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中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-[[(3R)-1-methylpiperidin-3-yl]methylsulfanyl]-N-[[(2S)-oxolan-2-yl]methyl]-1,3,4-thiadiazol-2-amine —— C14H24N4OS2
5-[[(3R)-1-methylpiperidin-3-yl]methylsulfanyl]-N-[[(2S)-oxolan-2-yl]methyl]-1,3,4-thiadiazol-2-amine
—— [(5R)-3-(3-fluorophenyl)-4,5-dihydro-1,2-oxazol-5-yl]methanamine —— C10H11FN2O
[(5R)-3-(3-fluorophenyl)-4,5-dihydro-1,2-oxazol-5-yl]methanamine
—— [(5R)-3-(4-chlorophenyl)-4,5-dihydro-1,2-oxazol-5-yl]methanamine —— C10H11ClN2O
[(5R)-3-(4-chlorophenyl)-4,5-dihydro-1,2-oxazol-5-yl]methanamine
—— [(5R)-3-(4-fluorophenyl)-4,5-dihydro-1,2-oxazol-5-yl]methanamine —— C10H11FN2O
[(5R)-3-(4-fluorophenyl)-4,5-dihydro-1,2-oxazol-5-yl]methanamine
—— [(5S)-3-(3-methoxyphenyl)-4,5-dihydro-1,2-oxazol-5-yl]methanamine —— C11H14N2O2
[(5S)-3-(3-methoxyphenyl)-4,5-dihydro-1,2-oxazol-5-yl]methanamine
—— [(5S)-3-(3-fluorophenyl)-4,5-dihydro-1,2-oxazol-5-yl]methanamine —— C10H11FN2O
[(5S)-3-(3-fluorophenyl)-4,5-dihydro-1,2-oxazol-5-yl]methanamine
—— [5-(2-fluorophenyl)-1,2-oxazol-3-yl]-[(3R)-3-imidazol-1-ylpiperidin-1-yl]methanone —— C18H17FN4O2
[5-(2-fluorophenyl)-1,2-oxazol-3-yl]-[(3R)-3-imidazol-1-ylpiperidin-1-yl]methanone
—— [(5S)-3-(4-fluorophenyl)-4,5-dihydro-1,2-oxazol-5-yl]methanamine —— C10H11FN2O
[(5S)-3-(4-fluorophenyl)-4,5-dihydro-1,2-oxazol-5-yl]methanamine
—— (5R)-1-[(4-fluorophenyl)methyl]-5-(3-imidazol-1-ylpropyliminomethyl)-2-sulfanylidene-1,3-diazinane-4,6-dione —— C18H18FN5O2S
(5R)-1-[(4-fluorophenyl)methyl]-5-(3-imidazol-1-ylpropyliminomethyl)-2-sulfanylidene-1,3-diazinane-4,6-dione
—— [(5R)-3-(2-chlorophenyl)-4,5-dihydro-1,2-oxazol-5-yl]methanamine —— C10H11ClN2O
[(5R)-3-(2-chlorophenyl)-4,5-dihydro-1,2-oxazol-5-yl]methanamine
—— 5-[[(3S)-1-methylpiperidin-3-yl]methylsulfanyl]-N-[[(2S)-oxolan-2-yl]methyl]-1,3,4-thiadiazol-2-amine —— C14H24N4OS2
5-[[(3S)-1-methylpiperidin-3-yl]methylsulfanyl]-N-[[(2S)-oxolan-2-yl]methyl]-1,3,4-thiadiazol-2-amine
—— 5-[[methyl-[(1R)-1-thiophen-2-ylethyl]amino]methyl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C14H16N4OS
5-[[methyl-[(1R)-1-thiophen-2-ylethyl]amino]methyl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-tert-butyl-2-[[(3R)-3-ethyl-4-(2-methoxyethyl)piperazin-1-yl]methyl]-1,3-oxazole —— C17H31N3O2
5-tert-butyl-2-[[(3R)-3-ethyl-4-(2-methoxyethyl)piperazin-1-yl]methyl]-1,3-oxazole
—— 5-tert-butyl-2-[[(3S)-3-ethyl-4-(2-methoxyethyl)piperazin-1-yl]methyl]-1,3-oxazole —— C17H31N3O2
5-tert-butyl-2-[[(3S)-3-ethyl-4-(2-methoxyethyl)piperazin-1-yl]methyl]-1,3-oxazole
—— (5S,10bS)-2-(3,4-dimethoxyphenyl)-5-(2-methylpropyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C22H26N2O3
(5S,10bS)-2-(3,4-dimethoxyphenyl)-5-(2-methylpropyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— 5-[[(3R)-oxolan-3-yl]methylsulfonyl]-3-(trifluoromethyl)-1,4,6,7-tetrahydropyrazolo[4,3-c]pyridine —— C12H16F3N3O3S
5-[[(3R)-oxolan-3-yl]methylsulfonyl]-3-(trifluoromethyl)-1,4,6,7-tetrahydropyrazolo[4,3-c]pyridine
—— 5-[(3R)-3-(3,5-dimethylpyrazol-1-yl)piperidine-1-carbonyl]-1,3-dihydrobenzimidazol-2-one —— C18H21N5O2
5-[(3R)-3-(3,5-dimethylpyrazol-1-yl)piperidine-1-carbonyl]-1,3-dihydrobenzimidazol-2-one
—— (5R,10bS)-2-(3,4-dimethoxyphenyl)-5-(2-methylpropyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C22H26N2O3
(5R,10bS)-2-(3,4-dimethoxyphenyl)-5-(2-methylpropyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— 5-methyl-1-(2-methyl-3,4-dihydro-1H-isoquinolin-5-yl)-N-[[(2S)-oxolan-2-yl]methyl]triazole-4-carboxamide —— C19H25N5O2
5-methyl-1-(2-methyl-3,4-dihydro-1H-isoquinolin-5-yl)-N-[[(2S)-oxolan-2-yl]methyl]triazole-4-carboxamide
—— 5-methyl-1-(2-methyl-3,4-dihydro-1H-isoquinolin-5-yl)-N-[[(2R)-oxolan-2-yl]methyl]triazole-4-carboxamide —— C19H25N5O2
5-methyl-1-(2-methyl-3,4-dihydro-1H-isoquinolin-5-yl)-N-[[(2R)-oxolan-2-yl]methyl]triazole-4-carboxamide
—— (5S,10bS)-2-(3-bromophenyl)-5-(2-methylsulfanylethyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C19H19BrN2OS
(5S,10bS)-2-(3-bromophenyl)-5-(2-methylsulfanylethyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— 5-[(3S)-3-(3,5-dimethylpyrazol-1-yl)piperidine-1-carbonyl]-1,3-dihydrobenzimidazol-2-one —— C18H21N5O2
5-[(3S)-3-(3,5-dimethylpyrazol-1-yl)piperidine-1-carbonyl]-1,3-dihydrobenzimidazol-2-one
—— (5S,10bS)-5-(3-methoxyphenyl)-2-(4-methylphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C24H22N2O2
(5S,10bS)-5-(3-methoxyphenyl)-2-(4-methylphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5S,10bR)-5-(3-methoxyphenyl)-2-(4-methylphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C24H22N2O2
(5S,10bR)-5-(3-methoxyphenyl)-2-(4-methylphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5S,10bS)-2-(1,3-benzodioxol-5-yl)-5-(3-nitrophenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C23H17N3O5
(5S,10bS)-2-(1,3-benzodioxol-5-yl)-5-(3-nitrophenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5-methoxy-1H-indol-3-yl)-[(2R)-2-phenylmorpholin-4-yl]methanone —— C20H20N2O3
(5-methoxy-1H-indol-3-yl)-[(2R)-2-phenylmorpholin-4-yl]methanone
—— (5-methoxy-1H-indol-3-yl)-[(2S)-2-phenylmorpholin-4-yl]methanone —— C20H20N2O3
(5-methoxy-1H-indol-3-yl)-[(2S)-2-phenylmorpholin-4-yl]methanone
—— 5-methyl-N-[(2S)-3-methylbutan-2-yl]-1-[2-(pyridin-3-ylmethyl)-3,4-dihydro-1H-isoquinolin-5-yl]triazole-4-carboxamide —— C24H30N6O
5-methyl-N-[(2S)-3-methylbutan-2-yl]-1-[2-(pyridin-3-ylmethyl)-3,4-dihydro-1H-isoquinolin-5-yl]triazole-4-carboxamide
—— (5S)-4-[hydroxy-[4-(2-methylpropoxy)phenyl]methylidene]-5-(4-hydroxyphenyl)-1-(2-methoxyethyl)pyrrolidine-2,3-dione —— C24H27NO6
(5S)-4-[hydroxy-[4-(2-methylpropoxy)phenyl]methylidene]-5-(4-hydroxyphenyl)-1-(2-methoxyethyl)pyrrolidine-2,3-dione
—— 5-fluoro-2-[[[1-[(2R)-2-hydroxypropyl]piperidin-4-yl]methyl-methylamino]methyl]benzonitrile —— C18H26FN3O
5-fluoro-2-[[[1-[(2R)-2-hydroxypropyl]piperidin-4-yl]methyl-methylamino]methyl]benzonitrile
—— 5-Methyl-3-[2-oxo-2-(5,6,7,8-tetrahydronaphthalen-2-yl)ethyl]-6-phenylthieno[2,3-d]pyrimidin-4-one —— C25H22N2O2S
5-Methyl-3-[2-oxo-2-(5,6,7,8-tetrahydronaphthalen-2-yl)ethyl]-6-phenylthieno[2,3-d]pyrimidin-4-one
—— (5R)-4-[hydroxy-[4-(2-methylpropoxy)phenyl]methylidene]-5-(4-hydroxyphenyl)-1-(2-methoxyethyl)pyrrolidine-2,3-dione —— C24H27NO6
(5R)-4-[hydroxy-[4-(2-methylpropoxy)phenyl]methylidene]-5-(4-hydroxyphenyl)-1-(2-methoxyethyl)pyrrolidine-2,3-dione
—— 5-methyl-N-[(2R)-3-methylbutan-2-yl]-1-[2-(pyridin-3-ylmethyl)-3,4-dihydro-1H-isoquinolin-5-yl]triazole-4-carboxamide —— C24H30N6O
5-methyl-N-[(2R)-3-methylbutan-2-yl]-1-[2-(pyridin-3-ylmethyl)-3,4-dihydro-1H-isoquinolin-5-yl]triazole-4-carboxamide
—— 5-Methyl-3-[2-oxo-2-(1,2,5-trimethylpyrrol-3-yl)ethyl]-6-phenylthieno[2,3-d]pyrimidin-4-one —— C22H21N3O2S
5-Methyl-3-[2-oxo-2-(1,2,5-trimethylpyrrol-3-yl)ethyl]-6-phenylthieno[2,3-d]pyrimidin-4-one
—— 5-Methyl-3-[2-oxo-2-(2,4,5-trimethylphenyl)ethyl]-6-phenylthieno[2,3-d]pyrimidin-4-one —— C24H22N2O2S
5-Methyl-3-[2-oxo-2-(2,4,5-trimethylphenyl)ethyl]-6-phenylthieno[2,3-d]pyrimidin-4-one
—— 5-fluoro-N-[2-[2-(3-fluorophenyl)-1,3-thiazol-4-yl]ethyl]-2-methoxybenzenesulfonamide —— C18H16F2N2O3S2
5-fluoro-N-[2-[2-(3-fluorophenyl)-1,3-thiazol-4-yl]ethyl]-2-methoxybenzenesulfonamide
—— 5-[(2,5-Dimethylphenyl)methyl]-1-phenyl-1H,4H,5H-pyrazolo[3,4-D]pyrimidin-4-one —— C20H18N4O
5-[(2,5-Dimethylphenyl)methyl]-1-phenyl-1H,4H,5H-pyrazolo[3,4-D]pyrimidin-4-one
—— 5-[(1R)-1-[(S)-(3-fluorophenyl)methylsulfinyl]ethyl]-3-thiophen-2-yl-1,2,4-oxadiazole —— C15H13FN2O2S2
5-[(1R)-1-[(S)-(3-fluorophenyl)methylsulfinyl]ethyl]-3-thiophen-2-yl-1,2,4-oxadiazole
—— 5-fluoro-2-[[[1-[(2S)-2-hydroxypropyl]piperidin-4-yl]methyl-methylamino]methyl]benzonitrile —— C18H26FN3O
5-fluoro-2-[[[1-[(2S)-2-hydroxypropyl]piperidin-4-yl]methyl-methylamino]methyl]benzonitrile
—— 5-[(1R)-1-[(R)-(3-fluorophenyl)methylsulfinyl]ethyl]-3-thiophen-2-yl-1,2,4-oxadiazole —— C15H13FN2O2S2
5-[(1R)-1-[(R)-(3-fluorophenyl)methylsulfinyl]ethyl]-3-thiophen-2-yl-1,2,4-oxadiazole
—— 5-[[(R)-cyclohexylmethylsulfinyl]methyl]-3-(2-methylphenyl)-1,2,4-oxadiazole —— C17H22N2O2S
5-[[(R)-cyclohexylmethylsulfinyl]methyl]-3-(2-methylphenyl)-1,2,4-oxadiazole
—— 5-[(1S)-1-[(S)-(3-fluorophenyl)methylsulfinyl]ethyl]-3-thiophen-2-yl-1,2,4-oxadiazole —— C15H13FN2O2S2
5-[(1S)-1-[(S)-(3-fluorophenyl)methylsulfinyl]ethyl]-3-thiophen-2-yl-1,2,4-oxadiazole
—— 5-methyl-N-[(2S)-3-methylbutan-2-yl]-1-(2-propan-2-ylsulfonyl-3,4-dihydro-1H-isoquinolin-5-yl)triazole-4-carboxamide —— C21H31N5O3S
5-methyl-N-[(2S)-3-methylbutan-2-yl]-1-(2-propan-2-ylsulfonyl-3,4-dihydro-1H-isoquinolin-5-yl)triazole-4-carboxamide
—— 5-[[(S)-cyclohexylmethylsulfinyl]methyl]-3-(2-methylphenyl)-1,2,4-oxadiazole —— C17H22N2O2S
5-[[(S)-cyclohexylmethylsulfinyl]methyl]-3-(2-methylphenyl)-1,2,4-oxadiazole
—— 5-[[(2R,3R)-3-pyrazol-1-ylbutan-2-yl]amino]pentanenitrile —— C12H20N4
5-[[(2R,3R)-3-pyrazol-1-ylbutan-2-yl]amino]pentanenitrile
—— 5-[(1S)-1-[(R)-(3-fluorophenyl)methylsulfinyl]ethyl]-3-thiophen-2-yl-1,2,4-oxadiazole —— C15H13FN2O2S2
5-[(1S)-1-[(R)-(3-fluorophenyl)methylsulfinyl]ethyl]-3-thiophen-2-yl-1,2,4-oxadiazole
—— 5-[[(2S,3R)-3-pyrazol-1-ylbutan-2-yl]amino]pentanenitrile —— C12H20N4
5-[[(2S,3R)-3-pyrazol-1-ylbutan-2-yl]amino]pentanenitrile
—— 5-[(Naphthalen-1-YL)methyl]-1-phenyl-1H,4H,5H-pyrazolo[3,4-D]pyrimidin-4-one —— C22H16N4O
5-[(Naphthalen-1-YL)methyl]-1-phenyl-1H,4H,5H-pyrazolo[3,4-D]pyrimidin-4-one
—— (5S)-5-[[(2S)-2-[(4-ethoxybenzoyl)amino]-3-methylbutanoyl]amino]-2-oxo-5,6,7,8-tetrahydro-1H-quinoline-3-carboxamide —— C24H30N4O5
(5S)-5-[[(2S)-2-[(4-ethoxybenzoyl)amino]-3-methylbutanoyl]amino]-2-oxo-5,6,7,8-tetrahydro-1H-quinoline-3-carboxamide
—— (5-chloro-3-methyl-1-benzofuran-2-yl)-[(3R)-3-[(dimethylamino)methyl]pyrrolidin-1-yl]methanone —— C17H21ClN2O2
(5-chloro-3-methyl-1-benzofuran-2-yl)-[(3R)-3-[(dimethylamino)methyl]pyrrolidin-1-yl]methanone