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—— 5-[(3-Bromophenyl)methylsulfanyl]-1-(2,4-dimethylphenyl)tetrazole —— C16H15BrN4S
5-[(3-Bromophenyl)methylsulfanyl]-1-(2,4-dimethylphenyl)tetrazole
—— 5-cyclopropyl-N-[5-[(2R)-pentan-2-yl]-1,3,4-thiadiazol-2-yl]-1H-pyrazole-4-carboxamide —— C14H19N5OS
5-cyclopropyl-N-[5-[(2R)-pentan-2-yl]-1,3,4-thiadiazol-2-yl]-1H-pyrazole-4-carboxamide
—— (5R)-5-(2,2-dimethylmorpholin-4-yl)-1-propyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C17H27N3O3
(5R)-5-(2,2-dimethylmorpholin-4-yl)-1-propyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— 5-[2-(4-Chlorophenyl)sulfanylethylsulfanyl]-1-(2,4-dimethylphenyl)tetrazole —— C17H17ClN4S2
5-[2-(4-Chlorophenyl)sulfanylethylsulfanyl]-1-(2,4-dimethylphenyl)tetrazole
—— (5S)-5-(3,4-dihydro-2H-chromen-6-ylmethylamino)-1-ethyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C20H25N3O3
(5S)-5-(3,4-dihydro-2H-chromen-6-ylmethylamino)-1-ethyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— 5-[2-(2,5-Dichlorophenyl)sulfanylethylsulfanyl]-1-(2,4-dimethylphenyl)tetrazole —— C17H16Cl2N4S2
5-[2-(2,5-Dichlorophenyl)sulfanylethylsulfanyl]-1-(2,4-dimethylphenyl)tetrazole
—— (5R)-2-(azepan-1-ylsulfonyl)-2,9-diazaspiro[4.5]decane —— C14H27N3O2S
(5R)-2-(azepan-1-ylsulfonyl)-2,9-diazaspiro[4.5]decane
—— 5,6,7-trimethoxy-3-[[(2R)-2-methyl-3-oxopiperazin-1-yl]methyl]-1H-quinolin-2-one —— C18H23N3O5
5,6,7-trimethoxy-3-[[(2R)-2-methyl-3-oxopiperazin-1-yl]methyl]-1H-quinolin-2-one
—— (5S)-5-(2,2-dimethylmorpholin-4-yl)-1-propyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C17H27N3O3
(5S)-5-(2,2-dimethylmorpholin-4-yl)-1-propyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— 5,6,7-trimethoxy-3-[[(2S)-2-methyl-3-oxopiperazin-1-yl]methyl]-1H-quinolin-2-one —— C18H23N3O5
5,6,7-trimethoxy-3-[[(2S)-2-methyl-3-oxopiperazin-1-yl]methyl]-1H-quinolin-2-one
—— 5-[(2S)-2-(aminomethyl)-5-methyl-2,3-dihydro-1-benzofuran-7-yl]-2-benzyl-N,N-dimethyl-1,2,4-triazol-3-amine —— C21H25N5O
5-[(2S)-2-(aminomethyl)-5-methyl-2,3-dihydro-1-benzofuran-7-yl]-2-benzyl-N,N-dimethyl-1,2,4-triazol-3-amine
—— 5-methyl-N-[[(3S)-1-(2-methylpropyl)pyrrolidin-3-yl]methyl]-1H-imidazole-4-carboxamide —— C14H24N4O
5-methyl-N-[[(3S)-1-(2-methylpropyl)pyrrolidin-3-yl]methyl]-1H-imidazole-4-carboxamide
—— [5-(imidazol-1-ylmethyl)furan-2-yl]-[(3R)-3-(1H-pyrazol-5-yl)piperidin-1-yl]methanone —— C17H19N5O2
[5-(imidazol-1-ylmethyl)furan-2-yl]-[(3R)-3-(1H-pyrazol-5-yl)piperidin-1-yl]methanone
—— (5-amino-4-cyano-2-ethoxycarbonylthiophen-3-yl)methyl 5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophene-2-carboxylate —— C19H20N2O4S2
(5-amino-4-cyano-2-ethoxycarbonylthiophen-3-yl)methyl 5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophene-2-carboxylate
—— (5R)-5-[3-(3-methylphenoxy)azetidin-1-yl]-1-propyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C21H27N3O3
(5R)-5-[3-(3-methylphenoxy)azetidin-1-yl]-1-propyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— 5-[(3S)-1-[(2-chloro-4-fluorophenyl)methyl]piperidin-3-yl]-4-ethyl-2-methyl-1,2,4-triazol-3-one —— C17H22ClFN4O
5-[(3S)-1-[(2-chloro-4-fluorophenyl)methyl]piperidin-3-yl]-4-ethyl-2-methyl-1,2,4-triazol-3-one
—— 5-[[benzyl(methyl)amino]methyl]-N-[(2S)-2-hydroxypropyl]-1,2-oxazole-3-carboxamide —— C16H21N3O3
5-[[benzyl(methyl)amino]methyl]-N-[(2S)-2-hydroxypropyl]-1,2-oxazole-3-carboxamide
—— 5-[(3-fluorophenoxy)methyl]-N-[(2R)-1-(methylamino)-1-oxopropan-2-yl]-1H-pyrazole-3-carboxamide —— C15H17FN4O3
5-[(3-fluorophenoxy)methyl]-N-[(2R)-1-(methylamino)-1-oxopropan-2-yl]-1H-pyrazole-3-carboxamide
—— 5-[(2,6-difluorophenoxy)methyl]-N-[(2R)-1-hydroxypropan-2-yl]-1,2-oxazole-3-carboxamide —— C14H14F2N2O4
5-[(2,6-difluorophenoxy)methyl]-N-[(2R)-1-hydroxypropan-2-yl]-1,2-oxazole-3-carboxamide
—— 5-[1-[[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]imidazol-2-yl]-2-pyrrolidin-1-ylpyrimidine —— C20H21N5O2
5-[1-[[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]imidazol-2-yl]-2-pyrrolidin-1-ylpyrimidine
—— (5S)-5-(2-methyl-4-oxo-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-7-yl)-1-propyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C20H27N5O3
(5S)-5-(2-methyl-4-oxo-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-7-yl)-1-propyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— 5-[(2,6-difluorophenoxy)methyl]-N-[(2S)-1-hydroxypropan-2-yl]-1,2-oxazole-3-carboxamide —— C14H14F2N2O4
5-[(2,6-difluorophenoxy)methyl]-N-[(2S)-1-hydroxypropan-2-yl]-1,2-oxazole-3-carboxamide
—— 5-[[(3S)-3-(2-chlorophenyl)pyrrolidin-1-yl]methyl]-2-methoxybenzoic acid —— C19H20ClNO3
5-[[(3S)-3-(2-chlorophenyl)pyrrolidin-1-yl]methyl]-2-methoxybenzoic acid
—— 5-[(3R)-1-[(2-chloro-4-fluorophenyl)methyl]piperidin-3-yl]-4-ethyl-2-methyl-1,2,4-triazol-3-one —— C17H22ClFN4O
5-[(3R)-1-[(2-chloro-4-fluorophenyl)methyl]piperidin-3-yl]-4-ethyl-2-methyl-1,2,4-triazol-3-one
—— 5-[1-[[(3S)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]imidazol-2-yl]-2-pyrrolidin-1-ylpyrimidine —— C20H21N5O2
5-[1-[[(3S)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]imidazol-2-yl]-2-pyrrolidin-1-ylpyrimidine
—— [5-[(2-fluorophenoxy)methyl]-1H-pyrazol-3-yl]-[(2S)-2-(2-methylphenyl)pyrrolidin-1-yl]methanone —— C22H22FN3O2
[5-[(2-fluorophenoxy)methyl]-1H-pyrazol-3-yl]-[(2S)-2-(2-methylphenyl)pyrrolidin-1-yl]methanone
—— [5-(imidazol-1-ylmethyl)furan-2-yl]-[(3S)-3-(1H-pyrazol-5-yl)piperidin-1-yl]methanone —— C17H19N5O2
[5-(imidazol-1-ylmethyl)furan-2-yl]-[(3S)-3-(1H-pyrazol-5-yl)piperidin-1-yl]methanone
—— 5-[[benzyl(methyl)amino]methyl]-N-[(2R)-2-hydroxypropyl]-1,2-oxazole-3-carboxamide —— C16H21N3O3
5-[[benzyl(methyl)amino]methyl]-N-[(2R)-2-hydroxypropyl]-1,2-oxazole-3-carboxamide
—— 5-[(2R)-2-(aminomethyl)-5-methyl-2,3-dihydro-1-benzofuran-7-yl]-2-benzyl-N,N-dimethyl-1,2,4-triazol-3-amine —— C21H25N5O
5-[(2R)-2-(aminomethyl)-5-methyl-2,3-dihydro-1-benzofuran-7-yl]-2-benzyl-N,N-dimethyl-1,2,4-triazol-3-amine
—— (5S)-5-[3-(3-methylphenoxy)azetidin-1-yl]-1-propyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C21H27N3O3
(5S)-5-[3-(3-methylphenoxy)azetidin-1-yl]-1-propyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— 5-[(3-fluorophenoxy)methyl]-N-[(2S)-1-(methylamino)-1-oxopropan-2-yl]-1H-pyrazole-3-carboxamide —— C15H17FN4O3
5-[(3-fluorophenoxy)methyl]-N-[(2S)-1-(methylamino)-1-oxopropan-2-yl]-1H-pyrazole-3-carboxamide
—— (5R)-N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-3-propan-2-yl-4,5-dihydro-1,2-oxazole-5-carboxamide —— C14H21N3O2S
(5R)-N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-3-propan-2-yl-4,5-dihydro-1,2-oxazole-5-carboxamide
—— 5-(benzimidazol-1-ylmethyl)-N-[(1R)-1-(3-methylpyridin-2-yl)propyl]-1H-pyrazole-3-carboxamide —— C21H22N6O
5-(benzimidazol-1-ylmethyl)-N-[(1R)-1-(3-methylpyridin-2-yl)propyl]-1H-pyrazole-3-carboxamide
—— 5-methyl-N-[[(3R)-1-(2-methylpropyl)pyrrolidin-3-yl]methyl]-1H-imidazole-4-carboxamide —— C14H24N4O
5-methyl-N-[[(3R)-1-(2-methylpropyl)pyrrolidin-3-yl]methyl]-1H-imidazole-4-carboxamide
—— 5-(benzimidazol-1-ylmethyl)-N-[(1S)-1-(3-methylpyridin-2-yl)propyl]-1H-pyrazole-3-carboxamide —— C21H22N6O
5-(benzimidazol-1-ylmethyl)-N-[(1S)-1-(3-methylpyridin-2-yl)propyl]-1H-pyrazole-3-carboxamide
—— (5S)-7-methyl-2-[2-[(6-methyl-1H-benzimidazol-2-yl)methoxy]acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C20H26N4O3
(5S)-7-methyl-2-[2-[(6-methyl-1H-benzimidazol-2-yl)methoxy]acetyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-5-(3,4-dihydro-2H-chromen-6-ylmethylamino)-1-ethyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C20H25N3O3
(5R)-5-(3,4-dihydro-2H-chromen-6-ylmethylamino)-1-ethyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— (5R)-7-methyl-2-[2-[(6-methyl-1H-benzimidazol-2-yl)methoxy]acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C20H26N4O3
(5R)-7-methyl-2-[2-[(6-methyl-1H-benzimidazol-2-yl)methoxy]acetyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-5-(2-methyl-4-oxo-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-7-yl)-1-propyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C20H27N5O3
(5R)-5-(2-methyl-4-oxo-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-7-yl)-1-propyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— 5,6-Bis(4-methylphenyl)-3-[(2-methylphenyl)methylsulfanyl]-1,2,4-triazine —— C25H23N3S
5,6-Bis(4-methylphenyl)-3-[(2-methylphenyl)methylsulfanyl]-1,2,4-triazine
—— 5,7-dimethyl-3-[(4S)-4,5,6,7-tetrahydro-1H-imidazo[4,5-c]pyridin-4-yl]pyrazolo[1,5-a]pyrimidine —— C14H16N6
5,7-dimethyl-3-[(4S)-4,5,6,7-tetrahydro-1H-imidazo[4,5-c]pyridin-4-yl]pyrazolo[1,5-a]pyrimidine
—— [(5-Chloropyridin-2-yl)carbamoyl]methyl 3,6-dichloropyridine-2-carboxylate —— C13H8Cl3N3O3
[(5-Chloropyridin-2-yl)carbamoyl]methyl 3,6-dichloropyridine-2-carboxylate
—— 5,7-dimethyl-3-[(4R)-4,5,6,7-tetrahydro-1H-imidazo[4,5-c]pyridin-4-yl]pyrazolo[1,5-a]pyrimidine —— C14H16N6
5,7-dimethyl-3-[(4R)-4,5,6,7-tetrahydro-1H-imidazo[4,5-c]pyridin-4-yl]pyrazolo[1,5-a]pyrimidine
—— (5-Phenyl-1,3,4-oxadiazol-2-yl)methyl 3,4,5-trichloropyridine-2-carboxylate —— C15H8Cl3N3O3
(5-Phenyl-1,3,4-oxadiazol-2-yl)methyl 3,4,5-trichloropyridine-2-carboxylate
—— [(5S)-2,9-diazaspiro[4.5]decan-2-yl]-(2,4-difluoro-3-methoxyphenyl)methanone —— C16H20F2N2O2
[(5S)-2,9-diazaspiro[4.5]decan-2-yl]-(2,4-difluoro-3-methoxyphenyl)methanone
—— (5S)-1-(cyclopropylmethyl)-5-[[1-(hydroxymethyl)cyclopentyl]methylamino]azepan-2-one —— C17H30N2O2
(5S)-1-(cyclopropylmethyl)-5-[[1-(hydroxymethyl)cyclopentyl]methylamino]azepan-2-one
—— 5-[(2,6-difluorophenoxy)methyl]-N-[[(2S)-oxan-2-yl]methyl]-1,2-oxazole-3-carboxamide —— C17H18F2N2O4
5-[(2,6-difluorophenoxy)methyl]-N-[[(2S)-oxan-2-yl]methyl]-1,2-oxazole-3-carboxamide
—— 5-methoxy-1-methyl-N-[[(3R)-1-methylpyrrolidin-3-yl]methyl]indole-2-carboxamide —— C17H23N3O2
5-methoxy-1-methyl-N-[[(3R)-1-methylpyrrolidin-3-yl]methyl]indole-2-carboxamide
—— 5-[(3R)-3-[[[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methylamino]methyl]pyrrolidin-1-yl]-2-methylpyridazin-3-one —— C20H23FN6O
5-[(3R)-3-[[[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methylamino]methyl]pyrrolidin-1-yl]-2-methylpyridazin-3-one
—— 5-[2-(3-chloro-1H-1,2,4-triazol-5-yl)ethyl]-3-[(3R)-3-(4-fluorophenyl)oxolan-3-yl]-1,2,4-oxadiazole —— C16H15ClFN5O2
5-[2-(3-chloro-1H-1,2,4-triazol-5-yl)ethyl]-3-[(3R)-3-(4-fluorophenyl)oxolan-3-yl]-1,2,4-oxadiazole