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—— 5-[(S)-(2,5-dimethoxyphenyl)-[(3S)-3-methylpiperidin-1-ium-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C20H27N4O3S+
5-[(S)-(2,5-dimethoxyphenyl)-[(3S)-3-methylpiperidin-1-ium-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-(2-methylphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C19H24N4O2S
5-[(S)-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-(2-methylphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-[(2S,6R)-2,6-dimethylmorpholin-4-yl]-(2-methylphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C19H24N4O2S
5-[(S)-[(2S,6R)-2,6-dimethylmorpholin-4-yl]-(2-methylphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-(4-ethylpiperazin-1-yl)-(2-methoxyphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C19H25N5O2S
5-[(S)-(4-ethylpiperazin-1-yl)-(2-methoxyphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-(2,4-dimethoxyphenyl)-[(3S)-3-methylpiperidin-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C20H26N4O3S
5-[(R)-(2,4-dimethoxyphenyl)-[(3S)-3-methylpiperidin-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-[(3S,5S)-3,5-dimethylpiperidin-1-ium-1-yl]-(2-methoxyphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C20H27N4O2S+
5-[(S)-[(3S,5S)-3,5-dimethylpiperidin-1-ium-1-yl]-(2-methoxyphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-(2,5-dimethoxyphenyl)-[(3S)-3-methylpiperidin-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C20H26N4O3S
5-[(R)-(2,5-dimethoxyphenyl)-[(3S)-3-methylpiperidin-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-(2-methoxyphenyl)-(4-methylpiperidin-1-ium-1-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C19H25N4O2S+
5-[(R)-(2-methoxyphenyl)-(4-methylpiperidin-1-ium-1-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-(Azepan-1-ylsulfonyl)-1,3-dimethylpyrimidine-2,4-dione —— C12H19N3O4S
5-(Azepan-1-ylsulfonyl)-1,3-dimethylpyrimidine-2,4-dione
—— 5-[(S)-(2,5-dimethoxyphenyl)-pyrrolidin-1-ium-1-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C18H23N4O3S+
5-[(S)-(2,5-dimethoxyphenyl)-pyrrolidin-1-ium-1-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-(2,5-dimethoxyphenyl)-[(3S,5R)-3,5-dimethylpiperidin-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C21H28N4O3S
5-[(R)-(2,5-dimethoxyphenyl)-[(3S,5R)-3,5-dimethylpiperidin-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-(2,5-dimethoxyphenyl)-(4-methylpiperidin-1-ium-1-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C20H27N4O3S+
5-[(R)-(2,5-dimethoxyphenyl)-(4-methylpiperidin-1-ium-1-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-(2-methoxyphenyl)-(4-methylpiperidin-1-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C19H24N4O2S
5-[(S)-(2-methoxyphenyl)-(4-methylpiperidin-1-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(2R)-2-ethylpiperidin-1-yl]sulfonyl-1,3,6-trimethylpyrimidine-2,4-dione —— C14H23N3O4S
5-[(2R)-2-ethylpiperidin-1-yl]sulfonyl-1,3,6-trimethylpyrimidine-2,4-dione
—— 5-[(R)-(2-methoxyphenyl)-piperidin-1-ium-1-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C18H23N4O2S+
5-[(R)-(2-methoxyphenyl)-piperidin-1-ium-1-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-(1,4-dioxa-8-azaspiro[4.5]decan-8-ylsulfonyl)-1,3,6-trimethylpyrimidine-2,4(1H,3H)-dione —— C14H21N3O6S
5-(1,4-dioxa-8-azaspiro[4.5]decan-8-ylsulfonyl)-1,3,6-trimethylpyrimidine-2,4(1H,3H)-dione
—— 5-[(2R,6S)-2,6-dimethylmorpholin-4-yl]sulfonyl-1,3,6-trimethylpyrimidine-2,4-dione —— C13H21N3O5S
5-[(2R,6S)-2,6-dimethylmorpholin-4-yl]sulfonyl-1,3,6-trimethylpyrimidine-2,4-dione
—— 5-[(3R,5R)-3,5-dimethylpiperidin-1-yl]sulfonyl-1,3-dimethylpyrimidine-2,4-dione —— C13H21N3O4S
5-[(3R,5R)-3,5-dimethylpiperidin-1-yl]sulfonyl-1,3-dimethylpyrimidine-2,4-dione
—— 5-[(3S,5S)-3,5-dimethylpiperidin-1-yl]sulfonyl-1,3-dimethylpyrimidine-2,4-dione —— C13H21N3O4S
5-[(3S,5S)-3,5-dimethylpiperidin-1-yl]sulfonyl-1,3-dimethylpyrimidine-2,4-dione
—— 5-[(2R,6R)-2,6-dimethylmorpholin-4-yl]sulfonyl-1,3,6-trimethylpyrimidine-2,4-dione —— C13H21N3O5S
5-[(2R,6R)-2,6-dimethylmorpholin-4-yl]sulfonyl-1,3,6-trimethylpyrimidine-2,4-dione
—— 5-[(R)-(2,4-dimethoxyphenyl)-pyrrolidin-1-ium-1-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C18H23N4O3S+
5-[(R)-(2,4-dimethoxyphenyl)-pyrrolidin-1-ium-1-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— (5-Methyl-2-propan-2-ylphenyl) 1,3,4-trimethyl-2,6-dioxopyrimidine-5-sulfonate —— C17H22N2O5S
(5-Methyl-2-propan-2-ylphenyl) 1,3,4-trimethyl-2,6-dioxopyrimidine-5-sulfonate
—— (5-chloro-1-methylimidazol-2-yl)methyl (2R)-2-methyl-3-oxo-4H-1,4-benzoxazine-8-carboxylate —— C15H14ClN3O4
(5-chloro-1-methylimidazol-2-yl)methyl (2R)-2-methyl-3-oxo-4H-1,4-benzoxazine-8-carboxylate
—— (5-chloro-1-methylimidazol-2-yl)methyl (2S)-2-methyl-3-oxo-4H-1,4-benzoxazine-8-carboxylate —— C15H14ClN3O4
(5-chloro-1-methylimidazol-2-yl)methyl (2S)-2-methyl-3-oxo-4H-1,4-benzoxazine-8-carboxylate
—— 5-[[(1S)-1-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]amino]-3H-1,3-benzoxazol-2-one —— C12H12N4O3
5-[[(1S)-1-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]amino]-3H-1,3-benzoxazol-2-one
—— (5R)-3-(4-bromophenyl)-7-(4-fluorophenyl)-1-oxa-2,7-diazaspiro[4.4]non-2-ene-6,8-dione —— C18H12BrFN2O3
(5R)-3-(4-bromophenyl)-7-(4-fluorophenyl)-1-oxa-2,7-diazaspiro[4.4]non-2-ene-6,8-dione
—— 5,6-dimethyl-4-[(3R)-3-(1,2,4-triazol-1-yl)piperidin-1-yl]thieno[2,3-d]pyrimidine —— C15H18N6S
5,6-dimethyl-4-[(3R)-3-(1,2,4-triazol-1-yl)piperidin-1-yl]thieno[2,3-d]pyrimidine
—— (5R)-7-naphthalen-2-yl-3-(3-nitrophenyl)-1-oxa-2,7-diazaspiro[4.4]non-2-ene-6,8-dione —— C22H15N3O5
(5R)-7-naphthalen-2-yl-3-(3-nitrophenyl)-1-oxa-2,7-diazaspiro[4.4]non-2-ene-6,8-dione
—— 5-[(2S)-6-(benzenesulfonyl)-6-azaspiro[2.5]octan-2-yl]-3-(3-chlorophenyl)-1,2,4-oxadiazole —— C21H20ClN3O3S
5-[(2S)-6-(benzenesulfonyl)-6-azaspiro[2.5]octan-2-yl]-3-(3-chlorophenyl)-1,2,4-oxadiazole
—— (5S)-5-(2-fluorophenyl)-4-[hydroxy-[(2S)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]methylidene]-1-(2-methoxyethyl)pyrrolidine-2,3-dione —— C23H22FNO5
(5S)-5-(2-fluorophenyl)-4-[hydroxy-[(2S)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]methylidene]-1-(2-methoxyethyl)pyrrolidine-2,3-dione
—— 5-[(2R)-6-(benzenesulfonyl)-6-azaspiro[2.5]octan-2-yl]-3-(3-chlorophenyl)-1,2,4-oxadiazole —— C21H20ClN3O3S
5-[(2R)-6-(benzenesulfonyl)-6-azaspiro[2.5]octan-2-yl]-3-(3-chlorophenyl)-1,2,4-oxadiazole
—— (5R)-7-(4-methylphenyl)-3-(4-nitrophenyl)-1-oxa-2,7-diazaspiro[4.4]non-2-ene-6,8-dione —— C19H15N3O5
(5R)-7-(4-methylphenyl)-3-(4-nitrophenyl)-1-oxa-2,7-diazaspiro[4.4]non-2-ene-6,8-dione
—— (5R)-5-(2-fluorophenyl)-4-[hydroxy-[(2S)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]methylidene]-1-(2-methoxyethyl)pyrrolidine-2,3-dione —— C23H22FNO5
(5R)-5-(2-fluorophenyl)-4-[hydroxy-[(2S)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]methylidene]-1-(2-methoxyethyl)pyrrolidine-2,3-dione
—— 5,6-dimethyl-4-[(3S)-3-(1,2,4-triazol-1-yl)piperidin-1-yl]thieno[2,3-d]pyrimidine —— C15H18N6S
5,6-dimethyl-4-[(3S)-3-(1,2,4-triazol-1-yl)piperidin-1-yl]thieno[2,3-d]pyrimidine
—— (5S)-4-[(4-chlorophenyl)-hydroxymethylidene]-1-(5-methyl-1,2-oxazol-3-yl)-5-pyridin-4-ylpyrrolidine-2,3-dione —— C20H14ClN3O4
(5S)-4-[(4-chlorophenyl)-hydroxymethylidene]-1-(5-methyl-1,2-oxazol-3-yl)-5-pyridin-4-ylpyrrolidine-2,3-dione
—— (5S)-5-(2-fluorophenyl)-4-[hydroxy-[(2R)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]methylidene]-1-(2-methoxyethyl)pyrrolidine-2,3-dione —— C23H22FNO5
(5S)-5-(2-fluorophenyl)-4-[hydroxy-[(2R)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]methylidene]-1-(2-methoxyethyl)pyrrolidine-2,3-dione
—— (5S)-4-[2,3-dihydro-1,4-benzodioxin-6-yl(hydroxy)methylidene]-1-(3-methoxypropyl)-5-(5-methylfuran-2-yl)pyrrolidine-2,3-dione —— C22H23NO7
(5S)-4-[2,3-dihydro-1,4-benzodioxin-6-yl(hydroxy)methylidene]-1-(3-methoxypropyl)-5-(5-methylfuran-2-yl)pyrrolidine-2,3-dione
—— (5R)-4-[2,3-dihydro-1,4-benzodioxin-6-yl(hydroxy)methylidene]-5-(2-fluorophenyl)-1-(2-methoxyethyl)pyrrolidine-2,3-dione —— C22H20FNO6
(5R)-4-[2,3-dihydro-1,4-benzodioxin-6-yl(hydroxy)methylidene]-5-(2-fluorophenyl)-1-(2-methoxyethyl)pyrrolidine-2,3-dione
—— (5R)-3-(2,5-difluorophenyl)-N-[3-(2-methylimidazol-1-yl)propyl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C17H18F2N4O2
(5R)-3-(2,5-difluorophenyl)-N-[3-(2-methylimidazol-1-yl)propyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5S)-7-(4-methylphenyl)-3-(4-nitrophenyl)-1-oxa-2,7-diazaspiro[4.4]non-2-ene-6,8-dione —— C19H15N3O5
(5S)-7-(4-methylphenyl)-3-(4-nitrophenyl)-1-oxa-2,7-diazaspiro[4.4]non-2-ene-6,8-dione
—— 5-bromo-6-oxo-N-(2-piperidin-1-ium-1-ylethyl)pyran-3-carboxamide —— C13H18BrN2O3+
5-bromo-6-oxo-N-(2-piperidin-1-ium-1-ylethyl)pyran-3-carboxamide
—— (5R)-1-[(2S)-butan-2-yl]-5-[2-(cyclohexen-1-yl)ethyliminomethyl]-2-sulfanylidene-1,3-diazinane-4,6-dione —— C17H25N3O2S
(5R)-1-[(2S)-butan-2-yl]-5-[2-(cyclohexen-1-yl)ethyliminomethyl]-2-sulfanylidene-1,3-diazinane-4,6-dione
—— (5R)-1-(4-methylphenyl)-5-(3-morpholin-4-ylpropyliminomethyl)-2-sulfanylidene-1,3-diazinane-4,6-dione —— C19H24N4O3S
(5R)-1-(4-methylphenyl)-5-(3-morpholin-4-ylpropyliminomethyl)-2-sulfanylidene-1,3-diazinane-4,6-dione
—— (5S)-3-(2,5-difluorophenyl)-N-[2-(pyrimidin-2-ylamino)ethyl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C16H15F2N5O2
(5S)-3-(2,5-difluorophenyl)-N-[2-(pyrimidin-2-ylamino)ethyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5R)-5-[2-(cyclohexen-1-yl)ethyliminomethyl]-1-[(4-fluorophenyl)methyl]-2-sulfanylidene-1,3-diazinane-4,6-dione —— C20H22FN3O2S
(5R)-5-[2-(cyclohexen-1-yl)ethyliminomethyl]-1-[(4-fluorophenyl)methyl]-2-sulfanylidene-1,3-diazinane-4,6-dione
—— 5-(C-ethyl-N-hexylcarbonimidoyl)-1,3-diazinane-2,4,6-trione —— C13H21N3O3
5-(C-ethyl-N-hexylcarbonimidoyl)-1,3-diazinane-2,4,6-trione
—— 5-[C-ethyl-N-(3-piperidin-1-ylpropyl)carbonimidoyl]-1-phenyl-1,3-diazinane-2,4,6-trione —— C21H28N4O3
5-[C-ethyl-N-(3-piperidin-1-ylpropyl)carbonimidoyl]-1-phenyl-1,3-diazinane-2,4,6-trione
—— 5,6-dimethyl-3-[(2S)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]pyridazine-4-carbonitrile —— C15H18N6
5,6-dimethyl-3-[(2S)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]pyridazine-4-carbonitrile
—— (5S)-4-[(4-fluorophenyl)-hydroxymethylidene]-1-(5-methyl-1,2-oxazol-3-yl)-5-pyridin-3-ylpyrrolidine-2,3-dione —— C20H14FN3O4
(5S)-4-[(4-fluorophenyl)-hydroxymethylidene]-1-(5-methyl-1,2-oxazol-3-yl)-5-pyridin-3-ylpyrrolidine-2,3-dione
—— (5R)-5-[[(1S,2R)-2-aminocyclohexyl]iminomethyl]-1-(2-methoxyphenyl)-2-sulfanylidene-1,3-diazinane-4,6-dione —— C18H22N4O3S
(5R)-5-[[(1S,2R)-2-aminocyclohexyl]iminomethyl]-1-(2-methoxyphenyl)-2-sulfanylidene-1,3-diazinane-4,6-dione