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—— (5-phenyl-1,3-oxazol-2-yl)methyl (3R)-1-(furan-2-ylmethyl)-5-oxopyrrolidine-3-carboxylate —— C20H18N2O5
(5-phenyl-1,3-oxazol-2-yl)methyl (3R)-1-(furan-2-ylmethyl)-5-oxopyrrolidine-3-carboxylate
—— (5S)-5-phenyl-1,5-dihydrothieno[3,2-e][1,4]thiazepin-2-one —— C13H11NOS2
(5S)-5-phenyl-1,5-dihydrothieno[3,2-e][1,4]thiazepin-2-one
—— (5S)-5-[4-(difluoromethoxy)-3-methoxyphenyl]-1,5-dihydrothieno[3,2-e][1,4]thiazepin-2-one —— C15H13F2NO3S2
(5S)-5-[4-(difluoromethoxy)-3-methoxyphenyl]-1,5-dihydrothieno[3,2-e][1,4]thiazepin-2-one
—— (5R)-5-phenyl-1,5-dihydrothieno[3,2-e][1,4]thiazepin-2-one —— C13H11NOS2
(5R)-5-phenyl-1,5-dihydrothieno[3,2-e][1,4]thiazepin-2-one
—— (5S)-5-(7-chloro-1,3-benzodioxol-5-yl)-1,5-dihydrothieno[3,2-e][1,4]thiazepin-2-one —— C14H10ClNO3S2
(5S)-5-(7-chloro-1,3-benzodioxol-5-yl)-1,5-dihydrothieno[3,2-e][1,4]thiazepin-2-one
—— (5R)-5-[4-(difluoromethoxy)-3-methoxyphenyl]-1,5-dihydrothieno[3,2-e][1,4]thiazepin-2-one —— C15H13F2NO3S2
(5R)-5-[4-(difluoromethoxy)-3-methoxyphenyl]-1,5-dihydrothieno[3,2-e][1,4]thiazepin-2-one
—— (5S)-5-(3-bromophenyl)-1,5-dihydrothieno[3,2-e][1,4]thiazepin-2-one —— C13H10BrNOS2
(5S)-5-(3-bromophenyl)-1,5-dihydrothieno[3,2-e][1,4]thiazepin-2-one
—— (5S)-5-(4-hydroxyphenyl)-1,5-dihydrothieno[3,2-e][1,4]thiazepin-2-one —— C13H11NO2S2
(5S)-5-(4-hydroxyphenyl)-1,5-dihydrothieno[3,2-e][1,4]thiazepin-2-one
—— (5R)-5-(4-propan-2-yloxyphenyl)-1,5-dihydrothieno[3,2-e][1,4]thiazepin-2-one —— C16H17NO2S2
(5R)-5-(4-propan-2-yloxyphenyl)-1,5-dihydrothieno[3,2-e][1,4]thiazepin-2-one
—— (5R)-1-ethyl-5-(ethylamino)-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C12H19N3O2
(5R)-1-ethyl-5-(ethylamino)-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— 5-(hydroxymethyl)-2-methyl-4-[[(2R)-2-(3-pyridin-4-yl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methyl]pyridin-3-ol —— C19H21N5O3
5-(hydroxymethyl)-2-methyl-4-[[(2R)-2-(3-pyridin-4-yl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methyl]pyridin-3-ol
—— [5-[[benzyl(methyl)amino]methyl]-1,2-oxazol-3-yl]-[(1S)-1-methyl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methanone —— C21H24N4O2
[5-[[benzyl(methyl)amino]methyl]-1,2-oxazol-3-yl]-[(1S)-1-methyl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methanone
—— 5-ethyl-N-[[(3S)-1-methylpiperidin-3-yl]methyl]-4-(pyrrolidin-1-ylmethyl)furan-2-carboxamide —— C19H31N3O2
5-ethyl-N-[[(3S)-1-methylpiperidin-3-yl]methyl]-4-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
—— 5-acetamido-N-[(2S)-2-cyclopropyl-2-hydroxyethyl]thiophene-2-carboxamide —— C12H16N2O3S
5-acetamido-N-[(2S)-2-cyclopropyl-2-hydroxyethyl]thiophene-2-carboxamide
—— (5R)-5-(2-fluorophenyl)-1,5-dihydrothieno[3,2-e][1,4]thiazepin-2-one —— C13H10FNOS2
(5R)-5-(2-fluorophenyl)-1,5-dihydrothieno[3,2-e][1,4]thiazepin-2-one
—— [5-[(4-ethylpiperazin-1-yl)methyl]-1,2-oxazol-3-yl]-[(2S)-2-methylpiperidin-1-yl]methanone —— C17H28N4O2
[5-[(4-ethylpiperazin-1-yl)methyl]-1,2-oxazol-3-yl]-[(2S)-2-methylpiperidin-1-yl]methanone
—— 5-(hydroxymethyl)-2-methyl-4-[[(2S)-2-(3-pyridin-4-yl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methyl]pyridin-3-ol —— C19H21N5O3
5-(hydroxymethyl)-2-methyl-4-[[(2S)-2-(3-pyridin-4-yl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methyl]pyridin-3-ol
—— (5S)-1-ethyl-5-(ethylamino)-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C12H19N3O2
(5S)-1-ethyl-5-(ethylamino)-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— 5-[(2R)-2-methyl-4-phenylpiperazine-1-carbonyl]-1H-pyrazin-2-one —— C16H18N4O2
5-[(2R)-2-methyl-4-phenylpiperazine-1-carbonyl]-1H-pyrazin-2-one
—— 5-[(1R)-1-[2-(3,5-difluorophenyl)imidazol-1-yl]ethyl]-3-(2-methoxyethyl)-1,2,4-oxadiazole —— C16H16F2N4O2
5-[(1R)-1-[2-(3,5-difluorophenyl)imidazol-1-yl]ethyl]-3-(2-methoxyethyl)-1,2,4-oxadiazole
—— 5-amino-2-bromo-N-[(2S)-2-cyclopropyl-2-hydroxyethyl]-4-fluorobenzamide —— C12H14BrFN2O2
5-amino-2-bromo-N-[(2S)-2-cyclopropyl-2-hydroxyethyl]-4-fluorobenzamide
—— (5S)-5-[(2-chloro-6-fluorophenyl)methylamino]-1-propyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C18H21ClFN3O2
(5S)-5-[(2-chloro-6-fluorophenyl)methylamino]-1-propyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— (5S)-5-(2,4-difluorophenyl)-1,5-dihydrothieno[3,2-e][1,4]thiazepin-2-one —— C13H9F2NOS2
(5S)-5-(2,4-difluorophenyl)-1,5-dihydrothieno[3,2-e][1,4]thiazepin-2-one
—— (5R)-5-(4-methoxy-3-phenylmethoxyphenyl)-1,5-dihydrothieno[3,2-e][1,4]thiazepin-2-one —— C21H19NO3S2
(5R)-5-(4-methoxy-3-phenylmethoxyphenyl)-1,5-dihydrothieno[3,2-e][1,4]thiazepin-2-one
—— (5R)-5-[[1-(ethylcarbamoyl)piperidin-4-yl]amino]-1-prop-2-enyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C19H29N5O3
(5R)-5-[[1-(ethylcarbamoyl)piperidin-4-yl]amino]-1-prop-2-enyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— (5S)-5-(3,5-dimethoxyphenyl)-1,5-dihydrothieno[3,2-e][1,4]thiazepin-2-one —— C15H15NO3S2
(5S)-5-(3,5-dimethoxyphenyl)-1,5-dihydrothieno[3,2-e][1,4]thiazepin-2-one
—— (5S)-5-(1-methyl-2-oxoquinolin-3-yl)-1,5-dihydrothieno[3,2-e][1,4]thiazepin-2-one —— C17H14N2O2S2
(5S)-5-(1-methyl-2-oxoquinolin-3-yl)-1,5-dihydrothieno[3,2-e][1,4]thiazepin-2-one
—— (5R)-5-(5-methoxy-2,3-dihydro-1,4-benzodioxin-7-yl)-1,5-dihydrothieno[3,2-e][1,4]thiazepin-2-one —— C16H15NO4S2
(5R)-5-(5-methoxy-2,3-dihydro-1,4-benzodioxin-7-yl)-1,5-dihydrothieno[3,2-e][1,4]thiazepin-2-one
—— (5R)-5-[4-(pyridin-2-ylmethoxy)phenyl]-1,5-dihydrothieno[3,2-e][1,4]thiazepin-2-one —— C19H16N2O2S2
(5R)-5-[4-(pyridin-2-ylmethoxy)phenyl]-1,5-dihydrothieno[3,2-e][1,4]thiazepin-2-one
—— (5S)-5-(2-fluorophenyl)-1,5-dihydrothieno[3,2-e][1,4]thiazepin-2-one —— C13H10FNOS2
(5S)-5-(2-fluorophenyl)-1,5-dihydrothieno[3,2-e][1,4]thiazepin-2-one
—— (5S)-5-(4-methoxy-3-phenylmethoxyphenyl)-1,5-dihydrothieno[3,2-e][1,4]thiazepin-2-one —— C21H19NO3S2
(5S)-5-(4-methoxy-3-phenylmethoxyphenyl)-1,5-dihydrothieno[3,2-e][1,4]thiazepin-2-one
—— (5R)-5-(3,5-dimethoxyphenyl)-1,5-dihydrothieno[3,2-e][1,4]thiazepin-2-one —— C15H15NO3S2
(5R)-5-(3,5-dimethoxyphenyl)-1,5-dihydrothieno[3,2-e][1,4]thiazepin-2-one
—— (5R)-5-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl-methylamino]-1-propyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C17H25N5O3
(5R)-5-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl-methylamino]-1-propyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— (5R)-5-[(2-chloro-6-fluorophenyl)methylamino]-1-propyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C18H21ClFN3O2
(5R)-5-[(2-chloro-6-fluorophenyl)methylamino]-1-propyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— (5R)-5-(2,4-difluorophenyl)-1,5-dihydrothieno[3,2-e][1,4]thiazepin-2-one —— C13H9F2NOS2
(5R)-5-(2,4-difluorophenyl)-1,5-dihydrothieno[3,2-e][1,4]thiazepin-2-one
—— (5-phenyl-1,3-oxazol-2-yl)methyl (3S)-1-(furan-2-ylmethyl)-5-oxopyrrolidine-3-carboxylate —— C20H18N2O5
(5-phenyl-1,3-oxazol-2-yl)methyl (3S)-1-(furan-2-ylmethyl)-5-oxopyrrolidine-3-carboxylate
—— (5S)-5-(1-benzyl-3,5-dimethylpyrazol-4-yl)-1,5-dihydrothieno[3,2-e][1,4]thiazepin-2-one —— C19H19N3OS2
(5S)-5-(1-benzyl-3,5-dimethylpyrazol-4-yl)-1,5-dihydrothieno[3,2-e][1,4]thiazepin-2-one
—— 5-[(4-benzylpiperidin-1-yl)methyl]-N-methyl-N-[(1S)-1-pyridin-2-ylethyl]-1,2-oxazole-3-carboxamide —— C25H30N4O2
5-[(4-benzylpiperidin-1-yl)methyl]-N-methyl-N-[(1S)-1-pyridin-2-ylethyl]-1,2-oxazole-3-carboxamide
—— (5R)-5-(1-benzyl-3,5-dimethylpyrazol-4-yl)-1,5-dihydrothieno[3,2-e][1,4]thiazepin-2-one —— C19H19N3OS2
(5R)-5-(1-benzyl-3,5-dimethylpyrazol-4-yl)-1,5-dihydrothieno[3,2-e][1,4]thiazepin-2-one
—— (5S)-5-[4-(pyridin-2-ylmethoxy)phenyl]-1,5-dihydrothieno[3,2-e][1,4]thiazepin-2-one —— C19H16N2O2S2
(5S)-5-[4-(pyridin-2-ylmethoxy)phenyl]-1,5-dihydrothieno[3,2-e][1,4]thiazepin-2-one
—— (5R)-5-(1-methyl-2-oxoquinolin-3-yl)-1,5-dihydrothieno[3,2-e][1,4]thiazepin-2-one —— C17H14N2O2S2
(5R)-5-(1-methyl-2-oxoquinolin-3-yl)-1,5-dihydrothieno[3,2-e][1,4]thiazepin-2-one
—— [5-[(4-ethylpiperazin-1-yl)methyl]-1,2-oxazol-3-yl]-[(2R)-2-methylpiperidin-1-yl]methanone —— C17H28N4O2
[5-[(4-ethylpiperazin-1-yl)methyl]-1,2-oxazol-3-yl]-[(2R)-2-methylpiperidin-1-yl]methanone
—— 5-indol-3-ylidene-3-[(1-methylpiperidin-4-yl)methyl]-2H-1,2,4-oxadiazole —— C17H20N4O
5-indol-3-ylidene-3-[(1-methylpiperidin-4-yl)methyl]-2H-1,2,4-oxadiazole
—— (5R)-5-(3-chlorophenyl)-1,5-dihydrothieno[3,2-e][1,4]thiazepin-2-one —— C13H10ClNOS2
(5R)-5-(3-chlorophenyl)-1,5-dihydrothieno[3,2-e][1,4]thiazepin-2-one
—— (5S)-5-(4-propan-2-yloxyphenyl)-1,5-dihydrothieno[3,2-e][1,4]thiazepin-2-one —— C16H17NO2S2
(5S)-5-(4-propan-2-yloxyphenyl)-1,5-dihydrothieno[3,2-e][1,4]thiazepin-2-one
—— 5-[(2S)-2-methyl-4-phenylpiperazine-1-carbonyl]-1H-pyrazin-2-one —— C16H18N4O2
5-[(2S)-2-methyl-4-phenylpiperazine-1-carbonyl]-1H-pyrazin-2-one
—— (5S)-5-(5-methoxy-2,3-dihydro-1,4-benzodioxin-7-yl)-1,5-dihydrothieno[3,2-e][1,4]thiazepin-2-one —— C16H15NO4S2
(5S)-5-(5-methoxy-2,3-dihydro-1,4-benzodioxin-7-yl)-1,5-dihydrothieno[3,2-e][1,4]thiazepin-2-one
—— (5R)-5-(2,3-dimethoxyphenyl)-1,5-dihydrothieno[3,2-e][1,4]thiazepin-2-one —— C15H15NO3S2
(5R)-5-(2,3-dimethoxyphenyl)-1,5-dihydrothieno[3,2-e][1,4]thiazepin-2-one
—— (5S)-1-ethyl-5-[2-(pyridin-3-ylamino)ethylamino]-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C17H23N5O2
(5S)-1-ethyl-5-[2-(pyridin-3-ylamino)ethylamino]-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— (5S)-5-[[1-(ethylcarbamoyl)piperidin-4-yl]amino]-1-prop-2-enyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C19H29N5O3
(5S)-5-[[1-(ethylcarbamoyl)piperidin-4-yl]amino]-1-prop-2-enyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid