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—— 5-[[(2S,3S)-3-pyrazol-1-ylbutan-2-yl]amino]pentanenitrile —— C12H20N4
5-[[(2S,3S)-3-pyrazol-1-ylbutan-2-yl]amino]pentanenitrile
—— 5-[(2R)-2-(pyrazol-1-ylmethyl)piperidine-1-carbonyl]-1,3-dihydrobenzimidazol-2-one —— C17H19N5O2
5-[(2R)-2-(pyrazol-1-ylmethyl)piperidine-1-carbonyl]-1,3-dihydrobenzimidazol-2-one
—— (5R)-5-[[(2S)-2-[(4-ethoxybenzoyl)amino]-3-methylbutanoyl]amino]-2-oxo-5,6,7,8-tetrahydro-1H-quinoline-3-carboxamide —— C24H30N4O5
(5R)-5-[[(2S)-2-[(4-ethoxybenzoyl)amino]-3-methylbutanoyl]amino]-2-oxo-5,6,7,8-tetrahydro-1H-quinoline-3-carboxamide
—— (5R)-5-[[(2R)-2-[(4-ethoxybenzoyl)amino]-3-methylbutanoyl]amino]-2-oxo-5,6,7,8-tetrahydro-1H-quinoline-3-carboxamide —— C24H30N4O5
(5R)-5-[[(2R)-2-[(4-ethoxybenzoyl)amino]-3-methylbutanoyl]amino]-2-oxo-5,6,7,8-tetrahydro-1H-quinoline-3-carboxamide
—— (5-methyl-1-phenylpyrazol-4-yl)-[(2S)-2-(pyrazol-1-ylmethyl)piperidin-1-yl]methanone —— C20H23N5O
(5-methyl-1-phenylpyrazol-4-yl)-[(2S)-2-(pyrazol-1-ylmethyl)piperidin-1-yl]methanone
—— (5-chloro-3-methyl-1-benzofuran-2-yl)-[(3S)-3-[(dimethylamino)methyl]pyrrolidin-1-yl]methanone —— C17H21ClN2O2
(5-chloro-3-methyl-1-benzofuran-2-yl)-[(3S)-3-[(dimethylamino)methyl]pyrrolidin-1-yl]methanone
—— 5-methyl-N-[(2R)-3-methylbutan-2-yl]-1-(2-propan-2-ylsulfonyl-3,4-dihydro-1H-isoquinolin-5-yl)triazole-4-carboxamide —— C21H31N5O3S
5-methyl-N-[(2R)-3-methylbutan-2-yl]-1-(2-propan-2-ylsulfonyl-3,4-dihydro-1H-isoquinolin-5-yl)triazole-4-carboxamide
—— 5-[(4-methylphenyl)methyl]-1-phenyl-1H,4H,5H-pyrazolo[3,4-d]pyrimidin-4-one —— C19H16N4O
5-[(4-methylphenyl)methyl]-1-phenyl-1H,4H,5H-pyrazolo[3,4-d]pyrimidin-4-one
—— 5-ethyl-N-{2-[2-(4-fluorophenyl)-1,3-thiazol-4-yl]ethyl}thiophene-2-sulfonamide —— C17H17FN2O2S3
5-ethyl-N-{2-[2-(4-fluorophenyl)-1,3-thiazol-4-yl]ethyl}thiophene-2-sulfonamide
—— 5-chloro-N-[2-[2-(3-fluorophenyl)-1,3-thiazol-4-yl]ethyl]-2-nitrobenzamide —— C18H13ClFN3O3S
5-chloro-N-[2-[2-(3-fluorophenyl)-1,3-thiazol-4-yl]ethyl]-2-nitrobenzamide
—— 5-chloro-N-{2-[2-(3-fluorophenyl)-1,3-thiazol-4-yl]ethyl}-2-methoxybenzamide —— C19H16ClFN2O2S
5-chloro-N-{2-[2-(3-fluorophenyl)-1,3-thiazol-4-yl]ethyl}-2-methoxybenzamide
—— 5-Methyl-3-(2-oxopropyl)-6-phenylthieno[2,3-d]pyrimidin-4-one —— C16H14N2O2S
5-Methyl-3-(2-oxopropyl)-6-phenylthieno[2,3-d]pyrimidin-4-one
—— 5-bromo-N-[2-[2-(4-chlorophenyl)-1,3-thiazol-4-yl]ethyl]furan-2-carboxamide —— C16H12BrClN2O2S
5-bromo-N-[2-[2-(4-chlorophenyl)-1,3-thiazol-4-yl]ethyl]furan-2-carboxamide
—— 5-chloro-N-[2-[2-(4-chlorophenyl)-1,3-thiazol-4-yl]ethyl]-2-methoxybenzamide —— C19H16Cl2N2O2S
5-chloro-N-[2-[2-(4-chlorophenyl)-1,3-thiazol-4-yl]ethyl]-2-methoxybenzamide
—— (5-methyl-1-phenylpyrazol-4-yl)-[(2R)-2-(pyrazol-1-ylmethyl)piperidin-1-yl]methanone —— C20H23N5O
(5-methyl-1-phenylpyrazol-4-yl)-[(2R)-2-(pyrazol-1-ylmethyl)piperidin-1-yl]methanone
—— 5-[(2S)-2-(pyrazol-1-ylmethyl)piperidine-1-carbonyl]-1,3-dihydrobenzimidazol-2-one —— C17H19N5O2
5-[(2S)-2-(pyrazol-1-ylmethyl)piperidine-1-carbonyl]-1,3-dihydrobenzimidazol-2-one
—— (5S)-5-[[(2R)-2-[(4-ethoxybenzoyl)amino]-3-methylbutanoyl]amino]-2-oxo-5,6,7,8-tetrahydro-1H-quinoline-3-carboxamide —— C24H30N4O5
(5S)-5-[[(2R)-2-[(4-ethoxybenzoyl)amino]-3-methylbutanoyl]amino]-2-oxo-5,6,7,8-tetrahydro-1H-quinoline-3-carboxamide
—— 5-chloro-N-{2-[2-(3-fluorophenyl)-4-methyl-1,3-thiazol-5-yl]ethyl}-2-methoxybenzamide —— C20H18ClFN2O2S
5-chloro-N-{2-[2-(3-fluorophenyl)-4-methyl-1,3-thiazol-5-yl]ethyl}-2-methoxybenzamide
—— 5-fluoro-2-methoxy-N-(1-methylsulfonyl-3,4-dihydro-2H-quinolin-7-yl)benzenesulfonamide —— C17H19FN2O5S2
5-fluoro-2-methoxy-N-(1-methylsulfonyl-3,4-dihydro-2H-quinolin-7-yl)benzenesulfonamide
—— 5-ethyl-N-{2-[2-(3-fluorophenyl)-4-methyl-1,3-thiazol-5-yl]ethyl}thiophene-2-sulfonamide —— C18H19FN2O2S3
5-ethyl-N-{2-[2-(3-fluorophenyl)-4-methyl-1,3-thiazol-5-yl]ethyl}thiophene-2-sulfonamide
—— 5-ethyl-N-(1-methylsulfonyl-3,4-dihydro-2H-quinolin-7-yl)thiophene-2-sulfonamide —— C16H20N2O4S3
5-ethyl-N-(1-methylsulfonyl-3,4-dihydro-2H-quinolin-7-yl)thiophene-2-sulfonamide
—— (5R)-5-(chloromethyl)-3-(2-phenylethyl)-4,5-dihydro-1,2-oxazole —— C12H14ClNO
(5R)-5-(chloromethyl)-3-(2-phenylethyl)-4,5-dihydro-1,2-oxazole
—— (5S)-5-(chloromethyl)-3-(4-fluorophenyl)-4,5-dihydro-1,2-oxazole —— C10H9ClFNO
(5S)-5-(chloromethyl)-3-(4-fluorophenyl)-4,5-dihydro-1,2-oxazole
—— 5-bromo-N-(1-methylsulfonyl-3,4-dihydro-2H-quinolin-7-yl)furan-2-carboxamide —— C15H15BrN2O4S
5-bromo-N-(1-methylsulfonyl-3,4-dihydro-2H-quinolin-7-yl)furan-2-carboxamide
—— [5-(diethylaminomethyl)furan-2-yl]-[(2R)-2-(pyrazol-1-ylmethyl)piperidin-1-yl]methanone —— C19H28N4O2
[5-(diethylaminomethyl)furan-2-yl]-[(2R)-2-(pyrazol-1-ylmethyl)piperidin-1-yl]methanone
—— [5-(diethylaminomethyl)furan-2-yl]-[(2S)-2-(pyrazol-1-ylmethyl)piperidin-1-yl]methanone —— C19H28N4O2
[5-(diethylaminomethyl)furan-2-yl]-[(2S)-2-(pyrazol-1-ylmethyl)piperidin-1-yl]methanone
—— (5S)-5-(chloromethyl)-3-(2-phenylethyl)-4,5-dihydro-1,2-oxazole —— C12H14ClNO
(5S)-5-(chloromethyl)-3-(2-phenylethyl)-4,5-dihydro-1,2-oxazole
—— [5-(5-methylfuran-2-yl)-1H-pyrazol-3-yl]-[(2R)-2-(pyrazol-1-ylmethyl)piperidin-1-yl]methanone —— C18H21N5O2
[5-(5-methylfuran-2-yl)-1H-pyrazol-3-yl]-[(2R)-2-(pyrazol-1-ylmethyl)piperidin-1-yl]methanone
—— 5-ethyl-N-(1-isobutyryl-1,2,3,4-tetrahydroquinolin-7-yl)thiophene-2-sulfonamide —— C19H24N2O3S2
5-ethyl-N-(1-isobutyryl-1,2,3,4-tetrahydroquinolin-7-yl)thiophene-2-sulfonamide
—— (5S)-5-(chloromethyl)-3-(4-chlorophenyl)-4,5-dihydro-1,2-oxazole —— C10H9Cl2NO
(5S)-5-(chloromethyl)-3-(4-chlorophenyl)-4,5-dihydro-1,2-oxazole
—— (5-chlorofuran-2-yl)-[4-[(2R)-2-hydroxybutyl]piperazin-1-yl]methanone —— C13H19ClN2O3
(5-chlorofuran-2-yl)-[4-[(2R)-2-hydroxybutyl]piperazin-1-yl]methanone
—— 5-chloro-2-methoxy-N-(1-(methylsulfonyl)-1,2,3,4-tetrahydroquinolin-7-yl)benzamide —— C18H19ClN2O4S
5-chloro-2-methoxy-N-(1-(methylsulfonyl)-1,2,3,4-tetrahydroquinolin-7-yl)benzamide
—— 5-chloro-N-(1-(methylsulfonyl)-1,2,3,4-tetrahydroquinolin-7-yl)-2-nitrobenzamide —— C17H16ClN3O5S
5-chloro-N-(1-(methylsulfonyl)-1,2,3,4-tetrahydroquinolin-7-yl)-2-nitrobenzamide
—— (5-chlorofuran-2-yl)-[4-[(2S)-2-hydroxybutyl]piperazin-1-yl]methanone —— C13H19ClN2O3
(5-chlorofuran-2-yl)-[4-[(2S)-2-hydroxybutyl]piperazin-1-yl]methanone
—— [5-(furan-2-yl)-1,2-oxazol-3-yl]-[(2S)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone —— C16H16N4O3
[5-(furan-2-yl)-1,2-oxazol-3-yl]-[(2S)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone
—— 5-[(1R)-1-(6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl)ethyl]-3-phenyl-1,2,4-oxadiazole —— C17H17N5O
5-[(1R)-1-(6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl)ethyl]-3-phenyl-1,2,4-oxadiazole
—— 5-[(1S)-1-(6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl)ethyl]-3-phenyl-1,2,4-oxadiazole —— C17H17N5O
5-[(1S)-1-(6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl)ethyl]-3-phenyl-1,2,4-oxadiazole
—— 5-ethyl-N-[1-(furan-2-carbonyl)-3,4-dihydro-2H-quinolin-7-yl]thiophene-2-sulfonamide —— C20H20N2O4S2
5-ethyl-N-[1-(furan-2-carbonyl)-3,4-dihydro-2H-quinolin-7-yl]thiophene-2-sulfonamide
—— 5-bromo-N-[1-(2-methylpropanoyl)-3,4-dihydro-2H-quinolin-7-yl]furan-2-carboxamide —— C18H19BrN2O3
5-bromo-N-[1-(2-methylpropanoyl)-3,4-dihydro-2H-quinolin-7-yl]furan-2-carboxamide
—— (5R)-5-(chloromethyl)-3-(4-chlorophenyl)-4,5-dihydro-1,2-oxazole —— C10H9Cl2NO
(5R)-5-(chloromethyl)-3-(4-chlorophenyl)-4,5-dihydro-1,2-oxazole
—— [5-(furan-2-yl)-1,2-oxazol-3-yl]-[(2R)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone —— C16H16N4O3
[5-(furan-2-yl)-1,2-oxazol-3-yl]-[(2R)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone
—— 5-chloro-N-(1-isobutyryl-1,2,3,4-tetrahydroquinolin-7-yl)-2-nitrobenzamide —— C20H20ClN3O4
5-chloro-N-(1-isobutyryl-1,2,3,4-tetrahydroquinolin-7-yl)-2-nitrobenzamide
—— 5-[(2R)-2-(1-methylpyrazol-4-yl)pyrrolidine-1-carbonyl]thiophene-2-carboxamide —— C14H16N4O2S
5-[(2R)-2-(1-methylpyrazol-4-yl)pyrrolidine-1-carbonyl]thiophene-2-carboxamide
—— 5-phenyl-2-[(1S)-1-[4-(pyridin-2-ylmethyl)piperazin-1-yl]ethyl]-1,3-oxazole —— C21H24N4O
5-phenyl-2-[(1S)-1-[4-(pyridin-2-ylmethyl)piperazin-1-yl]ethyl]-1,3-oxazole
—— 5-[(2S)-2-(1-methylpyrazol-4-yl)pyrrolidine-1-carbonyl]thiophene-2-carboxamide —— C14H16N4O2S
5-[(2S)-2-(1-methylpyrazol-4-yl)pyrrolidine-1-carbonyl]thiophene-2-carboxamide
—— (5-methyl-1,3,4-oxadiazol-2-yl)methyl (2S)-2-[4-(4-fluorophenyl)piperazin-1-yl]propanoate —— C17H21FN4O3
(5-methyl-1,3,4-oxadiazol-2-yl)methyl (2S)-2-[4-(4-fluorophenyl)piperazin-1-yl]propanoate
—— (5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)-[(2S)-2-(pyrazol-1-ylmethyl)piperidin-1-yl]methanone —— C17H21N7O
(5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)-[(2S)-2-(pyrazol-1-ylmethyl)piperidin-1-yl]methanone
—— (5-methyl-1,3,4-oxadiazol-2-yl)methyl (2R)-1-[(3-methylphenyl)methyl]piperidine-2-carboxylate —— C18H23N3O3
(5-methyl-1,3,4-oxadiazol-2-yl)methyl (2R)-1-[(3-methylphenyl)methyl]piperidine-2-carboxylate
—— (5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)-[(2R)-2-(pyrazol-1-ylmethyl)piperidin-1-yl]methanone —— C17H21N7O
(5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)-[(2R)-2-(pyrazol-1-ylmethyl)piperidin-1-yl]methanone
—— 5-chloro-N-(1-isobutyryl-1,2,3,4-tetrahydroquinolin-7-yl)-2-methoxybenzamide —— C21H23ClN2O3
5-chloro-N-(1-isobutyryl-1,2,3,4-tetrahydroquinolin-7-yl)-2-methoxybenzamide