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中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-chloro-N-[(1S)-1-(2,4-dimethyl-1,3-thiazol-5-yl)ethyl]-2-nitro-4-(trifluoromethyl)aniline —— C14H13ClF3N3O2S
5-chloro-N-[(1S)-1-(2,4-dimethyl-1,3-thiazol-5-yl)ethyl]-2-nitro-4-(trifluoromethyl)aniline
—— (5-chloro-2-propan-2-ylpyrimidin-4-yl)-[(2R)-2-(pyrazol-1-ylmethyl)piperidin-1-yl]methanone —— C17H22ClN5O
(5-chloro-2-propan-2-ylpyrimidin-4-yl)-[(2R)-2-(pyrazol-1-ylmethyl)piperidin-1-yl]methanone
—— 5-fluoro-2-[[(1S,2R)-2-methylcyclopropanecarbonyl]amino]-N-[(2R)-1,2,3,4-tetrahydronaphthalen-2-yl]benzamide —— C22H23FN2O2
5-fluoro-2-[[(1S,2R)-2-methylcyclopropanecarbonyl]amino]-N-[(2R)-1,2,3,4-tetrahydronaphthalen-2-yl]benzamide
—— 5-[(3R)-3-(3,5-dimethylpyrazol-1-yl)piperidine-1-carbonyl]-3,4-dimethyl-1H-pyridazin-6-one —— C17H23N5O2
5-[(3R)-3-(3,5-dimethylpyrazol-1-yl)piperidine-1-carbonyl]-3,4-dimethyl-1H-pyridazin-6-one
—— 5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl-[(2R)-2-(pyrazol-1-ylmethyl)piperidin-1-yl]methanone —— C17H21N3OS
5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl-[(2R)-2-(pyrazol-1-ylmethyl)piperidin-1-yl]methanone
—— 5-(4-methoxyphenyl)-2-[[(2S)-2-(1-methylpyrazol-4-yl)pyrrolidin-1-yl]methyl]-1,3-oxazole —— C19H22N4O2
5-(4-methoxyphenyl)-2-[[(2S)-2-(1-methylpyrazol-4-yl)pyrrolidin-1-yl]methyl]-1,3-oxazole
—— 5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl-[(2S)-2-(pyrazol-1-ylmethyl)piperidin-1-yl]methanone —— C17H21N3OS
5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl-[(2S)-2-(pyrazol-1-ylmethyl)piperidin-1-yl]methanone
—— 5-[[(2R)-2-[(2S)-1-benzylpyrrolidin-2-yl]pyrrolidin-1-yl]methyl]-3-butyl-1,2,4-oxadiazole —— C22H32N4O
5-[[(2R)-2-[(2S)-1-benzylpyrrolidin-2-yl]pyrrolidin-1-yl]methyl]-3-butyl-1,2,4-oxadiazole
—— 5-tert-butyl-3-[[(3S)-3-pyrimidin-4-ylpiperidin-1-yl]methyl]-1,2,4-oxadiazole —— C16H23N5O
5-tert-butyl-3-[[(3S)-3-pyrimidin-4-ylpiperidin-1-yl]methyl]-1,2,4-oxadiazole
—— (5-chloro-2-propan-2-ylpyrimidin-4-yl)-[(2S)-2-(pyrazol-1-ylmethyl)piperidin-1-yl]methanone —— C17H22ClN5O
(5-chloro-2-propan-2-ylpyrimidin-4-yl)-[(2S)-2-(pyrazol-1-ylmethyl)piperidin-1-yl]methanone
—— 5-fluoro-2-[[(1R,2S)-2-methylcyclopropanecarbonyl]amino]-N-[(2R)-1,2,3,4-tetrahydronaphthalen-2-yl]benzamide —— C22H23FN2O2
5-fluoro-2-[[(1R,2S)-2-methylcyclopropanecarbonyl]amino]-N-[(2R)-1,2,3,4-tetrahydronaphthalen-2-yl]benzamide
—— 5-[[(2S)-2-[(2S)-1-benzylpyrrolidin-2-yl]pyrrolidin-1-yl]methyl]-3-butyl-1,2,4-oxadiazole —— C22H32N4O
5-[[(2S)-2-[(2S)-1-benzylpyrrolidin-2-yl]pyrrolidin-1-yl]methyl]-3-butyl-1,2,4-oxadiazole
—— [5-(2-methylpropyl)-1H-pyrazol-3-yl]-[(2S)-2-(pyrazol-1-ylmethyl)piperidin-1-yl]methanone —— C17H25N5O
[5-(2-methylpropyl)-1H-pyrazol-3-yl]-[(2S)-2-(pyrazol-1-ylmethyl)piperidin-1-yl]methanone
—— 5-tert-butyl-3-[[(3R)-3-pyrimidin-4-ylpiperidin-1-yl]methyl]-1,2,4-oxadiazole —— C16H23N5O
5-tert-butyl-3-[[(3R)-3-pyrimidin-4-ylpiperidin-1-yl]methyl]-1,2,4-oxadiazole
—— (5-chlorofuran-2-yl)-[(6S)-6-methylspiro[2,3,6,8-tetrahydro-[1,4]dioxino[2,3-g]isoquinoline-9,1'-cyclopentane]-7-yl]methanone —— C21H22ClNO4
(5-chlorofuran-2-yl)-[(6S)-6-methylspiro[2,3,6,8-tetrahydro-[1,4]dioxino[2,3-g]isoquinoline-9,1'-cyclopentane]-7-yl]methanone
—— 5-[(3S)-3-(3,5-dimethylpyrazol-1-yl)piperidine-1-carbonyl]-3,4-dimethyl-1H-pyridazin-6-one —— C17H23N5O2
5-[(3S)-3-(3,5-dimethylpyrazol-1-yl)piperidine-1-carbonyl]-3,4-dimethyl-1H-pyridazin-6-one
—— (5-methyl-1-phenylpyrazol-4-yl)-[(2S)-2-[(4-methylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methanone —— C20H23N5O
(5-methyl-1-phenylpyrazol-4-yl)-[(2S)-2-[(4-methylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methanone
—— (5-chlorofuran-2-yl)-[(6R)-6-methylspiro[2,3,6,8-tetrahydro-[1,4]dioxino[2,3-g]isoquinoline-9,1'-cyclopentane]-7-yl]methanone —— C21H22ClNO4
(5-chlorofuran-2-yl)-[(6R)-6-methylspiro[2,3,6,8-tetrahydro-[1,4]dioxino[2,3-g]isoquinoline-9,1'-cyclopentane]-7-yl]methanone
—— (5-bromofuran-3-yl)-[(2R)-2-[(4-methylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methanone —— C14H16BrN3O2
(5-bromofuran-3-yl)-[(2R)-2-[(4-methylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methanone
—— (5-methyl-1-phenylpyrazol-4-yl)-[(2R)-2-[(4-methylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methanone —— C20H23N5O
(5-methyl-1-phenylpyrazol-4-yl)-[(2R)-2-[(4-methylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methanone
—— 5-bromo-N-[(2R)-1-(1H-indazol-5-ylamino)-1-oxopropan-2-yl]thiophene-2-carboxamide —— C15H13BrN4O2S
5-bromo-N-[(2R)-1-(1H-indazol-5-ylamino)-1-oxopropan-2-yl]thiophene-2-carboxamide
—— 5-bromo-N-[(2S)-1-(1H-indazol-5-ylamino)-1-oxopropan-2-yl]thiophene-2-carboxamide —— C15H13BrN4O2S
5-bromo-N-[(2S)-1-(1H-indazol-5-ylamino)-1-oxopropan-2-yl]thiophene-2-carboxamide
—— 5-methyl-3-[[4-[(2S)-2-methylpiperidin-1-yl]sulfonylpiperazin-1-yl]methyl]-1,2,4-oxadiazole —— C14H25N5O3S
5-methyl-3-[[4-[(2S)-2-methylpiperidin-1-yl]sulfonylpiperazin-1-yl]methyl]-1,2,4-oxadiazole
—— (5S,6S)-5-[(3R)-3-ethoxypiperidine-1-carbonyl]-1-methyl-6-(1-methylpyrazol-4-yl)piperidin-2-one —— C18H28N4O3
(5S,6S)-5-[(3R)-3-ethoxypiperidine-1-carbonyl]-1-methyl-6-(1-methylpyrazol-4-yl)piperidin-2-one
—— 5-methyl-3-[[4-[(2R)-2-methylpiperidin-1-yl]sulfonylpiperazin-1-yl]methyl]-1,2,4-oxadiazole —— C14H25N5O3S
5-methyl-3-[[4-[(2R)-2-methylpiperidin-1-yl]sulfonylpiperazin-1-yl]methyl]-1,2,4-oxadiazole
—— (5R)-N-[(4S)-1-tert-butyl-4,5,6,7-tetrahydroindazol-4-yl]-3-(5-chlorothiophen-2-yl)-4,5-dihydro-1,2-oxazole-5-carboxamide —— C19H23ClN4O2S
(5R)-N-[(4S)-1-tert-butyl-4,5,6,7-tetrahydroindazol-4-yl]-3-(5-chlorothiophen-2-yl)-4,5-dihydro-1,2-oxazole-5-carboxamide
—— 5-phenyl-3-[[(2S)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methyl]-1,2,4-oxadiazole —— C17H19N5O
5-phenyl-3-[[(2S)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methyl]-1,2,4-oxadiazole
—— 5-phenyl-3-[[(2R)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methyl]-1,2,4-oxadiazole —— C17H19N5O
5-phenyl-3-[[(2R)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methyl]-1,2,4-oxadiazole
—— (5R,6S)-5-[(3R)-3-ethoxypiperidine-1-carbonyl]-1-methyl-6-(1-methylpyrazol-4-yl)piperidin-2-one —— C18H28N4O3
(5R,6S)-5-[(3R)-3-ethoxypiperidine-1-carbonyl]-1-methyl-6-(1-methylpyrazol-4-yl)piperidin-2-one
—— (5S)-N-[(4S)-1-tert-butyl-4,5,6,7-tetrahydroindazol-4-yl]-3-(5-chlorothiophen-2-yl)-4,5-dihydro-1,2-oxazole-5-carboxamide —— C19H23ClN4O2S
(5S)-N-[(4S)-1-tert-butyl-4,5,6,7-tetrahydroindazol-4-yl]-3-(5-chlorothiophen-2-yl)-4,5-dihydro-1,2-oxazole-5-carboxamide
—— 5-cyclopropyl-3-[[(2S)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methyl]-1,2,4-oxadiazole —— C14H19N5O
5-cyclopropyl-3-[[(2S)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methyl]-1,2,4-oxadiazole
—— (5-methyl-1,2-oxazol-3-yl)-[(3R)-3-(2-propan-2-ylimidazol-1-yl)piperidin-1-yl]methanone —— C16H22N4O2
(5-methyl-1,2-oxazol-3-yl)-[(3R)-3-(2-propan-2-ylimidazol-1-yl)piperidin-1-yl]methanone
—— (5S,6S)-5-[(3S)-3-ethoxypiperidine-1-carbonyl]-1-methyl-6-(1-methylpyrazol-4-yl)piperidin-2-one —— C18H28N4O3
(5S,6S)-5-[(3S)-3-ethoxypiperidine-1-carbonyl]-1-methyl-6-(1-methylpyrazol-4-yl)piperidin-2-one
—— (5R,6S)-5-[(3S)-3-ethoxypiperidine-1-carbonyl]-1-methyl-6-(1-methylpyrazol-4-yl)piperidin-2-one —— C18H28N4O3
(5R,6S)-5-[(3S)-3-ethoxypiperidine-1-carbonyl]-1-methyl-6-(1-methylpyrazol-4-yl)piperidin-2-one
—— 5-cyclopropyl-3-[[(2R)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methyl]-1,2,4-oxadiazole —— C14H19N5O
5-cyclopropyl-3-[[(2R)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methyl]-1,2,4-oxadiazole
—— [(5R)-5-methyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-[4-(2-thiophen-2-ylethyl)piperazin-1-yl]methanone —— C20H26N2OS2
[(5R)-5-methyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-[4-(2-thiophen-2-ylethyl)piperazin-1-yl]methanone
—— (5-methyl-1,2-oxazol-3-yl)-[(3S)-3-(2-propan-2-ylimidazol-1-yl)piperidin-1-yl]methanone —— C16H22N4O2
(5-methyl-1,2-oxazol-3-yl)-[(3S)-3-(2-propan-2-ylimidazol-1-yl)piperidin-1-yl]methanone
—— (5R)-N-[(4R)-1-tert-butyl-4,5,6,7-tetrahydroindazol-4-yl]-3-(5-chlorothiophen-2-yl)-4,5-dihydro-1,2-oxazole-5-carboxamide —— C19H23ClN4O2S
(5R)-N-[(4R)-1-tert-butyl-4,5,6,7-tetrahydroindazol-4-yl]-3-(5-chlorothiophen-2-yl)-4,5-dihydro-1,2-oxazole-5-carboxamide
—— 5-chloro-2-methoxy-N-{2-oxo-1-azatricyclo[7.3.1.0^{5,13}]trideca-5,7,9(13)-trien-7-yl}benzamide —— C20H19ClN2O3
5-chloro-2-methoxy-N-{2-oxo-1-azatricyclo[7.3.1.0^{5,13}]trideca-5,7,9(13)-trien-7-yl}benzamide
—— 5-bromo-N-(3-oxo-1,2,3,5,6,7-hexahydropyrido[3,2,1-ij]quinolin-9-yl)furan-2-carboxamide —— C17H15BrN2O3
5-bromo-N-(3-oxo-1,2,3,5,6,7-hexahydropyrido[3,2,1-ij]quinolin-9-yl)furan-2-carboxamide
—— 5-[(3S)-3-(2-propan-2-ylimidazol-1-yl)piperidine-1-carbonyl]thiophene-3-carboxamide —— C17H22N4O2S
5-[(3S)-3-(2-propan-2-ylimidazol-1-yl)piperidine-1-carbonyl]thiophene-3-carboxamide
—— 5-[(3R)-3-(2-propan-2-ylimidazol-1-yl)piperidine-1-carbonyl]thiophene-3-carboxamide —— C17H22N4O2S
5-[(3R)-3-(2-propan-2-ylimidazol-1-yl)piperidine-1-carbonyl]thiophene-3-carboxamide
—— 5-fluoro-2-methoxy-N-[(3R)-3-methyl-2-oxo-1-azatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-trien-6-yl]benzenesulfonamide —— C19H19FN2O4S
5-fluoro-2-methoxy-N-[(3R)-3-methyl-2-oxo-1-azatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-trien-6-yl]benzenesulfonamide
—— 5-fluoro-2-methoxy-N-[(3S)-3-methyl-2-oxo-1-azatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-trien-6-yl]benzenesulfonamide —— C19H19FN2O4S
5-fluoro-2-methoxy-N-[(3S)-3-methyl-2-oxo-1-azatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-trien-6-yl]benzenesulfonamide
—— 5-[(4,5-dimethyl-1,3-oxazol-2-yl)methylsulfanyl]-N-[[(2S)-oxolan-2-yl]methyl]-1,3,4-thiadiazol-2-amine —— C13H18N4O2S2
5-[(4,5-dimethyl-1,3-oxazol-2-yl)methylsulfanyl]-N-[[(2S)-oxolan-2-yl]methyl]-1,3,4-thiadiazol-2-amine
—— [(5S)-5-methyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-[4-(2-thiophen-2-ylethyl)piperazin-1-yl]methanone —— C20H26N2OS2
[(5S)-5-methyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-[4-(2-thiophen-2-ylethyl)piperazin-1-yl]methanone
—— 5-bromo-N-[(3S)-3-methyl-2-oxo-1-azatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-trien-6-yl]furan-2-carboxamide —— C17H15BrN2O3
5-bromo-N-[(3S)-3-methyl-2-oxo-1-azatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-trien-6-yl]furan-2-carboxamide
—— 5-[[(2R)-2-[(4-methylpyrazol-1-yl)methyl]piperidin-1-yl]methyl]-3-pyridin-3-yl-1,2,4-oxadiazole —— C18H22N6O
5-[[(2R)-2-[(4-methylpyrazol-1-yl)methyl]piperidin-1-yl]methyl]-3-pyridin-3-yl-1,2,4-oxadiazole
—— 5-[[(2S)-2-[(4-methylpyrazol-1-yl)methyl]piperidin-1-yl]methyl]-3-pyridin-3-yl-1,2,4-oxadiazole —— C18H22N6O
5-[[(2S)-2-[(4-methylpyrazol-1-yl)methyl]piperidin-1-yl]methyl]-3-pyridin-3-yl-1,2,4-oxadiazole
—— 5-chloro-2-methoxy-N-[(3S)-3-methyl-2-oxo-1-azatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-trien-6-yl]benzamide —— C20H19ClN2O3
5-chloro-2-methoxy-N-[(3S)-3-methyl-2-oxo-1-azatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-trien-6-yl]benzamide