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中文名称 英文名称 CAS号 化学式 结构式图片
—— (5R)-5-morpholin-4-yl-1-propyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C15H23N3O3
(5R)-5-morpholin-4-yl-1-propyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— 5-[(3S)-3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl]-1H-pyrazin-2-one —— C20H21N5O2
5-[(3S)-3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl]-1H-pyrazin-2-one
—— 5-methyl-3-[[(3R)-3-(1H-pyrazol-5-yl)piperidin-1-yl]methyl]-1H-indole-2-carboxylic acid —— C19H22N4O2
5-methyl-3-[[(3R)-3-(1H-pyrazol-5-yl)piperidin-1-yl]methyl]-1H-indole-2-carboxylic acid
—— [(5R)-2,7-diazaspiro[4.5]decan-7-yl]-(6-methylpyrazolo[1,5-a]pyrimidin-3-yl)methanone —— C16H21N5O
[(5R)-2,7-diazaspiro[4.5]decan-7-yl]-(6-methylpyrazolo[1,5-a]pyrimidin-3-yl)methanone
—— 5-(3,4-dihydro-1H-isoquinolin-2-ylmethyl)-N-methyl-N-[(1R)-1-(1,2-oxazol-3-yl)ethyl]-1,2-oxazole-3-carboxamide —— C20H22N4O3
5-(3,4-dihydro-1H-isoquinolin-2-ylmethyl)-N-methyl-N-[(1R)-1-(1,2-oxazol-3-yl)ethyl]-1,2-oxazole-3-carboxamide
—— 5-[(2S)-2-(3,4-dihydro-1H-isoquinolin-2-yl)propanoyl]-1-methyl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-3-carboxylic acid —— C20H24N4O3
5-[(2S)-2-(3,4-dihydro-1H-isoquinolin-2-yl)propanoyl]-1-methyl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
—— 5-[[benzyl-[(2-fluorophenyl)methyl]amino]methyl]-N-[(2S)-butan-2-yl]furan-2-carboxamide —— C24H27FN2O2
5-[[benzyl-[(2-fluorophenyl)methyl]amino]methyl]-N-[(2S)-butan-2-yl]furan-2-carboxamide
—— 5-[(2R)-2-aminopropanoyl]-N-(pyridin-2-ylmethyl)-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine-2-carboxamide —— C16H20N6O2
5-[(2R)-2-aminopropanoyl]-N-(pyridin-2-ylmethyl)-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine-2-carboxamide
—— [(5R)-2,7-diazaspiro[4.5]decan-7-yl]-(4-ethylphenyl)methanone —— C17H24N2O
[(5R)-2,7-diazaspiro[4.5]decan-7-yl]-(4-ethylphenyl)methanone
—— (5S)-7-methyl-2-[2-(3-oxopiperazin-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C15H24N4O3
(5S)-7-methyl-2-[2-(3-oxopiperazin-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-(2,2-dimethylpropyl)-2,9-diazaspiro[4.5]decane —— C13H26N2
(5S)-2-(2,2-dimethylpropyl)-2,9-diazaspiro[4.5]decane
—— [5-[[(3S)-3-pyrrolidin-1-ylpiperidin-1-yl]methyl]furan-2-yl]methanol —— C15H24N2O2
[5-[[(3S)-3-pyrrolidin-1-ylpiperidin-1-yl]methyl]furan-2-yl]methanol
—— 5-[[benzyl(methyl)amino]methyl]-N-[(3R)-5-oxo-1-propan-2-ylpyrrolidin-3-yl]-1,2-oxazole-3-carboxamide —— C20H26N4O3
5-[[benzyl(methyl)amino]methyl]-N-[(3R)-5-oxo-1-propan-2-ylpyrrolidin-3-yl]-1,2-oxazole-3-carboxamide
—— 5-(benzimidazol-1-ylmethyl)-N-[(1R)-2-hydroxy-1-pyridin-3-ylethyl]-1H-pyrazole-3-carboxamide —— C19H18N6O2
5-(benzimidazol-1-ylmethyl)-N-[(1R)-2-hydroxy-1-pyridin-3-ylethyl]-1H-pyrazole-3-carboxamide
—— 5,7-Diphenyl-2-pyridin-2-yl-1,3-diazoniatricyclo[3.3.1.13,7]decan-6-one —— C25H25N3O+2
5,7-Diphenyl-2-pyridin-2-yl-1,3-diazoniatricyclo[3.3.1.13,7]decan-6-one
—— 5-chloro-N-(9-ethyl-9H-carbazol-3-yl)-2-methoxybenzamide —— C22H19ClN2O2
5-chloro-N-(9-ethyl-9H-carbazol-3-yl)-2-methoxybenzamide
—— (5R)-N-[2-(4-fluorophenyl)ethyl]-2,9-diazaspiro[4.5]decane-2-carboxamide —— C17H24FN3O
(5R)-N-[2-(4-fluorophenyl)ethyl]-2,9-diazaspiro[4.5]decane-2-carboxamide
—— [5-[[[(2R)-butan-2-yl]-(butylcarbamoyl)amino]methyl]-2-methoxyphenyl] methanesulfonate —— C18H30N2O5S
[5-[[[(2R)-butan-2-yl]-(butylcarbamoyl)amino]methyl]-2-methoxyphenyl] methanesulfonate
—— (5R)-5-(4-methylpiperazin-1-yl)-1-propyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C16H26N4O2
(5R)-5-(4-methylpiperazin-1-yl)-1-propyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— (5S)-N-[2-(4-fluorophenyl)ethyl]-2,9-diazaspiro[4.5]decane-2-carboxamide —— C17H24FN3O
(5S)-N-[2-(4-fluorophenyl)ethyl]-2,9-diazaspiro[4.5]decane-2-carboxamide
—— 5-[2-[4-[(2R)-2-phenylpropyl]triazol-1-yl]ethyl]-2H-tetrazole —— C14H17N7
5-[2-[4-[(2R)-2-phenylpropyl]triazol-1-yl]ethyl]-2H-tetrazole
—— (5-methyl-1,4,6,7-tetrahydropyrazolo[4,3-c]pyridin-3-yl)-[(4S)-spiro[azepane-4,2'-chromene]-1-yl]methanone —— C22H26N4O2
(5-methyl-1,4,6,7-tetrahydropyrazolo[4,3-c]pyridin-3-yl)-[(4S)-spiro[azepane-4,2'-chromene]-1-yl]methanone
—— (5R)-5-(1,3-dihydroisoindol-2-yl)-1-propyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C19H23N3O2
(5R)-5-(1,3-dihydroisoindol-2-yl)-1-propyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— (5-methyl-1H-imidazol-4-yl)-[(3S)-3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl]methanone —— C20H23N5O
(5-methyl-1H-imidazol-4-yl)-[(3S)-3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl]methanone
—— 5-nitro-2-[(2S)-4-oxo-1,2-dihydro-3,1-benzoxazin-2-yl]benzoate —— C15H9N2O6-
5-nitro-2-[(2S)-4-oxo-1,2-dihydro-3,1-benzoxazin-2-yl]benzoate
—— (5S)-5-(1,3-dihydroisoindol-2-yl)-1-propyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C19H23N3O2
(5S)-5-(1,3-dihydroisoindol-2-yl)-1-propyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— 5,7-Diphenyl-2-pyridin-3-yl-1,3-diazoniatricyclo[3.3.1.13,7]decan-6-one —— C25H25N3O+2
5,7-Diphenyl-2-pyridin-3-yl-1,3-diazoniatricyclo[3.3.1.13,7]decan-6-one
—— 5-[(2S)-5-oxopyrrolidine-2-carbonyl]-N-(pyridin-2-ylmethyl)-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine-2-carboxamide —— C18H20N6O3
5-[(2S)-5-oxopyrrolidine-2-carbonyl]-N-(pyridin-2-ylmethyl)-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine-2-carboxamide
—— 5-[(1S)-1-[5-(3,5-dimethylphenyl)-4-phenylimidazol-1-yl]ethyl]-2H-tetrazole —— C20H20N6
5-[(1S)-1-[5-(3,5-dimethylphenyl)-4-phenylimidazol-1-yl]ethyl]-2H-tetrazole
—— 5-nitro-2-[(2S)-4-oxo-1,2-dihydro-3,1-benzoxazin-2-yl]benzoic acid —— C15H10N2O6
5-nitro-2-[(2S)-4-oxo-1,2-dihydro-3,1-benzoxazin-2-yl]benzoic acid
—— 5-[(3R)-3-(1-methyl-5-oxo-4-phenyl-1,2,4-triazol-3-yl)piperidine-1-carbonyl]-1H-pyrazin-2-one —— C19H20N6O3
5-[(3R)-3-(1-methyl-5-oxo-4-phenyl-1,2,4-triazol-3-yl)piperidine-1-carbonyl]-1H-pyrazin-2-one
—— 5-[(2-methoxyphenoxy)methyl]-N-methyl-N-[(3S)-1-methylpyrrolidin-3-yl]-1H-pyrazole-3-carboxamide —— C18H24N4O3
5-[(2-methoxyphenoxy)methyl]-N-methyl-N-[(3S)-1-methylpyrrolidin-3-yl]-1H-pyrazole-3-carboxamide
—— [(5S)-12-methyl-1,4-diazatetracyclo[7.6.1.05,16.010,15]hexadeca-9(16),10(15),11,13-tetraen-4-yl]-(4,5,6,7-tetrahydro-1-benzothiophen-3-yl)methanone —— C24H26N2OS
[(5S)-12-methyl-1,4-diazatetracyclo[7.6.1.05,16.010,15]hexadeca-9(16),10(15),11,13-tetraen-4-yl]-(4,5,6,7-tetrahydro-1-benzothiophen-3-yl)methanone
—— (5-methyl-1H-imidazol-4-yl)-[(3R)-3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl]methanone —— C20H23N5O
(5-methyl-1H-imidazol-4-yl)-[(3R)-3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl]methanone
—— 5-(3,4-dihydro-1H-isoquinolin-2-ylmethyl)-N-methyl-N-[(1S)-1-(1,2-oxazol-3-yl)ethyl]-1,2-oxazole-3-carboxamide —— C20H22N4O3
5-(3,4-dihydro-1H-isoquinolin-2-ylmethyl)-N-methyl-N-[(1S)-1-(1,2-oxazol-3-yl)ethyl]-1,2-oxazole-3-carboxamide
—— (5R)-2-(2,2-dimethylpropyl)-2,9-diazaspiro[4.5]decane —— C13H26N2
(5R)-2-(2,2-dimethylpropyl)-2,9-diazaspiro[4.5]decane
—— (5R)-5-[4-(5-benzyl-1H-pyrazol-3-yl)piperidine-1-carbonyl]pyrrolidin-2-one —— C20H24N4O2
(5R)-5-[4-(5-benzyl-1H-pyrazol-3-yl)piperidine-1-carbonyl]pyrrolidin-2-one
—— (5S)-5-(4-methylpiperazin-1-yl)-1-propyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C16H26N4O2
(5S)-5-(4-methylpiperazin-1-yl)-1-propyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— (5R)-7-methyl-2-[2-(3-oxopiperazin-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C15H24N4O3
(5R)-7-methyl-2-[2-(3-oxopiperazin-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-[[benzyl(methyl)amino]methyl]-N-methyl-N-[(1S)-1-(1,3-thiazol-2-yl)ethyl]-1,2-oxazole-3-carboxamide —— C19H22N4O2S
5-[[benzyl(methyl)amino]methyl]-N-methyl-N-[(1S)-1-(1,3-thiazol-2-yl)ethyl]-1,2-oxazole-3-carboxamide
—— (5R)-1-phenyl-9-(2-phenylethyl)-1,3-diaza-9-azoniaspiro[4.5]decan-4-one —— C21H26N3O+
(5R)-1-phenyl-9-(2-phenylethyl)-1,3-diaza-9-azoniaspiro[4.5]decan-4-one
—— 5-[[benzyl(methyl)amino]methyl]-N-methyl-N-[(1R)-1-(1,3-thiazol-2-yl)ethyl]-1,2-oxazole-3-carboxamide —— C19H22N4O2S
5-[[benzyl(methyl)amino]methyl]-N-methyl-N-[(1R)-1-(1,3-thiazol-2-yl)ethyl]-1,2-oxazole-3-carboxamide
—— (5S)-5-[4-(5-benzyl-1H-pyrazol-3-yl)piperidine-1-carbonyl]pyrrolidin-2-one —— C20H24N4O2
(5S)-5-[4-(5-benzyl-1H-pyrazol-3-yl)piperidine-1-carbonyl]pyrrolidin-2-one
—— (5S)-2-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-2,9-diazaspiro[4.5]decane —— C14H17ClF3N3
(5S)-2-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-2,9-diazaspiro[4.5]decane
—— 5-[(4-benzylpiperidin-1-yl)methyl]-N-[(2S)-2-hydroxybutyl]-1,2-oxazole-3-carboxamide —— C21H29N3O3
5-[(4-benzylpiperidin-1-yl)methyl]-N-[(2S)-2-hydroxybutyl]-1,2-oxazole-3-carboxamide
—— 5-bromo-2-chloro-N-[(1R)-1-(3,4-difluorophenyl)ethyl]-N-methylpyridine-3-carboxamide —— C15H12BrClF2N2O
5-bromo-2-chloro-N-[(1R)-1-(3,4-difluorophenyl)ethyl]-N-methylpyridine-3-carboxamide
—— (5S)-1-phenyl-9-(2-phenylethyl)-1,3-diaza-9-azoniaspiro[4.5]decan-4-one —— C21H26N3O+
(5S)-1-phenyl-9-(2-phenylethyl)-1,3-diaza-9-azoniaspiro[4.5]decan-4-one
—— 5-[(1R)-1-[5-(3,5-dimethylphenyl)-4-phenylimidazol-1-yl]ethyl]-2H-tetrazole —— C20H20N6
5-[(1R)-1-[5-(3,5-dimethylphenyl)-4-phenylimidazol-1-yl]ethyl]-2H-tetrazole
—— (5S)-5-[[4-(3-chlorophenyl)piperazin-1-yl]methyl]-3-methyl-2-sulfanylidene-1,3-thiazolidin-4-one —— C15H18ClN3OS2
(5S)-5-[[4-(3-chlorophenyl)piperazin-1-yl]methyl]-3-methyl-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5S)-5-[2-butoxy-5-(4-methylphenyl)phenyl]-2-methyl-3,5-dihydropyrazolo[1,5-c]quinazoline —— C28H29N3O
(5S)-5-[2-butoxy-5-(4-methylphenyl)phenyl]-2-methyl-3,5-dihydropyrazolo[1,5-c]quinazoline