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—— 5-[(5-chloropyridin-3-yl)oxymethyl]-N-[(2R)-5-methylhexan-2-yl]-1,2-oxazole-3-carboxamide —— C17H22ClN3O3
5-[(5-chloropyridin-3-yl)oxymethyl]-N-[(2R)-5-methylhexan-2-yl]-1,2-oxazole-3-carboxamide
—— (5R)-1-ethyl-5-[2-[(3-methylpyridin-4-yl)amino]ethylamino]-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C18H25N5O2
(5R)-1-ethyl-5-[2-[(3-methylpyridin-4-yl)amino]ethylamino]-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— 5-(5-chloro-2-methoxyphenyl)-3-[[(2R)-2-methylpiperidin-1-ium-1-yl]methyl]-1,3,4-oxadiazole-2-thione —— C16H21ClN3O2S+
5-(5-chloro-2-methoxyphenyl)-3-[[(2R)-2-methylpiperidin-1-ium-1-yl]methyl]-1,3,4-oxadiazole-2-thione
—— (5R)-5-[(3,5-dimethyl-1-propan-2-ylpyrazol-4-yl)methyl-methylamino]-1-ethyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C20H31N5O2
(5R)-5-[(3,5-dimethyl-1-propan-2-ylpyrazol-4-yl)methyl-methylamino]-1-ethyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— (5E)-3-[[(2R,6R)-2,6-dimethylmorpholin-4-ium-4-yl]methyl]-5-[(2-methoxyphenyl)methylidene]-1,3-thiazolidine-2,4-dione —— C18H23N2O4S+
(5E)-3-[[(2R,6R)-2,6-dimethylmorpholin-4-ium-4-yl]methyl]-5-[(2-methoxyphenyl)methylidene]-1,3-thiazolidine-2,4-dione
—— (5E)-5-[(5-bromo-2-methoxyphenyl)methylidene]-2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-1,3-thiazol-4-one —— C17H19BrN2O3S
(5E)-5-[(5-bromo-2-methoxyphenyl)methylidene]-2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-1,3-thiazol-4-one
—— (5R)-7-[(3,5-difluoro-4-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decane —— C16H22F2N2O
(5R)-7-[(3,5-difluoro-4-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decane
—— 5-[(5,6-dimethylbenzimidazol-1-yl)methyl]-N-[[(2R)-oxolan-2-yl]methyl]-1H-pyrazole-3-carboxamide —— C19H23N5O2
5-[(5,6-dimethylbenzimidazol-1-yl)methyl]-N-[[(2R)-oxolan-2-yl]methyl]-1H-pyrazole-3-carboxamide
—— 5-(hydroxymethyl)-4-[[(4S)-4-(3-hydroxyphenyl)-1,4,6,7-tetrahydroimidazo[4,5-c]pyridin-5-yl]methyl]-2-methylpyridin-3-ol —— C20H22N4O3
5-(hydroxymethyl)-4-[[(4S)-4-(3-hydroxyphenyl)-1,4,6,7-tetrahydroimidazo[4,5-c]pyridin-5-yl]methyl]-2-methylpyridin-3-ol
—— 5-[(2,6-difluorophenoxy)methyl]-N-methyl-N-[[(3R)-piperidin-3-yl]methyl]-1,2-oxazole-3-carboxamide —— C18H21F2N3O3
5-[(2,6-difluorophenoxy)methyl]-N-methyl-N-[[(3R)-piperidin-3-yl]methyl]-1,2-oxazole-3-carboxamide
—— 5-methyl-N-[(S)-(2-methylphenyl)-thiophen-2-ylmethyl]-1,3,4-oxadiazole-2-carboxamide —— C16H15N3O2S
5-methyl-N-[(S)-(2-methylphenyl)-thiophen-2-ylmethyl]-1,3,4-oxadiazole-2-carboxamide
—— [(5S)-2,7-diazaspiro[4.5]decan-7-yl]-[5-[(4-methylpiperidin-1-yl)methyl]furan-2-yl]methanone —— C20H31N3O2
[(5S)-2,7-diazaspiro[4.5]decan-7-yl]-[5-[(4-methylpiperidin-1-yl)methyl]furan-2-yl]methanone
—— 5-[(2S)-5-oxopyrrolidine-2-carbonyl]-N-phenyl-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine-2-carboxamide —— C18H19N5O3
5-[(2S)-5-oxopyrrolidine-2-carbonyl]-N-phenyl-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine-2-carboxamide
—— 5-[(2R)-5-oxopyrrolidine-2-carbonyl]-N-phenyl-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine-2-carboxamide —— C18H19N5O3
5-[(2R)-5-oxopyrrolidine-2-carbonyl]-N-phenyl-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine-2-carboxamide
—— [(5R)-2,7-diazaspiro[4.5]decan-7-yl]-[5-[(4-methylpiperidin-1-yl)methyl]furan-2-yl]methanone —— C20H31N3O2
[(5R)-2,7-diazaspiro[4.5]decan-7-yl]-[5-[(4-methylpiperidin-1-yl)methyl]furan-2-yl]methanone
—— 5-[(2,6-difluorophenoxy)methyl]-N-methyl-N-[[(3S)-piperidin-3-yl]methyl]-1,2-oxazole-3-carboxamide —— C18H21F2N3O3
5-[(2,6-difluorophenoxy)methyl]-N-methyl-N-[[(3S)-piperidin-3-yl]methyl]-1,2-oxazole-3-carboxamide
—— (5R)-2-[(5-chloro-2,3-dimethoxyphenyl)methyl]-2,9-diazaspiro[4.5]decane —— C17H25ClN2O2
(5R)-2-[(5-chloro-2,3-dimethoxyphenyl)methyl]-2,9-diazaspiro[4.5]decane
—— (5E)-2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-5-[(3-ethoxy-4-hydroxyphenyl)methylidene]-1,3-thiazol-4-one —— C18H22N2O4S
(5E)-2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-5-[(3-ethoxy-4-hydroxyphenyl)methylidene]-1,3-thiazol-4-one
—— 5,6,7-trimethoxy-3-[(4R)-4,5,6,7-tetrahydro-1H-imidazo[4,5-c]pyridin-4-yl]-1H-quinolin-2-one —— C18H20N4O4
5,6,7-trimethoxy-3-[(4R)-4,5,6,7-tetrahydro-1H-imidazo[4,5-c]pyridin-4-yl]-1H-quinolin-2-one
—— [5-(1,3-benzodioxol-5-yloxymethyl)-1H-pyrazol-3-yl]-[(2R)-2-propyl-2,5-dihydropyrrol-1-yl]methanone —— C19H21N3O4
[5-(1,3-benzodioxol-5-yloxymethyl)-1H-pyrazol-3-yl]-[(2R)-2-propyl-2,5-dihydropyrrol-1-yl]methanone
—— 5-[(1R)-1-(4-nitropyrazol-1-yl)ethyl]-3-pyridin-4-yl-1,2,4-oxadiazole —— C12H10N6O3
5-[(1R)-1-(4-nitropyrazol-1-yl)ethyl]-3-pyridin-4-yl-1,2,4-oxadiazole
—— 5,6,7-trimethoxy-3-[(4S)-4,5,6,7-tetrahydro-1H-imidazo[4,5-c]pyridin-4-yl]-1H-quinolin-2-one —— C18H20N4O4
5,6,7-trimethoxy-3-[(4S)-4,5,6,7-tetrahydro-1H-imidazo[4,5-c]pyridin-4-yl]-1H-quinolin-2-one
—— (5S)-5-[5-(3-fluorophenyl)-1H-pyrazol-4-yl]-1,2,5,6-tetrahydropyrazolo[4,3-g]quinolin-7-one —— C19H14FN5O
(5S)-5-[5-(3-fluorophenyl)-1H-pyrazol-4-yl]-1,2,5,6-tetrahydropyrazolo[4,3-g]quinolin-7-one
—— (5S)-5-[(3,5-dimethyl-1-propan-2-ylpyrazol-4-yl)methyl-methylamino]-1-ethyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C20H31N5O2
(5S)-5-[(3,5-dimethyl-1-propan-2-ylpyrazol-4-yl)methyl-methylamino]-1-ethyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— [5-[[benzyl(methyl)amino]methyl]-1,2-oxazol-3-yl]-[(3R)-3-ethyl-4-methylpiperazin-1-yl]methanone —— C20H28N4O2
[5-[[benzyl(methyl)amino]methyl]-1,2-oxazol-3-yl]-[(3R)-3-ethyl-4-methylpiperazin-1-yl]methanone
—— 5-[(1S)-2,2-dimethylcyclopropanecarbonyl]-N-(pyridin-2-ylmethyl)-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine-2-carboxamide —— C19H23N5O2
5-[(1S)-2,2-dimethylcyclopropanecarbonyl]-N-(pyridin-2-ylmethyl)-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine-2-carboxamide
—— 5-[[5-(4-Methylpiperazin-4-ium-1-yl)furan-2-yl]methylidene]-2-sulfanylidene-1,3-diazinane-4,6-dione —— C14H17N4O3S+
5-[[5-(4-Methylpiperazin-4-ium-1-yl)furan-2-yl]methylidene]-2-sulfanylidene-1,3-diazinane-4,6-dione
—— 5-(hydroxymethyl)-4-[[(4R)-4-(3-hydroxyphenyl)-1,4,6,7-tetrahydroimidazo[4,5-c]pyridin-5-yl]methyl]-2-methylpyridin-3-ol —— C20H22N4O3
5-(hydroxymethyl)-4-[[(4R)-4-(3-hydroxyphenyl)-1,4,6,7-tetrahydroimidazo[4,5-c]pyridin-5-yl]methyl]-2-methylpyridin-3-ol
—— 5-chloro-N-[[(3R)-1-[(E)-2-methylpent-2-enyl]pyrrolidin-3-yl]methyl]-6-oxo-1H-pyridine-3-carboxamide —— C17H24ClN3O2
5-chloro-N-[[(3R)-1-[(E)-2-methylpent-2-enyl]pyrrolidin-3-yl]methyl]-6-oxo-1H-pyridine-3-carboxamide
—— 5-[(3R)-oxolane-3-carbonyl]-1-(3,3,3-trifluoropropyl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-3-carboxylic acid —— C15H18F3N3O4
5-[(3R)-oxolane-3-carbonyl]-1-(3,3,3-trifluoropropyl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
—— 5-[(1S)-1-(4-nitropyrazol-1-yl)ethyl]-3-pyridin-4-yl-1,2,4-oxadiazole —— C12H10N6O3
5-[(1S)-1-(4-nitropyrazol-1-yl)ethyl]-3-pyridin-4-yl-1,2,4-oxadiazole
—— (5S)-N-(3-acetamido-4-chlorophenyl)-3-(5-chlorothiophen-2-yl)-4,5-dihydro-1,2-oxazole-5-carboxamide —— C16H13Cl2N3O3S
(5S)-N-(3-acetamido-4-chlorophenyl)-3-(5-chlorothiophen-2-yl)-4,5-dihydro-1,2-oxazole-5-carboxamide
—— 5-[(3R)-3-(1H-pyrazol-5-yl)piperidine-1-carbonyl]-1H-pyrazin-2-one —— C13H15N5O2
5-[(3R)-3-(1H-pyrazol-5-yl)piperidine-1-carbonyl]-1H-pyrazin-2-one
—— (5S)-2-(6-amino-1H-pyrazolo[3,4-d]pyrimidin-4-yl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one —— C14H19N7O
(5S)-2-(6-amino-1H-pyrazolo[3,4-d]pyrimidin-4-yl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(1R)-2,2-dimethylcyclopropanecarbonyl]-N-(pyridin-2-ylmethyl)-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine-2-carboxamide —— C19H23N5O2
5-[(1R)-2,2-dimethylcyclopropanecarbonyl]-N-(pyridin-2-ylmethyl)-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine-2-carboxamide
—— (5S)-1-ethyl-5-[2-(1,2,3,5,6,7-hexahydropyrrolizin-8-yl)ethylamino]-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C19H30N4O2
(5S)-1-ethyl-5-[2-(1,2,3,5,6,7-hexahydropyrrolizin-8-yl)ethylamino]-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— (5S)-7-methyl-2-(6-phenylimidazo[2,1-b][1,3]thiazole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C21H22N4O2S
(5S)-7-methyl-2-(6-phenylimidazo[2,1-b][1,3]thiazole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-5-[5-(3-fluorophenyl)-1H-pyrazol-4-yl]-1,2,5,6-tetrahydropyrazolo[4,3-g]quinolin-7-one —— C19H14FN5O
(5R)-5-[5-(3-fluorophenyl)-1H-pyrazol-4-yl]-1,2,5,6-tetrahydropyrazolo[4,3-g]quinolin-7-one
—— 5-[(5,6-dimethylbenzimidazol-1-yl)methyl]-N-[[(2S)-oxolan-2-yl]methyl]-1H-pyrazole-3-carboxamide —— C19H23N5O2
5-[(5,6-dimethylbenzimidazol-1-yl)methyl]-N-[[(2S)-oxolan-2-yl]methyl]-1H-pyrazole-3-carboxamide
—— 5-[1-[(2S)-2-ethylsulfanylpropanoyl]piperidin-4-yl]-2-methyl-4-phenyl-1,2,4-triazol-3-one —— C19H26N4O2S
5-[1-[(2S)-2-ethylsulfanylpropanoyl]piperidin-4-yl]-2-methyl-4-phenyl-1,2,4-triazol-3-one
—— [5-(1,3-benzodioxol-5-yloxymethyl)-1H-pyrazol-3-yl]-[(2S)-2-propyl-2,5-dihydropyrrol-1-yl]methanone —— C19H21N3O4
[5-(1,3-benzodioxol-5-yloxymethyl)-1H-pyrazol-3-yl]-[(2S)-2-propyl-2,5-dihydropyrrol-1-yl]methanone
—— 5-[(3R)-oxolane-3-carbonyl]-1-(pyridin-2-ylmethyl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-3-carboxylic acid —— C18H20N4O4
5-[(3R)-oxolane-3-carbonyl]-1-(pyridin-2-ylmethyl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
—— [5-[[benzyl(methyl)amino]methyl]-1,2-oxazol-3-yl]-[(3S)-3-ethyl-4-methylpiperazin-1-yl]methanone —— C20H28N4O2
[5-[[benzyl(methyl)amino]methyl]-1,2-oxazol-3-yl]-[(3S)-3-ethyl-4-methylpiperazin-1-yl]methanone
—— (5R)-2-methyl-7-[(1-propylimidazol-2-yl)methyl]-2,7-diazaspiro[4.5]decane —— C16H28N4
(5R)-2-methyl-7-[(1-propylimidazol-2-yl)methyl]-2,7-diazaspiro[4.5]decane
—— 5-[(3S)-3-(1H-pyrazol-5-yl)piperidine-1-carbonyl]-1H-pyrazin-2-one —— C13H15N5O2
5-[(3S)-3-(1H-pyrazol-5-yl)piperidine-1-carbonyl]-1H-pyrazin-2-one
—— 5-(4-fluorophenyl)-2-methyl-N-pentyl-1-phenylpyrrole-3-carboxamide —— C23H25FN2O
5-(4-fluorophenyl)-2-methyl-N-pentyl-1-phenylpyrrole-3-carboxamide
—— 5-[[(2S)-2-ethylhexanoyl]amino]-N-(2-methoxyethyl)-2-pyrrolidin-1-ylbenzamide —— C22H35N3O3
5-[[(2S)-2-ethylhexanoyl]amino]-N-(2-methoxyethyl)-2-pyrrolidin-1-ylbenzamide
—— 5-(4-chlorophenyl)-N-hexyl-1-(3-methoxyphenyl)-2-methylpyrrole-3-carboxamide —— C25H29ClN2O2
5-(4-chlorophenyl)-N-hexyl-1-(3-methoxyphenyl)-2-methylpyrrole-3-carboxamide
—— [5-(4-Chlorophenyl)-2-methyl-1-phenylpyrrol-3-yl]-pyrrolidin-1-ylmethanone —— C22H21ClN2O
[5-(4-Chlorophenyl)-2-methyl-1-phenylpyrrol-3-yl]-pyrrolidin-1-ylmethanone
—— 5-[[2-[[(2-methoxyacetyl)-propylamino]methyl]pyrrol-1-yl]methyl]-N-propan-2-ylfuran-2-carboxamide —— C20H29N3O4
5-[[2-[[(2-methoxyacetyl)-propylamino]methyl]pyrrol-1-yl]methyl]-N-propan-2-ylfuran-2-carboxamide