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—— 5-[1-[2-[(3R)-1,1-dioxothiolan-3-yl]acetyl]piperidin-4-yl]-4-ethyl-2-methyl-1,2,4-triazol-3-one —— C16H26N4O4S
5-[1-[2-[(3R)-1,1-dioxothiolan-3-yl]acetyl]piperidin-4-yl]-4-ethyl-2-methyl-1,2,4-triazol-3-one
—— (5R)-5-(3-ethoxy-4-hydroxyphenyl)-8,8-dimethyl-5,7,9,10-tetrahydro-4H-[1,2,5]oxadiazolo[3,4-b][1,4]benzodiazepin-6-one —— C19H22N4O4
(5R)-5-(3-ethoxy-4-hydroxyphenyl)-8,8-dimethyl-5,7,9,10-tetrahydro-4H-[1,2,5]oxadiazolo[3,4-b][1,4]benzodiazepin-6-one
—— (5R)-1,3-dimethyl-5-(3,4,5-trimethoxyphenyl)-6,8-dihydro-5H-pyrido[2,3-d]pyrimidine-2,4,7-trione —— C18H21N3O6
(5R)-1,3-dimethyl-5-(3,4,5-trimethoxyphenyl)-6,8-dihydro-5H-pyrido[2,3-d]pyrimidine-2,4,7-trione
—— (5R)-2,4-diamino-8,8-dimethyl-6-oxo-5-phenyl-7,9-dihydro-5H-chromeno[2,3-b]pyridine-3-carbonitrile —— C21H20N4O2
(5R)-2,4-diamino-8,8-dimethyl-6-oxo-5-phenyl-7,9-dihydro-5H-chromeno[2,3-b]pyridine-3-carbonitrile
—— (5-Oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl 2-(2,4-dimethylphenyl)sulfanylacetate —— C17H16N2O3S2
(5-Oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl 2-(2,4-dimethylphenyl)sulfanylacetate
—— (5R)-2,4-diamino-8,8-dimethyl-6-oxo-5-phenyl-7,9-dihydro-5H-chromeno[2,3-b]pyridin-1-ium-3-carbonitrile —— C21H21N4O2+
(5R)-2,4-diamino-8,8-dimethyl-6-oxo-5-phenyl-7,9-dihydro-5H-chromeno[2,3-b]pyridin-1-ium-3-carbonitrile
—— (5-Phenyl-1,3,4-oxadiazol-2-yl)methyl 2-(2,4-dimethylphenyl)sulfanylacetate —— C19H18N2O3S
(5-Phenyl-1,3,4-oxadiazol-2-yl)methyl 2-(2,4-dimethylphenyl)sulfanylacetate
—— 5-fluoro-2-methoxy-N-[[(3R)-1-methylpiperidin-3-yl]methyl]benzamide —— C15H21FN2O2
5-fluoro-2-methoxy-N-[[(3R)-1-methylpiperidin-3-yl]methyl]benzamide
—— 5-(benzimidazol-1-ylmethyl)-N-[(2R)-2-(3,5-dimethylpyrazol-1-yl)propyl]-1H-pyrazole-3-carboxamide —— C20H23N7O
5-(benzimidazol-1-ylmethyl)-N-[(2R)-2-(3,5-dimethylpyrazol-1-yl)propyl]-1H-pyrazole-3-carboxamide
—— 5-[(3R)-1-[4-(aminomethyl)benzoyl]piperidin-3-yl]-4-ethyl-2-methyl-1,2,4-triazol-3-one —— C18H25N5O2
5-[(3R)-1-[4-(aminomethyl)benzoyl]piperidin-3-yl]-4-ethyl-2-methyl-1,2,4-triazol-3-one
—— 5-[(3S)-1-(2-hydroxyacetyl)piperidin-3-yl]-2-methyl-4-phenyl-1,2,4-triazol-3-one —— C16H20N4O3
5-[(3S)-1-(2-hydroxyacetyl)piperidin-3-yl]-2-methyl-4-phenyl-1,2,4-triazol-3-one
—— [(5S)-2,9-diazaspiro[4.5]decan-2-yl]-[4-(1H-pyrazol-5-yl)phenyl]methanone —— C18H22N4O
[(5S)-2,9-diazaspiro[4.5]decan-2-yl]-[4-(1H-pyrazol-5-yl)phenyl]methanone
—— (5S)-1-(2-methylpropyl)-5-pyrrolidin-1-yl-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C16H25N3O2
(5S)-1-(2-methylpropyl)-5-pyrrolidin-1-yl-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— (5R)-1-ethyl-5-[(3-methoxy-3-oxopropyl)amino]-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C14H21N3O4
(5R)-1-ethyl-5-[(3-methoxy-3-oxopropyl)amino]-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— (5S)-2-[(4-chlorophenyl)methylsulfonyl]-2,9-diazaspiro[4.5]decane —— C15H21ClN2O2S
(5S)-2-[(4-chlorophenyl)methylsulfonyl]-2,9-diazaspiro[4.5]decane
—— 5-[1-[2-[(3S)-1,1-dioxothiolan-3-yl]acetyl]piperidin-4-yl]-4-ethyl-2-methyl-1,2,4-triazol-3-one —— C16H26N4O4S
5-[1-[2-[(3S)-1,1-dioxothiolan-3-yl]acetyl]piperidin-4-yl]-4-ethyl-2-methyl-1,2,4-triazol-3-one
—— 5-[(3-acetylphenoxy)methyl]-N-[(3R)-3-hydroxybutyl]-1,2-oxazole-3-carboxamide —— C17H20N2O5
5-[(3-acetylphenoxy)methyl]-N-[(3R)-3-hydroxybutyl]-1,2-oxazole-3-carboxamide
—— (5R)-5-[4-[(2-cyanophenyl)methyl]piperazin-1-yl]-1-ethyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C22H27N5O2
(5R)-5-[4-[(2-cyanophenyl)methyl]piperazin-1-yl]-1-ethyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— (5R)-5-(2,3-dimethyl-4-oxo-5,7-dihydropyrrolo[3,4-d]pyrimidin-6-yl)-1-propyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C19H25N5O3
(5R)-5-(2,3-dimethyl-4-oxo-5,7-dihydropyrrolo[3,4-d]pyrimidin-6-yl)-1-propyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— 5-[(3R)-1-[2-(1H-benzimidazol-2-yl)acetyl]piperidin-3-yl]-4-ethyl-2-methyl-1,2,4-triazol-3-one —— C19H24N6O2
5-[(3R)-1-[2-(1H-benzimidazol-2-yl)acetyl]piperidin-3-yl]-4-ethyl-2-methyl-1,2,4-triazol-3-one
—— 5-[(3S)-1-[4-(aminomethyl)benzoyl]piperidin-3-yl]-4-ethyl-2-methyl-1,2,4-triazol-3-one —— C18H25N5O2
5-[(3S)-1-[4-(aminomethyl)benzoyl]piperidin-3-yl]-4-ethyl-2-methyl-1,2,4-triazol-3-one
—— (5R)-5-(2-morpholin-4-ylethylamino)-1-prop-2-enyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C17H26N4O3
(5R)-5-(2-morpholin-4-ylethylamino)-1-prop-2-enyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— 5-(3-fluorophenyl)-N-[2-[(2R)-2-(hydroxymethyl)piperidin-1-yl]ethyl]-1H-pyrazole-4-carboxamide —— C18H23FN4O2
5-(3-fluorophenyl)-N-[2-[(2R)-2-(hydroxymethyl)piperidin-1-yl]ethyl]-1H-pyrazole-4-carboxamide
—— [(5R)-2,9-diazaspiro[4.5]decan-2-yl]-[4-(1H-pyrazol-5-yl)phenyl]methanone —— C18H22N4O
[(5R)-2,9-diazaspiro[4.5]decan-2-yl]-[4-(1H-pyrazol-5-yl)phenyl]methanone
—— 5-[(3R)-1-(2-hydroxyacetyl)piperidin-3-yl]-2-methyl-4-phenyl-1,2,4-triazol-3-one —— C16H20N4O3
5-[(3R)-1-(2-hydroxyacetyl)piperidin-3-yl]-2-methyl-4-phenyl-1,2,4-triazol-3-one
—— (5S)-5-(2-morpholin-4-ylethylamino)-1-prop-2-enyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C17H26N4O3
(5S)-5-(2-morpholin-4-ylethylamino)-1-prop-2-enyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— 5-[(3S)-1-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]piperidin-3-yl]-4-ethyl-2-methyl-1,2,4-triazol-3-one —— C18H28N6O2
5-[(3S)-1-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]piperidin-3-yl]-4-ethyl-2-methyl-1,2,4-triazol-3-one
—— (5S)-7-(7-chloroquinolin-4-yl)-2,7-diazaspiro[4.5]decane —— C17H20ClN3
(5S)-7-(7-chloroquinolin-4-yl)-2,7-diazaspiro[4.5]decane
—— (5R)-7-(7-chloroquinolin-4-yl)-2,7-diazaspiro[4.5]decane —— C17H20ClN3
(5R)-7-(7-chloroquinolin-4-yl)-2,7-diazaspiro[4.5]decane
—— [5-(morpholin-4-ylmethyl)-1,2-oxazol-3-yl]-[(3S)-3-propylmorpholin-4-yl]methanone —— C16H25N3O4
[5-(morpholin-4-ylmethyl)-1,2-oxazol-3-yl]-[(3S)-3-propylmorpholin-4-yl]methanone
—— 5-[(2R)-2-(aminomethyl)-7-chloro-2,3-dihydro-1-benzofuran-5-yl]-1,3-benzothiazol-2-amine —— C16H14ClN3OS
5-[(2R)-2-(aminomethyl)-7-chloro-2,3-dihydro-1-benzofuran-5-yl]-1,3-benzothiazol-2-amine
—— 5-[(4-ethylpiperazin-1-yl)methyl]-N-methyl-N-[[(2S)-1-methylpiperidin-2-yl]methyl]-1,2-oxazole-3-carboxamide —— C19H33N5O2
5-[(4-ethylpiperazin-1-yl)methyl]-N-methyl-N-[[(2S)-1-methylpiperidin-2-yl]methyl]-1,2-oxazole-3-carboxamide
—— [(5S)-2-methyl-2,7-diazaspiro[4.5]decan-7-yl]-(5-methyl-1H-pyrazol-3-yl)methanone —— C14H22N4O
[(5S)-2-methyl-2,7-diazaspiro[4.5]decan-7-yl]-(5-methyl-1H-pyrazol-3-yl)methanone
—— 5-[(3R)-1-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]piperidin-3-yl]-4-ethyl-2-methyl-1,2,4-triazol-3-one —— C18H28N6O2
5-[(3R)-1-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]piperidin-3-yl]-4-ethyl-2-methyl-1,2,4-triazol-3-one
—— (5S)-5-(3-phenoxyphenoxy)-1-azabicyclo[3.2.1]octane —— C19H21NO2
(5S)-5-(3-phenoxyphenoxy)-1-azabicyclo[3.2.1]octane
—— (5S)-5-(2-cyano-4,6,7,8-tetrahydropyrazolo[1,5-a][1,4]diazepin-5-yl)-1-prop-2-enyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C19H22N6O2
(5S)-5-(2-cyano-4,6,7,8-tetrahydropyrazolo[1,5-a][1,4]diazepin-5-yl)-1-prop-2-enyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— 5-[(2S)-2-(aminomethyl)-7-chloro-2,3-dihydro-1-benzofuran-5-yl]-1,3-benzothiazol-2-amine —— C16H14ClN3OS
5-[(2S)-2-(aminomethyl)-7-chloro-2,3-dihydro-1-benzofuran-5-yl]-1,3-benzothiazol-2-amine
—— [5-(morpholin-4-ylmethyl)-1,2-oxazol-3-yl]-[(3R)-3-propylmorpholin-4-yl]methanone —— C16H25N3O4
[5-(morpholin-4-ylmethyl)-1,2-oxazol-3-yl]-[(3R)-3-propylmorpholin-4-yl]methanone
—— 5-(5-methylthiophen-2-yl)-N-[[5-[(2R)-oxolan-2-yl]-1,2,4-oxadiazol-3-yl]methyl]-1H-pyrazole-3-carboxamide —— C16H17N5O3S
5-(5-methylthiophen-2-yl)-N-[[5-[(2R)-oxolan-2-yl]-1,2,4-oxadiazol-3-yl]methyl]-1H-pyrazole-3-carboxamide
—— [(5R)-2-methyl-2,7-diazaspiro[4.5]decan-7-yl]-(5-methyl-1H-pyrazol-3-yl)methanone —— C14H22N4O
[(5R)-2-methyl-2,7-diazaspiro[4.5]decan-7-yl]-(5-methyl-1H-pyrazol-3-yl)methanone
—— (5R)-5-(2-cyano-4,6,7,8-tetrahydropyrazolo[1,5-a][1,4]diazepin-5-yl)-1-prop-2-enyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C19H22N6O2
(5R)-5-(2-cyano-4,6,7,8-tetrahydropyrazolo[1,5-a][1,4]diazepin-5-yl)-1-prop-2-enyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— 5-cyclopropyl-N-[5-[(2S)-pentan-2-yl]-1,3,4-thiadiazol-2-yl]-1H-pyrazole-4-carboxamide —— C14H19N5OS
5-cyclopropyl-N-[5-[(2S)-pentan-2-yl]-1,3,4-thiadiazol-2-yl]-1H-pyrazole-4-carboxamide
—— (5S)-5-[4-(dimethylsulfamoyl)piperazin-1-yl]-1-ethyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C16H27N5O4S
(5S)-5-[4-(dimethylsulfamoyl)piperazin-1-yl]-1-ethyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— (5S)-2-(azepan-1-ylsulfonyl)-2,9-diazaspiro[4.5]decane —— C14H27N3O2S
(5S)-2-(azepan-1-ylsulfonyl)-2,9-diazaspiro[4.5]decane
—— 5-(5-methylthiophen-2-yl)-N-[[5-[(2S)-oxolan-2-yl]-1,2,4-oxadiazol-3-yl]methyl]-1H-pyrazole-3-carboxamide —— C16H17N5O3S
5-(5-methylthiophen-2-yl)-N-[[5-[(2S)-oxolan-2-yl]-1,2,4-oxadiazol-3-yl]methyl]-1H-pyrazole-3-carboxamide
—— (5R)-5-(3-phenoxyphenoxy)-1-azabicyclo[3.2.1]octane —— C19H21NO2
(5R)-5-(3-phenoxyphenoxy)-1-azabicyclo[3.2.1]octane
—— 5-[(2S)-2-imidazol-1-ylpropanoyl]-1-methyl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-3-carboxylic acid —— C14H17N5O3
5-[(2S)-2-imidazol-1-ylpropanoyl]-1-methyl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
—— 5-[(2R)-2-imidazol-1-ylpropanoyl]-1-methyl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-3-carboxylic acid —— C14H17N5O3
5-[(2R)-2-imidazol-1-ylpropanoyl]-1-methyl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
—— 5-[(3,4-Dichlorophenyl)methylsulfanyl]-1-(2,4-dimethylphenyl)tetrazole —— C16H14Cl2N4S
5-[(3,4-Dichlorophenyl)methylsulfanyl]-1-(2,4-dimethylphenyl)tetrazole
—— (5R)-5-[4-(dimethylsulfamoyl)piperazin-1-yl]-1-ethyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C16H27N5O4S
(5R)-5-[4-(dimethylsulfamoyl)piperazin-1-yl]-1-ethyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid