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—— (5S)-4-[(4-butoxy-2-methylphenyl)-hydroxymethylidene]-1-(2-methoxyethyl)-5-pyridin-4-ylpyrrolidine-2,3-dione —— C24H28N2O5
(5S)-4-[(4-butoxy-2-methylphenyl)-hydroxymethylidene]-1-(2-methoxyethyl)-5-pyridin-4-ylpyrrolidine-2,3-dione
—— (5S,10bS)-2-(4-fluorophenyl)-5-(3-methoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C23H19FN2O2
(5S,10bS)-2-(4-fluorophenyl)-5-(3-methoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— 5-oxo-5-[[(7R)-5-oxo-7-phenyl-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl]amino]pentanoate —— C16H16N5O4-
5-oxo-5-[[(7R)-5-oxo-7-phenyl-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl]amino]pentanoate
—— 5-oxo-5-[[(7S)-5-oxo-7-phenyl-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl]amino]pentanoic acid —— C16H17N5O4
5-oxo-5-[[(7S)-5-oxo-7-phenyl-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl]amino]pentanoic acid
—— 5-oxo-5-[[(7S)-5-oxo-7-phenyl-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl]amino]pentanoate —— C16H16N5O4-
5-oxo-5-[[(7S)-5-oxo-7-phenyl-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl]amino]pentanoate
—— 5-oxo-5-[[(7R)-5-oxo-7-phenyl-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl]amino]pentanoic acid —— C16H17N5O4
5-oxo-5-[[(7R)-5-oxo-7-phenyl-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl]amino]pentanoic acid
—— 5-chloro-N-[3-chloro-4-(4-methylpiperazin-4-ium-1-yl)phenyl]-2-methoxybenzamide —— C19H22Cl2N3O2+
5-chloro-N-[3-chloro-4-(4-methylpiperazin-4-ium-1-yl)phenyl]-2-methoxybenzamide
—— 5-[(1S)-1-[4-[(1R)-1-(2,6-difluorophenyl)ethyl]piperazin-1-yl]ethyl]-3-methyl-1,2,4-oxadiazole —— C17H22F2N4O
5-[(1S)-1-[4-[(1R)-1-(2,6-difluorophenyl)ethyl]piperazin-1-yl]ethyl]-3-methyl-1,2,4-oxadiazole
—— 5-[(1R)-1-[4-(1H-imidazo[4,5-b]pyridin-2-ylmethyl)piperazin-1-yl]ethyl]-3-methyl-1,2,4-oxadiazole —— C16H21N7O
5-[(1R)-1-[4-(1H-imidazo[4,5-b]pyridin-2-ylmethyl)piperazin-1-yl]ethyl]-3-methyl-1,2,4-oxadiazole
—— 5-[(1R)-1-[4-[(1R)-1-(2,6-difluorophenyl)ethyl]piperazin-1-yl]ethyl]-3-methyl-1,2,4-oxadiazole —— C17H22F2N4O
5-[(1R)-1-[4-[(1R)-1-(2,6-difluorophenyl)ethyl]piperazin-1-yl]ethyl]-3-methyl-1,2,4-oxadiazole
—— 5-[(1R)-1-[4-[(1S)-1-(2,6-difluorophenyl)ethyl]piperazin-1-yl]ethyl]-3-methyl-1,2,4-oxadiazole —— C17H22F2N4O
5-[(1R)-1-[4-[(1S)-1-(2,6-difluorophenyl)ethyl]piperazin-1-yl]ethyl]-3-methyl-1,2,4-oxadiazole
—— 5-[(1S)-1-[4-[(1S)-1-(2,6-difluorophenyl)ethyl]piperazin-1-yl]ethyl]-3-methyl-1,2,4-oxadiazole —— C17H22F2N4O
5-[(1S)-1-[4-[(1S)-1-(2,6-difluorophenyl)ethyl]piperazin-1-yl]ethyl]-3-methyl-1,2,4-oxadiazole
—— (5S)-1-butyl-4-[(4-chlorophenyl)-hydroxymethylidene]-5-(4-fluorophenyl)pyrrolidine-2,3-dione —— C21H19ClFNO3
(5S)-1-butyl-4-[(4-chlorophenyl)-hydroxymethylidene]-5-(4-fluorophenyl)pyrrolidine-2,3-dione
—— 5-propyl-N-[(2S,3R)-3-pyrazol-1-ylbutan-2-yl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine —— C15H21N7
5-propyl-N-[(2S,3R)-3-pyrazol-1-ylbutan-2-yl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine
—— 5-propyl-N-[(2S,3S)-3-pyrazol-1-ylbutan-2-yl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine —— C15H21N7
5-propyl-N-[(2S,3S)-3-pyrazol-1-ylbutan-2-yl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine
—— 5-cyclohexyl-N-[(2S)-1-(1,2,4-triazol-1-yl)propan-2-yl]-1H-pyrazole-4-carboxamide —— C15H22N6O
5-cyclohexyl-N-[(2S)-1-(1,2,4-triazol-1-yl)propan-2-yl]-1H-pyrazole-4-carboxamide
—— 5-cyclohexyl-N-[(2R)-1-(1,2,4-triazol-1-yl)propan-2-yl]-1H-pyrazole-4-carboxamide —— C15H22N6O
5-cyclohexyl-N-[(2R)-1-(1,2,4-triazol-1-yl)propan-2-yl]-1H-pyrazole-4-carboxamide
—— 5-propyl-N-[(2R,3S)-3-pyrazol-1-ylbutan-2-yl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine —— C15H21N7
5-propyl-N-[(2R,3S)-3-pyrazol-1-ylbutan-2-yl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine
—— 5-[(1S)-1-[4-(1H-imidazo[4,5-b]pyridin-2-ylmethyl)piperazin-1-yl]ethyl]-3-methyl-1,2,4-oxadiazole —— C16H21N7O
5-[(1S)-1-[4-(1H-imidazo[4,5-b]pyridin-2-ylmethyl)piperazin-1-yl]ethyl]-3-methyl-1,2,4-oxadiazole
—— 5-propyl-N-[(2R,3R)-3-pyrazol-1-ylbutan-2-yl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine —— C15H21N7
5-propyl-N-[(2R,3R)-3-pyrazol-1-ylbutan-2-yl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine
—— (5S)-5-hydroxy-5-(trifluoromethyl)-4H-pyrazole-1-carbothioamide —— C5H6F3N3OS
(5S)-5-hydroxy-5-(trifluoromethyl)-4H-pyrazole-1-carbothioamide
—— 5-[(1S)-1-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]ethyl]-3-methyl-1,2,4-oxadiazole —— C16H19N5OS
5-[(1S)-1-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]ethyl]-3-methyl-1,2,4-oxadiazole
—— 5-[(1R)-1-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]ethyl]-3-methyl-1,2,4-oxadiazole —— C16H19N5OS
5-[(1R)-1-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]ethyl]-3-methyl-1,2,4-oxadiazole
—— (5S,10bR)-2-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-(3-fluorophenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C24H19FN2O3
(5S,10bR)-2-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-(3-fluorophenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5R)-5-(4-fluorospiro[2H-indole-3,1'-cyclopentane]-1-carbonyl)piperidin-2-one —— C18H21FN2O2
(5R)-5-(4-fluorospiro[2H-indole-3,1'-cyclopentane]-1-carbonyl)piperidin-2-one
—— (5S,10bS)-2-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-(3-methoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C25H22N2O4
(5S,10bS)-2-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-(3-methoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5S,10bS)-2-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-(4-ethylphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C26H24N2O3
(5S,10bS)-2-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-(4-ethylphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— 5-methyl-N-(3-morpholin-4-ium-4-ylpropyl)-N-[3-oxo-3-(propan-2-ylamino)propyl]pyrazine-2-carboxamide —— C19H32N5O3+
5-methyl-N-(3-morpholin-4-ium-4-ylpropyl)-N-[3-oxo-3-(propan-2-ylamino)propyl]pyrazine-2-carboxamide
—— (5S)-5-(4-fluorospiro[2H-indole-3,1'-cyclopentane]-1-carbonyl)piperidin-2-one —— C18H21FN2O2
(5S)-5-(4-fluorospiro[2H-indole-3,1'-cyclopentane]-1-carbonyl)piperidin-2-one
—— (5R,10bS)-2-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-(3-methoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C25H22N2O4
(5R,10bS)-2-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-(3-methoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— 5-[[(3-fluorophenyl)methyl-propan-2-ylamino]methyl]-N-[3-[(2R)-2-methylpiperidin-1-yl]propyl]furan-2-carboxamide —— C25H36FN3O2
5-[[(3-fluorophenyl)methyl-propan-2-ylamino]methyl]-N-[3-[(2R)-2-methylpiperidin-1-yl]propyl]furan-2-carboxamide
—— (5S,10bS)-2-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-(3-fluorophenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C24H19FN2O3
(5S,10bS)-2-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-(3-fluorophenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— 5-methyl-N-[3-[3-[(2R)-2-methylpiperidin-1-ium-1-yl]propylamino]-3-oxopropyl]-N-propylpyrazine-2-carboxamide —— C21H36N5O2+
5-methyl-N-[3-[3-[(2R)-2-methylpiperidin-1-ium-1-yl]propylamino]-3-oxopropyl]-N-propylpyrazine-2-carboxamide
—— 5-[[(3-fluorophenyl)methyl-propan-2-ylamino]methyl]-N-[3-[(2S)-2-methylpiperidin-1-yl]propyl]furan-2-carboxamide —— C25H36FN3O2
5-[[(3-fluorophenyl)methyl-propan-2-ylamino]methyl]-N-[3-[(2S)-2-methylpiperidin-1-yl]propyl]furan-2-carboxamide
—— 5-[(1S)-1-[(2-chlorophenyl)methylsulfonyl]ethyl]-3-methyl-1,2,4-oxadiazole —— C12H13ClN2O3S
5-[(1S)-1-[(2-chlorophenyl)methylsulfonyl]ethyl]-3-methyl-1,2,4-oxadiazole
—— 5-methyl-N-(2-morpholin-4-ium-4-ylethyl)-N-(3-oxo-3-pyrrolidin-1-ylpropyl)pyrazine-2-carboxamide —— C19H30N5O3+
5-methyl-N-(2-morpholin-4-ium-4-ylethyl)-N-(3-oxo-3-pyrrolidin-1-ylpropyl)pyrazine-2-carboxamide
—— (5R,10bS)-2-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-(4-ethylphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C26H24N2O3
(5R,10bS)-2-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-(4-ethylphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— 5-(4-methoxyphenyl)-2-(3-methylphenyl)-N-(2-piperidin-1-ium-1-ylethyl)pyrazole-3-carboxamide —— C25H31N4O2+
5-(4-methoxyphenyl)-2-(3-methylphenyl)-N-(2-piperidin-1-ium-1-ylethyl)pyrazole-3-carboxamide
—— 5-[[(3-fluorophenyl)methyl-propan-2-ylamino]methyl]-N-[(2S)-4-phenylbutan-2-yl]furan-2-carboxamide —— C26H31FN2O2
5-[[(3-fluorophenyl)methyl-propan-2-ylamino]methyl]-N-[(2S)-4-phenylbutan-2-yl]furan-2-carboxamide
—— 5-cyclohexyl-N-[(2R)-2-(3,4-difluorophenyl)-2-hydroxyethyl]-1H-pyrazole-4-carboxamide —— C18H21F2N3O2
5-cyclohexyl-N-[(2R)-2-(3,4-difluorophenyl)-2-hydroxyethyl]-1H-pyrazole-4-carboxamide
—— 5-chloro-2-(methanesulfonamido)-N-[(2S)-1-methoxypropan-2-yl]benzamide —— C12H17ClN2O4S
5-chloro-2-(methanesulfonamido)-N-[(2S)-1-methoxypropan-2-yl]benzamide
—— 5-[(3S)-3-pyrazol-1-ylpiperidine-1-carbonyl]thiophene-3-carboxamide —— C14H16N4O2S
5-[(3S)-3-pyrazol-1-ylpiperidine-1-carbonyl]thiophene-3-carboxamide
—— 5-methyl-N-[3-(3-methylbutylamino)-3-oxopropyl]-N-[[(2S)-oxolan-2-yl]methyl]pyrazine-2-carboxamide —— C19H30N4O3
5-methyl-N-[3-(3-methylbutylamino)-3-oxopropyl]-N-[[(2S)-oxolan-2-yl]methyl]pyrazine-2-carboxamide
—— [5-[[[(2S)-butan-2-yl]-[(2S)-2-ethylhexanoyl]amino]methyl]-2-methoxyphenyl] methanesulfonate —— C21H35NO5S
[5-[[[(2S)-butan-2-yl]-[(2S)-2-ethylhexanoyl]amino]methyl]-2-methoxyphenyl] methanesulfonate
—— (5S)-2-[[4-(4-methylbenzoyl)piperidin-1-yl]methyl]-7-thia-2-azaspiro[4.4]nonane-1,3-dione —— C21H26N2O3S
(5S)-2-[[4-(4-methylbenzoyl)piperidin-1-yl]methyl]-7-thia-2-azaspiro[4.4]nonane-1,3-dione
—— (5S,7R)-3-[5-chloro-4-(furan-2-ylmethylamino)-6-oxopyridazin-1-yl]adamantane-1-carboxylic acid —— C20H22ClN3O4
(5S,7R)-3-[5-chloro-4-(furan-2-ylmethylamino)-6-oxopyridazin-1-yl]adamantane-1-carboxylic acid
—— (5S,7R)-N-(4-bromophenyl)-3-(5-methyltetrazol-2-yl)adamantane-1-carboxamide —— C19H22BrN5O
(5S,7R)-N-(4-bromophenyl)-3-(5-methyltetrazol-2-yl)adamantane-1-carboxamide
—— (5S,7R)-3-[5-chloro-4-(4-fluoroanilino)-6-oxopyridazin-1-yl]adamantane-1-carboxylate —— C21H20ClFN3O3-
(5S,7R)-3-[5-chloro-4-(4-fluoroanilino)-6-oxopyridazin-1-yl]adamantane-1-carboxylate
—— [5-(4-Nitrophenyl)-1,3,4-oxadiazol-2-yl]methyl 5-methyl-4-propylthiophene-2-carboxylate —— C18H17N3O5S
[5-(4-Nitrophenyl)-1,3,4-oxadiazol-2-yl]methyl 5-methyl-4-propylthiophene-2-carboxylate
—— 5-[(3R)-3-pyrazol-1-ylpiperidine-1-carbonyl]thiophene-3-carboxamide —— C14H16N4O2S
5-[(3R)-3-pyrazol-1-ylpiperidine-1-carbonyl]thiophene-3-carboxamide