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—— 5,5-dioxo-N-[(2R)-2-phenylpropyl]-4H-[1,2,4]triazolo[5,1-c][1,2,4]benzothiadiazine-2-carboxamide —— C18H17N5O3S
5,5-dioxo-N-[(2R)-2-phenylpropyl]-4H-[1,2,4]triazolo[5,1-c][1,2,4]benzothiadiazine-2-carboxamide
—— 5-methyl-3-[[(2S)-2-(1,2,4-triazol-1-ylmethyl)pyrrolidin-1-yl]methyl]-1,2,4-oxadiazole —— C11H16N6O
5-methyl-3-[[(2S)-2-(1,2,4-triazol-1-ylmethyl)pyrrolidin-1-yl]methyl]-1,2,4-oxadiazole
—— 5-methyl-3-[[(2R)-2-(1,2,4-triazol-1-ylmethyl)pyrrolidin-1-yl]methyl]-1,2,4-oxadiazole —— C11H16N6O
5-methyl-3-[[(2R)-2-(1,2,4-triazol-1-ylmethyl)pyrrolidin-1-yl]methyl]-1,2,4-oxadiazole
—— 5-(4-methylphenyl)-3-[[(3S)-3-(1,2,4-triazol-1-ylmethyl)piperidin-1-yl]methyl]-1,2,4-oxadiazole —— C18H22N6O
5-(4-methylphenyl)-3-[[(3S)-3-(1,2,4-triazol-1-ylmethyl)piperidin-1-yl]methyl]-1,2,4-oxadiazole
—— 5-[(1R)-1-[4-[[(2S)-oxan-2-yl]methyl]piperazin-1-yl]ethyl]-3-propan-2-yl-1,2,4-oxadiazole —— C17H30N4O2
5-[(1R)-1-[4-[[(2S)-oxan-2-yl]methyl]piperazin-1-yl]ethyl]-3-propan-2-yl-1,2,4-oxadiazole
—— 5-(4-methylphenyl)-3-[[(3R)-3-(1,2,4-triazol-1-ylmethyl)piperidin-1-yl]methyl]-1,2,4-oxadiazole —— C18H22N6O
5-(4-methylphenyl)-3-[[(3R)-3-(1,2,4-triazol-1-ylmethyl)piperidin-1-yl]methyl]-1,2,4-oxadiazole
—— 5,5-dioxo-N-[(2S)-2-phenylpropyl]-4H-[1,2,4]triazolo[5,1-c][1,2,4]benzothiadiazine-2-carboxamide —— C18H17N5O3S
5,5-dioxo-N-[(2S)-2-phenylpropyl]-4H-[1,2,4]triazolo[5,1-c][1,2,4]benzothiadiazine-2-carboxamide
—— 5-[(1S)-1-[4-[[(2S)-oxan-2-yl]methyl]piperazin-1-yl]ethyl]-3-propan-2-yl-1,2,4-oxadiazole —— C17H30N4O2
5-[(1S)-1-[4-[[(2S)-oxan-2-yl]methyl]piperazin-1-yl]ethyl]-3-propan-2-yl-1,2,4-oxadiazole
—— 5-[(1R)-1-(3-propan-2-yl-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl)ethyl]-3-thiophen-2-yl-1,2,4-oxadiazole —— C16H20N6OS
5-[(1R)-1-(3-propan-2-yl-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl)ethyl]-3-thiophen-2-yl-1,2,4-oxadiazole
—— 5-phenyl-2-[[(3R)-3-(1,2,4-triazol-1-ylmethyl)piperidin-1-yl]methyl]-1,3-oxazole —— C18H21N5O
5-phenyl-2-[[(3R)-3-(1,2,4-triazol-1-ylmethyl)piperidin-1-yl]methyl]-1,3-oxazole
—— 5-[(1S)-1-[4-[[(2R)-oxan-2-yl]methyl]piperazin-1-yl]ethyl]-3-propan-2-yl-1,2,4-oxadiazole —— C17H30N4O2
5-[(1S)-1-[4-[[(2R)-oxan-2-yl]methyl]piperazin-1-yl]ethyl]-3-propan-2-yl-1,2,4-oxadiazole
—— 5-[(1R)-1-[4-[[(2R)-oxan-2-yl]methyl]piperazin-1-yl]ethyl]-3-propan-2-yl-1,2,4-oxadiazole —— C17H30N4O2
5-[(1R)-1-[4-[[(2R)-oxan-2-yl]methyl]piperazin-1-yl]ethyl]-3-propan-2-yl-1,2,4-oxadiazole
—— (5-chloro-2-fluorophenyl)-[4-[(2R)-2-hydroxybutyl]piperazin-1-yl]methanone —— C15H20ClFN2O2
(5-chloro-2-fluorophenyl)-[4-[(2R)-2-hydroxybutyl]piperazin-1-yl]methanone
—— 5-phenyl-2-[[(3S)-3-(1,2,4-triazol-1-ylmethyl)piperidin-1-yl]methyl]-1,3-oxazole —— C18H21N5O
5-phenyl-2-[[(3S)-3-(1,2,4-triazol-1-ylmethyl)piperidin-1-yl]methyl]-1,3-oxazole
—— (5-chloro-2-fluorophenyl)-[4-[(2S)-2-hydroxybutyl]piperazin-1-yl]methanone —— C15H20ClFN2O2
(5-chloro-2-fluorophenyl)-[4-[(2S)-2-hydroxybutyl]piperazin-1-yl]methanone
—— 5,6-dimethoxy-N-(6-nitrobenzo[d]thiazol-2-yl)benzo[d]thiazol-2-amine —— C16H12N4O4S2
5,6-dimethoxy-N-(6-nitrobenzo[d]thiazol-2-yl)benzo[d]thiazol-2-amine
—— 5,6-dimethyl-3-[[(3R)-1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-3-yl]amino]pyridazine-4-carbonitrile —— C16H21N7O
5,6-dimethyl-3-[[(3R)-1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-3-yl]amino]pyridazine-4-carbonitrile
—— 5,6-dimethoxy-N-(6-methoxy-1,3-benzothiazol-2-yl)-1,3-benzothiazol-2-amine —— C17H15N3O3S2
5,6-dimethoxy-N-(6-methoxy-1,3-benzothiazol-2-yl)-1,3-benzothiazol-2-amine
—— 5-chloro-N-[3-(dimethylamino)propyl]-N-(4,6-dimethyl-1,3-benzothiazol-2-yl)thiophene-2-carboxamide —— C19H22ClN3OS2
5-chloro-N-[3-(dimethylamino)propyl]-N-(4,6-dimethyl-1,3-benzothiazol-2-yl)thiophene-2-carboxamide
—— 5-methyl-N-[(S)-(5-methyl-1H-1,2,4-triazol-3-yl)-phenylmethyl]furan-2-carboxamide —— C16H16N4O2
5-methyl-N-[(S)-(5-methyl-1H-1,2,4-triazol-3-yl)-phenylmethyl]furan-2-carboxamide
—— 5-methyl-N-[(3S)-1-pyridazin-3-ylpiperidin-3-yl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine —— C15H18N8
5-methyl-N-[(3S)-1-pyridazin-3-ylpiperidin-3-yl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine
—— 5-methoxy-N-(4-methoxybenzo[d]thiazol-2-yl)benzo[d]thiazol-2-amine —— C16H13N3O2S2
5-methoxy-N-(4-methoxybenzo[d]thiazol-2-yl)benzo[d]thiazol-2-amine
—— (5S)-5-[(3-chlorophenyl)methylsulfanylmethyl]-1,3-oxazolidin-2-one —— C11H12ClNO2S
(5S)-5-[(3-chlorophenyl)methylsulfanylmethyl]-1,3-oxazolidin-2-one
—— (5-tert-butyl-1H-pyrazol-3-yl)-[4-[(2R)-2-hydroxypropyl]piperazin-1-yl]methanone —— C15H26N4O2
(5-tert-butyl-1H-pyrazol-3-yl)-[4-[(2R)-2-hydroxypropyl]piperazin-1-yl]methanone
—— (5-fluoro-1-benzothiophen-2-yl)-[(2S)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone —— C17H16FN3OS
(5-fluoro-1-benzothiophen-2-yl)-[(2S)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone
—— 5-chloro-N-[3-(dimethylamino)propyl]-N-(4,5-dimethyl-1,3-benzothiazol-2-yl)thiophene-2-carboxamide —— C19H22ClN3OS2
5-chloro-N-[3-(dimethylamino)propyl]-N-(4,5-dimethyl-1,3-benzothiazol-2-yl)thiophene-2-carboxamide
—— [(5R)-5-methyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-(3-propan-2-yl-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl)methanone —— C18H24N4OS
[(5R)-5-methyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-(3-propan-2-yl-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl)methanone
—— 5,6-dimethyl-3-[[(3S)-1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-3-yl]amino]pyridazine-4-carbonitrile —— C16H21N7O
5,6-dimethyl-3-[[(3S)-1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-3-yl]amino]pyridazine-4-carbonitrile
—— [(5S)-5-methyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-(3-propan-2-yl-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl)methanone —— C18H24N4OS
[(5S)-5-methyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-(3-propan-2-yl-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl)methanone
—— 5-methyl-N-[(2S)-3-methylbutan-2-yl]-1-(2-methyl-3,4-dihydro-1H-isoquinolin-5-yl)triazole-4-carboxamide —— C19H27N5O
5-methyl-N-[(2S)-3-methylbutan-2-yl]-1-(2-methyl-3,4-dihydro-1H-isoquinolin-5-yl)triazole-4-carboxamide
—— 5-methyl-N-[(2R)-3-methylbutan-2-yl]-1-(2-methyl-3,4-dihydro-1H-isoquinolin-5-yl)triazole-4-carboxamide —— C19H27N5O
5-methyl-N-[(2R)-3-methylbutan-2-yl]-1-(2-methyl-3,4-dihydro-1H-isoquinolin-5-yl)triazole-4-carboxamide
—— (5R)-5-[(3-chlorophenyl)methylsulfanylmethyl]-1,3-oxazolidin-2-one —— C11H12ClNO2S
(5R)-5-[(3-chlorophenyl)methylsulfanylmethyl]-1,3-oxazolidin-2-one
—— 5,6-dimethoxy-N-(6-methylbenzo[d]thiazol-2-yl)benzo[d]thiazol-2-amine —— C17H15N3O2S2
5,6-dimethoxy-N-(6-methylbenzo[d]thiazol-2-yl)benzo[d]thiazol-2-amine
—— 5-methoxy-N-[(6S)-6-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]-1,3-benzothiazol-2-amine —— C16H17N3OS2
5-methoxy-N-[(6S)-6-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]-1,3-benzothiazol-2-amine
—— 5,5-dioxo-N-[(1R)-1-pyridin-2-ylethyl]-4H-[1,2,4]triazolo[5,1-c][1,2,4]benzothiadiazine-2-carboxamide —— C16H14N6O3S
5,5-dioxo-N-[(1R)-1-pyridin-2-ylethyl]-4H-[1,2,4]triazolo[5,1-c][1,2,4]benzothiadiazine-2-carboxamide
—— 5-tert-butyl-2-[[(3S)-4-(2-ethoxyethyl)-3-methylpiperazin-1-yl]methyl]-1,3-oxazole —— C17H31N3O2
5-tert-butyl-2-[[(3S)-4-(2-ethoxyethyl)-3-methylpiperazin-1-yl]methyl]-1,3-oxazole
—— 5-chloro-N-(4-chloro-1,3-benzothiazol-2-yl)-N-[3-(dimethylamino)propyl]thiophene-2-carboxamide —— C17H17Cl2N3OS2
5-chloro-N-(4-chloro-1,3-benzothiazol-2-yl)-N-[3-(dimethylamino)propyl]thiophene-2-carboxamide
—— 5-methyl-N-[(3R)-1-pyridazin-3-ylpiperidin-3-yl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine —— C15H18N8
5-methyl-N-[(3R)-1-pyridazin-3-ylpiperidin-3-yl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine
—— 5-methyl-N-[(R)-(5-methyl-1H-1,2,4-triazol-3-yl)-phenylmethyl]furan-2-carboxamide —— C16H16N4O2
5-methyl-N-[(R)-(5-methyl-1H-1,2,4-triazol-3-yl)-phenylmethyl]furan-2-carboxamide
—— (5-fluoro-1-benzothiophen-2-yl)-[(2R)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone —— C17H16FN3OS
(5-fluoro-1-benzothiophen-2-yl)-[(2R)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone
—— [5-(5-methylfuran-2-yl)-1H-pyrazol-3-yl]-[(3S)-3-(2-methylimidazol-1-yl)piperidin-1-yl]methanone —— C18H21N5O2
[5-(5-methylfuran-2-yl)-1H-pyrazol-3-yl]-[(3S)-3-(2-methylimidazol-1-yl)piperidin-1-yl]methanone
—— 5-chloro-N-(6-chloro-1,3-benzothiazol-2-yl)-N-[3-(dimethylamino)propyl]thiophene-2-carboxamide —— C17H17Cl2N3OS2
5-chloro-N-(6-chloro-1,3-benzothiazol-2-yl)-N-[3-(dimethylamino)propyl]thiophene-2-carboxamide
—— 5-methoxy-N-(6-nitrobenzo[d]thiazol-2-yl)benzo[d]thiazol-2-amine —— C15H10N4O3S2
5-methoxy-N-(6-nitrobenzo[d]thiazol-2-yl)benzo[d]thiazol-2-amine
—— 5,5-dioxo-N-[(1S)-1-pyridin-2-ylethyl]-4H-[1,2,4]triazolo[5,1-c][1,2,4]benzothiadiazine-2-carboxamide —— C16H14N6O3S
5,5-dioxo-N-[(1S)-1-pyridin-2-ylethyl]-4H-[1,2,4]triazolo[5,1-c][1,2,4]benzothiadiazine-2-carboxamide
—— (5-tert-butyl-1H-pyrazol-3-yl)-[4-[(2S)-2-hydroxypropyl]piperazin-1-yl]methanone —— C15H26N4O2
(5-tert-butyl-1H-pyrazol-3-yl)-[4-[(2S)-2-hydroxypropyl]piperazin-1-yl]methanone
—— 5-fluoro-2-[[(3S)-3-(1,2,4-triazol-1-ylmethyl)piperidin-1-yl]methyl]benzonitrile —— C16H18FN5
5-fluoro-2-[[(3S)-3-(1,2,4-triazol-1-ylmethyl)piperidin-1-yl]methyl]benzonitrile
—— [5-(2-fluorophenyl)furan-2-yl]-[(2R)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone —— C19H18FN3O2
[5-(2-fluorophenyl)furan-2-yl]-[(2R)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone
—— [5-(2-fluorophenyl)furan-2-yl]-[(2S)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone —— C19H18FN3O2
[5-(2-fluorophenyl)furan-2-yl]-[(2S)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone
—— 5,7-dimethyl-6-[2-[(2S)-2-methylthiomorpholin-4-yl]-2-oxoethyl]-1H-pyrazolo[1,5-a]pyrimidin-2-one —— C15H20N4O2S
5,7-dimethyl-6-[2-[(2S)-2-methylthiomorpholin-4-yl]-2-oxoethyl]-1H-pyrazolo[1,5-a]pyrimidin-2-one
—— 5-[(2S)-2-[(2R)-1-ethylpyrrolidin-2-yl]pyrrolidine-1-carbonyl]thiophene-2-carboxamide —— C16H23N3O2S
5-[(2S)-2-[(2R)-1-ethylpyrrolidin-2-yl]pyrrolidine-1-carbonyl]thiophene-2-carboxamide