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—— (5S)-1-ethyl-5-[[5-(methylcarbamoyl)furan-2-yl]methylamino]-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C17H22N4O4
(5S)-1-ethyl-5-[[5-(methylcarbamoyl)furan-2-yl]methylamino]-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— (5R)-1-ethyl-5-[methyl-[(3-pyridin-3-yl-1,2-oxazol-5-yl)methyl]amino]-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C20H23N5O3
(5R)-1-ethyl-5-[methyl-[(3-pyridin-3-yl-1,2-oxazol-5-yl)methyl]amino]-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— 5-[(4-benzylpiperidin-1-yl)methyl]-N-methyl-N-[(1R)-1-pyridin-2-ylethyl]-1,2-oxazole-3-carboxamide —— C25H30N4O2
5-[(4-benzylpiperidin-1-yl)methyl]-N-methyl-N-[(1R)-1-pyridin-2-ylethyl]-1,2-oxazole-3-carboxamide
—— (5S)-5-(3-chlorophenyl)-1,5-dihydrothieno[3,2-e][1,4]thiazepin-2-one —— C13H10ClNOS2
(5S)-5-(3-chlorophenyl)-1,5-dihydrothieno[3,2-e][1,4]thiazepin-2-one
—— 5-amino-N-[(2R)-2-cyclopropyl-2-hydroxyethyl]-2-methoxybenzamide —— C13H18N2O3
5-amino-N-[(2R)-2-cyclopropyl-2-hydroxyethyl]-2-methoxybenzamide
—— (5S)-5-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl-methylamino]-1-propyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C17H25N5O3
(5S)-5-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl-methylamino]-1-propyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— (5R)-1-ethyl-5-[[5-(methylcarbamoyl)furan-2-yl]methylamino]-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C17H22N4O4
(5R)-1-ethyl-5-[[5-(methylcarbamoyl)furan-2-yl]methylamino]-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— 5-[(1S)-1-[2-(3,5-difluorophenyl)imidazol-1-yl]ethyl]-3-(2-methoxyethyl)-1,2,4-oxadiazole —— C16H16F2N4O2
5-[(1S)-1-[2-(3,5-difluorophenyl)imidazol-1-yl]ethyl]-3-(2-methoxyethyl)-1,2,4-oxadiazole
—— (5S)-9-[(2,3-difluorophenyl)methyl]-2-[(1-ethylpyrazol-4-yl)methyl]-2,9-diazaspiro[4.5]decane —— C21H28F2N4
(5S)-9-[(2,3-difluorophenyl)methyl]-2-[(1-ethylpyrazol-4-yl)methyl]-2,9-diazaspiro[4.5]decane
—— 5-[[(4S)-4-(4-ethylphenyl)-1,4,6,7-tetrahydroimidazo[4,5-c]pyridin-5-yl]methyl]-3-propan-2-yl-1,2-oxazole —— C21H26N4O
5-[[(4S)-4-(4-ethylphenyl)-1,4,6,7-tetrahydroimidazo[4,5-c]pyridin-5-yl]methyl]-3-propan-2-yl-1,2-oxazole
—— 5-amino-2-bromo-N-[(2R)-2-cyclopropyl-2-hydroxyethyl]-4-fluorobenzamide —— C12H14BrFN2O2
5-amino-2-bromo-N-[(2R)-2-cyclopropyl-2-hydroxyethyl]-4-fluorobenzamide
—— (5S,7S)-7-methyl-N-[(1-methylimidazol-2-yl)methyl]-3-thia-1-azaspiro[4.5]dec-1-en-2-amine —— C14H22N4S
(5S,7S)-7-methyl-N-[(1-methylimidazol-2-yl)methyl]-3-thia-1-azaspiro[4.5]dec-1-en-2-amine
—— 5-[2-(benzimidazol-1-yl)ethyl]-3-[(3S)-3-(4-fluorophenyl)oxolan-3-yl]-1,2,4-oxadiazole —— C21H19FN4O2
5-[2-(benzimidazol-1-yl)ethyl]-3-[(3S)-3-(4-fluorophenyl)oxolan-3-yl]-1,2,4-oxadiazole
—— 5-[2-(benzimidazol-1-yl)ethyl]-3-[(3R)-3-(4-fluorophenyl)oxolan-3-yl]-1,2,4-oxadiazole —— C21H19FN4O2
5-[2-(benzimidazol-1-yl)ethyl]-3-[(3R)-3-(4-fluorophenyl)oxolan-3-yl]-1,2,4-oxadiazole
—— 5-ethyl-N-[[(3R)-1-methylpiperidin-3-yl]methyl]-4-(pyrrolidin-1-ylmethyl)furan-2-carboxamide —— C19H31N3O2
5-ethyl-N-[[(3R)-1-methylpiperidin-3-yl]methyl]-4-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
—— (5S)-1-ethyl-5-[methyl-[(3-pyridin-3-yl-1,2-oxazol-5-yl)methyl]amino]-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C20H23N5O3
(5S)-1-ethyl-5-[methyl-[(3-pyridin-3-yl-1,2-oxazol-5-yl)methyl]amino]-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— 5-acetamido-N-[(2R)-2-cyclopropyl-2-hydroxyethyl]thiophene-2-carboxamide —— C12H16N2O3S
5-acetamido-N-[(2R)-2-cyclopropyl-2-hydroxyethyl]thiophene-2-carboxamide
—— 5-bromo-N-[(2R)-2-cyclopropyl-2-hydroxyethyl]-2-fluorobenzamide —— C12H13BrFNO2
5-bromo-N-[(2R)-2-cyclopropyl-2-hydroxyethyl]-2-fluorobenzamide
—— 5-[(1R)-1-(2-chlorophenyl)ethyl]sulfanyl-1-[4-(trifluoromethoxy)phenyl]tetrazole —— C16H12ClF3N4OS
5-[(1R)-1-(2-chlorophenyl)ethyl]sulfanyl-1-[4-(trifluoromethoxy)phenyl]tetrazole
—— (5-amino-4-cyano-2-ethoxycarbonylthiophen-3-yl)methyl (3S)-1-(furan-2-ylmethyl)-5-oxopyrrolidine-3-carboxylate —— C19H19N3O6S
(5-amino-4-cyano-2-ethoxycarbonylthiophen-3-yl)methyl (3S)-1-(furan-2-ylmethyl)-5-oxopyrrolidine-3-carboxylate
—— 5-[(1R)-1-(4-fluorophenyl)ethyl]sulfanyl-1-[4-(trifluoromethoxy)phenyl]tetrazole —— C16H12F4N4OS
5-[(1R)-1-(4-fluorophenyl)ethyl]sulfanyl-1-[4-(trifluoromethoxy)phenyl]tetrazole
—— (5S,7R)-7-methyl-N-[(1-methylimidazol-2-yl)methyl]-3-thia-1-azaspiro[4.5]dec-1-en-2-amine —— C14H22N4S
(5S,7R)-7-methyl-N-[(1-methylimidazol-2-yl)methyl]-3-thia-1-azaspiro[4.5]dec-1-en-2-amine
—— 5-amino-N-[(2S)-2-cyclopropyl-2-hydroxyethyl]-2-methylpyridine-3-carboxamide —— C12H17N3O2
5-amino-N-[(2S)-2-cyclopropyl-2-hydroxyethyl]-2-methylpyridine-3-carboxamide
—— 5-bromo-N-[(2S)-2-cyclopropyl-2-hydroxyethyl]-2-fluorobenzamide —— C12H13BrFNO2
5-bromo-N-[(2S)-2-cyclopropyl-2-hydroxyethyl]-2-fluorobenzamide
—— (5-amino-4-cyano-2-ethoxycarbonylthiophen-3-yl)methyl (3R)-1-(furan-2-ylmethyl)-5-oxopyrrolidine-3-carboxylate —— C19H19N3O6S
(5-amino-4-cyano-2-ethoxycarbonylthiophen-3-yl)methyl (3R)-1-(furan-2-ylmethyl)-5-oxopyrrolidine-3-carboxylate
—— 5-amino-N-[(2S)-2-cyclopropyl-2-hydroxyethyl]-2-methoxybenzamide —— C13H18N2O3
5-amino-N-[(2S)-2-cyclopropyl-2-hydroxyethyl]-2-methoxybenzamide
—— 5-[(3-Methylphenyl)methylsulfanyl]-1-[4-(trifluoromethoxy)phenyl]tetrazole —— C16H13F3N4OS
5-[(3-Methylphenyl)methylsulfanyl]-1-[4-(trifluoromethoxy)phenyl]tetrazole
—— 5-amino-N-[(2R)-2-cyclopropyl-2-hydroxyethyl]-2-methylpyridine-3-carboxamide —— C12H17N3O2
5-amino-N-[(2R)-2-cyclopropyl-2-hydroxyethyl]-2-methylpyridine-3-carboxamide
—— 5-bromo-2-[[(2R)-1-thiophen-2-ylpropan-2-yl]amino]pyridine-3-carboxylic acid —— C13H13BrN2O2S
5-bromo-2-[[(2R)-1-thiophen-2-ylpropan-2-yl]amino]pyridine-3-carboxylic acid
—— 5-bromo-2-[[(2S)-1-thiophen-2-ylpropan-2-yl]amino]pyridine-3-carboxylic acid —— C13H13BrN2O2S
5-bromo-2-[[(2S)-1-thiophen-2-ylpropan-2-yl]amino]pyridine-3-carboxylic acid
—— 5-amino-2-[[(2R)-1-thiophen-2-ylpropan-2-yl]amino]benzonitrile —— C14H15N3S
5-amino-2-[[(2R)-1-thiophen-2-ylpropan-2-yl]amino]benzonitrile
—— 5-amino-2-[[(2S)-1-thiophen-2-ylpropan-2-yl]amino]benzonitrile —— C14H15N3S
5-amino-2-[[(2S)-1-thiophen-2-ylpropan-2-yl]amino]benzonitrile
—— 5-[[(2R)-1-thiophen-2-ylpropan-2-yl]amino]furan-2-carboxylic acid —— C12H13NO3S
5-[[(2R)-1-thiophen-2-ylpropan-2-yl]amino]furan-2-carboxylic acid
—— 5-fluoro-1-[(2R)-1-thiophen-2-ylpropan-2-yl]benzimidazol-2-amine —— C14H14FN3S
5-fluoro-1-[(2R)-1-thiophen-2-ylpropan-2-yl]benzimidazol-2-amine
—— 5-[[(2S)-1-thiophen-2-ylpropan-2-yl]amino]furan-2-carboxylic acid —— C12H13NO3S
5-[[(2S)-1-thiophen-2-ylpropan-2-yl]amino]furan-2-carboxylic acid
—— 5-N-[(2S)-1-thiophen-2-ylpropan-2-yl]-1,3-benzothiazole-4,5-diamine —— C14H15N3S2
5-N-[(2S)-1-thiophen-2-ylpropan-2-yl]-1,3-benzothiazole-4,5-diamine
—— 5-fluoro-1-[(2S)-1-thiophen-2-ylpropan-2-yl]benzimidazol-2-amine —— C14H14FN3S
5-fluoro-1-[(2S)-1-thiophen-2-ylpropan-2-yl]benzimidazol-2-amine
—— 5-fluoro-2-[[(3S)-3-(2-hydroxyethyl)piperidin-1-yl]methyl]benzonitrile —— C15H19FN2O
5-fluoro-2-[[(3S)-3-(2-hydroxyethyl)piperidin-1-yl]methyl]benzonitrile
—— 5-fluoro-N'-hydroxy-2-[[(2S)-2-methylmorpholin-4-yl]methyl]benzenecarboximidamide —— C13H18FN3O2
5-fluoro-N'-hydroxy-2-[[(2S)-2-methylmorpholin-4-yl]methyl]benzenecarboximidamide
—— 5,6-Dimethyl-2-(2-methyl-allylsulfanyl)-3H-thieno[2,3-d]pyrimidin-4-one —— C12H14N2OS2
5,6-Dimethyl-2-(2-methyl-allylsulfanyl)-3H-thieno[2,3-d]pyrimidin-4-one
—— 5-fluoro-2-[[methyl-[(2S)-pentan-2-yl]amino]methyl]benzenecarboximidamide —— C14H22FN3
5-fluoro-2-[[methyl-[(2S)-pentan-2-yl]amino]methyl]benzenecarboximidamide
—— 5-fluoro-2-[[(3R)-3-hydroxypiperidin-1-yl]methyl]benzenecarbothioamide —— C13H17FN2OS
5-fluoro-2-[[(3R)-3-hydroxypiperidin-1-yl]methyl]benzenecarbothioamide
—— 5-fluoro-2-[[(3R)-3-(2-hydroxyethyl)piperidin-1-yl]methyl]benzonitrile —— C15H19FN2O
5-fluoro-2-[[(3R)-3-(2-hydroxyethyl)piperidin-1-yl]methyl]benzonitrile
—— 5-fluoro-2-[[[(2S)-1-methoxypropan-2-yl]-methylamino]methyl]benzenecarboximidamide —— C13H20FN3O
5-fluoro-2-[[[(2S)-1-methoxypropan-2-yl]-methylamino]methyl]benzenecarboximidamide
—— 5-fluoro-N'-hydroxy-2-(2-methylpropoxymethyl)benzenecarboximidamide —— C12H17FN2O2
5-fluoro-N'-hydroxy-2-(2-methylpropoxymethyl)benzenecarboximidamide
—— 5-fluoro-2-[[methyl-[(2S)-2-methylbutyl]amino]methyl]benzenecarboximidamide —— C14H22FN3
5-fluoro-2-[[methyl-[(2S)-2-methylbutyl]amino]methyl]benzenecarboximidamide
—— 5-fluoro-N'-hydroxy-2-[[(2S)-2-methylpiperidin-1-yl]methyl]benzenecarboximidamide —— C14H20FN3O
5-fluoro-N'-hydroxy-2-[[(2S)-2-methylpiperidin-1-yl]methyl]benzenecarboximidamide
—— [5-fluoro-2-[[(1S,2S)-2-methylcyclohexyl]oxymethyl]phenyl]methanamine —— C15H22FNO
[5-fluoro-2-[[(1S,2S)-2-methylcyclohexyl]oxymethyl]phenyl]methanamine
—— 5-fluoro-N'-hydroxy-2-(thiophen-2-ylmethoxymethyl)benzenecarboximidamide —— C13H13FN2O2S
5-fluoro-N'-hydroxy-2-(thiophen-2-ylmethoxymethyl)benzenecarboximidamide
—— 5-fluoro-2-[[(3R)-3-(hydroxymethyl)piperidin-1-yl]methyl]benzonitrile —— C14H17FN2O
5-fluoro-2-[[(3R)-3-(hydroxymethyl)piperidin-1-yl]methyl]benzonitrile