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—— (5R)-4-[hydroxy-(4-methoxy-3-methylphenyl)methylidene]-1-(3-methoxypropyl)-5-(4-methylphenyl)pyrrolidine-2,3-dione —— C24H27NO5
(5R)-4-[hydroxy-(4-methoxy-3-methylphenyl)methylidene]-1-(3-methoxypropyl)-5-(4-methylphenyl)pyrrolidine-2,3-dione
—— (5S)-N-[(Z)-(2-chloro-6-fluorophenyl)methylideneamino]-5-ethyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C18H18ClFN2OS
(5S)-N-[(Z)-(2-chloro-6-fluorophenyl)methylideneamino]-5-ethyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— (5S)-5-ethyl-N-(heptan-4-ylideneamino)-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C18H28N2OS
(5S)-5-ethyl-N-(heptan-4-ylideneamino)-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— (5R)-N-[(Z)-(1-benzyl-3,5-dimethylpyrazol-4-yl)methylideneamino]-5-ethyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C24H28N4OS
(5R)-N-[(Z)-(1-benzyl-3,5-dimethylpyrazol-4-yl)methylideneamino]-5-ethyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— (5S)-5-ethyl-N-[(Z)-(6-fluoro-2,3-dihydrothiochromen-4-ylidene)amino]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C20H21FN2OS2
(5S)-5-ethyl-N-[(Z)-(6-fluoro-2,3-dihydrothiochromen-4-ylidene)amino]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— (5S)-7-(3,5-dimethylphenyl)-1,2,7-triazaspiro[4.4]non-1-ene-6,8-dione —— C14H15N3O2
(5S)-7-(3,5-dimethylphenyl)-1,2,7-triazaspiro[4.4]non-1-ene-6,8-dione
—— (5R)-5-ethyl-N'-[(3-methoxy-5-nitro-4-oxocyclohexa-2,5-dien-1-ylidene)methyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carbohydrazide —— C19H21N3O5S
(5R)-5-ethyl-N'-[(3-methoxy-5-nitro-4-oxocyclohexa-2,5-dien-1-ylidene)methyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carbohydrazide
—— (5S)-N-[(Z)-(3,5-dimethyl-1-phenylpyrazol-4-yl)methylideneamino]-5-ethyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C23H26N4OS
(5S)-N-[(Z)-(3,5-dimethyl-1-phenylpyrazol-4-yl)methylideneamino]-5-ethyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— (5S)-5-ethyl-N'-[(2-oxonaphthalen-1-ylidene)methyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carbohydrazide —— C22H22N2O2S
(5S)-5-ethyl-N'-[(2-oxonaphthalen-1-ylidene)methyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carbohydrazide
—— (5R)-N-[(Z)-[4-(2-amino-2-oxoethoxy)-3-methoxyphenyl]methylideneamino]-5-ethyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C21H25N3O4S
(5R)-N-[(Z)-[4-(2-amino-2-oxoethoxy)-3-methoxyphenyl]methylideneamino]-5-ethyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— (5R)-N-[(Z)-(3,5-dimethyl-1-phenylpyrazol-4-yl)methylideneamino]-5-ethyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C23H26N4OS
(5R)-N-[(Z)-(3,5-dimethyl-1-phenylpyrazol-4-yl)methylideneamino]-5-ethyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— (5S)-5-ethyl-N'-[(3-nitro-6-oxocyclohexa-2,4-dien-1-ylidene)methyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carbohydrazide —— C18H19N3O4S
(5S)-5-ethyl-N'-[(3-nitro-6-oxocyclohexa-2,4-dien-1-ylidene)methyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carbohydrazide
—— (5R)-N-[(Z)-[4-(dimethylamino)phenyl]methylideneamino]-5-ethyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C20H25N3OS
(5R)-N-[(Z)-[4-(dimethylamino)phenyl]methylideneamino]-5-ethyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— 5-methyl-3-[[(3R)-3-methyl-4-[(1-methylimidazol-2-yl)methyl]piperazin-1-yl]methyl]-1,2-oxazole —— C15H23N5O
5-methyl-3-[[(3R)-3-methyl-4-[(1-methylimidazol-2-yl)methyl]piperazin-1-yl]methyl]-1,2-oxazole
—— (5R)-5-ethyl-N-[(Z)-thiophen-2-ylmethylideneamino]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C16H18N2OS2
(5R)-5-ethyl-N-[(Z)-thiophen-2-ylmethylideneamino]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— (5-ethyl-1H-pyrazol-4-yl)-[(3S)-3-(4-methylpyrazol-1-yl)piperidin-1-yl]methanone —— C15H21N5O
(5-ethyl-1H-pyrazol-4-yl)-[(3S)-3-(4-methylpyrazol-1-yl)piperidin-1-yl]methanone
—— (5S)-5-ethyl-N-[(Z)-naphthalen-2-ylmethylideneamino]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C22H22N2OS
(5S)-5-ethyl-N-[(Z)-naphthalen-2-ylmethylideneamino]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— (5S)-N-[(Z)-(4-acetamidophenyl)methylideneamino]-5-ethyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C20H23N3O2S
(5S)-N-[(Z)-(4-acetamidophenyl)methylideneamino]-5-ethyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— 5-[(1R)-1-[4-[(5-ethoxy-1,3,4-thiadiazol-2-yl)methyl]piperazin-1-yl]ethyl]-3-methyl-1,2,4-oxadiazole —— C14H22N6O2S
5-[(1R)-1-[4-[(5-ethoxy-1,3,4-thiadiazol-2-yl)methyl]piperazin-1-yl]ethyl]-3-methyl-1,2,4-oxadiazole
—— (5-tert-butyl-1H-pyrazol-3-yl)-[(3S)-3-pyrazol-1-ylpiperidin-1-yl]methanone —— C16H23N5O
(5-tert-butyl-1H-pyrazol-3-yl)-[(3S)-3-pyrazol-1-ylpiperidin-1-yl]methanone
—— 5-fluoro-8-[[4-[[(2S)-oxolan-2-yl]methyl]-1,4-diazepan-1-yl]methyl]quinoline —— C20H26FN3O
5-fluoro-8-[[4-[[(2S)-oxolan-2-yl]methyl]-1,4-diazepan-1-yl]methyl]quinoline
—— (5-ethyl-1H-pyrazol-4-yl)-[(3R)-3-(4-methylpyrazol-1-yl)piperidin-1-yl]methanone —— C15H21N5O
(5-ethyl-1H-pyrazol-4-yl)-[(3R)-3-(4-methylpyrazol-1-yl)piperidin-1-yl]methanone
—— (5-methyl-1H-pyrazol-4-yl)-[(3R)-3-(4-methylpyrazol-1-yl)piperidin-1-yl]methanone —— C14H19N5O
(5-methyl-1H-pyrazol-4-yl)-[(3R)-3-(4-methylpyrazol-1-yl)piperidin-1-yl]methanone
—— 5-[(1S)-1-[4-[(5-ethoxy-1,3,4-thiadiazol-2-yl)methyl]piperazin-1-yl]ethyl]-3-methyl-1,2,4-oxadiazole —— C14H22N6O2S
5-[(1S)-1-[4-[(5-ethoxy-1,3,4-thiadiazol-2-yl)methyl]piperazin-1-yl]ethyl]-3-methyl-1,2,4-oxadiazole
—— (5-tert-butyl-1H-pyrazol-3-yl)-[(3R)-3-pyrazol-1-ylpiperidin-1-yl]methanone —— C16H23N5O
(5-tert-butyl-1H-pyrazol-3-yl)-[(3R)-3-pyrazol-1-ylpiperidin-1-yl]methanone
—— (5-methyl-1H-pyrazol-4-yl)-[(3S)-3-(4-methylpyrazol-1-yl)piperidin-1-yl]methanone —— C14H19N5O
(5-methyl-1H-pyrazol-4-yl)-[(3S)-3-(4-methylpyrazol-1-yl)piperidin-1-yl]methanone
—— 5,5-Dimethyl-2-[2-[4-(2-phenylacetyl)piperazin-1-yl]ethyliminomethyl]cyclohexane-1,3-dione —— C23H31N3O3
5,5-Dimethyl-2-[2-[4-(2-phenylacetyl)piperazin-1-yl]ethyliminomethyl]cyclohexane-1,3-dione
—— 5,5-Dimethyl-2-[2-[4-(2-phenylacetyl)piperazin-1-ium-1-yl]ethyliminomethyl]cyclohexane-1,3-dione —— C23H32N3O3+
5,5-Dimethyl-2-[2-[4-(2-phenylacetyl)piperazin-1-ium-1-yl]ethyliminomethyl]cyclohexane-1,3-dione
—— (5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)-[(3S)-3-(4-methylpyrazol-1-yl)piperidin-1-yl]methanone —— C17H21N7O
(5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)-[(3S)-3-(4-methylpyrazol-1-yl)piperidin-1-yl]methanone
—— 5-[(1S)-1-[4-(6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)piperazin-1-yl]ethyl]-3-ethyl-1,2,4-oxadiazole —— C17H24N6O
5-[(1S)-1-[4-(6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)piperazin-1-yl]ethyl]-3-ethyl-1,2,4-oxadiazole
—— [5-(5-methylthiophen-2-yl)-1H-pyrazol-3-yl]-[(3R)-3-pyrazol-1-ylpiperidin-1-yl]methanone —— C17H19N5OS
[5-(5-methylthiophen-2-yl)-1H-pyrazol-3-yl]-[(3R)-3-pyrazol-1-ylpiperidin-1-yl]methanone
—— (5R)-1-ethyl-5-[2-(1H-indol-3-yl)ethyliminomethyl]-2-sulfanylidene-1,3-diazinane-4,6-dione —— C17H18N4O2S
(5R)-1-ethyl-5-[2-(1H-indol-3-yl)ethyliminomethyl]-2-sulfanylidene-1,3-diazinane-4,6-dione
—— (5S)-1-ethyl-5-(furan-2-ylmethyliminomethyl)-2-sulfanylidene-1,3-diazinane-4,6-dione —— C12H13N3O3S
(5S)-1-ethyl-5-(furan-2-ylmethyliminomethyl)-2-sulfanylidene-1,3-diazinane-4,6-dione
—— 5-[(1R)-1-[4-(6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)piperazin-1-yl]ethyl]-3-ethyl-1,2,4-oxadiazole —— C17H24N6O
5-[(1R)-1-[4-(6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)piperazin-1-yl]ethyl]-3-ethyl-1,2,4-oxadiazole
—— (5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)-[(3R)-3-(4-methylpyrazol-1-yl)piperidin-1-yl]methanone —— C17H21N7O
(5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)-[(3R)-3-(4-methylpyrazol-1-yl)piperidin-1-yl]methanone
—— (5R)-5-(cyclopentyliminomethyl)-1-methyl-2-sulfanylidene-1,3-diazinane-4,6-dione —— C11H15N3O2S
(5R)-5-(cyclopentyliminomethyl)-1-methyl-2-sulfanylidene-1,3-diazinane-4,6-dione
—— (5R)-N-[(1R,8aR)-1,2,3,5,6,7,8,8a-octahydroindolizin-1-yl]-3-(3-fluorophenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide —— C18H22FN3O2
(5R)-N-[(1R,8aR)-1,2,3,5,6,7,8,8a-octahydroindolizin-1-yl]-3-(3-fluorophenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5S)-N-[(1S,8aR)-1,2,3,5,6,7,8,8a-octahydroindolizin-1-yl]-3-(3-fluorophenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide —— C18H22FN3O2
(5S)-N-[(1S,8aR)-1,2,3,5,6,7,8,8a-octahydroindolizin-1-yl]-3-(3-fluorophenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
—— 5-(4-fluorophenyl)-N-[(3R)-1-methyl-5-oxopyrrolidin-3-yl]-5-oxopentanamide —— C16H19FN2O3
5-(4-fluorophenyl)-N-[(3R)-1-methyl-5-oxopyrrolidin-3-yl]-5-oxopentanamide
—— 5-chloro-N-[[(3R)-1-(2-methoxyphenyl)pyrrolidin-3-yl]methyl]furan-2-carboxamide —— C17H19ClN2O3
5-chloro-N-[[(3R)-1-(2-methoxyphenyl)pyrrolidin-3-yl]methyl]furan-2-carboxamide
—— 5-chloro-N-[[(3S)-1-(2-methoxyphenyl)pyrrolidin-3-yl]methyl]furan-2-carboxamide —— C17H19ClN2O3
5-chloro-N-[[(3S)-1-(2-methoxyphenyl)pyrrolidin-3-yl]methyl]furan-2-carboxamide
—— 5-imino-2-[(1R)-1-phenylpropyl]-6-(thiophen-2-ylmethylidene)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C19H16N4OS2
5-imino-2-[(1R)-1-phenylpropyl]-6-(thiophen-2-ylmethylidene)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 5-(4-fluorophenyl)-N-[(3S)-1-methyl-5-oxopyrrolidin-3-yl]-5-oxopentanamide —— C16H19FN2O3
5-(4-fluorophenyl)-N-[(3S)-1-methyl-5-oxopyrrolidin-3-yl]-5-oxopentanamide
—— 5-[(4aS,8aR)-3,4,4a,5,6,7,8,8a-octahydro-2H-quinoline-1-carbonyl]-4-methylthiophene-2-sulfonamide —— C15H22N2O3S2
5-[(4aS,8aR)-3,4,4a,5,6,7,8,8a-octahydro-2H-quinoline-1-carbonyl]-4-methylthiophene-2-sulfonamide
—— 5,6-dimethyl-2-[(2R)-1-(4-methylpiperidin-1-yl)-1-oxopropan-2-yl]sulfanyl-3-propan-2-ylthieno[2,3-d]pyrimidin-4-one —— C20H29N3O2S2
5,6-dimethyl-2-[(2R)-1-(4-methylpiperidin-1-yl)-1-oxopropan-2-yl]sulfanyl-3-propan-2-ylthieno[2,3-d]pyrimidin-4-one
—— 5-[(1S)-1-(4-propan-2-ylpiperazin-1-yl)ethyl]-3-propyl-1,2,4-oxadiazole —— C14H26N4O
5-[(1S)-1-(4-propan-2-ylpiperazin-1-yl)ethyl]-3-propyl-1,2,4-oxadiazole
—— 5-[(4aS,8aS)-3,4,4a,5,6,7,8,8a-octahydro-2H-quinoline-1-carbonyl]-4-methylthiophene-2-sulfonamide —— C15H22N2O3S2
5-[(4aS,8aS)-3,4,4a,5,6,7,8,8a-octahydro-2H-quinoline-1-carbonyl]-4-methylthiophene-2-sulfonamide
—— 5-bromo-N-[(1S)-1-cyanobutyl]-2,3-dihydro-1,4-benzodioxine-7-carboxamide —— C14H15BrN2O3
5-bromo-N-[(1S)-1-cyanobutyl]-2,3-dihydro-1,4-benzodioxine-7-carboxamide
—— 5,6-dimethyl-2-[2-[(2S)-2-methylpiperidin-1-yl]-2-oxoethyl]sulfanyl-3-propan-2-ylthieno[2,3-d]pyrimidin-4-one —— C19H27N3O2S2
5,6-dimethyl-2-[2-[(2S)-2-methylpiperidin-1-yl]-2-oxoethyl]sulfanyl-3-propan-2-ylthieno[2,3-d]pyrimidin-4-one
—— (5S)-5-(3,4-dichlorophenyl)-1,5,7,8,9,10-hexahydropyrimido[4,5-b]quinoline-2,4,6-trione —— C17H13Cl2N3O3
(5S)-5-(3,4-dichlorophenyl)-1,5,7,8,9,10-hexahydropyrimido[4,5-b]quinoline-2,4,6-trione