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—— 5,6-dimethyl-2-[2-[(2R)-2-methylpiperidin-1-yl]-2-oxoethyl]sulfanyl-3-propan-2-ylthieno[2,3-d]pyrimidin-4-one —— C19H27N3O2S2
5,6-dimethyl-2-[2-[(2R)-2-methylpiperidin-1-yl]-2-oxoethyl]sulfanyl-3-propan-2-ylthieno[2,3-d]pyrimidin-4-one
—— 5-bromo-N-[(1R)-1-cyanobutyl]-2,3-dihydro-1,4-benzodioxine-7-carboxamide —— C14H15BrN2O3
5-bromo-N-[(1R)-1-cyanobutyl]-2,3-dihydro-1,4-benzodioxine-7-carboxamide
—— 5-[(4aR,8aS)-3,4,4a,5,6,7,8,8a-octahydro-2H-quinoline-1-carbonyl]-4-methylthiophene-2-sulfonamide —— C15H22N2O3S2
5-[(4aR,8aS)-3,4,4a,5,6,7,8,8a-octahydro-2H-quinoline-1-carbonyl]-4-methylthiophene-2-sulfonamide
—— 5-bromo-3-(2H-tetrazol-5-ylhydrazinylidene)indol-2-olate —— C9H5BrN7O-
5-bromo-3-(2H-tetrazol-5-ylhydrazinylidene)indol-2-olate
—— 5-(2,5-dimethoxyphenyl)-N-[(2S)-2-(dimethylamino)propyl]-1,2-oxazole-3-carboxamide —— C17H23N3O4
5-(2,5-dimethoxyphenyl)-N-[(2S)-2-(dimethylamino)propyl]-1,2-oxazole-3-carboxamide
—— (5-methyl-1-phenylpyrazol-4-yl)-[(3S)-3-(4-methylpyrazol-1-yl)piperidin-1-yl]methanone —— C20H23N5O
(5-methyl-1-phenylpyrazol-4-yl)-[(3S)-3-(4-methylpyrazol-1-yl)piperidin-1-yl]methanone
—— 5-[(4aR,8aR)-3,4,4a,5,6,7,8,8a-octahydro-2H-quinoline-1-carbonyl]-4-methylthiophene-2-sulfonamide —— C15H22N2O3S2
5-[(4aR,8aR)-3,4,4a,5,6,7,8,8a-octahydro-2H-quinoline-1-carbonyl]-4-methylthiophene-2-sulfonamide
—— 5-cyclopropyl-N-ethyl-N-[[(3S)-oxolan-3-yl]methyl]-1-phenyl-1,2,4-triazole-3-carboxamide —— C19H24N4O2
5-cyclopropyl-N-ethyl-N-[[(3S)-oxolan-3-yl]methyl]-1-phenyl-1,2,4-triazole-3-carboxamide
—— (5R)-8,8-dimethyl-5-[4-(trifluoromethyl)phenyl]-5,7,9,10-tetrahydro-1H-pyrimido[4,5-b]quinoline-2,4,6-trione —— C20H18F3N3O3
(5R)-8,8-dimethyl-5-[4-(trifluoromethyl)phenyl]-5,7,9,10-tetrahydro-1H-pyrimido[4,5-b]quinoline-2,4,6-trione
—— (5-methyl-1-phenylpyrazol-4-yl)-[(3R)-3-(4-methylpyrazol-1-yl)piperidin-1-yl]methanone —— C20H23N5O
(5-methyl-1-phenylpyrazol-4-yl)-[(3R)-3-(4-methylpyrazol-1-yl)piperidin-1-yl]methanone
—— (5S)-8,8-dimethyl-5-[4-(trifluoromethyl)phenyl]-5,7,9,10-tetrahydro-1H-pyrimido[4,5-b]quinoline-2,4,6-trione —— C20H18F3N3O3
(5S)-8,8-dimethyl-5-[4-(trifluoromethyl)phenyl]-5,7,9,10-tetrahydro-1H-pyrimido[4,5-b]quinoline-2,4,6-trione
—— (5S)-5-methyl-2-nitro-6H-[1,3]oxazolo[3,2-b][1,2,4]triazole-5-carbonitrile —— C6H5N5O3
(5S)-5-methyl-2-nitro-6H-[1,3]oxazolo[3,2-b][1,2,4]triazole-5-carbonitrile
—— 5-fluoro-2-[[(2R)-2-[(4-methylpyrazol-1-yl)methyl]morpholin-4-yl]methyl]benzonitrile —— C17H19FN4O
5-fluoro-2-[[(2R)-2-[(4-methylpyrazol-1-yl)methyl]morpholin-4-yl]methyl]benzonitrile
—— 5-methyl-N-[(2R,3R)-3-(4-methylpyrazol-1-yl)butan-2-yl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine —— C14H19N7
5-methyl-N-[(2R,3R)-3-(4-methylpyrazol-1-yl)butan-2-yl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine
—— 5-[(1S)-1-[4-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]piperazin-1-yl]ethyl]-3-methyl-1,2,4-oxadiazole —— C18H27N5O2
5-[(1S)-1-[4-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]piperazin-1-yl]ethyl]-3-methyl-1,2,4-oxadiazole
—— 5-fluoro-2-[[(2S)-2-[(4-methylpyrazol-1-yl)methyl]morpholin-4-yl]methyl]benzonitrile —— C17H19FN4O
5-fluoro-2-[[(2S)-2-[(4-methylpyrazol-1-yl)methyl]morpholin-4-yl]methyl]benzonitrile
—— 5-[(1R)-1-[4-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]piperazin-1-yl]ethyl]-3-methyl-1,2,4-oxadiazole —— C18H27N5O2
5-[(1R)-1-[4-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]piperazin-1-yl]ethyl]-3-methyl-1,2,4-oxadiazole
—— 5-methyl-4-[[(3S)-3-(2-methylpyrazol-3-yl)piperidin-1-yl]methyl]-2-thiophen-3-yl-1,3-oxazole —— C18H22N4OS
5-methyl-4-[[(3S)-3-(2-methylpyrazol-3-yl)piperidin-1-yl]methyl]-2-thiophen-3-yl-1,3-oxazole
—— 5-[(1S)-1-[4-[(5-chlorothiadiazol-4-yl)methyl]piperazin-1-yl]ethyl]-3-ethyl-1,2,4-oxadiazole —— C13H19ClN6OS
5-[(1S)-1-[4-[(5-chlorothiadiazol-4-yl)methyl]piperazin-1-yl]ethyl]-3-ethyl-1,2,4-oxadiazole
—— 5-methyl-N-[(2S,3R)-3-(4-methylpyrazol-1-yl)butan-2-yl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine —— C14H19N7
5-methyl-N-[(2S,3R)-3-(4-methylpyrazol-1-yl)butan-2-yl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine
—— 5-methyl-4-[[(3R)-3-(2-methylpyrazol-3-yl)piperidin-1-yl]methyl]-2-thiophen-3-yl-1,3-oxazole —— C18H22N4OS
5-methyl-4-[[(3R)-3-(2-methylpyrazol-3-yl)piperidin-1-yl]methyl]-2-thiophen-3-yl-1,3-oxazole
—— 5-[(1R)-1-(1-cyclopropyl-6,7-dihydro-4H-imidazo[4,5-c]pyridin-5-yl)ethyl]-3-thiophen-2-yl-1,2,4-oxadiazole —— C17H19N5OS
5-[(1R)-1-(1-cyclopropyl-6,7-dihydro-4H-imidazo[4,5-c]pyridin-5-yl)ethyl]-3-thiophen-2-yl-1,2,4-oxadiazole
—— 5-(N-benzyl-C-methylcarbonimidoyl)-1,3-diazinane-2,4,6-trione —— C13H13N3O3
5-(N-benzyl-C-methylcarbonimidoyl)-1,3-diazinane-2,4,6-trione
—— 5-bromo-N-[(1R)-2-methyl-1-(1,2,4-triazol-1-yl)propyl]pyridin-1-ium-2-amine —— C11H15BrN5+
5-bromo-N-[(1R)-2-methyl-1-(1,2,4-triazol-1-yl)propyl]pyridin-1-ium-2-amine
—— (5R)-5-(2,6-dichlorophenyl)-2-prop-2-enylsulfanyl-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-4,7-dione —— C16H13Cl2N3O2S
(5R)-5-(2,6-dichlorophenyl)-2-prop-2-enylsulfanyl-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-4,7-dione
—— 5-[(1S)-1-(1-cyclopropyl-6,7-dihydro-4H-imidazo[4,5-c]pyridin-5-yl)ethyl]-3-thiophen-2-yl-1,2,4-oxadiazole —— C17H19N5OS
5-[(1S)-1-(1-cyclopropyl-6,7-dihydro-4H-imidazo[4,5-c]pyridin-5-yl)ethyl]-3-thiophen-2-yl-1,2,4-oxadiazole
—— (5S)-2-ethylsulfanyl-5-naphthalen-2-yl-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-4,7-dione —— C19H17N3O2S
(5S)-2-ethylsulfanyl-5-naphthalen-2-yl-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-4,7-dione
—— (5S)-1-butyl-4-[(4-chlorophenyl)-hydroxymethylidene]-5-(4-methoxyphenyl)pyrrolidine-2,3-dione —— C22H22ClNO4
(5S)-1-butyl-4-[(4-chlorophenyl)-hydroxymethylidene]-5-(4-methoxyphenyl)pyrrolidine-2,3-dione
—— (5R)-5-(3-bromophenyl)-2-prop-2-enylsulfanyl-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-4,7-dione —— C16H14BrN3O2S
(5R)-5-(3-bromophenyl)-2-prop-2-enylsulfanyl-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-4,7-dione
—— 5-methyl-N-[(2R,3S)-3-(4-methylpyrazol-1-yl)butan-2-yl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine —— C14H19N7
5-methyl-N-[(2R,3S)-3-(4-methylpyrazol-1-yl)butan-2-yl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine
—— (5S)-5-(4-methylsulfanylphenyl)-2-prop-2-enylsulfanyl-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-4,7-dione —— C17H17N3O2S2
(5S)-5-(4-methylsulfanylphenyl)-2-prop-2-enylsulfanyl-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-4,7-dione
—— (5S)-2-ethylsulfanyl-5-(4-methylsulfanylphenyl)-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-4,7-dione —— C16H17N3O2S2
(5S)-2-ethylsulfanyl-5-(4-methylsulfanylphenyl)-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-4,7-dione
—— (5R)-5-(3,4-dichlorophenyl)-2-methylsulfanyl-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-4,7-dione —— C14H11Cl2N3O2S
(5R)-5-(3,4-dichlorophenyl)-2-methylsulfanyl-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-4,7-dione
—— (5R)-5-(3,4-dichlorophenyl)-2-ethylsulfanyl-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-4,7-dione —— C15H13Cl2N3O2S
(5R)-5-(3,4-dichlorophenyl)-2-ethylsulfanyl-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-4,7-dione
—— 5,5-dimethyl-2-[[(1R)-1-phenylethyl]iminomethyl]cyclohexane-1,3-dione —— C17H21NO2
5,5-dimethyl-2-[[(1R)-1-phenylethyl]iminomethyl]cyclohexane-1,3-dione
—— 5-bromo-N-[(1S)-2-methyl-1-(1,2,4-triazol-1-yl)propyl]pyridin-2-amine —— C11H14BrN5
5-bromo-N-[(1S)-2-methyl-1-(1,2,4-triazol-1-yl)propyl]pyridin-2-amine
—— 5,5-dimethyl-2-(C-methyl-N-prop-2-enylcarbonimidoyl)cyclohexane-1,3-dione —— C13H19NO2
5,5-dimethyl-2-(C-methyl-N-prop-2-enylcarbonimidoyl)cyclohexane-1,3-dione
—— (5R)-1-butyl-4-[(4-chlorophenyl)-hydroxymethylidene]-5-(4-methoxyphenyl)pyrrolidine-2,3-dione —— C22H22ClNO4
(5R)-1-butyl-4-[(4-chlorophenyl)-hydroxymethylidene]-5-(4-methoxyphenyl)pyrrolidine-2,3-dione
—— (5E)-5-benzylidene-3-(benzyliminomethyl)pyrrolidine-2,4-dione —— C19H16N2O2
(5E)-5-benzylidene-3-(benzyliminomethyl)pyrrolidine-2,4-dione
—— (5S,6R)-2,7-diamino-4-oxo-5-phenyl-5,6-dihydro-3H-pyrido[2,3-d]pyrimidine-6-carbonitrile —— C14H12N6O
(5S,6R)-2,7-diamino-4-oxo-5-phenyl-5,6-dihydro-3H-pyrido[2,3-d]pyrimidine-6-carbonitrile
—— (5-methyl-1-benzofuran-2-yl)-[(3R)-3-pyrazol-1-ylpiperidin-1-yl]methanone —— C18H19N3O2
(5-methyl-1-benzofuran-2-yl)-[(3R)-3-pyrazol-1-ylpiperidin-1-yl]methanone
—— 5-chloro-6-[[(2S)-2-hydroxy-2-phenylethyl]amino]pyridine-3-carbonitrile —— C14H12ClN3O
5-chloro-6-[[(2S)-2-hydroxy-2-phenylethyl]amino]pyridine-3-carbonitrile
—— (5-methyl-1,2-oxazol-3-yl)-[(3R)-3-pyrazol-1-ylpiperidin-1-yl]methanone —— C13H16N4O2
(5-methyl-1,2-oxazol-3-yl)-[(3R)-3-pyrazol-1-ylpiperidin-1-yl]methanone
—— (5-methylfuro[3,2-b]pyridin-2-yl)-[(3S)-3-pyrazol-1-ylpiperidin-1-yl]methanone —— C17H18N4O2
(5-methylfuro[3,2-b]pyridin-2-yl)-[(3S)-3-pyrazol-1-ylpiperidin-1-yl]methanone
—— (5-methyl-1,2-oxazol-3-yl)-[(3S)-3-pyrazol-1-ylpiperidin-1-yl]methanone —— C13H16N4O2
(5-methyl-1,2-oxazol-3-yl)-[(3S)-3-pyrazol-1-ylpiperidin-1-yl]methanone
—— (5R,6R)-2,7-diamino-4-oxo-5-phenyl-5,6-dihydro-3H-pyrido[2,3-d]pyrimidine-6-carbonitrile —— C14H12N6O
(5R,6R)-2,7-diamino-4-oxo-5-phenyl-5,6-dihydro-3H-pyrido[2,3-d]pyrimidine-6-carbonitrile
—— (5-methyl-1-benzofuran-2-yl)-[(3S)-3-pyrazol-1-ylpiperidin-1-yl]methanone —— C18H19N3O2
(5-methyl-1-benzofuran-2-yl)-[(3S)-3-pyrazol-1-ylpiperidin-1-yl]methanone
—— (5R,6S)-2,7-diamino-5-(4-fluorophenyl)-4-oxo-5,6-dihydro-3H-pyrido[2,3-d]pyrimidine-6-carbonitrile —— C14H11FN6O
(5R,6S)-2,7-diamino-5-(4-fluorophenyl)-4-oxo-5,6-dihydro-3H-pyrido[2,3-d]pyrimidine-6-carbonitrile
—— (5S,6S)-2-amino-4,7-dioxo-5-phenyl-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-6-carbonitrile —— C14H11N5O2
(5S,6S)-2-amino-4,7-dioxo-5-phenyl-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-6-carbonitrile
—— (5R,6R)-2-amino-4,7-dioxo-5-phenyl-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-6-carbonitrile —— C14H11N5O2
(5R,6R)-2-amino-4,7-dioxo-5-phenyl-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-6-carbonitrile