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—— (5R)-3-(2,5-difluorophenyl)-N-[3-(4-methylpyrazol-1-yl)propyl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C17H18F2N4O2
(5R)-3-(2,5-difluorophenyl)-N-[3-(4-methylpyrazol-1-yl)propyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— 5-[(R)-1,4-dioxa-8-azaspiro[4.5]decan-8-yl-(2-methoxyphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C20H24N4O4S
5-[(R)-1,4-dioxa-8-azaspiro[4.5]decan-8-yl-(2-methoxyphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-[(3S,5R)-3,5-dimethylpiperidin-1-yl]-(2-methylphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C20H26N4OS
5-[(S)-[(3S,5R)-3,5-dimethylpiperidin-1-yl]-(2-methylphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-(2,5-dimethoxyphenyl)-[(3S,5R)-3,5-dimethylpiperidin-1-ium-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C21H29N4O3S+
5-[(R)-(2,5-dimethoxyphenyl)-[(3S,5R)-3,5-dimethylpiperidin-1-ium-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-(2,4-dimethoxyphenyl)-[(3S,5R)-3,5-dimethylpiperidin-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C21H28N4O3S
5-[(R)-(2,4-dimethoxyphenyl)-[(3S,5R)-3,5-dimethylpiperidin-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-[(2S,6R)-2,6-dimethylmorpholin-4-yl]-(2-methoxyphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C19H24N4O3S
5-[(R)-[(2S,6R)-2,6-dimethylmorpholin-4-yl]-(2-methoxyphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-bromo-N-[[(2R)-oxolan-2-yl]methyl]-1H-indazole-3-carboxamide —— C13H14BrN3O2
5-bromo-N-[[(2R)-oxolan-2-yl]methyl]-1H-indazole-3-carboxamide
—— 5-[(S)-(2,5-dimethoxyphenyl)-[(3S)-3-methylpiperidin-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C20H26N4O3S
5-[(S)-(2,5-dimethoxyphenyl)-[(3S)-3-methylpiperidin-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— [(5S)-2-morpholin-4-yl-4,5-dihydro-1,3-thiazol-5-yl]methyl pyrrolidine-1-carbodithioate —— C13H21N3OS3
[(5S)-2-morpholin-4-yl-4,5-dihydro-1,3-thiazol-5-yl]methyl pyrrolidine-1-carbodithioate
—— 5-[(S)-1,4-dioxa-8-azoniaspiro[4.5]decan-8-yl-(2-methylphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C20H25N4O3S+
5-[(S)-1,4-dioxa-8-azoniaspiro[4.5]decan-8-yl-(2-methylphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-(3-methylthiophen-2-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C18H24N4OS2
5-[(R)-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-(3-methylthiophen-2-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-(2,4-dimethoxyphenyl)-(4-methylpiperazin-1-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C19H25N5O3S
5-[(R)-(2,4-dimethoxyphenyl)-(4-methylpiperazin-1-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-[(3S,5R)-3,5-dimethylpiperidin-1-ium-1-yl]-(3-methylthiophen-2-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C18H25N4OS2+
5-[(S)-[(3S,5R)-3,5-dimethylpiperidin-1-ium-1-yl]-(3-methylthiophen-2-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— (5R)-N-[(3R)-3-cyanothiolan-3-yl]-3-(2,5-difluorophenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide —— C15H13F2N3O2S
(5R)-N-[(3R)-3-cyanothiolan-3-yl]-3-(2,5-difluorophenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
—— 5-[(S)-(2,5-dimethoxyphenyl)-morpholin-4-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C18H22N4O4S
5-[(S)-(2,5-dimethoxyphenyl)-morpholin-4-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-(2-methoxyphenyl)-morpholin-4-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C17H20N4O3S
5-[(S)-(2-methoxyphenyl)-morpholin-4-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-(2-methoxyphenyl)-(4-methylpiperidin-1-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C19H24N4O2S
5-[(R)-(2-methoxyphenyl)-(4-methylpiperidin-1-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-(2,5-dimethoxyphenyl)-[(3S)-3-methylpiperidin-1-ium-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C20H27N4O3S+
5-[(R)-(2,5-dimethoxyphenyl)-[(3S)-3-methylpiperidin-1-ium-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-(2-methylphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C20H26N4OS
5-[(R)-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-(2-methylphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— (5S)-N-[(3R)-3-cyanothiolan-3-yl]-3-(2,5-difluorophenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide —— C15H13F2N3O2S
(5S)-N-[(3R)-3-cyanothiolan-3-yl]-3-(2,5-difluorophenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
—— 5-[(R)-(2,5-dimethoxyphenyl)-piperidin-1-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C19H24N4O3S
5-[(R)-(2,5-dimethoxyphenyl)-piperidin-1-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[[(S)-[1-(3-fluorophenyl)pyrazol-3-yl]methylsulfinyl]methyl]-3-propan-2-yl-1,2,4-oxadiazole —— C16H17FN4O2S
5-[[(S)-[1-(3-fluorophenyl)pyrazol-3-yl]methylsulfinyl]methyl]-3-propan-2-yl-1,2,4-oxadiazole
—— 5-[[(R)-[1-(3-fluorophenyl)pyrazol-3-yl]methylsulfinyl]methyl]-3-propan-2-yl-1,2,4-oxadiazole —— C16H17FN4O2S
5-[[(R)-[1-(3-fluorophenyl)pyrazol-3-yl]methylsulfinyl]methyl]-3-propan-2-yl-1,2,4-oxadiazole
—— 5-[(S)-(2,4-dimethoxyphenyl)-pyrrolidin-1-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C18H22N4O3S
5-[(S)-(2,4-dimethoxyphenyl)-pyrrolidin-1-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-(2-methoxyphenyl)-pyrrolidin-1-ium-1-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C17H21N4O2S+
5-[(S)-(2-methoxyphenyl)-pyrrolidin-1-ium-1-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-(2,4-dimethoxyphenyl)-[(3S,5R)-3,5-dimethylpiperidin-1-ium-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C21H29N4O3S+
5-[(R)-(2,4-dimethoxyphenyl)-[(3S,5R)-3,5-dimethylpiperidin-1-ium-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-(2,4-dimethoxyphenyl)-(4-methylpiperidin-1-ium-1-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C20H27N4O3S+
5-[(S)-(2,4-dimethoxyphenyl)-(4-methylpiperidin-1-ium-1-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-(2,4-dimethoxyphenyl)-piperidin-1-ium-1-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C19H25N4O3S+
5-[(R)-(2,4-dimethoxyphenyl)-piperidin-1-ium-1-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-[4-(2-hydroxyethyl)piperazine-1,4-diium-1-yl]-(2-methylphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C19H27N5O2S+2
5-[(R)-[4-(2-hydroxyethyl)piperazine-1,4-diium-1-yl]-(2-methylphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-(2,5-dimethoxyphenyl)-(4-methylpiperidin-1-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C20H26N4O3S
5-[(S)-(2,5-dimethoxyphenyl)-(4-methylpiperidin-1-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-(2-methoxyphenyl)-piperidin-1-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C18H22N4O2S
5-[(R)-(2-methoxyphenyl)-piperidin-1-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-[(2S,6R)-2,6-dimethylmorpholin-4-ium-4-yl]-(2-methoxyphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C19H25N4O3S+
5-[(R)-[(2S,6R)-2,6-dimethylmorpholin-4-ium-4-yl]-(2-methoxyphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-(2,4-dimethoxyphenyl)-(4-methylpiperidin-1-ium-1-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C20H27N4O3S+
5-[(R)-(2,4-dimethoxyphenyl)-(4-methylpiperidin-1-ium-1-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-(2,5-dimethoxyphenyl)-piperidin-1-ium-1-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C19H25N4O3S+
5-[(S)-(2,5-dimethoxyphenyl)-piperidin-1-ium-1-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-(2-methoxyphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C20H26N4O2S
5-[(S)-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-(2-methoxyphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-(4-ethylpiperazine-1,4-diium-1-yl)-(3-methylthiophen-2-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C17H25N5OS2+2
5-[(S)-(4-ethylpiperazine-1,4-diium-1-yl)-(3-methylthiophen-2-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-[(3S,5S)-3,5-dimethylpiperidin-1-ium-1-yl]-(3-methylthiophen-2-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C18H25N4OS2+
5-[(R)-[(3S,5S)-3,5-dimethylpiperidin-1-ium-1-yl]-(3-methylthiophen-2-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-[(3S,5S)-3,5-dimethylpiperidin-1-ium-1-yl]-(2-methoxyphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C20H27N4O2S+
5-[(R)-[(3S,5S)-3,5-dimethylpiperidin-1-ium-1-yl]-(2-methoxyphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-(2,4-dimethoxyphenyl)-(4-methylpiperazine-1,4-diium-1-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C19H27N5O3S+2
5-[(S)-(2,4-dimethoxyphenyl)-(4-methylpiperazine-1,4-diium-1-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-(2,5-dimethoxyphenyl)-[(3S,5S)-3,5-dimethylpiperidin-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C21H28N4O3S
5-[(R)-(2,5-dimethoxyphenyl)-[(3S,5S)-3,5-dimethylpiperidin-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-[(3S,5S)-3,5-dimethylpiperidin-1-ium-1-yl]-(3-methylthiophen-2-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C18H25N4OS2+
5-[(S)-[(3S,5S)-3,5-dimethylpiperidin-1-ium-1-yl]-(3-methylthiophen-2-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-(2,5-dimethoxyphenyl)-piperidin-1-ium-1-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C19H25N4O3S+
5-[(R)-(2,5-dimethoxyphenyl)-piperidin-1-ium-1-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-(2-methoxyphenyl)-[(3S)-3-methylpiperidin-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C19H24N4O2S
5-[(S)-(2-methoxyphenyl)-[(3S)-3-methylpiperidin-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-(2,5-dimethoxyphenyl)-[(3S,5S)-3,5-dimethylpiperidin-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C21H28N4O3S
5-[(S)-(2,5-dimethoxyphenyl)-[(3S,5S)-3,5-dimethylpiperidin-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-(2,5-dimethoxyphenyl)-morpholin-4-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C18H22N4O4S
5-[(R)-(2,5-dimethoxyphenyl)-morpholin-4-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-(2,4-dimethoxyphenyl)-[(3S)-3-methylpiperidin-1-ium-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C20H27N4O3S+
5-[(R)-(2,4-dimethoxyphenyl)-[(3S)-3-methylpiperidin-1-ium-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-(2,5-dimethoxyphenyl)-[(2R,6R)-2,6-dimethylmorpholin-4-ium-4-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C20H27N4O4S+
5-[(R)-(2,5-dimethoxyphenyl)-[(2R,6R)-2,6-dimethylmorpholin-4-ium-4-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-(2,4-dimethoxyphenyl)-(4-ethylpiperazine-1,4-diium-1-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C20H29N5O3S+2
5-[(R)-(2,4-dimethoxyphenyl)-(4-ethylpiperazine-1,4-diium-1-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-(2,5-dimethoxyphenyl)-(4-methylpiperazin-1-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C19H25N5O3S
5-[(S)-(2,5-dimethoxyphenyl)-(4-methylpiperazin-1-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-[4-(2-hydroxyethyl)piperazine-1,4-diium-1-yl]-(3-methylthiophen-2-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C17H25N5O2S2+2
5-[(R)-[4-(2-hydroxyethyl)piperazine-1,4-diium-1-yl]-(3-methylthiophen-2-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol