxo-2-[[3-(2-phenoxyethoxy)phenyl]methylidene]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2Z,5R)-2-[[4-[2-[4-[(2R)-butan-2-yl]phenoxy]ethoxy]phenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C36H38N2O6S
ethyl (2Z,5R)-2-[[4-[2-[4-[(2R)-butan-2-yl]phenoxy]ethoxy]phenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E)-2-cyano-N-(2,3-dimethylcyclohexyl)-3-phenylprop-2-enamide —— C18H22N2O
(E)-2-cyano-N-(2,3-dimethylcyclohexyl)-3-phenylprop-2-enamide
—— ethyl (2Z,5R)-2-[[4-[2-(3,5-dimethylphenoxy)ethoxy]-3-methoxyphenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C35H36N2O7S
ethyl (2Z,5R)-2-[[4-[2-(3,5-dimethylphenoxy)ethoxy]-3-methoxyphenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E)-2-cyano-3-[3-(cyanomethoxy)phenyl]-N-(3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)prop-2-enamide —— C21H16N4O2S
(E)-2-cyano-3-[3-(cyanomethoxy)phenyl]-N-(3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)prop-2-enamide
—— (E)-3-(3,4-dimethoxyphenyl)-1-(2-phenyl-4-propylimidazo[1,2-a]benzimidazol-1-yl)prop-2-en-1-one —— C29H27N3O3
(E)-3-(3,4-dimethoxyphenyl)-1-(2-phenyl-4-propylimidazo[1,2-a]benzimidazol-1-yl)prop-2-en-1-one
—— ethyl (2Z,5S)-2-[[4-[2-(3,5-dimethylphenoxy)ethoxy]-3-methoxyphenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C35H36N2O7S
ethyl (2Z,5S)-2-[[4-[2-(3,5-dimethylphenoxy)ethoxy]-3-methoxyphenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2Z,5R)-5-(4-methoxyphenyl)-7-methyl-3-oxo-2-[[3-(2-phenoxyethoxy)phenyl]methylidene]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C32H30N2O6S
ethyl (2Z,5R)-5-(4-methoxyphenyl)-7-methyl-3-oxo-2-[[3-(2-phenoxyethoxy)phenyl]methylidene]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2Z,5S)-2-[[3-ethoxy-4-[2-(4-methylphenoxy)ethoxy]phenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C35H36N2O7S
ethyl (2Z,5S)-2-[[3-ethoxy-4-[2-(4-methylphenoxy)ethoxy]phenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E)-1-(5-bromo-2-hydroxyphenyl)-3-(6-chloro-4H-1,3-benzodioxin-8-yl)prop-2-en-1-one —— C17H12BrClO4
(E)-1-(5-bromo-2-hydroxyphenyl)-3-(6-chloro-4H-1,3-benzodioxin-8-yl)prop-2-en-1-one
—— ethyl (2Z,5S)-5-(4-methoxyphenyl)-7-methyl-2-[[3-[2-(4-methylphenoxy)ethoxy]phenyl]methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C33H32N2O6S
ethyl (2Z,5S)-5-(4-methoxyphenyl)-7-methyl-2-[[3-[2-(4-methylphenoxy)ethoxy]phenyl]methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl 8-(trifluoromethyl)-4-[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]quinoline-3-carboxylate —— C23H27F3N2O2
ethyl 8-(trifluoromethyl)-4-[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]quinoline-3-carboxylate
—— ethyl (2Z,5R)-2-[[4-[2-(4-chloro-3-methylphenoxy)ethoxy]phenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C33H31ClN2O6S
ethyl (2Z,5R)-2-[[4-[2-(4-chloro-3-methylphenoxy)ethoxy]phenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2Z,5S)-2-[[4-(benzenesulfonyloxy)-3-methoxyphenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C31H28N2O8S2
ethyl (2Z,5S)-2-[[4-(benzenesulfonyloxy)-3-methoxyphenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E)-N-[[5-benzylsulfanyl-4-(2,4-dichlorophenyl)-1,2,4-triazol-3-yl]methyl]-3-phenylprop-2-enamide —— C25H20Cl2N4OS
(E)-N-[[5-benzylsulfanyl-4-(2,4-dichlorophenyl)-1,2,4-triazol-3-yl]methyl]-3-phenylprop-2-enamide
—— ethyl (2Z,5S)-2-[[3-ethoxy-4-(2-phenoxyethoxy)phenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C34H34N2O7S
ethyl (2Z,5S)-2-[[3-ethoxy-4-(2-phenoxyethoxy)phenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E)-N-[4-chloro-3-[(4-chlorophenyl)sulfamoyl]phenyl]-3-phenylprop-2-enamide —— C21H16Cl2N2O3S
(E)-N-[4-chloro-3-[(4-chlorophenyl)sulfamoyl]phenyl]-3-phenylprop-2-enamide
—— ethyl (2Z,5R)-2-[[3-ethoxy-4-[2-(4-methylphenoxy)ethoxy]phenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C35H36N2O7S
ethyl (2Z,5R)-2-[[3-ethoxy-4-[2-(4-methylphenoxy)ethoxy]phenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (6R)-6-methyl-2-[[2-[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]acetyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C24H36N2O3S
ethyl (6R)-6-methyl-2-[[2-[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]acetyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— [(E)-[(1S,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanylidene]amino] hydrogen carbonate —— C11H17NO3
[(E)-[(1S,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanylidene]amino] hydrogen carbonate
—— ethyl (2Z,5R)-2-[[3-methoxy-4-[2-(4-methylphenoxy)ethoxy]phenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C34H34N2O7S
ethyl (2Z,5R)-2-[[3-methoxy-4-[2-(4-methylphenoxy)ethoxy]phenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2Z,5S)-2-[[4-[2-[4-[(2R)-butan-2-yl]phenoxy]ethoxy]phenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C36H38N2O6S
ethyl (2Z,5S)-2-[[4-[2-[4-[(2R)-butan-2-yl]phenoxy]ethoxy]phenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2Z,5S)-5-(4-methoxyphenyl)-7-methyl-3-oxo-2-[[2-(2-phenoxyethoxy)phenyl]methylidene]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C32H30N2O6S
ethyl (2Z,5S)-5-(4-methoxyphenyl)-7-methyl-3-oxo-2-[[2-(2-phenoxyethoxy)phenyl]methylidene]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl 3-[[(1S,4S)-4,7,7-trimethyl-3-oxo-2-oxabicyclo[2.2.1]heptane-1-carbonyl]amino]benzoate —— C19H23NO5
ethyl 3-[[(1S,4S)-4,7,7-trimethyl-3-oxo-2-oxabicyclo[2.2.1]heptane-1-carbonyl]amino]benzoate
—— ethyl (2Z,5S)-2-[[3-methoxy-4-(2-phenoxyethoxy)phenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C33H32N2O7S
ethyl (2Z,5S)-2-[[3-methoxy-4-(2-phenoxyethoxy)phenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2Z,5S)-2-[[3-methoxy-4-[2-(3-methoxyphenoxy)ethoxy]phenyl]methylidene]-7-methyl-3-oxo-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C33H32N2O7S
ethyl (2Z,5S)-2-[[3-methoxy-4-[2-(3-methoxyphenoxy)ethoxy]phenyl]methylidene]-7-methyl-3-oxo-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2Z,5R)-2-[[3-ethoxy-4-(2-phenoxyethoxy)phenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C34H34N2O7S
ethyl (2Z,5R)-2-[[3-ethoxy-4-(2-phenoxyethoxy)phenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E)-2-(2-(benzo[d][1,3]dioxol-5-yl)vinyl)-3-ethylquinazolin-4(3H)-one —— C19H16N2O3
(E)-2-(2-(benzo[d][1,3]dioxol-5-yl)vinyl)-3-ethylquinazolin-4(3H)-one
—— (E)-1-[(7E)-3-(4-chlorophenyl)-7-[(4-chlorophenyl)methylidene]-3a,4,5,6-tetrahydro-3H-indazol-2-yl]-3-[4-(difluoromethylsulfanyl)phenyl]prop-2-en-1-one —— C30H24Cl2F2N2OS
(E)-1-[(7E)-3-(4-chlorophenyl)-7-[(4-chlorophenyl)methylidene]-3a,4,5,6-tetrahydro-3H-indazol-2-yl]-3-[4-(difluoromethylsulfanyl)phenyl]prop-2-en-1-one
—— ethyl (2Z,5R)-2-[[4-(benzenesulfonyloxy)-3-methoxyphenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C31H28N2O8S2
ethyl (2Z,5R)-2-[[4-(benzenesulfonyloxy)-3-methoxyphenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2Z,5R)-2-[[4-[2-(4-tert-butylphenoxy)ethoxy]phenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C36H38N2O6S
ethyl (2Z,5R)-2-[[4-[2-(4-tert-butylphenoxy)ethoxy]phenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2Z,5R)-2-[[3-methoxy-4-(2-phenoxyethoxy)phenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C33H32N2O7S
ethyl (2Z,5R)-2-[[3-methoxy-4-(2-phenoxyethoxy)phenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl 2-[[(1S,4S)-4,7,7-trimethyl-3-oxo-2-oxabicyclo[2.2.1]heptane-1-carbonyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C21H27NO5S
ethyl 2-[[(1S,4S)-4,7,7-trimethyl-3-oxo-2-oxabicyclo[2.2.1]heptane-1-carbonyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— (E)-N-(3-benzylsulfanyl-5-methyl-1,2,4-triazol-4-yl)-1-[2-(4-methylpiperazin-1-yl)-5-nitrophenyl]methanimine —— C22H25N7O2S
(E)-N-(3-benzylsulfanyl-5-methyl-1,2,4-triazol-4-yl)-1-[2-(4-methylpiperazin-1-yl)-5-nitrophenyl]methanimine
—— ethyl (2Z,5S)-2-[[4-[2-(4-chloro-3-methylphenoxy)ethoxy]phenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C33H31ClN2O6S
ethyl (2Z,5S)-2-[[4-[2-(4-chloro-3-methylphenoxy)ethoxy]phenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2Z,5S)-2-[[4-[2-[4-[(2S)-butan-2-yl]phenoxy]ethoxy]phenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C36H38N2O6S
ethyl (2Z,5S)-2-[[4-[2-[4-[(2S)-butan-2-yl]phenoxy]ethoxy]phenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E)-1-[(1S,5S)-3-methyl-3,8-diazabicyclo[3.2.1]octan-8-yl]-3-phenylprop-2-en-1-one —— C16H20N2O
(E)-1-[(1S,5S)-3-methyl-3,8-diazabicyclo[3.2.1]octan-8-yl]-3-phenylprop-2-en-1-one
—— ethyl (2Z,5S)-2-[[3-methoxy-4-[2-(4-methylphenoxy)ethoxy]phenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C34H34N2O7S
ethyl (2Z,5S)-2-[[3-methoxy-4-[2-(4-methylphenoxy)ethoxy]phenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2Z,5R)-2-[[4-[2-[4-[(2S)-butan-2-yl]phenoxy]ethoxy]phenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C36H38N2O6S
ethyl (2Z,5R)-2-[[4-[2-[4-[(2S)-butan-2-yl]phenoxy]ethoxy]phenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2Z,5S)-2-[[4-[2-(4-tert-butylphenoxy)ethoxy]phenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C36H38N2O6S
ethyl (2Z,5S)-2-[[4-[2-(4-tert-butylphenoxy)ethoxy]phenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (3S,5S)-2-imino-5-methylthiane-3-carboxylate —— C9H15NO2S
ethyl (3S,5S)-2-imino-5-methylthiane-3-carboxylate
—— ethyl (2Z,5R)-5-(4-methoxyphenyl)-7-methyl-3-oxo-2-[[4-(2-phenoxyethoxy)phenyl]methylidene]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C32H30N2O6S
ethyl (2Z,5R)-5-(4-methoxyphenyl)-7-methyl-3-oxo-2-[[4-(2-phenoxyethoxy)phenyl]methylidene]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2Z)-2-[(1-benzylindol-3-yl)methylidene]-5-(4-chlorophenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C32H26ClN3O3S
ethyl (2Z)-2-[(1-benzylindol-3-yl)methylidene]-5-(4-chlorophenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2Z)-3-amino-2-[(2-phenylpropanethioyl)amino]but-2-enoate —— C15H20N2O2S
ethyl (2Z)-3-amino-2-[(2-phenylpropanethioyl)amino]but-2-enoate
—— (E)-N-[4-[5-[2-(4-acetamidoanilino)-2-oxoethyl]sulfanyl-4-ethyl-1,2,4-triazol-3-yl]phenyl]-3-phenylprop-2-enamide —— C29H28N6O3S
(E)-N-[4-[5-[2-(4-acetamidoanilino)-2-oxoethyl]sulfanyl-4-ethyl-1,2,4-triazol-3-yl]phenyl]-3-phenylprop-2-enamide
—— ethyl 4-[[(1R,4S)-3,3-dimethyl-2-methylidenebicyclo[2.2.1]heptane-1-carbonyl]amino]benzoate —— C20H25NO3
ethyl 4-[[(1R,4S)-3,3-dimethyl-2-methylidenebicyclo[2.2.1]heptane-1-carbonyl]amino]benzoate
—— (E)-N-(3-benzylsulfanyl-1,2,4-triazol-4-yl)-1-[2-(4-methylpiperazin-1-yl)-5-nitrophenyl]methanimine —— C21H23N7O2S
(E)-N-(3-benzylsulfanyl-1,2,4-triazol-4-yl)-1-[2-(4-methylpiperazin-1-yl)-5-nitrophenyl]methanimine
—— (E)-N-[4-(hexylsulfamoyl)phenyl]-3-(3-nitrophenyl)prop-2-enamide —— C21H25N3O5S
(E)-N-[4-(hexylsulfamoyl)phenyl]-3-(3-nitrophenyl)prop-2-enamide
—— ethyl 4-[(1S,4S)-4,7,7-trimethyl-3-oxo-2-oxabicyclo[2.2.1]heptane-1-carbonyl]piperazine-1-carboxylate —— C17H26N2O5
ethyl 4-[(1S,4S)-4,7,7-trimethyl-3-oxo-2-oxabicyclo[2.2.1]heptane-1-carbonyl]piperazine-1-carboxylate
—— (E)-N-[[5-(5-butan-2-yl-1,3-benzoxazol-2-yl)-2-chlorophenyl]carbamothioyl]-3-phenylprop-2-enamide —— C27H24ClN3O2S
(E)-N-[[5-(5-butan-2-yl-1,3-benzoxazol-2-yl)-2-chlorophenyl]carbamothioyl]-3-phenylprop-2-enamide