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—— 5,6-dimethyl-3-[[(6S)-3-propan-2-yl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-6-yl]methylamino]pyridazine-4-carbonitrile —— C17H23N7
5,6-dimethyl-3-[[(6S)-3-propan-2-yl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-6-yl]methylamino]pyridazine-4-carbonitrile
—— 5,6-dimethyl-3-[[(6R)-3-propan-2-yl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-6-yl]methylamino]pyridazine-4-carbonitrile —— C17H23N7
5,6-dimethyl-3-[[(6R)-3-propan-2-yl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-6-yl]methylamino]pyridazine-4-carbonitrile
—— 5-chloro-N-[(2R)-1-cyanopropan-2-yl]-2-pyrrolidin-1-ylpyrimidine-4-carboxamide —— C13H16ClN5O
5-chloro-N-[(2R)-1-cyanopropan-2-yl]-2-pyrrolidin-1-ylpyrimidine-4-carboxamide
—— 5-[(2S)-2-[(2S)-1-ethylpyrrolidin-2-yl]pyrrolidine-1-carbonyl]thiophene-2-carboxamide —— C16H23N3O2S
5-[(2S)-2-[(2S)-1-ethylpyrrolidin-2-yl]pyrrolidine-1-carbonyl]thiophene-2-carboxamide
—— 5-fluoro-8-[[(2S)-2-(1-methylpyrazol-4-yl)pyrrolidin-1-yl]methyl]quinoline —— C18H19FN4
5-fluoro-8-[[(2S)-2-(1-methylpyrazol-4-yl)pyrrolidin-1-yl]methyl]quinoline
—— 5-[(1S)-1-[(3S)-3-ethyl-4-(2-methoxyethyl)piperazin-1-yl]ethyl]-3-methyl-1,2,4-oxadiazole —— C14H26N4O2
5-[(1S)-1-[(3S)-3-ethyl-4-(2-methoxyethyl)piperazin-1-yl]ethyl]-3-methyl-1,2,4-oxadiazole
—— 5,7-dimethyl-6-[2-[(2R)-2-methylthiomorpholin-4-yl]-2-oxoethyl]-1H-pyrazolo[1,5-a]pyrimidin-2-one —— C15H20N4O2S
5,7-dimethyl-6-[2-[(2R)-2-methylthiomorpholin-4-yl]-2-oxoethyl]-1H-pyrazolo[1,5-a]pyrimidin-2-one
—— 5-[[(1S)-1-(3-fluorophenyl)ethyl]sulfonylmethyl]-3-phenyl-1,2-oxazole —— C18H16FNO3S
5-[[(1S)-1-(3-fluorophenyl)ethyl]sulfonylmethyl]-3-phenyl-1,2-oxazole
—— 5-[[(1R)-1-(3-fluorophenyl)ethyl]sulfonylmethyl]-3-phenyl-1,2-oxazole —— C18H16FNO3S
5-[[(1R)-1-(3-fluorophenyl)ethyl]sulfonylmethyl]-3-phenyl-1,2-oxazole
—— 5-[(1S)-1-[(4-ethoxyphenyl)methylamino]ethyl]-1,3-dihydrobenzimidazol-2-one —— C18H21N3O2
5-[(1S)-1-[(4-ethoxyphenyl)methylamino]ethyl]-1,3-dihydrobenzimidazol-2-one
—— 5-[(1R)-1-[(4-ethoxyphenyl)methylamino]ethyl]-1,3-dihydrobenzimidazol-2-one —— C18H21N3O2
5-[(1R)-1-[(4-ethoxyphenyl)methylamino]ethyl]-1,3-dihydrobenzimidazol-2-one
—— (5S)-N-[(4,5-dimethyl-1,2,4-triazol-3-yl)methyl]-5-phenyl-4,5-dihydro-1,2-oxazole-3-carboxamide —— C15H17N5O2
(5S)-N-[(4,5-dimethyl-1,2,4-triazol-3-yl)methyl]-5-phenyl-4,5-dihydro-1,2-oxazole-3-carboxamide
—— 5,6-diethyl-2-[(2R)-2-hydroxy-2-(4-propan-2-ylphenyl)ethyl]-3-oxopyridazine-4-carbonitrile —— C20H25N3O2
5,6-diethyl-2-[(2R)-2-hydroxy-2-(4-propan-2-ylphenyl)ethyl]-3-oxopyridazine-4-carbonitrile
—— (5S)-5-[(2S)-2-(4-chlorophenyl)morpholine-4-carbonyl]pyrrolidin-2-one —— C15H17ClN2O3
(5S)-5-[(2S)-2-(4-chlorophenyl)morpholine-4-carbonyl]pyrrolidin-2-one
—— (5R)-N-[(4,5-dimethyl-1,2,4-triazol-3-yl)methyl]-5-phenyl-4,5-dihydro-1,2-oxazole-3-carboxamide —— C15H17N5O2
(5R)-N-[(4,5-dimethyl-1,2,4-triazol-3-yl)methyl]-5-phenyl-4,5-dihydro-1,2-oxazole-3-carboxamide
—— (5-fluoro-1-benzothiophen-2-yl)-[(3R)-3-imidazol-1-ylpiperidin-1-yl]methanone —— C17H16FN3OS
(5-fluoro-1-benzothiophen-2-yl)-[(3R)-3-imidazol-1-ylpiperidin-1-yl]methanone
—— 5-methyl-2-thiophen-3-yl-4-[[(3S)-3-(1,2,4-triazol-1-ylmethyl)piperidin-1-yl]methyl]-1,3-oxazole —— C17H21N5OS
5-methyl-2-thiophen-3-yl-4-[[(3S)-3-(1,2,4-triazol-1-ylmethyl)piperidin-1-yl]methyl]-1,3-oxazole
—— 5-chloro-N-[2-(diethylamino)ethyl]-N-(4-fluoro-1,3-benzothiazol-2-yl)thiophene-2-carboxamide —— C18H19ClFN3OS2
5-chloro-N-[2-(diethylamino)ethyl]-N-(4-fluoro-1,3-benzothiazol-2-yl)thiophene-2-carboxamide
—— (5S)-5-[(2R)-2-(4-chlorophenyl)morpholine-4-carbonyl]pyrrolidin-2-one —— C15H17ClN2O3
(5S)-5-[(2R)-2-(4-chlorophenyl)morpholine-4-carbonyl]pyrrolidin-2-one
—— 5-chloro-N-[2-(diethylamino)ethyl]-N-(6-fluoro-1,3-benzothiazol-2-yl)thiophene-2-carboxamide —— C18H19ClFN3OS2
5-chloro-N-[2-(diethylamino)ethyl]-N-(6-fluoro-1,3-benzothiazol-2-yl)thiophene-2-carboxamide
—— 5-chloro-N-[2-(diethylamino)ethyl]-N-(4-methyl-1,3-benzothiazol-2-yl)thiophene-2-carboxamide —— C19H22ClN3OS2
5-chloro-N-[2-(diethylamino)ethyl]-N-(4-methyl-1,3-benzothiazol-2-yl)thiophene-2-carboxamide
—— (5-chloroquinolin-8-yl)-[(3R)-3-imidazol-1-ylpiperidin-1-yl]methanone —— C18H17ClN4O
(5-chloroquinolin-8-yl)-[(3R)-3-imidazol-1-ylpiperidin-1-yl]methanone
—— (5-chloroquinolin-8-yl)-[(3S)-3-imidazol-1-ylpiperidin-1-yl]methanone —— C18H17ClN4O
(5-chloroquinolin-8-yl)-[(3S)-3-imidazol-1-ylpiperidin-1-yl]methanone
—— (5R)-5-[(2R)-2-(4-chlorophenyl)morpholine-4-carbonyl]pyrrolidin-2-one —— C15H17ClN2O3
(5R)-5-[(2R)-2-(4-chlorophenyl)morpholine-4-carbonyl]pyrrolidin-2-one
—— 5,6-diethyl-2-[(2S)-2-hydroxy-2-(4-propan-2-ylphenyl)ethyl]-3-oxopyridazine-4-carbonitrile —— C20H25N3O2
5,6-diethyl-2-[(2S)-2-hydroxy-2-(4-propan-2-ylphenyl)ethyl]-3-oxopyridazine-4-carbonitrile
—— 5-phenyl-3-[[(3R)-3-(1,2,4-triazol-1-ylmethyl)piperidin-1-yl]methyl]-1,2,4-oxadiazole —— C17H20N6O
5-phenyl-3-[[(3R)-3-(1,2,4-triazol-1-ylmethyl)piperidin-1-yl]methyl]-1,2,4-oxadiazole
—— 5-(4-fluorophenyl)-3-[[(2R)-4-propan-2-ylmorpholin-2-yl]methyl]-1,3,4-oxadiazol-2-one —— C16H20FN3O3
5-(4-fluorophenyl)-3-[[(2R)-4-propan-2-ylmorpholin-2-yl]methyl]-1,3,4-oxadiazol-2-one
—— 5-methyl-2-thiophen-3-yl-4-[[(3R)-3-(1,2,4-triazol-1-ylmethyl)piperidin-1-yl]methyl]-1,3-oxazole —— C17H21N5OS
5-methyl-2-thiophen-3-yl-4-[[(3R)-3-(1,2,4-triazol-1-ylmethyl)piperidin-1-yl]methyl]-1,3-oxazole
—— 5-phenyl-3-[[(3S)-3-(1,2,4-triazol-1-ylmethyl)piperidin-1-yl]methyl]-1,2,4-oxadiazole —— C17H20N6O
5-phenyl-3-[[(3S)-3-(1,2,4-triazol-1-ylmethyl)piperidin-1-yl]methyl]-1,2,4-oxadiazole
—— 5-phenyl-2-[(1S)-1-(1-prop-2-enyltetrazol-5-yl)sulfanylethyl]-1,3-oxazole —— C15H15N5OS
5-phenyl-2-[(1S)-1-(1-prop-2-enyltetrazol-5-yl)sulfanylethyl]-1,3-oxazole
—— (5-fluoro-1-benzothiophen-2-yl)-[(3S)-3-imidazol-1-ylpiperidin-1-yl]methanone —— C17H16FN3OS
(5-fluoro-1-benzothiophen-2-yl)-[(3S)-3-imidazol-1-ylpiperidin-1-yl]methanone
—— 5-chloro-N-[2-(dimethylamino)ethyl]-N-(5,7-dimethyl-1,3-benzothiazol-2-yl)thiophene-2-carboxamide —— C18H20ClN3OS2
5-chloro-N-[2-(dimethylamino)ethyl]-N-(5,7-dimethyl-1,3-benzothiazol-2-yl)thiophene-2-carboxamide
—— 5-phenyl-2-[(1R)-1-(1-prop-2-enyltetrazol-5-yl)sulfanylethyl]-1,3-oxazole —— C15H15N5OS
5-phenyl-2-[(1R)-1-(1-prop-2-enyltetrazol-5-yl)sulfanylethyl]-1,3-oxazole
—— (5-chloro-2-propan-2-ylpyrimidin-4-yl)-[(3R)-3-imidazol-1-ylpiperidin-1-yl]methanone —— C16H20ClN5O
(5-chloro-2-propan-2-ylpyrimidin-4-yl)-[(3R)-3-imidazol-1-ylpiperidin-1-yl]methanone
—— 5-[(2R)-2-[(3,5-dimethylpyrazol-1-yl)methyl]piperidine-1-carbonyl]thiophene-3-carboxamide —— C17H22N4O2S
5-[(2R)-2-[(3,5-dimethylpyrazol-1-yl)methyl]piperidine-1-carbonyl]thiophene-3-carboxamide
—— 5-[cyclohexyl-[(2S)-2-hydroxypropyl]amino]pentanenitrile —— C14H26N2O
5-[cyclohexyl-[(2S)-2-hydroxypropyl]amino]pentanenitrile
—— (5-chloro-2-propan-2-ylpyrimidin-4-yl)-[(3S)-3-imidazol-1-ylpiperidin-1-yl]methanone —— C16H20ClN5O
(5-chloro-2-propan-2-ylpyrimidin-4-yl)-[(3S)-3-imidazol-1-ylpiperidin-1-yl]methanone
—— 5-[(3R)-3-(2-ethylimidazol-1-yl)piperidine-1-carbonyl]-N-methylpyridine-2-carboxamide —— C18H23N5O2
5-[(3R)-3-(2-ethylimidazol-1-yl)piperidine-1-carbonyl]-N-methylpyridine-2-carboxamide
—— (5-phenyl-1,2-oxazol-3-yl)-[(2R)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone —— C18H18N4O2
(5-phenyl-1,2-oxazol-3-yl)-[(2R)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone
—— 5-[(2R)-2-(2-chlorophenyl)morpholin-4-yl]pentanenitrile —— C15H19ClN2O
5-[(2R)-2-(2-chlorophenyl)morpholin-4-yl]pentanenitrile
—— 5-chloro-N-[2-(dimethylamino)ethyl]-N-(5-methoxy-1,3-benzothiazol-2-yl)thiophene-2-carboxamide —— C17H18ClN3O2S2
5-chloro-N-[2-(dimethylamino)ethyl]-N-(5-methoxy-1,3-benzothiazol-2-yl)thiophene-2-carboxamide
—— 5-[cyclohexyl-[(2R)-2-hydroxypropyl]amino]pentanenitrile —— C14H26N2O
5-[cyclohexyl-[(2R)-2-hydroxypropyl]amino]pentanenitrile
—— (5-phenyl-1,2-oxazol-3-yl)-[(2S)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone —— C18H18N4O2
(5-phenyl-1,2-oxazol-3-yl)-[(2S)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone
—— 5-[(2S)-6-(4-methoxy-3-methylphenyl)sulfonyl-6-azaspiro[2.5]octan-2-yl]-3-pyridin-3-yl-1,2,4-oxadiazole —— C22H24N4O4S
5-[(2S)-6-(4-methoxy-3-methylphenyl)sulfonyl-6-azaspiro[2.5]octan-2-yl]-3-pyridin-3-yl-1,2,4-oxadiazole
—— (5-methylfuran-2-yl)-[(2S)-2-[(4-methylpyrazol-1-yl)methyl]piperidin-1-yl]methanone —— C16H21N3O2
(5-methylfuran-2-yl)-[(2S)-2-[(4-methylpyrazol-1-yl)methyl]piperidin-1-yl]methanone
—— 5-bromo-2-ethoxy-N-(4-fluoro-2-methylphenyl)benzenesulfonamide —— C15H15BrFNO3S
5-bromo-2-ethoxy-N-(4-fluoro-2-methylphenyl)benzenesulfonamide
—— (5-fluoro-1H-indol-2-yl)-[(3R)-3-imidazol-1-ylpiperidin-1-yl]methanone —— C17H17FN4O
(5-fluoro-1H-indol-2-yl)-[(3R)-3-imidazol-1-ylpiperidin-1-yl]methanone
—— [5-(4-fluorophenyl)furan-2-yl]-[(3R)-3-imidazol-1-ylpiperidin-1-yl]methanone —— C19H18FN3O2
[5-(4-fluorophenyl)furan-2-yl]-[(3R)-3-imidazol-1-ylpiperidin-1-yl]methanone
—— 5,7-dimethyl-2-[[(2S)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methyl]imidazo[1,2-a]pyrimidine —— C17H22N6
5,7-dimethyl-2-[[(2S)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methyl]imidazo[1,2-a]pyrimidine
—— 5,7-dimethyl-2-[[(2R)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methyl]imidazo[1,2-a]pyrimidine —— C17H22N6
5,7-dimethyl-2-[[(2R)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methyl]imidazo[1,2-a]pyrimidine