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中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-bromo-N-[(1R)-1-pyridin-2-ylethyl]-1H-indazole-3-carboxamide —— C15H13BrN4O
5-bromo-N-[(1R)-1-pyridin-2-ylethyl]-1H-indazole-3-carboxamide
—— 5-[[(2S)-2-[(3,5-dimethylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methyl]-3-pyridin-2-yl-1,2,4-oxadiazole —— C18H22N6O
5-[[(2S)-2-[(3,5-dimethylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methyl]-3-pyridin-2-yl-1,2,4-oxadiazole
—— 5-[(1S)-1-[(R)-(4-fluorophenyl)methylsulfinyl]ethyl]-3-thiophen-2-yl-1,2,4-oxadiazole —— C15H13FN2O2S2
5-[(1S)-1-[(R)-(4-fluorophenyl)methylsulfinyl]ethyl]-3-thiophen-2-yl-1,2,4-oxadiazole
—— (5-chloro-3-methyl-1-benzofuran-2-yl)-[(2S)-2-[[(2R,6R)-2,6-dimethylmorpholin-4-yl]methyl]pyrrolidin-1-yl]methanone —— C21H27ClN2O3
(5-chloro-3-methyl-1-benzofuran-2-yl)-[(2S)-2-[[(2R,6R)-2,6-dimethylmorpholin-4-yl]methyl]pyrrolidin-1-yl]methanone
—— 5-methyl-N-[(6R)-2-propan-2-yl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-yl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine —— C15H20N8
5-methyl-N-[(6R)-2-propan-2-yl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-yl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine
—— (5S)-4-amino-3-(2-hydroxyethyl)-5-(4-methoxyphenyl)-8,8-dimethyl-7,9-dihydro-5H-chromeno[2,3-d]pyrimidin-3-ium-6-one —— C22H26N3O4+
(5S)-4-amino-3-(2-hydroxyethyl)-5-(4-methoxyphenyl)-8,8-dimethyl-7,9-dihydro-5H-chromeno[2,3-d]pyrimidin-3-ium-6-one
—— (5-bromothiophen-3-yl)-[(2R)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone —— C13H14BrN3OS
(5-bromothiophen-3-yl)-[(2R)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone
—— 5-[[(2R)-2-[(3,5-dimethylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methyl]-3-methyl-1,2-oxazole —— C15H22N4O
5-[[(2R)-2-[(3,5-dimethylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methyl]-3-methyl-1,2-oxazole
—— 5-[[(2S)-2-[(3,5-dimethylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methyl]-3-pyridin-3-yl-1,2,4-oxadiazole —— C18H22N6O
5-[[(2S)-2-[(3,5-dimethylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methyl]-3-pyridin-3-yl-1,2,4-oxadiazole
—— (5S)-5-[4-[2-[benzyl(methyl)amino]ethyl]piperazine-1-carbonyl]pyrrolidin-2-one —— C19H28N4O2
(5S)-5-[4-[2-[benzyl(methyl)amino]ethyl]piperazine-1-carbonyl]pyrrolidin-2-one
—— 5-[[(2S)-2-[(3,5-dimethylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methyl]-3-methyl-1,2-oxazole —— C15H22N4O
5-[[(2S)-2-[(3,5-dimethylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methyl]-3-methyl-1,2-oxazole
—— 5-[[(2R)-2-[(3,5-dimethylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methyl]-3-pyridin-2-yl-1,2,4-oxadiazole —— C18H22N6O
5-[[(2R)-2-[(3,5-dimethylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methyl]-3-pyridin-2-yl-1,2,4-oxadiazole
—— (5-chloro-3-methyl-1-benzofuran-2-yl)-[(2R)-2-[[(2R,6R)-2,6-dimethylmorpholin-4-yl]methyl]pyrrolidin-1-yl]methanone —— C21H27ClN2O3
(5-chloro-3-methyl-1-benzofuran-2-yl)-[(2R)-2-[[(2R,6R)-2,6-dimethylmorpholin-4-yl]methyl]pyrrolidin-1-yl]methanone
—— (5R)-5-(4-chlorophenyl)-4-[hydroxy-(4-methoxyphenyl)methylidene]-1-(2-methoxyethyl)pyrrolidine-2,3-dione —— C21H20ClNO5
(5R)-5-(4-chlorophenyl)-4-[hydroxy-(4-methoxyphenyl)methylidene]-1-(2-methoxyethyl)pyrrolidine-2,3-dione
—— 5-[(2S,6R)-2,6-dimethylmorpholin-4-yl]-2-[(Z)-(3-methyl-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene)methyl]-1,3-oxazole-4-carbonitrile —— C15H16N4O3S2
5-[(2S,6R)-2,6-dimethylmorpholin-4-yl]-2-[(Z)-(3-methyl-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene)methyl]-1,3-oxazole-4-carbonitrile
—— (5S)-N-[3-(cyclohexylamino)-3-oxopropyl]-3-(3-fluorophenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide —— C19H24FN3O3
(5S)-N-[3-(cyclohexylamino)-3-oxopropyl]-3-(3-fluorophenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
—— 5-(2-fluorophenyl)-N-[(3R)-1-methylsulfonylpiperidin-3-yl]furan-2-carboxamide —— C17H19FN2O4S
5-(2-fluorophenyl)-N-[(3R)-1-methylsulfonylpiperidin-3-yl]furan-2-carboxamide
—— (5S,10bS)-5-(2-methylpropyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C18H20N2OS
(5S,10bS)-5-(2-methylpropyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— 5-bromo-N-[(1S)-1-pyridin-2-ylethyl]-1H-indazole-3-carboxamide —— C15H13BrN4O
5-bromo-N-[(1S)-1-pyridin-2-ylethyl]-1H-indazole-3-carboxamide
—— (5S)-3-(5-chlorothiophen-2-yl)-N-[2-[(3S,5S)-3,5-dimethylpiperidin-1-yl]ethyl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C17H24ClN3O2S
(5S)-3-(5-chlorothiophen-2-yl)-N-[2-[(3S,5S)-3,5-dimethylpiperidin-1-yl]ethyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— 5-[(1R)-1-[(R)-(4-fluorophenyl)methylsulfinyl]ethyl]-3-thiophen-2-yl-1,2,4-oxadiazole —— C15H13FN2O2S2
5-[(1R)-1-[(R)-(4-fluorophenyl)methylsulfinyl]ethyl]-3-thiophen-2-yl-1,2,4-oxadiazole
—— 5-[[(2R)-2-[(3,5-dimethylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methyl]-3-(2-methoxyethyl)-1,2,4-oxadiazole —— C16H25N5O2
5-[[(2R)-2-[(3,5-dimethylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methyl]-3-(2-methoxyethyl)-1,2,4-oxadiazole
—— (5R)-5-(furan-2-yl)-4-[hydroxy(pyridin-4-yl)methylidene]-1-(3-morpholin-4-ylpropyl)pyrrolidine-2,3-dione —— C21H23N3O5
(5R)-5-(furan-2-yl)-4-[hydroxy(pyridin-4-yl)methylidene]-1-(3-morpholin-4-ylpropyl)pyrrolidine-2,3-dione
—— (5R)-5-(furan-2-yl)-4-[hydroxy(pyridin-4-yl)methylidene]-1-(3-morpholin-4-ium-4-ylpropyl)pyrrolidine-2,3-dione —— C21H24N3O5+
(5R)-5-(furan-2-yl)-4-[hydroxy(pyridin-4-yl)methylidene]-1-(3-morpholin-4-ium-4-ylpropyl)pyrrolidine-2,3-dione
—— 5-[[(2S)-2-[(3,5-dimethylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methyl]-3-(2-methoxyethyl)-1,2,4-oxadiazole —— C16H25N5O2
5-[[(2S)-2-[(3,5-dimethylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methyl]-3-(2-methoxyethyl)-1,2,4-oxadiazole
—— 5-[[(2R)-2-[(3,5-dimethylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methyl]-3-(furan-3-yl)-1,2,4-oxadiazole —— C17H21N5O2
5-[[(2R)-2-[(3,5-dimethylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methyl]-3-(furan-3-yl)-1,2,4-oxadiazole
—— (5R)-5-[4-[2-[benzyl(methyl)amino]ethyl]piperazine-1-carbonyl]pyrrolidin-2-one —— C19H28N4O2
(5R)-5-[4-[2-[benzyl(methyl)amino]ethyl]piperazine-1-carbonyl]pyrrolidin-2-one
—— (5S,10bR)-2-(3,4-dimethylphenyl)-5-(2-methylsulfanylethyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C21H24N2OS
(5S,10bR)-2-(3,4-dimethylphenyl)-5-(2-methylsulfanylethyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— 5-[[(2S)-2-[(3,5-dimethylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methyl]-3-(furan-3-yl)-1,2,4-oxadiazole —— C17H21N5O2
5-[[(2S)-2-[(3,5-dimethylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methyl]-3-(furan-3-yl)-1,2,4-oxadiazole
—— 5-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-2-[(Z)-(3-methyl-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene)methyl]-1,3-oxazole-4-carbonitrile —— C15H16N4O3S2
5-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-2-[(Z)-(3-methyl-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene)methyl]-1,3-oxazole-4-carbonitrile
—— 5-(4-fluorophenyl)-2-[[(2S)-2-[(4-methylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methyl]-1,3-oxazole —— C19H21FN4O
5-(4-fluorophenyl)-2-[[(2S)-2-[(4-methylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methyl]-1,3-oxazole
—— (5-bromothiophen-3-yl)-[4-[(2S)-2-hydroxybutyl]piperazin-1-yl]methanone —— C13H19BrN2O2S
(5-bromothiophen-3-yl)-[4-[(2S)-2-hydroxybutyl]piperazin-1-yl]methanone
—— 5-(4-fluorophenyl)-2-[[(2R)-2-[(4-methylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methyl]-1,3-oxazole —— C19H21FN4O
5-(4-fluorophenyl)-2-[[(2R)-2-[(4-methylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methyl]-1,3-oxazole
—— (5R)-5-methyl-N-[3-[(5-methylpyridin-2-yl)amino]-3-oxopropyl]-6-oxo-1-phenyl-2,5-dihydro-1,2,4-triazine-3-carboxamide —— C20H22N6O3
(5R)-5-methyl-N-[3-[(5-methylpyridin-2-yl)amino]-3-oxopropyl]-6-oxo-1-phenyl-2,5-dihydro-1,2,4-triazine-3-carboxamide
—— 5-[(1S)-1-[(S)-(2-methoxy-5-methylphenyl)methylsulfinyl]ethyl]-3-propan-2-yl-1,2,4-oxadiazole —— C16H22N2O3S
5-[(1S)-1-[(S)-(2-methoxy-5-methylphenyl)methylsulfinyl]ethyl]-3-propan-2-yl-1,2,4-oxadiazole
—— 5-[(1R)-1-[(S)-(2-methoxy-5-methylphenyl)methylsulfinyl]ethyl]-3-propan-2-yl-1,2,4-oxadiazole —— C16H22N2O3S
5-[(1R)-1-[(S)-(2-methoxy-5-methylphenyl)methylsulfinyl]ethyl]-3-propan-2-yl-1,2,4-oxadiazole
—— (5-methyl-1H-indol-2-yl)-[(2S)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone —— C18H20N4O
(5-methyl-1H-indol-2-yl)-[(2S)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone
—— (5-bromothiophen-3-yl)-[4-[(2R)-2-hydroxybutyl]piperazin-1-yl]methanone —— C13H19BrN2O2S
(5-bromothiophen-3-yl)-[4-[(2R)-2-hydroxybutyl]piperazin-1-yl]methanone
—— (5-methyl-1H-indol-2-yl)-[(2R)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone —— C18H20N4O
(5-methyl-1H-indol-2-yl)-[(2R)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone
—— (5-chloro-2-fluorophenyl)-[(2R)-2-[(4-methylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methanone —— C16H17ClFN3O
(5-chloro-2-fluorophenyl)-[(2R)-2-[(4-methylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methanone
—— 5-[(1R)-1-[(R)-(2-methoxy-5-methylphenyl)methylsulfinyl]ethyl]-3-propan-2-yl-1,2,4-oxadiazole —— C16H22N2O3S
5-[(1R)-1-[(R)-(2-methoxy-5-methylphenyl)methylsulfinyl]ethyl]-3-propan-2-yl-1,2,4-oxadiazole
—— 5-[(1S)-1-[(R)-(2-methoxy-5-methylphenyl)methylsulfinyl]ethyl]-3-propan-2-yl-1,2,4-oxadiazole —— C16H22N2O3S
5-[(1S)-1-[(R)-(2-methoxy-5-methylphenyl)methylsulfinyl]ethyl]-3-propan-2-yl-1,2,4-oxadiazole
—— (5-chloro-2-fluorophenyl)-[(2S)-2-[(4-methylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methanone —— C16H17ClFN3O
(5-chloro-2-fluorophenyl)-[(2S)-2-[(4-methylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methanone
—— (5-methyl-1H-indol-2-yl)-[(2R)-2-(1-methylpyrazol-4-yl)pyrrolidin-1-yl]methanone —— C18H20N4O
(5-methyl-1H-indol-2-yl)-[(2R)-2-(1-methylpyrazol-4-yl)pyrrolidin-1-yl]methanone
—— (5S)-5-methyl-N-[3-[(5-methylpyridin-2-yl)amino]-3-oxopropyl]-6-oxo-1-phenyl-2,5-dihydro-1,2,4-triazine-3-carboxamide —— C20H22N6O3
(5S)-5-methyl-N-[3-[(5-methylpyridin-2-yl)amino]-3-oxopropyl]-6-oxo-1-phenyl-2,5-dihydro-1,2,4-triazine-3-carboxamide
—— (5-methyl-1H-indol-2-yl)-[(2S)-2-(1-methylpyrazol-4-yl)pyrrolidin-1-yl]methanone —— C18H20N4O
(5-methyl-1H-indol-2-yl)-[(2S)-2-(1-methylpyrazol-4-yl)pyrrolidin-1-yl]methanone
—— (5-chloro-1-benzofuran-2-yl)-[(2S)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone —— C17H16ClN3O2
(5-chloro-1-benzofuran-2-yl)-[(2S)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone
—— (5S)-5-(4-hydroxyphenyl)-4-[hydroxy-(4-propan-2-yloxyphenyl)methylidene]-1-(3-methoxypropyl)pyrrolidine-2,3-dione —— C24H27NO6
(5S)-5-(4-hydroxyphenyl)-4-[hydroxy-(4-propan-2-yloxyphenyl)methylidene]-1-(3-methoxypropyl)pyrrolidine-2,3-dione
—— (5-chloro-1-benzofuran-2-yl)-[(2R)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone —— C17H16ClN3O2
(5-chloro-1-benzofuran-2-yl)-[(2R)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone
—— (5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)-[(2R)-2-[(4-methylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methanone —— C17H21N7O
(5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)-[(2R)-2-[(4-methylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methanone