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—— (5R)-N-methyl-3-propan-2-yl-N-[(3-pyridin-4-yl-1,2-oxazol-5-yl)methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C17H20N4O3
(5R)-N-methyl-3-propan-2-yl-N-[(3-pyridin-4-yl-1,2-oxazol-5-yl)methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5R)-2-[(5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl)methyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one —— C18H25N5O
(5R)-2-[(5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl)methyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-1-ethyl-5-[methyl-[(3-pyridin-4-yl-1,2-oxazol-5-yl)methyl]amino]-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C20H23N5O3
(5R)-1-ethyl-5-[methyl-[(3-pyridin-4-yl-1,2-oxazol-5-yl)methyl]amino]-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— 5-benzyl-N-[(3S)-pyrrolidin-3-yl]-4,6,7,8-tetrahydropyrazolo[1,5-a][1,4]diazepine-2-carboxamide —— C19H25N5O
5-benzyl-N-[(3S)-pyrrolidin-3-yl]-4,6,7,8-tetrahydropyrazolo[1,5-a][1,4]diazepine-2-carboxamide
—— (5S)-1-ethyl-5-[methyl-[(3-pyridin-4-yl-1,2-oxazol-5-yl)methyl]amino]-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C20H23N5O3
(5S)-1-ethyl-5-[methyl-[(3-pyridin-4-yl-1,2-oxazol-5-yl)methyl]amino]-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— (5R)-5-[4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl]piperidin-2-one —— C20H23FN4O2
(5R)-5-[4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl]piperidin-2-one
—— 5-[4-[[(5R)-2,9-diazaspiro[4.5]decan-2-yl]sulfonyl]phenyl]-1,3-oxazole —— C17H21N3O3S
5-[4-[[(5R)-2,9-diazaspiro[4.5]decan-2-yl]sulfonyl]phenyl]-1,3-oxazole
—— 5-N-[(1S)-1-(2,5-dimethyl-1,3-thiazol-4-yl)ethyl]-6-N-(2-methoxyethyl)-5-N-methyl-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine —— C15H21N7O2S
5-N-[(1S)-1-(2,5-dimethyl-1,3-thiazol-4-yl)ethyl]-6-N-(2-methoxyethyl)-5-N-methyl-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
—— 5-chloro-N-[2-[(3S)-1-ethylpiperidin-3-yl]ethyl]-1,3-dimethylpyrazole-4-sulfonamide —— C14H25ClN4O2S
5-chloro-N-[2-[(3S)-1-ethylpiperidin-3-yl]ethyl]-1,3-dimethylpyrazole-4-sulfonamide
—— (5S)-2-[(5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl)methyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one —— C18H25N5O
(5S)-2-[(5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl)methyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
—— 5-(benzimidazol-1-ylmethyl)-N-methyl-N-[(1S)-1-pyrimidin-4-ylethyl]-1H-pyrazole-3-carboxamide —— C19H19N7O
5-(benzimidazol-1-ylmethyl)-N-methyl-N-[(1S)-1-pyrimidin-4-ylethyl]-1H-pyrazole-3-carboxamide
—— 5-chloro-N-[2-[(3R)-1-ethylpiperidin-3-yl]ethyl]-1,3-dimethylpyrazole-4-sulfonamide —— C14H25ClN4O2S
5-chloro-N-[2-[(3R)-1-ethylpiperidin-3-yl]ethyl]-1,3-dimethylpyrazole-4-sulfonamide
—— 5-[(2,6-dimethylphenoxy)methyl]-N-[(3S)-1,1-dioxothiolan-3-yl]-N-ethyl-1,2-oxazole-3-carboxamide —— C19H24N2O5S
5-[(2,6-dimethylphenoxy)methyl]-N-[(3S)-1,1-dioxothiolan-3-yl]-N-ethyl-1,2-oxazole-3-carboxamide
—— (5S)-N-methyl-3-propan-2-yl-N-[(3-pyridin-4-yl-1,2-oxazol-5-yl)methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C17H20N4O3
(5S)-N-methyl-3-propan-2-yl-N-[(3-pyridin-4-yl-1,2-oxazol-5-yl)methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5S,7R)-3-(4-methylphenyl)-N'-[(6-oxocyclohexa-2,4-dien-1-ylidene)methyl]adamantane-1-carbohydrazide —— C25H28N2O2
(5S,7R)-3-(4-methylphenyl)-N'-[(6-oxocyclohexa-2,4-dien-1-ylidene)methyl]adamantane-1-carbohydrazide
—— [(5S)-2,7-diazaspiro[4.5]decan-7-yl]-(5-phenyl-1H-pyrrol-2-yl)methanone —— C19H23N3O
[(5S)-2,7-diazaspiro[4.5]decan-7-yl]-(5-phenyl-1H-pyrrol-2-yl)methanone
—— 5-benzyl-N-[(3R)-pyrrolidin-3-yl]-4,6,7,8-tetrahydropyrazolo[1,5-a][1,4]diazepine-2-carboxamide —— C19H25N5O
5-benzyl-N-[(3R)-pyrrolidin-3-yl]-4,6,7,8-tetrahydropyrazolo[1,5-a][1,4]diazepine-2-carboxamide
—— (5R)-5-(7-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)-1,2,5,6-tetrahydropyrazolo[4,3-g]quinolin-7-one —— C20H19N3O4
(5R)-5-(7-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)-1,2,5,6-tetrahydropyrazolo[4,3-g]quinolin-7-one
—— 5-chloro-N'-[(1E)-1-(4-ethylphenyl)ethylidene]-3-methyl-1H-indole-2-carbohydrazide —— C20H20ClN3O
5-chloro-N'-[(1E)-1-(4-ethylphenyl)ethylidene]-3-methyl-1H-indole-2-carbohydrazide
—— 5-(4-methylphenyl)-N-[[(3R)-1-methylpyrrolidin-3-yl]methyl]furan-2-carboxamide —— C18H22N2O2
5-(4-methylphenyl)-N-[[(3R)-1-methylpyrrolidin-3-yl]methyl]furan-2-carboxamide
—— 5-[(4-ethylpiperazin-1-yl)methyl]-N-methyl-N-[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]-1,2-oxazole-3-carboxamide —— C22H30N4O2
5-[(4-ethylpiperazin-1-yl)methyl]-N-methyl-N-[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]-1,2-oxazole-3-carboxamide
—— (5S)-1-ethyl-5-[4-(3-methoxyphenyl)piperazin-1-yl]-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C21H28N4O3
(5S)-1-ethyl-5-[4-(3-methoxyphenyl)piperazin-1-yl]-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— (5S,7R)-3-(dimethylamino)adamantane-1-thiol —— C12H21NS
(5S,7R)-3-(dimethylamino)adamantane-1-thiol
—— (5S,7R)-3-(4-methylphenyl)-N-[(Z)-(3-nitrophenyl)methylideneamino]adamantane-1-carboxamide —— C25H27N3O3
(5S,7R)-3-(4-methylphenyl)-N-[(Z)-(3-nitrophenyl)methylideneamino]adamantane-1-carboxamide
—— (5S)-5-(7-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)-1,2,5,6-tetrahydropyrazolo[4,3-g]quinolin-7-one —— C20H19N3O4
(5S)-5-(7-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)-1,2,5,6-tetrahydropyrazolo[4,3-g]quinolin-7-one
—— 5-(benzimidazol-1-ylmethyl)-N-[[(3R)-5-oxo-1-propan-2-ylpyrrolidin-3-yl]methyl]-1,2-oxazole-3-carboxamide —— C20H23N5O3
5-(benzimidazol-1-ylmethyl)-N-[[(3R)-5-oxo-1-propan-2-ylpyrrolidin-3-yl]methyl]-1,2-oxazole-3-carboxamide
—— 5-(3-chlorobenzyl)-2-[(4,6-dimethylquinazolin-2-yl)amino]-6-methylpyrimidin-4(3H)-one —— C22H20ClN5O
5-(3-chlorobenzyl)-2-[(4,6-dimethylquinazolin-2-yl)amino]-6-methylpyrimidin-4(3H)-one
—— 5-[[[(2R)-1-(3,5-dimethylpyrazol-1-yl)propan-2-yl]amino]methyl]-1,3-dimethylbenzimidazol-2-one —— C18H25N5O
5-[[[(2R)-1-(3,5-dimethylpyrazol-1-yl)propan-2-yl]amino]methyl]-1,3-dimethylbenzimidazol-2-one
—— 5-(benzimidazol-1-ylmethyl)-N-ethyl-N-[[(3S)-1-methylpyrrolidin-3-yl]methyl]-1H-pyrazole-3-carboxamide —— C20H26N6O
5-(benzimidazol-1-ylmethyl)-N-ethyl-N-[[(3S)-1-methylpyrrolidin-3-yl]methyl]-1H-pyrazole-3-carboxamide
—— 5-(4-methylphenyl)-N-[[(3S)-1-methylpyrrolidin-3-yl]methyl]furan-2-carboxamide —— C18H22N2O2
5-(4-methylphenyl)-N-[[(3S)-1-methylpyrrolidin-3-yl]methyl]furan-2-carboxamide
—— (5-ethylfuran-2-yl)-[(3R)-3-(5-ethyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]methanone —— C16H21N3O3
(5-ethylfuran-2-yl)-[(3R)-3-(5-ethyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]methanone
—— 5-[(4-ethylpiperazin-1-yl)methyl]-N-methyl-N-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]-1,2-oxazole-3-carboxamide —— C22H30N4O2
5-[(4-ethylpiperazin-1-yl)methyl]-N-methyl-N-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]-1,2-oxazole-3-carboxamide
—— (5-ethylfuran-2-yl)-[(3S)-3-(5-ethyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]methanone —— C16H21N3O3
(5-ethylfuran-2-yl)-[(3S)-3-(5-ethyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]methanone
—— 5-(benzimidazol-1-ylmethyl)-N-ethyl-N-[[(3R)-1-methylpyrrolidin-3-yl]methyl]-1H-pyrazole-3-carboxamide —— C20H26N6O
5-(benzimidazol-1-ylmethyl)-N-ethyl-N-[[(3R)-1-methylpyrrolidin-3-yl]methyl]-1H-pyrazole-3-carboxamide
—— 5-(benzimidazol-1-ylmethyl)-N-[[(3S)-5-oxo-1-propan-2-ylpyrrolidin-3-yl]methyl]-1,2-oxazole-3-carboxamide —— C20H23N5O3
5-(benzimidazol-1-ylmethyl)-N-[[(3S)-5-oxo-1-propan-2-ylpyrrolidin-3-yl]methyl]-1,2-oxazole-3-carboxamide
—— (5S,7R)-N-[(Z)-furan-2-ylmethylideneamino]-3-(4-methylphenyl)adamantane-1-carboxamide —— C23H26N2O2
(5S,7R)-N-[(Z)-furan-2-ylmethylideneamino]-3-(4-methylphenyl)adamantane-1-carboxamide
—— 5-[(4-hydroxypiperidin-1-yl)methyl]-N-[(2S)-1-thiophen-3-ylpropan-2-yl]-1,2-oxazole-3-carboxamide —— C17H23N3O3S
5-[(4-hydroxypiperidin-1-yl)methyl]-N-[(2S)-1-thiophen-3-ylpropan-2-yl]-1,2-oxazole-3-carboxamide
—— (5S)-7-(5-chloropyridin-2-yl)-2-methyl-2,7-diazaspiro[4.5]decane —— C14H20ClN3
(5S)-7-(5-chloropyridin-2-yl)-2-methyl-2,7-diazaspiro[4.5]decane
—— (5R)-7-(5-chloropyridin-2-yl)-2-methyl-2,7-diazaspiro[4.5]decane —— C14H20ClN3
(5R)-7-(5-chloropyridin-2-yl)-2-methyl-2,7-diazaspiro[4.5]decane
—— (5R)-3-[(3-benzylsulfanyl-1H-1,2,4-triazol-5-yl)amino]-5-phenylcyclohex-2-en-1-one —— C21H20N4OS
(5R)-3-[(3-benzylsulfanyl-1H-1,2,4-triazol-5-yl)amino]-5-phenylcyclohex-2-en-1-one
—— (5R)-2-[(1-propan-2-ylbenzimidazol-2-yl)methyl]-2,9-diazaspiro[4.5]decane —— C19H28N4
(5R)-2-[(1-propan-2-ylbenzimidazol-2-yl)methyl]-2,9-diazaspiro[4.5]decane
—— (5R)-3-ethyl-5-nitroso-2-sulfanylidene-1,3-thiazolidin-4-one —— C5H6N2O2S2
(5R)-3-ethyl-5-nitroso-2-sulfanylidene-1,3-thiazolidin-4-one
—— 5-[(4-hydroxypiperidin-1-yl)methyl]-N-[(2R)-1-thiophen-3-ylpropan-2-yl]-1,2-oxazole-3-carboxamide —— C17H23N3O3S
5-[(4-hydroxypiperidin-1-yl)methyl]-N-[(2R)-1-thiophen-3-ylpropan-2-yl]-1,2-oxazole-3-carboxamide
—— (5S)-2-[(1-propan-2-ylbenzimidazol-2-yl)methyl]-2,9-diazaspiro[4.5]decane —— C19H28N4
(5S)-2-[(1-propan-2-ylbenzimidazol-2-yl)methyl]-2,9-diazaspiro[4.5]decane
—— 5-[(4-benzylpiperidin-1-yl)methyl]-N-[[(2S)-1-ethylpyrrolidin-2-yl]methyl]-1,2-oxazole-3-carboxamide —— C24H34N4O2
5-[(4-benzylpiperidin-1-yl)methyl]-N-[[(2S)-1-ethylpyrrolidin-2-yl]methyl]-1,2-oxazole-3-carboxamide
—— 5-[(2-chloro-4-methoxyphenoxy)methyl]-N-[(2R)-2,3-dihydroxypropyl]-1H-pyrazole-3-carboxamide —— C15H18ClN3O5
5-[(2-chloro-4-methoxyphenoxy)methyl]-N-[(2R)-2,3-dihydroxypropyl]-1H-pyrazole-3-carboxamide
—— (5S)-5-[4-hydroxy-4-(pyrrolidin-1-ylmethyl)piperidin-1-yl]-1-prop-2-enyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C21H32N4O3
(5S)-5-[4-hydroxy-4-(pyrrolidin-1-ylmethyl)piperidin-1-yl]-1-prop-2-enyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— (5S,7R)-3-(4-methylphenyl)-N'-[(4-oxocyclohexa-2,5-dien-1-ylidene)methyl]adamantane-1-carbohydrazide —— C25H28N2O2
(5S,7R)-3-(4-methylphenyl)-N'-[(4-oxocyclohexa-2,5-dien-1-ylidene)methyl]adamantane-1-carbohydrazide
—— 5-(Furan-2-ylmethyl)-1,3-diphenyl-1,3,5-triazinane-2-thione —— C20H19N3OS
5-(Furan-2-ylmethyl)-1,3-diphenyl-1,3,5-triazinane-2-thione
—— 5-cyclopropyl-N-[(3S)-1-(furan-2-carbonyl)piperidin-3-yl]-1H-pyrazole-3-carboxamide —— C17H20N4O3
5-cyclopropyl-N-[(3S)-1-(furan-2-carbonyl)piperidin-3-yl]-1H-pyrazole-3-carboxamide