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—— 5-methoxy-1-methyl-N-[(4S)-1-methyl-4,5,6,7-tetrahydroindazol-4-yl]pyrazole-3-carboxamide —— C14H19N5O2
5-methoxy-1-methyl-N-[(4S)-1-methyl-4,5,6,7-tetrahydroindazol-4-yl]pyrazole-3-carboxamide
—— 5-ethyl-2-methyl-N-[(4S)-1-pyridin-2-yl-4,5,6,7-tetrahydroindazol-4-yl]pyrazole-3-carboxamide —— C19H22N6O
5-ethyl-2-methyl-N-[(4S)-1-pyridin-2-yl-4,5,6,7-tetrahydroindazol-4-yl]pyrazole-3-carboxamide
—— 5-propan-2-yl-N-[(4R)-1-pyridin-2-yl-4,5,6,7-tetrahydroindazol-4-yl]-1,2-oxazole-3-carboxamide —— C19H21N5O2
5-propan-2-yl-N-[(4R)-1-pyridin-2-yl-4,5,6,7-tetrahydroindazol-4-yl]-1,2-oxazole-3-carboxamide
—— 5-methyl-N-[(5R)-2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl]-1H-pyrazole-3-carboxamide —— C19H19N5O
5-methyl-N-[(5R)-2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl]-1H-pyrazole-3-carboxamide
—— (5-methyl-1,2-oxazol-3-yl)methyl (2S)-2-[(4-acetamidophenyl)sulfonylamino]propanoate —— C16H19N3O6S
(5-methyl-1,2-oxazol-3-yl)methyl (2S)-2-[(4-acetamidophenyl)sulfonylamino]propanoate
—— 5-methyl-N-[(5S)-2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl]-1H-pyrazole-3-carboxamide —— C19H19N5O
5-methyl-N-[(5S)-2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl]-1H-pyrazole-3-carboxamide
—— 5-chloro-1-methyl-N-[(4S)-1-pyridin-2-yl-4,5,6,7-tetrahydroindazol-4-yl]pyrazole-4-carboxamide —— C17H17ClN6O
5-chloro-1-methyl-N-[(4S)-1-pyridin-2-yl-4,5,6,7-tetrahydroindazol-4-yl]pyrazole-4-carboxamide
—— 5-chloro-1-methyl-N-[(4R)-1-pyridin-2-yl-4,5,6,7-tetrahydroindazol-4-yl]pyrazole-4-carboxamide —— C17H17ClN6O
5-chloro-1-methyl-N-[(4R)-1-pyridin-2-yl-4,5,6,7-tetrahydroindazol-4-yl]pyrazole-4-carboxamide
—— (5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl (2S)-2-[(3aR,7aS)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]propanoate —— C18H17N3O5S
(5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl (2S)-2-[(3aR,7aS)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]propanoate
—— 5-[(3,5-dimethylpyrazol-1-yl)methyl]-N-[(4S)-1-methyl-4,5,6,7-tetrahydroindazol-4-yl]furan-2-carboxamide —— C19H23N5O2
5-[(3,5-dimethylpyrazol-1-yl)methyl]-N-[(4S)-1-methyl-4,5,6,7-tetrahydroindazol-4-yl]furan-2-carboxamide
—— 5-propan-2-yl-N-[(4S)-1-pyridin-2-yl-4,5,6,7-tetrahydroindazol-4-yl]-1,2-oxazole-3-carboxamide —— C19H21N5O2
5-propan-2-yl-N-[(4S)-1-pyridin-2-yl-4,5,6,7-tetrahydroindazol-4-yl]-1,2-oxazole-3-carboxamide
—— 5-(4-fluorophenyl)-N-[(4R)-1-methyl-4,5,6,7-tetrahydroindazol-4-yl]-1,2-oxazole-3-carboxamide —— C18H17FN4O2
5-(4-fluorophenyl)-N-[(4R)-1-methyl-4,5,6,7-tetrahydroindazol-4-yl]-1,2-oxazole-3-carboxamide
—— 5-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]-N-[(4R)-1-methyl-4,5,6,7-tetrahydroindazol-4-yl]furan-2-carboxamide —— C19H22N4O3
5-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]-N-[(4R)-1-methyl-4,5,6,7-tetrahydroindazol-4-yl]furan-2-carboxamide
—— 5-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]-N-[(4S)-1-methyl-4,5,6,7-tetrahydroindazol-4-yl]furan-2-carboxamide —— C19H22N4O3
5-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]-N-[(4S)-1-methyl-4,5,6,7-tetrahydroindazol-4-yl]furan-2-carboxamide
—— 5-[(3,5-dimethylpyrazol-1-yl)methyl]-N-[(4R)-1-methyl-4,5,6,7-tetrahydroindazol-4-yl]furan-2-carboxamide —— C19H23N5O2
5-[(3,5-dimethylpyrazol-1-yl)methyl]-N-[(4R)-1-methyl-4,5,6,7-tetrahydroindazol-4-yl]furan-2-carboxamide
—— (5-phenyl-1,3,4-oxadiazol-2-yl)methyl (2S)-2-[(3aR,7aS)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]propanoate —— C20H19N3O5
(5-phenyl-1,3,4-oxadiazol-2-yl)methyl (2S)-2-[(3aR,7aS)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]propanoate
—— 5-chloro-1-methyl-N-[(4S)-1-methyl-4,5,6,7-tetrahydroindazol-4-yl]pyrazole-4-carboxamide —— C13H16ClN5O
5-chloro-1-methyl-N-[(4S)-1-methyl-4,5,6,7-tetrahydroindazol-4-yl]pyrazole-4-carboxamide
—— 5-chloro-1-methyl-N-[(4R)-1-methyl-4,5,6,7-tetrahydroindazol-4-yl]pyrazole-4-carboxamide —— C13H16ClN5O
5-chloro-1-methyl-N-[(4R)-1-methyl-4,5,6,7-tetrahydroindazol-4-yl]pyrazole-4-carboxamide
—— 5-fluoro-N-[(4R)-1-methyl-4,5,6,7-tetrahydroindazol-4-yl]-1H-indole-2-carboxamide —— C17H17FN4O
5-fluoro-N-[(4R)-1-methyl-4,5,6,7-tetrahydroindazol-4-yl]-1H-indole-2-carboxamide
—— 5-ethoxy-1-methyl-N-[(4S)-1-pyridin-2-yl-4,5,6,7-tetrahydroindazol-4-yl]pyrazole-3-carboxamide —— C19H22N6O2
5-ethoxy-1-methyl-N-[(4S)-1-pyridin-2-yl-4,5,6,7-tetrahydroindazol-4-yl]pyrazole-3-carboxamide
—— 5-cyclopropyl-2-methyl-N-[(4S)-1-methyl-4,5,6,7-tetrahydroindazol-4-yl]pyrazole-3-carboxamide —— C16H21N5O
5-cyclopropyl-2-methyl-N-[(4S)-1-methyl-4,5,6,7-tetrahydroindazol-4-yl]pyrazole-3-carboxamide
—— 5-ethoxy-1-methyl-N-[(4R)-1-pyridin-2-yl-4,5,6,7-tetrahydroindazol-4-yl]pyrazole-3-carboxamide —— C19H22N6O2
5-ethoxy-1-methyl-N-[(4R)-1-pyridin-2-yl-4,5,6,7-tetrahydroindazol-4-yl]pyrazole-3-carboxamide
—— [5-(4-methylphenyl)thiadiazol-4-yl]-[(3S)-3-methylpiperidin-1-yl]methanone —— C16H19N3OS
[5-(4-methylphenyl)thiadiazol-4-yl]-[(3S)-3-methylpiperidin-1-yl]methanone
—— 5-(4-fluorophenyl)-N-[(4S)-1-methyl-4,5,6,7-tetrahydroindazol-4-yl]-1,2-oxazole-3-carboxamide —— C18H17FN4O2
5-(4-fluorophenyl)-N-[(4S)-1-methyl-4,5,6,7-tetrahydroindazol-4-yl]-1,2-oxazole-3-carboxamide
—— 5-(3,4-difluorophenyl)-N-[(2S)-2-phenylpentyl]-1,2-oxazole-3-carboxamide —— C21H20F2N2O2
5-(3,4-difluorophenyl)-N-[(2S)-2-phenylpentyl]-1,2-oxazole-3-carboxamide
—— (5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl (2S)-2-benzamidopropanoate —— C17H15N3O4S
(5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl (2S)-2-benzamidopropanoate
—— (5-phenyl-1,3,4-oxadiazol-2-yl)methyl 2-[2-(4-oxocyclohexa-2,5-dien-1-ylidene)hydrazinyl]benzoate —— C22H16N4O4
(5-phenyl-1,3,4-oxadiazol-2-yl)methyl 2-[2-(4-oxocyclohexa-2,5-dien-1-ylidene)hydrazinyl]benzoate
—— (5-Phenyl-1,3,4-oxadiazol-2-yl)methyl 3-aminopyrazine-2-carboxylate —— C14H11N5O3
(5-Phenyl-1,3,4-oxadiazol-2-yl)methyl 3-aminopyrazine-2-carboxylate
—— 5-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-[(2S)-2-phenylbutyl]-1,2-oxazole-3-carboxamide —— C22H22N2O4
5-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-[(2S)-2-phenylbutyl]-1,2-oxazole-3-carboxamide
—— 5-[(2R)-2-hydroxy-3-(methylamino)propyl]-1-methylpyrazolo[3,4-d]pyrimidin-4-one —— C10H15N5O2
5-[(2R)-2-hydroxy-3-(methylamino)propyl]-1-methylpyrazolo[3,4-d]pyrimidin-4-one
—— 5-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-[(2R)-2-(dimethylamino)-2-thiophen-3-ylethyl]-1,2-oxazole-3-carboxamide —— C20H21N3O4S
5-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-[(2R)-2-(dimethylamino)-2-thiophen-3-ylethyl]-1,2-oxazole-3-carboxamide
—— 5-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-[(2R)-2-phenylbutyl]-1,2-oxazole-3-carboxamide —— C22H22N2O4
5-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-[(2R)-2-phenylbutyl]-1,2-oxazole-3-carboxamide
—— 5-(3,5-dimethyl-6-oxocyclohexa-2,4-dien-1-ylidene)-N-(4-ethoxyphenyl)-1,2-dihydropyrazole-3-carboxamide —— C20H21N3O3
5-(3,5-dimethyl-6-oxocyclohexa-2,4-dien-1-ylidene)-N-(4-ethoxyphenyl)-1,2-dihydropyrazole-3-carboxamide
—— 5-[(4S)-4-(ethylamino)pentyl]-1-methylpyrazolo[3,4-d]pyrimidin-4-one —— C13H21N5O
5-[(4S)-4-(ethylamino)pentyl]-1-methylpyrazolo[3,4-d]pyrimidin-4-one
—— 5-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-[(2S)-2-(dimethylamino)-2-thiophen-3-ylethyl]-1,2-oxazole-3-carboxamide —— C20H21N3O4S
5-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-[(2S)-2-(dimethylamino)-2-thiophen-3-ylethyl]-1,2-oxazole-3-carboxamide
—— 5-[(2R)-2-hydroxy-3-(propylamino)propyl]-1-methylpyrazolo[3,4-d]pyrimidin-4-one —— C12H19N5O2
5-[(2R)-2-hydroxy-3-(propylamino)propyl]-1-methylpyrazolo[3,4-d]pyrimidin-4-one
—— 5-[(2S)-2-(ethylamino)pentyl]-1-methylpyrazolo[3,4-d]pyrimidin-4-one —— C13H21N5O
5-[(2S)-2-(ethylamino)pentyl]-1-methylpyrazolo[3,4-d]pyrimidin-4-one
—— 5-bromo-N-methyl-N-[[(3S)-1-methylpyrrolidin-3-yl]methyl]thiophene-2-sulfonamide —— C11H17BrN2O2S2
5-bromo-N-methyl-N-[[(3S)-1-methylpyrrolidin-3-yl]methyl]thiophene-2-sulfonamide
—— 5-(3,4-difluorophenyl)-N-[(2R)-2-phenylpentyl]-1,2-oxazole-3-carboxamide —— C21H20F2N2O2
5-(3,4-difluorophenyl)-N-[(2R)-2-phenylpentyl]-1,2-oxazole-3-carboxamide
—— 5-(3,4-difluorophenyl)-N-[(2S)-2-phenylbutyl]-1,2-oxazole-3-carboxamide —— C20H18F2N2O2
5-(3,4-difluorophenyl)-N-[(2S)-2-phenylbutyl]-1,2-oxazole-3-carboxamide
—— 5-[(2S)-2-hydroxy-3-(propylamino)propyl]-1-methylpyrazolo[3,4-d]pyrimidin-4-one —— C12H19N5O2
5-[(2S)-2-hydroxy-3-(propylamino)propyl]-1-methylpyrazolo[3,4-d]pyrimidin-4-one
—— 5-(aminomethyl)-N-methyl-N-[[(3S)-1-methylpyrrolidin-3-yl]methyl]-4-propyl-1,3-thiazol-2-amine —— C14H26N4S
5-(aminomethyl)-N-methyl-N-[[(3S)-1-methylpyrrolidin-3-yl]methyl]-4-propyl-1,3-thiazol-2-amine
—— 5-bromo-N-methyl-N-[[(3S)-1-methylpyrrolidin-3-yl]methyl]-3-nitropyridin-2-amine —— C12H17BrN4O2
5-bromo-N-methyl-N-[[(3S)-1-methylpyrrolidin-3-yl]methyl]-3-nitropyridin-2-amine
—— 5-bromo-N-methyl-N-[[(3R)-1-methylpyrrolidin-3-yl]methyl]-3-nitropyridin-2-amine —— C12H17BrN4O2
5-bromo-N-methyl-N-[[(3R)-1-methylpyrrolidin-3-yl]methyl]-3-nitropyridin-2-amine
—— 5-[(4R)-4-(ethylamino)pentyl]-1-methylpyrazolo[3,4-d]pyrimidin-4-one —— C13H21N5O
5-[(4R)-4-(ethylamino)pentyl]-1-methylpyrazolo[3,4-d]pyrimidin-4-one
—— 5-[(cyclopropylamino)methyl]-N-methyl-N-[[(3S)-1-methylpyrrolidin-3-yl]methyl]-1,3-thiazol-2-amine —— C14H24N4S
5-[(cyclopropylamino)methyl]-N-methyl-N-[[(3S)-1-methylpyrrolidin-3-yl]methyl]-1,3-thiazol-2-amine
—— 5-(aminomethyl)-N-methyl-N-[[(3R)-1-methylpyrrolidin-3-yl]methyl]-4-propyl-1,3-thiazol-2-amine —— C14H26N4S
5-(aminomethyl)-N-methyl-N-[[(3R)-1-methylpyrrolidin-3-yl]methyl]-4-propyl-1,3-thiazol-2-amine
—— 5-chloro-2-hydroxy-N-methyl-N-[[(3R)-1-methylpyrrolidin-3-yl]methyl]benzamide —— C14H19ClN2O2
5-chloro-2-hydroxy-N-methyl-N-[[(3R)-1-methylpyrrolidin-3-yl]methyl]benzamide
—— 5-[(2R)-2-(ethylamino)pentyl]-1-methylpyrazolo[3,4-d]pyrimidin-4-one —— C13H21N5O
5-[(2R)-2-(ethylamino)pentyl]-1-methylpyrazolo[3,4-d]pyrimidin-4-one
—— 5-[(cyclopropylamino)methyl]-N-methyl-N-[[(3R)-1-methylpyrrolidin-3-yl]methyl]-1,3-thiazol-2-amine —— C14H24N4S
5-[(cyclopropylamino)methyl]-N-methyl-N-[[(3R)-1-methylpyrrolidin-3-yl]methyl]-1,3-thiazol-2-amine