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—— 5-[(2S)-3-(2,4-dichlorophenoxy)-2-hydroxypropyl]-1-(2-nitrophenyl)pyrazolo[3,4-d]pyrimidin-4-one —— C20H15Cl2N5O5
5-[(2S)-3-(2,4-dichlorophenoxy)-2-hydroxypropyl]-1-(2-nitrophenyl)pyrazolo[3,4-d]pyrimidin-4-one
—— 5-[(2R)-3-(4-bromophenoxy)-2-hydroxypropyl]-1-(2-nitrophenyl)pyrazolo[3,4-d]pyrimidin-4-one —— C20H16BrN5O5
5-[(2R)-3-(4-bromophenoxy)-2-hydroxypropyl]-1-(2-nitrophenyl)pyrazolo[3,4-d]pyrimidin-4-one
—— 5-bromo-N-[(2R)-1-oxo-1-[4-(pyridin-3-ylmethylsulfanyl)anilino]propan-2-yl]thiophene-2-carboxamide —— C20H18BrN3O2S2
5-bromo-N-[(2R)-1-oxo-1-[4-(pyridin-3-ylmethylsulfanyl)anilino]propan-2-yl]thiophene-2-carboxamide
—— 5-bromo-N-[(2R)-1-[[(2R)-2-(diethylamino)-2-(3-methoxyphenyl)ethyl]amino]-1-oxopropan-2-yl]thiophene-2-carboxamide —— C21H28BrN3O3S
5-bromo-N-[(2R)-1-[[(2R)-2-(diethylamino)-2-(3-methoxyphenyl)ethyl]amino]-1-oxopropan-2-yl]thiophene-2-carboxamide
—— 5-[(2R)-3-(2,4-dichlorophenoxy)-2-hydroxypropyl]-1-(2-nitrophenyl)pyrazolo[3,4-d]pyrimidin-4-one —— C20H15Cl2N5O5
5-[(2R)-3-(2,4-dichlorophenoxy)-2-hydroxypropyl]-1-(2-nitrophenyl)pyrazolo[3,4-d]pyrimidin-4-one
—— 5-bromo-N-[(2R)-1-[[(2S)-2-(diethylamino)-2-(3-methoxyphenyl)ethyl]amino]-1-oxopropan-2-yl]thiophene-2-carboxamide —— C21H28BrN3O3S
5-bromo-N-[(2R)-1-[[(2S)-2-(diethylamino)-2-(3-methoxyphenyl)ethyl]amino]-1-oxopropan-2-yl]thiophene-2-carboxamide
—— 5-bromo-N-[(2S)-1-oxo-1-[4-(pyridin-3-ylmethylsulfanyl)anilino]propan-2-yl]thiophene-2-carboxamide —— C20H18BrN3O2S2
5-bromo-N-[(2S)-1-oxo-1-[4-(pyridin-3-ylmethylsulfanyl)anilino]propan-2-yl]thiophene-2-carboxamide
—— 5-[(2S)-3-(4-bromophenoxy)-2-hydroxypropyl]-1-(2-nitrophenyl)pyrazolo[3,4-d]pyrimidin-4-one —— C20H16BrN5O5
5-[(2S)-3-(4-bromophenoxy)-2-hydroxypropyl]-1-(2-nitrophenyl)pyrazolo[3,4-d]pyrimidin-4-one
—— 5-bromo-N-[(2S)-1-[[(2R)-2-(diethylamino)-2-(3-methoxyphenyl)ethyl]amino]-1-oxopropan-2-yl]thiophene-2-carboxamide —— C21H28BrN3O3S
5-bromo-N-[(2S)-1-[[(2R)-2-(diethylamino)-2-(3-methoxyphenyl)ethyl]amino]-1-oxopropan-2-yl]thiophene-2-carboxamide
—— 5-bromo-N-[(2S)-1-[[5-[(2-chlorophenyl)methyl]-1,3-thiazol-2-yl]amino]-1-oxopropan-2-yl]thiophene-2-carboxamide —— C18H15BrClN3O2S2
5-bromo-N-[(2S)-1-[[5-[(2-chlorophenyl)methyl]-1,3-thiazol-2-yl]amino]-1-oxopropan-2-yl]thiophene-2-carboxamide
—— 5-[(2R)-3-(2,5-dichlorophenoxy)-2-hydroxypropyl]-1-(2-nitrophenyl)pyrazolo[3,4-d]pyrimidin-4-one —— C20H15Cl2N5O5
5-[(2R)-3-(2,5-dichlorophenoxy)-2-hydroxypropyl]-1-(2-nitrophenyl)pyrazolo[3,4-d]pyrimidin-4-one
—— 5-bromo-N-[(2R)-1-[[4-(4-fluorophenyl)-5-methyl-1,3-thiazol-2-yl]amino]-1-oxopropan-2-yl]thiophene-2-carboxamide —— C18H15BrFN3O2S2
5-bromo-N-[(2R)-1-[[4-(4-fluorophenyl)-5-methyl-1,3-thiazol-2-yl]amino]-1-oxopropan-2-yl]thiophene-2-carboxamide
—— 5-bromo-N-[(2S)-1-[[4-(4-fluorophenyl)-5-methyl-1,3-thiazol-2-yl]amino]-1-oxopropan-2-yl]thiophene-2-carboxamide —— C18H15BrFN3O2S2
5-bromo-N-[(2S)-1-[[4-(4-fluorophenyl)-5-methyl-1,3-thiazol-2-yl]amino]-1-oxopropan-2-yl]thiophene-2-carboxamide
—— 5-bromo-N-[(2R)-1-[[1-(2,3-dihydro-1,4-benzodioxin-6-yl)cyclopentyl]methylamino]-1-oxopropan-2-yl]thiophene-2-carboxamide —— C22H25BrN2O4S
5-bromo-N-[(2R)-1-[[1-(2,3-dihydro-1,4-benzodioxin-6-yl)cyclopentyl]methylamino]-1-oxopropan-2-yl]thiophene-2-carboxamide
—— 5-bromo-N-[(2S)-1-[[4-(4-methoxyphenyl)-5-methyl-1,3-thiazol-2-yl]amino]-1-oxopropan-2-yl]thiophene-2-carboxamide —— C19H18BrN3O3S2
5-bromo-N-[(2S)-1-[[4-(4-methoxyphenyl)-5-methyl-1,3-thiazol-2-yl]amino]-1-oxopropan-2-yl]thiophene-2-carboxamide
—— 5-bromo-N-[(2S)-1-[[1-(2,3-dihydro-1,4-benzodioxin-6-yl)cyclopentyl]methylamino]-1-oxopropan-2-yl]thiophene-2-carboxamide —— C22H25BrN2O4S
5-bromo-N-[(2S)-1-[[1-(2,3-dihydro-1,4-benzodioxin-6-yl)cyclopentyl]methylamino]-1-oxopropan-2-yl]thiophene-2-carboxamide
—— 5-bromo-N-[(2S)-1-[[4-(3-fluoro-4-methoxyphenyl)-1,3-thiazol-2-yl]amino]-1-oxopropan-2-yl]thiophene-2-carboxamide —— C18H15BrFN3O3S2
5-bromo-N-[(2S)-1-[[4-(3-fluoro-4-methoxyphenyl)-1,3-thiazol-2-yl]amino]-1-oxopropan-2-yl]thiophene-2-carboxamide
—— 5-bromo-N-[(2R)-1-oxo-1-[2-(5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophene-2-carbonyl)hydrazinyl]propan-2-yl]thiophene-2-carboxamide —— C18H20BrN3O3S2
5-bromo-N-[(2R)-1-oxo-1-[2-(5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophene-2-carbonyl)hydrazinyl]propan-2-yl]thiophene-2-carboxamide
—— 5-bromo-N-[(2R)-1-[[4-(3-fluoro-4-methoxyphenyl)-1,3-thiazol-2-yl]amino]-1-oxopropan-2-yl]thiophene-2-carboxamide —— C18H15BrFN3O3S2
5-bromo-N-[(2R)-1-[[4-(3-fluoro-4-methoxyphenyl)-1,3-thiazol-2-yl]amino]-1-oxopropan-2-yl]thiophene-2-carboxamide
—— 5-bromo-N-[(2R)-1-[2-(4,5,6,7,8,9-hexahydrocycloocta[b]thiophene-2-carbonyl)hydrazinyl]-1-oxopropan-2-yl]thiophene-2-carboxamide —— C19H22BrN3O3S2
5-bromo-N-[(2R)-1-[2-(4,5,6,7,8,9-hexahydrocycloocta[b]thiophene-2-carbonyl)hydrazinyl]-1-oxopropan-2-yl]thiophene-2-carboxamide
—— 5-bromo-N-[(2S)-1-oxo-1-[2-(5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophene-2-carbonyl)hydrazinyl]propan-2-yl]thiophene-2-carboxamide —— C18H20BrN3O3S2
5-bromo-N-[(2S)-1-oxo-1-[2-(5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophene-2-carbonyl)hydrazinyl]propan-2-yl]thiophene-2-carboxamide
—— 5-bromo-N-[(2S)-1-[2-(4,5,6,7,8,9-hexahydrocycloocta[b]thiophene-2-carbonyl)hydrazinyl]-1-oxopropan-2-yl]thiophene-2-carboxamide —— C19H22BrN3O3S2
5-bromo-N-[(2S)-1-[2-(4,5,6,7,8,9-hexahydrocycloocta[b]thiophene-2-carbonyl)hydrazinyl]-1-oxopropan-2-yl]thiophene-2-carboxamide
—— 5-[[2-(2-Methoxyethyl)-1,3-dioxoisoindole-5-carbonyl]amino]benzene-1,3-dicarboxylate —— C20H14N2O8-2
5-[[2-(2-Methoxyethyl)-1,3-dioxoisoindole-5-carbonyl]amino]benzene-1,3-dicarboxylate
—— [(5S)-3-(5-chloro-2,4-dimethoxyphenyl)-4,5-dihydro-1,2-oxazol-5-yl]-(4-methylpiperazin-4-ium-1-yl)methanone —— C17H23ClN3O4+
[(5S)-3-(5-chloro-2,4-dimethoxyphenyl)-4,5-dihydro-1,2-oxazol-5-yl]-(4-methylpiperazin-4-ium-1-yl)methanone
—— [(5R)-3-(5-chloro-2,4-dimethoxyphenyl)-4,5-dihydro-1,2-oxazol-5-yl]-(4-methylpiperazin-4-ium-1-yl)methanone —— C17H23ClN3O4+
[(5R)-3-(5-chloro-2,4-dimethoxyphenyl)-4,5-dihydro-1,2-oxazol-5-yl]-(4-methylpiperazin-4-ium-1-yl)methanone
—— (5R)-3-(5-chloro-2,4-dimethoxyphenyl)-N-(3-morpholin-4-ylpropyl)-4,5-dihydro-1,2-oxazole-5-carboxamide —— C19H26ClN3O5
(5R)-3-(5-chloro-2,4-dimethoxyphenyl)-N-(3-morpholin-4-ylpropyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
—— 5-bromo-N-[(2S)-1-[2-[5-(4-fluorophenyl)thiophene-2-carbonyl]hydrazinyl]-1-oxopropan-2-yl]thiophene-2-carboxamide —— C19H15BrFN3O3S2
5-bromo-N-[(2S)-1-[2-[5-(4-fluorophenyl)thiophene-2-carbonyl]hydrazinyl]-1-oxopropan-2-yl]thiophene-2-carboxamide
—— 5-bromo-N-[(2R)-1-[2-[5-(4-fluorophenyl)thiophene-2-carbonyl]hydrazinyl]-1-oxopropan-2-yl]thiophene-2-carboxamide —— C19H15BrFN3O3S2
5-bromo-N-[(2R)-1-[2-[5-(4-fluorophenyl)thiophene-2-carbonyl]hydrazinyl]-1-oxopropan-2-yl]thiophene-2-carboxamide
—— 5-[[2-(4-Methylphenyl)-5-phenylpyrazol-3-yl]amino]-5-oxopentanoate —— C21H20N3O3-
5-[[2-(4-Methylphenyl)-5-phenylpyrazol-3-yl]amino]-5-oxopentanoate
—— 5-[[2-[[cyclopropanecarbonyl(propyl)amino]methyl]pyrrol-1-yl]methyl]-N-cyclopropylfuran-2-carboxamide —— C21H27N3O3
5-[[2-[[cyclopropanecarbonyl(propyl)amino]methyl]pyrrol-1-yl]methyl]-N-cyclopropylfuran-2-carboxamide
—— 5-nitro-2-[4-[(1R)-1-[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]benzonitrile —— C22H19F3N6O3
5-nitro-2-[4-[(1R)-1-[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]benzonitrile
—— (5R)-3-(5-chloro-2,4-dimethoxyphenyl)-N-(3-morpholin-4-ium-4-ylpropyl)-4,5-dihydro-1,2-oxazole-5-carboxamide —— C19H27ClN3O5+
(5R)-3-(5-chloro-2,4-dimethoxyphenyl)-N-(3-morpholin-4-ium-4-ylpropyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5S)-3-(5-chloro-2,4-dimethoxyphenyl)-N-(3-morpholin-4-ylpropyl)-4,5-dihydro-1,2-oxazole-5-carboxamide —— C19H26ClN3O5
(5S)-3-(5-chloro-2,4-dimethoxyphenyl)-N-(3-morpholin-4-ylpropyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
—— 5-(1,3-benzothiazol-2-yl)-N-[[(2S)-1-ethylpyrrolidin-2-yl]methyl]thiophene-2-carboxamide —— C19H21N3OS2
5-(1,3-benzothiazol-2-yl)-N-[[(2S)-1-ethylpyrrolidin-2-yl]methyl]thiophene-2-carboxamide
—— 5-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-[[(2S)-1-ethylpyrrolidin-2-yl]methyl]thiophene-2-carboxamide —— C20H24N2O3S
5-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-[[(2S)-1-ethylpyrrolidin-2-yl]methyl]thiophene-2-carboxamide
—— 5-bromo-N-[(2S)-1-oxo-1-[4-(2-oxo-3H-benzimidazol-1-yl)piperidin-1-yl]propan-2-yl]thiophene-2-carboxamide —— C20H21BrN4O3S
5-bromo-N-[(2S)-1-oxo-1-[4-(2-oxo-3H-benzimidazol-1-yl)piperidin-1-yl]propan-2-yl]thiophene-2-carboxamide
—— 5-(1,3-benzothiazol-2-yl)-N-[[(2R)-1-ethylpyrrolidin-2-yl]methyl]thiophene-2-carboxamide —— C19H21N3OS2
5-(1,3-benzothiazol-2-yl)-N-[[(2R)-1-ethylpyrrolidin-2-yl]methyl]thiophene-2-carboxamide
—— (5S)-3-(5-chloro-2,4-dimethoxyphenyl)-N-(3-morpholin-4-ium-4-ylpropyl)-4,5-dihydro-1,2-oxazole-5-carboxamide —— C19H27ClN3O5+
(5S)-3-(5-chloro-2,4-dimethoxyphenyl)-N-(3-morpholin-4-ium-4-ylpropyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5S,7R)-5-(2-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxylate —— C15H13F3N3O3-
(5S,7R)-5-(2-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxylate
—— 5-Benzyl-2-[(4-fluorophenyl)methylsulfanyl]-3,6-dimethylpyrimidin-4-one —— C20H19FN2OS
5-Benzyl-2-[(4-fluorophenyl)methylsulfanyl]-3,6-dimethylpyrimidin-4-one
—— 5-[(1R)-1-[4-(2,4-dinitrophenyl)piperazin-1-yl]ethyl]-3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazole —— C21H19F3N6O5
5-[(1R)-1-[4-(2,4-dinitrophenyl)piperazin-1-yl]ethyl]-3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazole
—— (5R,7S)-5-(2-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxylate —— C15H13F3N3O3-
(5R,7S)-5-(2-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxylate
—— (5R,7R)-5-(2-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxylate —— C15H13F3N3O3-
(5R,7R)-5-(2-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxylate
—— (5R,7R)-5-(2-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxylic acid —— C15H14F3N3O3
(5R,7R)-5-(2-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxylic acid
—— (5S,7R)-5-(2-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxylic acid —— C15H14F3N3O3
(5S,7R)-5-(2-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxylic acid
—— (5S,7S)-5-(2-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxylate —— C15H13F3N3O3-
(5S,7S)-5-(2-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxylate
—— (5S)-3-(2-chlorophenyl)-N-[[(2S)-oxolan-2-yl]methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C15H17ClN2O3
(5S)-3-(2-chlorophenyl)-N-[[(2S)-oxolan-2-yl]methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5R)-3-(2-chlorophenyl)-N-[[(2R)-oxolan-2-yl]methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C15H17ClN2O3
(5R)-3-(2-chlorophenyl)-N-[[(2R)-oxolan-2-yl]methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5R)-3-(2-chlorophenyl)-N-[[(2S)-oxolan-2-yl]methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C15H17ClN2O3
(5R)-3-(2-chlorophenyl)-N-[[(2S)-oxolan-2-yl]methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5S)-3-(2-chlorophenyl)-N-[[(2R)-oxolan-2-yl]methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C15H17ClN2O3
(5S)-3-(2-chlorophenyl)-N-[[(2R)-oxolan-2-yl]methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide