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—— 5-chloro-N-[(2R)-2-(4-chlorophenyl)-2-morpholin-4-ylethyl]-1,3-dimethylpyrazole-4-carboxamide —— C18H22Cl2N4O2
5-chloro-N-[(2R)-2-(4-chlorophenyl)-2-morpholin-4-ylethyl]-1,3-dimethylpyrazole-4-carboxamide
—— 5-[(3R)-dithiolan-3-yl]-N-[4-(1-methylimidazole-2-carbonyl)phenyl]pentanamide —— C19H23N3O2S2
5-[(3R)-dithiolan-3-yl]-N-[4-(1-methylimidazole-2-carbonyl)phenyl]pentanamide
—— 5-sulfamoyl-N-[(2S)-1-thiophen-2-ylpropan-2-yl]thiophene-3-carboxamide —— C12H14N2O3S3
5-sulfamoyl-N-[(2S)-1-thiophen-2-ylpropan-2-yl]thiophene-3-carboxamide
—— 5-fluoro-2-(methanesulfonamido)-N-[(1S)-1-(2-methoxy-5-methylphenyl)ethyl]benzamide —— C18H21FN2O4S
5-fluoro-2-(methanesulfonamido)-N-[(1S)-1-(2-methoxy-5-methylphenyl)ethyl]benzamide
—— 5-fluoro-2-(methanesulfonamido)-N-[(1R)-1-(2-methylphenyl)ethyl]benzamide —— C17H19FN2O3S
5-fluoro-2-(methanesulfonamido)-N-[(1R)-1-(2-methylphenyl)ethyl]benzamide
—— 5-(ethylsulfamoyl)-2-fluoro-N-[(1S)-1-pyridin-4-ylethyl]benzamide —— C16H18FN3O3S
5-(ethylsulfamoyl)-2-fluoro-N-[(1S)-1-pyridin-4-ylethyl]benzamide
—— (5-Oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl 2-(2-fluorophenyl)sulfanylacetate —— C15H11FN2O3S2
(5-Oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl 2-(2-fluorophenyl)sulfanylacetate
—— 5-(ethylsulfamoyl)-2-fluoro-N-[(1R)-1-pyridin-4-ylethyl]benzamide —— C16H18FN3O3S
5-(ethylsulfamoyl)-2-fluoro-N-[(1R)-1-pyridin-4-ylethyl]benzamide
—— 5-[[(2R)-2-(3,4-dimethylphenyl)pyrrolidin-1-yl]methyl]-1-propyltetrazole —— C17H25N5
5-[[(2R)-2-(3,4-dimethylphenyl)pyrrolidin-1-yl]methyl]-1-propyltetrazole
—— 5-[[benzyl(methyl)amino]methyl]-N-[(4S)-2-oxo-3,4-dihydro-1H-quinolin-4-yl]-1,2-oxazole-3-carboxamide —— C22H22N4O3
5-[[benzyl(methyl)amino]methyl]-N-[(4S)-2-oxo-3,4-dihydro-1H-quinolin-4-yl]-1,2-oxazole-3-carboxamide
—— [(5S)-2,9-diazaspiro[4.5]decan-2-yl]-[4-(tetrazol-1-yl)phenyl]methanone —— C16H20N6O
[(5S)-2,9-diazaspiro[4.5]decan-2-yl]-[4-(tetrazol-1-yl)phenyl]methanone
—— 5-methyl-3-[(2R)-1-[(3-phenylpyrazolo[1,5-a]pyrimidin-6-yl)methyl]pyrrolidin-2-yl]-1,2-oxazole —— C21H21N5O
5-methyl-3-[(2R)-1-[(3-phenylpyrazolo[1,5-a]pyrimidin-6-yl)methyl]pyrrolidin-2-yl]-1,2-oxazole
—— 5-(3-Bromophenyl)-3-(2,6-difluorophenyl)-1,2,4-oxadiazole —— C14H7BrF2N2O
5-(3-Bromophenyl)-3-(2,6-difluorophenyl)-1,2,4-oxadiazole
—— 5-methyl-3-[(2S)-1-[(3-phenylpyrazolo[1,5-a]pyrimidin-6-yl)methyl]pyrrolidin-2-yl]-1,2-oxazole —— C21H21N5O
5-methyl-3-[(2S)-1-[(3-phenylpyrazolo[1,5-a]pyrimidin-6-yl)methyl]pyrrolidin-2-yl]-1,2-oxazole
—— (5S)-1-ethyl-5-[methyl-[(5-phenyl-1,2-oxazol-3-yl)methyl]amino]-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C21H24N4O3
(5S)-1-ethyl-5-[methyl-[(5-phenyl-1,2-oxazol-3-yl)methyl]amino]-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— 5-[(3,4-difluorophenoxy)methyl]-N-[(1R)-2-hydroxy-1-pyridin-3-ylethyl]-1,2-oxazole-3-carboxamide —— C18H15F2N3O4
5-[(3,4-difluorophenoxy)methyl]-N-[(1R)-2-hydroxy-1-pyridin-3-ylethyl]-1,2-oxazole-3-carboxamide
—— 5-[[(2S)-2-(3,4-dimethylphenyl)pyrrolidin-1-yl]methyl]-1-propyltetrazole —— C17H25N5
5-[[(2S)-2-(3,4-dimethylphenyl)pyrrolidin-1-yl]methyl]-1-propyltetrazole
—— 5-(2-Chloro-6-fluorobenzyl)-3-(2-fluorophenyl)-1,2,4-oxadiazole —— C15H9ClF2N2O
5-(2-Chloro-6-fluorobenzyl)-3-(2-fluorophenyl)-1,2,4-oxadiazole
—— (5R)-1-ethyl-5-[methyl-[(5-phenyl-1,2-oxazol-3-yl)methyl]amino]-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C21H24N4O3
(5R)-1-ethyl-5-[methyl-[(5-phenyl-1,2-oxazol-3-yl)methyl]amino]-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— (5S)-5-[(2-methyl-1H-indol-5-yl)methylamino]-1-propyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C21H26N4O2
(5S)-5-[(2-methyl-1H-indol-5-yl)methylamino]-1-propyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— (5S)-N-(4-methoxy-2-methylphenyl)-2,9-diazaspiro[4.5]decane-2-carboxamide —— C17H25N3O2
(5S)-N-(4-methoxy-2-methylphenyl)-2,9-diazaspiro[4.5]decane-2-carboxamide
—— (5R)-5-[(2-methyl-1H-indol-5-yl)methylamino]-1-propyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C21H26N4O2
(5R)-5-[(2-methyl-1H-indol-5-yl)methylamino]-1-propyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— (5S)-5-[methyl(quinoxalin-2-ylmethyl)amino]-1-prop-2-enyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C21H23N5O2
(5S)-5-[methyl(quinoxalin-2-ylmethyl)amino]-1-prop-2-enyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— 5-methyl-4-[[(2R)-1-pyrazin-2-ylpropan-2-yl]amino]thieno[2,3-d]pyrimidine-6-carboxylic acid —— C15H15N5O2S
5-methyl-4-[[(2R)-1-pyrazin-2-ylpropan-2-yl]amino]thieno[2,3-d]pyrimidine-6-carboxylic acid
—— 5-[(2-methoxyphenoxy)methyl]-N-[(2R)-2-methylbutyl]-1H-pyrazole-3-carboxamide —— C17H23N3O3
5-[(2-methoxyphenoxy)methyl]-N-[(2R)-2-methylbutyl]-1H-pyrazole-3-carboxamide
—— (5-chlorothiophen-2-yl)-[(2S)-2-(1-methylbenzimidazol-2-yl)pyrrolidin-1-yl]methanone —— C17H16ClN3OS
(5-chlorothiophen-2-yl)-[(2S)-2-(1-methylbenzimidazol-2-yl)pyrrolidin-1-yl]methanone
—— (5-chlorothiophen-2-yl)-[(2R)-2-(1-methylbenzimidazol-2-yl)pyrrolidin-1-yl]methanone —— C17H16ClN3OS
(5-chlorothiophen-2-yl)-[(2R)-2-(1-methylbenzimidazol-2-yl)pyrrolidin-1-yl]methanone
—— 5-fluoro-3-methyl-2-[[(3R)-3-(1H-pyrazol-5-yl)piperidin-1-yl]methyl]-1H-indole —— C18H21FN4
5-fluoro-3-methyl-2-[[(3R)-3-(1H-pyrazol-5-yl)piperidin-1-yl]methyl]-1H-indole
—— 5-(2-Methoxy-4-nitrophenyl)furan-2-carboxylate —— C12H8NO6-
5-(2-Methoxy-4-nitrophenyl)furan-2-carboxylate
—— (5R)-5-(5-methoxy-2-pyrazol-1-ylphenyl)-1,2,5,6-tetrahydropyrazolo[4,3-g]quinolin-7-one —— C20H17N5O2
(5R)-5-(5-methoxy-2-pyrazol-1-ylphenyl)-1,2,5,6-tetrahydropyrazolo[4,3-g]quinolin-7-one
—— 5-methyl-N-[[(3S)-1-[(E)-3-phenylprop-2-enyl]pyrrolidin-3-yl]methyl]pyrazine-2-carboxamide —— C20H24N4O
5-methyl-N-[[(3S)-1-[(E)-3-phenylprop-2-enyl]pyrrolidin-3-yl]methyl]pyrazine-2-carboxamide
—— 5-[(2-methoxyphenoxy)methyl]-N-[(2S)-2-methylbutyl]-1H-pyrazole-3-carboxamide —— C17H23N3O3
5-[(2-methoxyphenoxy)methyl]-N-[(2S)-2-methylbutyl]-1H-pyrazole-3-carboxamide
—— (5S)-5-(5-methoxy-2-pyrazol-1-ylphenyl)-1,2,5,6-tetrahydropyrazolo[4,3-g]quinolin-7-one —— C20H17N5O2
(5S)-5-(5-methoxy-2-pyrazol-1-ylphenyl)-1,2,5,6-tetrahydropyrazolo[4,3-g]quinolin-7-one
—— 5-methyl-N-[[(3R)-1-[(E)-3-phenylprop-2-enyl]pyrrolidin-3-yl]methyl]pyrazine-2-carboxamide —— C20H24N4O
5-methyl-N-[[(3R)-1-[(E)-3-phenylprop-2-enyl]pyrrolidin-3-yl]methyl]pyrazine-2-carboxamide
—— 5-fluoro-3-methyl-2-[[(3S)-3-(1H-pyrazol-5-yl)piperidin-1-yl]methyl]-1H-indole —— C18H21FN4
5-fluoro-3-methyl-2-[[(3S)-3-(1H-pyrazol-5-yl)piperidin-1-yl]methyl]-1H-indole
—— 5-[[benzyl(methyl)amino]methyl]-N-[(4R)-2-oxo-3,4-dihydro-1H-quinolin-4-yl]-1,2-oxazole-3-carboxamide —— C22H22N4O3
5-[[benzyl(methyl)amino]methyl]-N-[(4R)-2-oxo-3,4-dihydro-1H-quinolin-4-yl]-1,2-oxazole-3-carboxamide
—— 5-[(3,4-difluorophenoxy)methyl]-N-[(1S)-2-hydroxy-1-pyridin-3-ylethyl]-1,2-oxazole-3-carboxamide —— C18H15F2N3O4
5-[(3,4-difluorophenoxy)methyl]-N-[(1S)-2-hydroxy-1-pyridin-3-ylethyl]-1,2-oxazole-3-carboxamide
—— (5S)-5-(4,6-dimethyl-2-propan-2-ylpyrimidin-5-yl)oxy-1-azabicyclo[3.2.1]octane —— C16H25N3O
(5S)-5-(4,6-dimethyl-2-propan-2-ylpyrimidin-5-yl)oxy-1-azabicyclo[3.2.1]octane
—— 5-methyl-4-[[(2S)-1-pyrazin-2-ylpropan-2-yl]amino]thieno[2,3-d]pyrimidine-6-carboxylic acid —— C15H15N5O2S
5-methyl-4-[[(2S)-1-pyrazin-2-ylpropan-2-yl]amino]thieno[2,3-d]pyrimidine-6-carboxylic acid
—— [(5R)-2,9-diazaspiro[4.5]decan-2-yl]-[4-(tetrazol-1-yl)phenyl]methanone —— C16H20N6O
[(5R)-2,9-diazaspiro[4.5]decan-2-yl]-[4-(tetrazol-1-yl)phenyl]methanone
—— [5-[[benzyl(methyl)amino]methyl]-1,2-oxazol-3-yl]-[(2S)-2-butyl-2,5-dihydropyrrol-1-yl]methanone —— C21H27N3O2
[5-[[benzyl(methyl)amino]methyl]-1,2-oxazol-3-yl]-[(2S)-2-butyl-2,5-dihydropyrrol-1-yl]methanone
—— (5R)-3-methyl-N-[[2-[methyl(2-pyridin-2-ylethyl)amino]pyridin-3-yl]methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C19H23N5O2
(5R)-3-methyl-N-[[2-[methyl(2-pyridin-2-ylethyl)amino]pyridin-3-yl]methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— 5-(hydroxymethyl)-2-methyl-4-[[methyl-[(1R)-1-pyridin-3-ylpropyl]amino]methyl]pyridin-3-ol —— C17H23N3O2
5-(hydroxymethyl)-2-methyl-4-[[methyl-[(1R)-1-pyridin-3-ylpropyl]amino]methyl]pyridin-3-ol
—— 5-methyl-N-[[(3S)-1-[(2-methyl-1H-imidazol-5-yl)methyl]pyrrolidin-3-yl]methyl]pyrazine-2-carboxamide —— C16H22N6O
5-methyl-N-[[(3S)-1-[(2-methyl-1H-imidazol-5-yl)methyl]pyrrolidin-3-yl]methyl]pyrazine-2-carboxamide
—— (5-chloropyridin-3-yl)-[(3R)-3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl]methanone —— C21H21ClN4O
(5-chloropyridin-3-yl)-[(3R)-3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl]methanone
—— [5-[(2-methoxyphenoxy)methyl]-1H-pyrazol-3-yl]-[(2S)-2-methylpyrrolidin-1-yl]methanone —— C17H21N3O3
[5-[(2-methoxyphenoxy)methyl]-1H-pyrazol-3-yl]-[(2S)-2-methylpyrrolidin-1-yl]methanone
—— (5R)-5-(6-methoxy-3,4-dihydro-1H-isoquinolin-2-yl)-1-propyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C21H27N3O3
(5R)-5-(6-methoxy-3,4-dihydro-1H-isoquinolin-2-yl)-1-propyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— (5S)-1,3-dimethyl-5-thiophen-2-yl-6,8-dihydro-5H-pyrido[2,3-d]pyrimidine-2,4,7-trione —— C13H13N3O3S
(5S)-1,3-dimethyl-5-thiophen-2-yl-6,8-dihydro-5H-pyrido[2,3-d]pyrimidine-2,4,7-trione
—— (5S)-5-[4-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]phenoxy]-1-azabicyclo[3.2.1]octane —— C22H29N5O
(5S)-5-[4-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]phenoxy]-1-azabicyclo[3.2.1]octane
—— (5R)-1-ethyl-5-[methyl-[(4-pyrazol-1-ylphenyl)methyl]amino]-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C21H25N5O2
(5R)-1-ethyl-5-[methyl-[(4-pyrazol-1-ylphenyl)methyl]amino]-4,5,6,7-tetrahydroindazole-3-carboxylic acid