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—— 5-[(3-fluorophenoxy)methyl]-N-methyl-N-[(1R)-1-(1,3-thiazol-5-yl)ethyl]-1H-pyrazole-3-carboxamide —— C17H17FN4O2S
5-[(3-fluorophenoxy)methyl]-N-methyl-N-[(1R)-1-(1,3-thiazol-5-yl)ethyl]-1H-pyrazole-3-carboxamide
—— 5-[(2S)-1-(1H-imidazol-2-ylmethyl)pyrrolidin-2-yl]-3-pyridin-2-yl-1,2,4-oxadiazole —— C15H16N6O
5-[(2S)-1-(1H-imidazol-2-ylmethyl)pyrrolidin-2-yl]-3-pyridin-2-yl-1,2,4-oxadiazole
—— 5-(4-Bromophenyl)-2-formylpyrazole-3-carboxylate —— C11H6BrN2O3-
5-(4-Bromophenyl)-2-formylpyrazole-3-carboxylate
—— (5S)-5-[2-[methyl(methylsulfonyl)amino]ethylamino]-1-prop-2-enyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C15H24N4O4S
(5S)-5-[2-[methyl(methylsulfonyl)amino]ethylamino]-1-prop-2-enyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— 5-[(2R)-butan-2-yl]-1-(2-methylpropyl)-2H-imidazo[4,5-c]pyrazole —— C12H20N4
5-[(2R)-butan-2-yl]-1-(2-methylpropyl)-2H-imidazo[4,5-c]pyrazole
—— (5S)-5-(3-propan-2-ylphenoxy)-1-azabicyclo[3.2.1]octane —— C16H23NO
(5S)-5-(3-propan-2-ylphenoxy)-1-azabicyclo[3.2.1]octane
—— (5R)-5-[2-[methyl(methylsulfonyl)amino]ethylamino]-1-prop-2-enyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C15H24N4O4S
(5R)-5-[2-[methyl(methylsulfonyl)amino]ethylamino]-1-prop-2-enyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— (5S)-5-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methylamino]-1-prop-2-enyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C21H27N5O2
(5S)-5-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methylamino]-1-prop-2-enyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— 5-[(2-fluorophenoxy)methyl]-N-[(1S)-2-hydroxy-1-pyridin-3-ylethyl]-1H-pyrazole-3-carboxamide —— C18H17FN4O3
5-[(2-fluorophenoxy)methyl]-N-[(1S)-2-hydroxy-1-pyridin-3-ylethyl]-1H-pyrazole-3-carboxamide
—— 5-(phenoxymethyl)-N-[(1R)-1-(4-propan-2-yl-1,2,4-triazol-3-yl)ethyl]-1H-pyrazole-3-carboxamide —— C18H22N6O2
5-(phenoxymethyl)-N-[(1R)-1-(4-propan-2-yl-1,2,4-triazol-3-yl)ethyl]-1H-pyrazole-3-carboxamide
—— (5R)-5-[methyl-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino]-1-(2-methylpropyl)-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C17H25N5O3
(5R)-5-[methyl-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino]-1-(2-methylpropyl)-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— 5-[[benzyl(methyl)amino]methyl]-N-[2-[(2S)-piperidin-2-yl]ethyl]-1,2-oxazole-3-carboxamide —— C20H28N4O2
5-[[benzyl(methyl)amino]methyl]-N-[2-[(2S)-piperidin-2-yl]ethyl]-1,2-oxazole-3-carboxamide
—— 5-(phenoxymethyl)-N-[(1S)-1-(4-propan-2-yl-1,2,4-triazol-3-yl)ethyl]-1H-pyrazole-3-carboxamide —— C18H22N6O2
5-(phenoxymethyl)-N-[(1S)-1-(4-propan-2-yl-1,2,4-triazol-3-yl)ethyl]-1H-pyrazole-3-carboxamide
—— 5-[(3R)-1-(2-methoxyacetyl)piperidin-3-yl]-2-methyl-4-phenyl-1,2,4-triazol-3-one —— C17H22N4O3
5-[(3R)-1-(2-methoxyacetyl)piperidin-3-yl]-2-methyl-4-phenyl-1,2,4-triazol-3-one
—— 5-acetyl-N-[(1R)-1-(1-ethyl-3,5-dimethylpyrazol-4-yl)ethyl]-2,4-dimethyl-1H-pyrrole-3-carboxamide —— C18H26N4O2
5-acetyl-N-[(1R)-1-(1-ethyl-3,5-dimethylpyrazol-4-yl)ethyl]-2,4-dimethyl-1H-pyrrole-3-carboxamide
—— 5-acetyl-N-[(1S)-1-(1-ethyl-3,5-dimethylpyrazol-4-yl)ethyl]-2,4-dimethyl-1H-pyrrole-3-carboxamide —— C18H26N4O2
5-acetyl-N-[(1S)-1-(1-ethyl-3,5-dimethylpyrazol-4-yl)ethyl]-2,4-dimethyl-1H-pyrrole-3-carboxamide
—— (5R)-1-(2-methylpropyl)-5-(pyridin-3-ylmethylamino)-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C18H24N4O2
(5R)-1-(2-methylpropyl)-5-(pyridin-3-ylmethylamino)-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— (5R)-5-[methyl-[(4-methylthiadiazol-5-yl)methyl]amino]-1-(2-methylpropyl)-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C17H25N5O2S
(5R)-5-[methyl-[(4-methylthiadiazol-5-yl)methyl]amino]-1-(2-methylpropyl)-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— (5S)-1,3-dimethyl-5-(3,4,5-trimethoxyphenyl)-6,8-dihydro-5H-pyrido[2,3-d]pyrimidine-2,4,7-trione —— C18H21N3O6
(5S)-1,3-dimethyl-5-(3,4,5-trimethoxyphenyl)-6,8-dihydro-5H-pyrido[2,3-d]pyrimidine-2,4,7-trione
—— 5-[(2R)-1-(1H-imidazol-2-ylmethyl)pyrrolidin-2-yl]-3-propan-2-yl-1,2,4-oxadiazole —— C13H19N5O
5-[(2R)-1-(1H-imidazol-2-ylmethyl)pyrrolidin-2-yl]-3-propan-2-yl-1,2,4-oxadiazole
—— (5S)-1-ethyl-5-[[4-(1,2,4-triazol-1-yl)phenyl]methylamino]-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C19H22N6O2
(5S)-1-ethyl-5-[[4-(1,2,4-triazol-1-yl)phenyl]methylamino]-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— 5-[(2R)-1-(1H-imidazol-2-ylmethyl)pyrrolidin-2-yl]-3-pyridin-2-yl-1,2,4-oxadiazole —— C15H16N6O
5-[(2R)-1-(1H-imidazol-2-ylmethyl)pyrrolidin-2-yl]-3-pyridin-2-yl-1,2,4-oxadiazole
—— 5-[(3-fluorophenoxy)methyl]-N-methyl-N-[(1S)-1-(1,3-thiazol-5-yl)ethyl]-1H-pyrazole-3-carboxamide —— C17H17FN4O2S
5-[(3-fluorophenoxy)methyl]-N-methyl-N-[(1S)-1-(1,3-thiazol-5-yl)ethyl]-1H-pyrazole-3-carboxamide
—— (5R)-5-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methylamino]-1-prop-2-enyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C21H27N5O2
(5R)-5-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methylamino]-1-prop-2-enyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— (5R)-1-ethyl-5-[[4-(1,2,4-triazol-1-yl)phenyl]methylamino]-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C19H22N6O2
(5R)-1-ethyl-5-[[4-(1,2,4-triazol-1-yl)phenyl]methylamino]-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— [(5R)-2,7-diazaspiro[4.5]decan-7-yl]-[2-(2-methylprop-2-enoxy)phenyl]methanone —— C19H26N2O2
[(5R)-2,7-diazaspiro[4.5]decan-7-yl]-[2-(2-methylprop-2-enoxy)phenyl]methanone
—— (5S)-5-[methyl-[(4-methylthiadiazol-5-yl)methyl]amino]-1-(2-methylpropyl)-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C17H25N5O2S
(5S)-5-[methyl-[(4-methylthiadiazol-5-yl)methyl]amino]-1-(2-methylpropyl)-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— 5-[[(2S)-2-(aminomethyl)morpholin-4-yl]methyl]-N-benzylpyrimidin-2-amine —— C17H23N5O
5-[[(2S)-2-(aminomethyl)morpholin-4-yl]methyl]-N-benzylpyrimidin-2-amine
—— 5-[(4-hydroxypiperidin-1-yl)methyl]-N-[(1R)-1-phenylethyl]-N-propyl-1,2-oxazole-3-carboxamide —— C21H29N3O3
5-[(4-hydroxypiperidin-1-yl)methyl]-N-[(1R)-1-phenylethyl]-N-propyl-1,2-oxazole-3-carboxamide
—— 5-[(2S)-1-(1H-imidazol-2-ylmethyl)pyrrolidin-2-yl]-3-propan-2-yl-1,2,4-oxadiazole —— C13H19N5O
5-[(2S)-1-(1H-imidazol-2-ylmethyl)pyrrolidin-2-yl]-3-propan-2-yl-1,2,4-oxadiazole
—— 5-[[(2R)-2-(aminomethyl)morpholin-4-yl]methyl]-N-benzylpyrimidin-2-amine —— C17H23N5O
5-[[(2R)-2-(aminomethyl)morpholin-4-yl]methyl]-N-benzylpyrimidin-2-amine
—— (5R)-2-(3-azaspiro[5.5]undecan-9-yl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one —— C19H33N3O
(5R)-2-(3-azaspiro[5.5]undecan-9-yl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-(3-azaspiro[5.5]undecan-9-yl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one —— C19H33N3O
(5S)-2-(3-azaspiro[5.5]undecan-9-yl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(3S)-1-(1-benzofuran-2-ylmethyl)piperidin-3-yl]-4-ethyl-2-methyl-1,2,4-triazol-3-one —— C19H24N4O2
5-[(3S)-1-(1-benzofuran-2-ylmethyl)piperidin-3-yl]-4-ethyl-2-methyl-1,2,4-triazol-3-one
—— [(5S)-2,7-diazaspiro[4.5]decan-7-yl]-[2-(2-methylprop-2-enoxy)phenyl]methanone —— C19H26N2O2
[(5S)-2,7-diazaspiro[4.5]decan-7-yl]-[2-(2-methylprop-2-enoxy)phenyl]methanone
—— 5-[(4-hydroxypiperidin-1-yl)methyl]-N-[(1S)-1-phenylethyl]-N-propyl-1,2-oxazole-3-carboxamide —— C21H29N3O3
5-[(4-hydroxypiperidin-1-yl)methyl]-N-[(1S)-1-phenylethyl]-N-propyl-1,2-oxazole-3-carboxamide
—— 5-[[benzyl(methyl)amino]methyl]-N-[2-[(2R)-piperidin-2-yl]ethyl]-1,2-oxazole-3-carboxamide —— C20H28N4O2
5-[[benzyl(methyl)amino]methyl]-N-[2-[(2R)-piperidin-2-yl]ethyl]-1,2-oxazole-3-carboxamide
—— 5-methyl-N-[[(3R)-1-propan-2-ylpyrrolidin-3-yl]methyl]-1-propylpyrazole-4-carboxamide —— C16H28N4O
5-methyl-N-[[(3R)-1-propan-2-ylpyrrolidin-3-yl]methyl]-1-propylpyrazole-4-carboxamide
—— 5-chloro-N-[[(3R)-1-(furan-2-ylmethyl)pyrrolidin-3-yl]methyl]-2-oxo-1H-pyridine-3-carboxamide —— C16H18ClN3O3
5-chloro-N-[[(3R)-1-(furan-2-ylmethyl)pyrrolidin-3-yl]methyl]-2-oxo-1H-pyridine-3-carboxamide
—— (5S)-1-ethyl-5-[(3-methoxy-3-oxopropyl)amino]-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C14H21N3O4
(5S)-1-ethyl-5-[(3-methoxy-3-oxopropyl)amino]-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— 5-fluoro-2-methoxy-N-[[(3S)-1-methylpiperidin-3-yl]methyl]benzamide —— C15H21FN2O2
5-fluoro-2-methoxy-N-[[(3S)-1-methylpiperidin-3-yl]methyl]benzamide
—— (5S)-N-(2,3-dihydro-1H-inden-2-yl)-N,5-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide —— C19H23N3O
(5S)-N-(2,3-dihydro-1H-inden-2-yl)-N,5-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
—— 5-(3-fluorophenyl)-N-[2-[(2S)-2-(hydroxymethyl)piperidin-1-yl]ethyl]-1H-pyrazole-4-carboxamide —— C18H23FN4O2
5-(3-fluorophenyl)-N-[2-[(2S)-2-(hydroxymethyl)piperidin-1-yl]ethyl]-1H-pyrazole-4-carboxamide
—— (5R)-5-[2-(4,6-dimethyl-2-oxopyrimidin-1-yl)ethylamino]-1-ethyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C18H25N5O3
(5R)-5-[2-(4,6-dimethyl-2-oxopyrimidin-1-yl)ethylamino]-1-ethyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— (5S)-5-[4-[(2-cyanophenyl)methyl]piperazin-1-yl]-1-ethyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C22H27N5O2
(5S)-5-[4-[(2-cyanophenyl)methyl]piperazin-1-yl]-1-ethyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— (5R)-2-[(4-chlorophenyl)methylsulfonyl]-2,9-diazaspiro[4.5]decane —— C15H21ClN2O2S
(5R)-2-[(4-chlorophenyl)methylsulfonyl]-2,9-diazaspiro[4.5]decane
—— (5R)-N-(2,3-dihydro-1H-inden-2-yl)-N,5-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide —— C19H23N3O
(5R)-N-(2,3-dihydro-1H-inden-2-yl)-N,5-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
—— 5-[(3S)-1-[2-(1H-benzimidazol-2-yl)acetyl]piperidin-3-yl]-4-ethyl-2-methyl-1,2,4-triazol-3-one —— C19H24N6O2
5-[(3S)-1-[2-(1H-benzimidazol-2-yl)acetyl]piperidin-3-yl]-4-ethyl-2-methyl-1,2,4-triazol-3-one
—— 5-[(3-acetylphenoxy)methyl]-N-[(3S)-3-hydroxybutyl]-1,2-oxazole-3-carboxamide —— C17H20N2O5
5-[(3-acetylphenoxy)methyl]-N-[(3S)-3-hydroxybutyl]-1,2-oxazole-3-carboxamide
—— 5-(benzimidazol-1-ylmethyl)-N-[(2S)-2-(3,5-dimethylpyrazol-1-yl)propyl]-1H-pyrazole-3-carboxamide —— C20H23N7O
5-(benzimidazol-1-ylmethyl)-N-[(2S)-2-(3,5-dimethylpyrazol-1-yl)propyl]-1H-pyrazole-3-carboxamide