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—— (5R)-5-[1-[bis(2-chlorophenyl)methyl]tetrazol-5-yl]-4-methoxy-6-methyl-7,8-dihydro-5H-[1,3]dioxolo[4,5-g]isoquinoline —— C26H23Cl2N5O3
(5R)-5-[1-[bis(2-chlorophenyl)methyl]tetrazol-5-yl]-4-methoxy-6-methyl-7,8-dihydro-5H-[1,3]dioxolo[4,5-g]isoquinoline
—— 5-[(2R)-1-[(1R,4aS,8aS)-1-(4-chlorophenyl)-4a-hydroxy-1,3,4,5,6,7,8,8a-octahydroisoquinolin-2-yl]-1-oxopropan-2-yl]oxy-3-benzyl-4,7-dimethylchromen-2-one —— C36H38ClNO5
5-[(2R)-1-[(1R,4aS,8aS)-1-(4-chlorophenyl)-4a-hydroxy-1,3,4,5,6,7,8,8a-octahydroisoquinolin-2-yl]-1-oxopropan-2-yl]oxy-3-benzyl-4,7-dimethylchromen-2-one
—— (5S)-5-[1-[bis(2-chlorophenyl)methyl]tetrazol-5-yl]-4-methoxy-6-methyl-7,8-dihydro-5H-[1,3]dioxolo[4,5-g]isoquinoline —— C26H23Cl2N5O3
(5S)-5-[1-[bis(2-chlorophenyl)methyl]tetrazol-5-yl]-4-methoxy-6-methyl-7,8-dihydro-5H-[1,3]dioxolo[4,5-g]isoquinoline
—— (5R)-7,7-dimethyl-2-azaspiro[4.5]decane —— C11H21N
(5R)-7,7-dimethyl-2-azaspiro[4.5]decane
—— 5-chloro-N-(3-chloro-2-fluorophenyl)-3-methyl-1-phenylpyrazole-4-carboxamide —— C17H12Cl2FN3O
5-chloro-N-(3-chloro-2-fluorophenyl)-3-methyl-1-phenylpyrazole-4-carboxamide
—— (5S)-7,7-dimethyl-2-azaspiro[4.5]decane —— C11H21N
(5S)-7,7-dimethyl-2-azaspiro[4.5]decane
—— 5-[[(3aS,6aS)-3-(3-methoxyphenyl)-5,5-dioxo-3a,4,6,6a-tetrahydrothieno[3,4-d][1,3]thiazol-2-ylidene]amino]-5-oxopentanoate —— C17H19N2O6S2-
5-[[(3aS,6aS)-3-(3-methoxyphenyl)-5,5-dioxo-3a,4,6,6a-tetrahydrothieno[3,4-d][1,3]thiazol-2-ylidene]amino]-5-oxopentanoate
—— (5E)-1-(4-bromophenyl)-5-[[[(5R)-4-methoxy-6-methyl-7,8-dihydro-5H-[1,3]dioxolo[4,5-g]isoquinolin-5-yl]methylamino]methylidene]-2-sulfanylidene-1,3-diazinane-4,6-dione —— C24H23BrN4O5S
(5E)-1-(4-bromophenyl)-5-[[[(5R)-4-methoxy-6-methyl-7,8-dihydro-5H-[1,3]dioxolo[4,5-g]isoquinolin-5-yl]methylamino]methylidene]-2-sulfanylidene-1,3-diazinane-4,6-dione
—— [5-[(4-fluorophenoxy)methyl]furan-2-yl]-[(2S)-2-methylpiperidin-1-yl]methanone —— C18H20FNO3
[5-[(4-fluorophenoxy)methyl]furan-2-yl]-[(2S)-2-methylpiperidin-1-yl]methanone
—— (5'R)-5'-(1,3-dimethyl-2,4,6-trioxo-5-prop-2-enyl-1,3-diazinan-5-yl)-4'-methoxy-1,3-dimethylspiro[1,3-diazinane-5,6'-7,8-dihydro-5H-benzo[f][1,3]benzodioxole]-2,4,6-trione —— C26H28N4O9
(5'R)-5'-(1,3-dimethyl-2,4,6-trioxo-5-prop-2-enyl-1,3-diazinan-5-yl)-4'-methoxy-1,3-dimethylspiro[1,3-diazinane-5,6'-7,8-dihydro-5H-benzo[f][1,3]benzodioxole]-2,4,6-trione
—— [5-[(4-fluorophenoxy)methyl]furan-2-yl]-[(2R)-2-methylpiperidin-1-yl]methanone —— C18H20FNO3
[5-[(4-fluorophenoxy)methyl]furan-2-yl]-[(2R)-2-methylpiperidin-1-yl]methanone
—— (5'S)-5'-(1,3-dimethyl-2,4,6-trioxo-5-prop-2-enyl-1,3-diazinan-5-yl)-4'-methoxy-1,3-dimethylspiro[1,3-diazinane-5,6'-7,8-dihydro-5H-benzo[f][1,3]benzodioxole]-2,4,6-trione —— C26H28N4O9
(5'S)-5'-(1,3-dimethyl-2,4,6-trioxo-5-prop-2-enyl-1,3-diazinan-5-yl)-4'-methoxy-1,3-dimethylspiro[1,3-diazinane-5,6'-7,8-dihydro-5H-benzo[f][1,3]benzodioxole]-2,4,6-trione
—— (5E)-1-(4-bromophenyl)-5-[[[(5S)-4-methoxy-6-methyl-7,8-dihydro-5H-[1,3]dioxolo[4,5-g]isoquinolin-5-yl]methylamino]methylidene]-2-sulfanylidene-1,3-diazinane-4,6-dione —— C24H23BrN4O5S
(5E)-1-(4-bromophenyl)-5-[[[(5S)-4-methoxy-6-methyl-7,8-dihydro-5H-[1,3]dioxolo[4,5-g]isoquinolin-5-yl]methylamino]methylidene]-2-sulfanylidene-1,3-diazinane-4,6-dione
—— 5-[[(3aR,6aR)-3-(3-methoxyphenyl)-5,5-dioxo-3a,4,6,6a-tetrahydrothieno[3,4-d][1,3]thiazol-2-ylidene]amino]-5-oxopentanoate —— C17H19N2O6S2-
5-[[(3aR,6aR)-3-(3-methoxyphenyl)-5,5-dioxo-3a,4,6,6a-tetrahydrothieno[3,4-d][1,3]thiazol-2-ylidene]amino]-5-oxopentanoate
—— (5S)-5-[[(1S)-6,7-dimethoxy-1-methyl-3,4-dihydro-1H-isoquinolin-2-yl]methyl]-5-[(4-methoxyphenyl)methyl]-1-phenyl-1,3-diazinane-2,4,6-trione —— C31H33N3O6
(5S)-5-[[(1S)-6,7-dimethoxy-1-methyl-3,4-dihydro-1H-isoquinolin-2-yl]methyl]-5-[(4-methoxyphenyl)methyl]-1-phenyl-1,3-diazinane-2,4,6-trione
—— 5-[[4-[(2S)-2-hydroxy-2-phenylethoxy]phenyl]methyl]-1,3-dimethyl-5-[[(1R,9S)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]methyl]-1,3-diazinane-2,4,6-trione —— C33H36N4O6
5-[[4-[(2S)-2-hydroxy-2-phenylethoxy]phenyl]methyl]-1,3-dimethyl-5-[[(1R,9S)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]methyl]-1,3-diazinane-2,4,6-trione
—— (5S)-1-(4-ethylphenyl)-5-[[(1S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]methyl]-5-[(3,4,5-trimethoxyphenyl)methyl]-1,3-diazinane-2,4,6-trione —— C34H38N4O7
(5S)-1-(4-ethylphenyl)-5-[[(1S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]methyl]-5-[(3,4,5-trimethoxyphenyl)methyl]-1,3-diazinane-2,4,6-trione
—— (5E)-1-(4-bromophenyl)-5-[[[(5S)-4-methoxy-6-methyl-7,8-dihydro-5H-[1,3]dioxolo[4,5-g]isoquinolin-5-yl]methylamino]methylidene]-1,3-diazinane-2,4,6-trione —— C24H23BrN4O6
(5E)-1-(4-bromophenyl)-5-[[[(5S)-4-methoxy-6-methyl-7,8-dihydro-5H-[1,3]dioxolo[4,5-g]isoquinolin-5-yl]methylamino]methylidene]-1,3-diazinane-2,4,6-trione
—— (5E)-3-[(3R)-1,1-dioxothiolan-3-yl]-5-[[(2R)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C17H17NO4S3
(5E)-3-[(3R)-1,1-dioxothiolan-3-yl]-5-[[(2R)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— 5-[(5-bromo-2-methoxyphenyl)methyl]-1,3-dimethyl-5-[[(1S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]methyl]-1,3-diazinane-2,4,6-trione —— C26H29BrN4O5
5-[(5-bromo-2-methoxyphenyl)methyl]-1,3-dimethyl-5-[[(1S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]methyl]-1,3-diazinane-2,4,6-trione
—— 5-[[(3aR,6aS)-3-(3-methoxyphenyl)-5,5-dioxo-3a,4,6,6a-tetrahydrothieno[3,4-d][1,3]thiazol-2-ylidene]amino]-5-oxopentanoate —— C17H19N2O6S2-
5-[[(3aR,6aS)-3-(3-methoxyphenyl)-5,5-dioxo-3a,4,6,6a-tetrahydrothieno[3,4-d][1,3]thiazol-2-ylidene]amino]-5-oxopentanoate
—— (5E)-5-[4-(2-phenoxyethoxy)benzylidene]-2-thioxo-1,3-thiazolidin-4-one —— C18H15NO3S2
(5E)-5-[4-(2-phenoxyethoxy)benzylidene]-2-thioxo-1,3-thiazolidin-4-one
—— 5-[(4-bromophenyl)methyl]-1,3-dimethyl-5-[[(1R,9S)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]methyl]-1,3-diazinane-2,4,6-trione —— C25H27BrN4O4
5-[(4-bromophenyl)methyl]-1,3-dimethyl-5-[[(1R,9S)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]methyl]-1,3-diazinane-2,4,6-trione
—— 5-(dimethylsulfamoyl)-N-[4-[ethyl(propan-2-yl)amino]phenyl]-2-methylbenzamide —— C21H29N3O3S
5-(dimethylsulfamoyl)-N-[4-[ethyl(propan-2-yl)amino]phenyl]-2-methylbenzamide
—— 5-[[(3aS,6aS)-3-(3-methoxyphenyl)-5,5-dioxo-3a,4,6,6a-tetrahydrothieno[3,4-d][1,3]thiazol-2-ylidene]amino]-5-oxopentanoic acid —— C17H20N2O6S2
5-[[(3aS,6aS)-3-(3-methoxyphenyl)-5,5-dioxo-3a,4,6,6a-tetrahydrothieno[3,4-d][1,3]thiazol-2-ylidene]amino]-5-oxopentanoic acid
—— 5-Thia-3,8-diaza-1-azoniatricyclo[7.4.0.02,6]trideca-1(13),2(6),7,9,11-pentaen-4-one —— C9H6N3OS+
5-Thia-3,8-diaza-1-azoniatricyclo[7.4.0.02,6]trideca-1(13),2(6),7,9,11-pentaen-4-one
—— (5E)-2-[(2-chlorophenyl)amino]-5-(naphthalen-1-ylmethylidene)-1,3-thiazol-4(5H)-one —— C20H13ClN2OS
(5E)-2-[(2-chlorophenyl)amino]-5-(naphthalen-1-ylmethylidene)-1,3-thiazol-4(5H)-one
—— (5R)-1-benzyl-5-(naphthalen-1-ylmethyl)-5-[[(1S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]methyl]-1,3-diazinane-2,4,6-trione —— C34H32N4O4
(5R)-1-benzyl-5-(naphthalen-1-ylmethyl)-5-[[(1S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]methyl]-1,3-diazinane-2,4,6-trione
—— 5-[[(3aS,6aR)-3-(3-methoxyphenyl)-5,5-dioxo-3a,4,6,6a-tetrahydrothieno[3,4-d][1,3]thiazol-2-ylidene]amino]-5-oxopentanoic acid —— C17H20N2O6S2
5-[[(3aS,6aR)-3-(3-methoxyphenyl)-5,5-dioxo-3a,4,6,6a-tetrahydrothieno[3,4-d][1,3]thiazol-2-ylidene]amino]-5-oxopentanoic acid
—— 5-[(3-bromo-5-ethoxy-4-hydroxyphenyl)methyl]-1,3-dimethyl-5-[[(1S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]methyl]-2-sulfanylidene-1,3-diazinane-4,6-dione —— C27H31BrN4O5S
5-[(3-bromo-5-ethoxy-4-hydroxyphenyl)methyl]-1,3-dimethyl-5-[[(1S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]methyl]-2-sulfanylidene-1,3-diazinane-4,6-dione
—— (5R)-5-tert-butyl-N-[(3R)-1,1-dioxothiolan-3-yl]-N-propyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C20H31NO3S2
(5R)-5-tert-butyl-N-[(3R)-1,1-dioxothiolan-3-yl]-N-propyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— (5E)-2-[(2-chlorophenyl)amino]-5-(4-ethoxybenzylidene)-1,3-thiazol-4(5H)-one —— C18H15ClN2O2S
(5E)-2-[(2-chlorophenyl)amino]-5-(4-ethoxybenzylidene)-1,3-thiazol-4(5H)-one
—— (5S,7S)-N-(2-methoxyethyl)-5-(4-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C18H21F3N4O3
(5S,7S)-N-(2-methoxyethyl)-5-(4-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5R,7S)-N-(2-methoxyethyl)-5-(4-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C18H21F3N4O3
(5R,7S)-N-(2-methoxyethyl)-5-(4-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— 5-[[(3aR,6aR)-3-(3-methoxyphenyl)-5,5-dioxo-3a,4,6,6a-tetrahydrothieno[3,4-d][1,3]thiazol-2-ylidene]amino]-5-oxopentanoic acid —— C17H20N2O6S2
5-[[(3aR,6aR)-3-(3-methoxyphenyl)-5,5-dioxo-3a,4,6,6a-tetrahydrothieno[3,4-d][1,3]thiazol-2-ylidene]amino]-5-oxopentanoic acid
—— 5-[(1-benzylindol-3-yl)methyl]-1,3-dimethyl-5-[[(1S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]methyl]-1,3-diazinane-2,4,6-trione —— C34H35N5O4
5-[(1-benzylindol-3-yl)methyl]-1,3-dimethyl-5-[[(1S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]methyl]-1,3-diazinane-2,4,6-trione
—— (5E)-3-[(3S)-1,1-dioxothiolan-3-yl]-5-[[(2S)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C17H17NO4S3
(5E)-3-[(3S)-1,1-dioxothiolan-3-yl]-5-[[(2S)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5R)-5-tert-butyl-N-[(3S)-1,1-dioxothiolan-3-yl]-N-propyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C20H31NO3S2
(5R)-5-tert-butyl-N-[(3S)-1,1-dioxothiolan-3-yl]-N-propyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— (5S)-5-tert-butyl-N-[(3S)-1,1-dioxothiolan-3-yl]-N-propyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C20H31NO3S2
(5S)-5-tert-butyl-N-[(3S)-1,1-dioxothiolan-3-yl]-N-propyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— 5-[(4-hydroxy-3-iodo-5-methoxyphenyl)methyl]-1,3-dimethyl-5-[[(1S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]methyl]-1,3-diazinane-2,4,6-trione —— C26H29IN4O6
5-[(4-hydroxy-3-iodo-5-methoxyphenyl)methyl]-1,3-dimethyl-5-[[(1S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]methyl]-1,3-diazinane-2,4,6-trione
—— (5R,7R)-N-(2-methoxyethyl)-5-(4-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C18H21F3N4O3
(5R,7R)-N-(2-methoxyethyl)-5-(4-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5S)-1-[3-(dimethylamino)propyl]-4-[hydroxy-[2-methyl-4-(2-methylpropoxy)phenyl]methylidene]-5-(3,4,5-trimethoxyphenyl)pyrrolidine-2,3-dione —— C30H40N2O7
(5S)-1-[3-(dimethylamino)propyl]-4-[hydroxy-[2-methyl-4-(2-methylpropoxy)phenyl]methylidene]-5-(3,4,5-trimethoxyphenyl)pyrrolidine-2,3-dione
—— 5-(dimethylsulfamoyl)-N-(2-ethoxyphenyl)-2-pyrrolidin-1-ylbenzamide —— C21H27N3O4S
5-(dimethylsulfamoyl)-N-(2-ethoxyphenyl)-2-pyrrolidin-1-ylbenzamide
—— (5S)-5-tert-butyl-N-[(3R)-1,1-dioxothiolan-3-yl]-N-propyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C20H31NO3S2
(5S)-5-tert-butyl-N-[(3R)-1,1-dioxothiolan-3-yl]-N-propyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— (5-Amino-4-cyano-2-ethoxycarbonylthiophen-3-yl)methyl 3-(methoxymethyl)-1-benzofuran-2-carboxylate —— C20H18N2O6S
(5-Amino-4-cyano-2-ethoxycarbonylthiophen-3-yl)methyl 3-(methoxymethyl)-1-benzofuran-2-carboxylate
—— 5-(dimethylsulfamoyl)-N-(5-ethyl-1,3,4-thiadiazol-2-yl)-2-pyrrolidin-1-ylbenzamide —— C17H23N5O3S2
5-(dimethylsulfamoyl)-N-(5-ethyl-1,3,4-thiadiazol-2-yl)-2-pyrrolidin-1-ylbenzamide
—— (5R)-1-[3-(dimethylamino)propyl]-4-[hydroxy-[2-methyl-4-(2-methylpropoxy)phenyl]methylidene]-5-(3,4,5-trimethoxyphenyl)pyrrolidine-2,3-dione —— C30H40N2O7
(5R)-1-[3-(dimethylamino)propyl]-4-[hydroxy-[2-methyl-4-(2-methylpropoxy)phenyl]methylidene]-5-(3,4,5-trimethoxyphenyl)pyrrolidine-2,3-dione
—— (5-Methoxy-3-methyl-1-benzofuran-2-yl)-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]methanone —— C22H21F3N2O3
(5-Methoxy-3-methyl-1-benzofuran-2-yl)-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]methanone
—— 5-[[4-[(2R)-2-hydroxy-2-phenylethoxy]phenyl]methyl]-1,3-dimethyl-5-[[(1R,9S)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]methyl]-1,3-diazinane-2,4,6-trione —— C33H36N4O6
5-[[4-[(2R)-2-hydroxy-2-phenylethoxy]phenyl]methyl]-1,3-dimethyl-5-[[(1R,9S)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]methyl]-1,3-diazinane-2,4,6-trione
—— 5-(dimethylsulfamoyl)-N-[(4-fluorophenyl)methyl]-2-morpholin-4-ylbenzamide —— C20H24FN3O4S
5-(dimethylsulfamoyl)-N-[(4-fluorophenyl)methyl]-2-morpholin-4-ylbenzamide