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—— (5-fluoro-1H-indol-2-yl)-[(2R)-2-(pyrazol-1-ylmethyl)piperidin-1-yl]methanone —— C18H19FN4O
(5-fluoro-1H-indol-2-yl)-[(2R)-2-(pyrazol-1-ylmethyl)piperidin-1-yl]methanone
—— (5-methyl-1,3,4-oxadiazol-2-yl)methyl (2R)-2-[4-(4-fluorophenyl)piperazin-1-yl]propanoate —— C17H21FN4O3
(5-methyl-1,3,4-oxadiazol-2-yl)methyl (2R)-2-[4-(4-fluorophenyl)piperazin-1-yl]propanoate
—— (5-methoxy-3-methyl-1-benzofuran-2-yl)-[(2S)-2-(1-methylpyrazol-4-yl)pyrrolidin-1-yl]methanone —— C19H21N3O3
(5-methoxy-3-methyl-1-benzofuran-2-yl)-[(2S)-2-(1-methylpyrazol-4-yl)pyrrolidin-1-yl]methanone
—— 5-phenyl-2-[(1R)-1-[4-(pyridin-2-ylmethyl)piperazin-1-yl]ethyl]-1,3-oxazole —— C21H24N4O
5-phenyl-2-[(1R)-1-[4-(pyridin-2-ylmethyl)piperazin-1-yl]ethyl]-1,3-oxazole
—— (5-fluoro-1H-indol-2-yl)-[(2S)-2-(pyrazol-1-ylmethyl)piperidin-1-yl]methanone —— C18H19FN4O
(5-fluoro-1H-indol-2-yl)-[(2S)-2-(pyrazol-1-ylmethyl)piperidin-1-yl]methanone
—— (5S)-N-[(3-methoxy-4-methylsulfanylphenyl)methyl]-N-methyl-5-phenyl-4,5-dihydro-1,2-oxazole-3-carboxamide —— C20H22N2O3S
(5S)-N-[(3-methoxy-4-methylsulfanylphenyl)methyl]-N-methyl-5-phenyl-4,5-dihydro-1,2-oxazole-3-carboxamide
—— (5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl (2S)-2-(3-fluorophenyl)-2-hydroxypropanoate —— C16H13FN2O4S
(5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl (2S)-2-(3-fluorophenyl)-2-hydroxypropanoate
—— [5-(diethylaminomethyl)furan-2-yl]-[4-[(2R)-2-hydroxypropyl]piperazin-1-yl]methanone —— C17H29N3O3
[5-(diethylaminomethyl)furan-2-yl]-[4-[(2R)-2-hydroxypropyl]piperazin-1-yl]methanone
—— 5-chloro-6-[4-[(2S)-1-(2-methoxyacetyl)azepan-2-yl]piperidin-1-yl]pyridine-3-carboxamide —— C20H29ClN4O3
5-chloro-6-[4-[(2S)-1-(2-methoxyacetyl)azepan-2-yl]piperidin-1-yl]pyridine-3-carboxamide
—— 5-[(1R)-1-[[4-cyclohexyl-5-(3,4-dimethoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]ethyl]-3-phenyl-1,2,4-oxadiazole —— C26H29N5O3S
5-[(1R)-1-[[4-cyclohexyl-5-(3,4-dimethoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]ethyl]-3-phenyl-1,2,4-oxadiazole
—— 5-[[(3R)-3-[(3,5-dimethyl-1,2,4-triazol-1-yl)methyl]piperidin-1-yl]methyl]-3-(furan-2-yl)-1,2,4-oxadiazole —— C17H22N6O2
5-[[(3R)-3-[(3,5-dimethyl-1,2,4-triazol-1-yl)methyl]piperidin-1-yl]methyl]-3-(furan-2-yl)-1,2,4-oxadiazole
—— (5-bromopyridin-2-yl)-[(3R)-3-(2-methylimidazol-1-yl)piperidin-1-yl]methanone —— C15H17BrN4O
(5-bromopyridin-2-yl)-[(3R)-3-(2-methylimidazol-1-yl)piperidin-1-yl]methanone
—— (5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl (2R)-2-(3-fluorophenyl)-2-hydroxypropanoate —— C16H13FN2O4S
(5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl (2R)-2-(3-fluorophenyl)-2-hydroxypropanoate
—— 5-[[(6S)-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-yl]amino]pentanenitrile —— C11H17N5
5-[[(6S)-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-yl]amino]pentanenitrile
—— (5-methylpyrazolo[1,5-a]pyrimidin-3-yl)-[(2S)-2-(pyrazol-1-ylmethyl)piperidin-1-yl]methanone —— C17H20N6O
(5-methylpyrazolo[1,5-a]pyrimidin-3-yl)-[(2S)-2-(pyrazol-1-ylmethyl)piperidin-1-yl]methanone
—— (5-phenyl-1,2-oxazol-3-yl)-[(2S)-2-(pyrazol-1-ylmethyl)piperidin-1-yl]methanone —— C19H20N4O2
(5-phenyl-1,2-oxazol-3-yl)-[(2S)-2-(pyrazol-1-ylmethyl)piperidin-1-yl]methanone
—— 5-[(1S)-1-[[4-cyclohexyl-5-(3,4-dimethoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]ethyl]-3-phenyl-1,2,4-oxadiazole —— C26H29N5O3S
5-[(1S)-1-[[4-cyclohexyl-5-(3,4-dimethoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]ethyl]-3-phenyl-1,2,4-oxadiazole
—— 5-[(1S)-1-[[5-(2-methoxyphenyl)-4-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]ethyl]-3-phenyl-1,2,4-oxadiazole —— C26H23N5O3S
5-[(1S)-1-[[5-(2-methoxyphenyl)-4-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]ethyl]-3-phenyl-1,2,4-oxadiazole
—— [5-(diethylaminomethyl)furan-2-yl]-[4-[(2S)-2-hydroxypropyl]piperazin-1-yl]methanone —— C17H29N3O3
[5-(diethylaminomethyl)furan-2-yl]-[4-[(2S)-2-hydroxypropyl]piperazin-1-yl]methanone
—— 5-chloro-6-[4-[(2R)-1-(2-methoxyacetyl)azepan-2-yl]piperidin-1-yl]pyridine-3-carboxamide —— C20H29ClN4O3
5-chloro-6-[4-[(2R)-1-(2-methoxyacetyl)azepan-2-yl]piperidin-1-yl]pyridine-3-carboxamide
—— 5-[[(3S)-3-[(3,5-dimethyl-1,2,4-triazol-1-yl)methyl]piperidin-1-yl]methyl]-3-(furan-2-yl)-1,2,4-oxadiazole —— C17H22N6O2
5-[[(3S)-3-[(3,5-dimethyl-1,2,4-triazol-1-yl)methyl]piperidin-1-yl]methyl]-3-(furan-2-yl)-1,2,4-oxadiazole
—— (5-methylpyrazolo[1,5-a]pyrimidin-3-yl)-[(2R)-2-(pyrazol-1-ylmethyl)piperidin-1-yl]methanone —— C17H20N6O
(5-methylpyrazolo[1,5-a]pyrimidin-3-yl)-[(2R)-2-(pyrazol-1-ylmethyl)piperidin-1-yl]methanone
—— 5-[(E)-2-[4-(4-methylphenyl)-1,3-thiazol-2-yl]ethenyl]-6-phenylimidazo[2,1-b][1,3]thiazole —— C23H17N3S2
5-[(E)-2-[4-(4-methylphenyl)-1,3-thiazol-2-yl]ethenyl]-6-phenylimidazo[2,1-b][1,3]thiazole
—— 5-[[(2S)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methyl]-3-thiophen-3-yl-1,2,4-oxadiazole —— C15H17N5OS
5-[[(2S)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methyl]-3-thiophen-3-yl-1,2,4-oxadiazole
—— (5-bromothiophen-2-yl)-[4-[(2S)-2-hydroxybutyl]piperazin-1-yl]methanone —— C13H19BrN2O2S
(5-bromothiophen-2-yl)-[4-[(2S)-2-hydroxybutyl]piperazin-1-yl]methanone
—— 5-[[(2R)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methyl]-3-thiophen-3-yl-1,2,4-oxadiazole —— C15H17N5OS
5-[[(2R)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methyl]-3-thiophen-3-yl-1,2,4-oxadiazole
—— 5-[[(2R)-2-ethoxypropanoyl]amino]-N-[(4-methoxyphenyl)methyl]-1H-pyrazole-4-carboxamide —— C17H22N4O4
5-[[(2R)-2-ethoxypropanoyl]amino]-N-[(4-methoxyphenyl)methyl]-1H-pyrazole-4-carboxamide
—— (5-methyl-1,2-oxazol-3-yl)methyl (2R)-2-[4-(4-fluorophenyl)piperazin-1-yl]propanoate —— C18H22FN3O3
(5-methyl-1,2-oxazol-3-yl)methyl (2R)-2-[4-(4-fluorophenyl)piperazin-1-yl]propanoate
—— 5-[[4-[(2S)-1-(benzenesulfonyl)azepan-2-yl]piperidin-1-yl]methyl]-3-propan-2-yl-1,2,4-oxadiazole —— C23H34N4O3S
5-[[4-[(2S)-1-(benzenesulfonyl)azepan-2-yl]piperidin-1-yl]methyl]-3-propan-2-yl-1,2,4-oxadiazole
—— 5-[[4-[(2R)-1-(benzenesulfonyl)azepan-2-yl]piperidin-1-yl]methyl]-3-propan-2-yl-1,2,4-oxadiazole —— C23H34N4O3S
5-[[4-[(2R)-1-(benzenesulfonyl)azepan-2-yl]piperidin-1-yl]methyl]-3-propan-2-yl-1,2,4-oxadiazole
—— (5-methyl-1,2-oxazol-3-yl)methyl (2S)-2-[4-(4-fluorophenyl)piperazin-1-yl]propanoate —— C18H22FN3O3
(5-methyl-1,2-oxazol-3-yl)methyl (2S)-2-[4-(4-fluorophenyl)piperazin-1-yl]propanoate
—— 5-[[(2S)-2-ethoxypropanoyl]amino]-N-[(4-methoxyphenyl)methyl]-1H-pyrazole-4-carboxamide —— C17H22N4O4
5-[[(2S)-2-ethoxypropanoyl]amino]-N-[(4-methoxyphenyl)methyl]-1H-pyrazole-4-carboxamide
—— (5-methyl-1,2-oxazol-3-yl)-[(2R)-2-[(4-methylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methanone —— C14H18N4O2
(5-methyl-1,2-oxazol-3-yl)-[(2R)-2-[(4-methylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methanone
—— 5-chloro-N-[(1S)-2-methyl-1-(3-methyl-1,2,4-oxadiazol-5-yl)propyl]thiophene-2-sulfonamide —— C11H14ClN3O3S2
5-chloro-N-[(1S)-2-methyl-1-(3-methyl-1,2,4-oxadiazol-5-yl)propyl]thiophene-2-sulfonamide
—— (5Z)-5-[(4-ethylphenyl)methylidene]-3-pyridin-3-yl-2-sulfanylidene-1,3-thiazolidin-4-one —— C17H14N2OS2
(5Z)-5-[(4-ethylphenyl)methylidene]-3-pyridin-3-yl-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5-fluoro-3-methyl-1-benzofuran-2-yl)-[4-[(2R)-2-hydroxybutyl]piperazin-1-yl]methanone —— C18H23FN2O3
(5-fluoro-3-methyl-1-benzofuran-2-yl)-[4-[(2R)-2-hydroxybutyl]piperazin-1-yl]methanone
—— (5-bromofuran-3-yl)-[(2R)-2-(pyrazol-1-ylmethyl)piperidin-1-yl]methanone —— C14H16BrN3O2
(5-bromofuran-3-yl)-[(2R)-2-(pyrazol-1-ylmethyl)piperidin-1-yl]methanone
—— 5-fluoro-2-[[[(2R)-1-pyrazol-1-ylpropan-2-yl]amino]methyl]benzonitrile —— C14H15FN4
5-fluoro-2-[[[(2R)-1-pyrazol-1-ylpropan-2-yl]amino]methyl]benzonitrile
—— (5-methyl-1,2-oxazol-3-yl)-[(2S)-2-[(4-methylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methanone —— C14H18N4O2
(5-methyl-1,2-oxazol-3-yl)-[(2S)-2-[(4-methylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methanone
—— (5-fluoro-3-methyl-1-benzofuran-2-yl)-[4-[(2S)-2-hydroxybutyl]piperazin-1-yl]methanone —— C18H23FN2O3
(5-fluoro-3-methyl-1-benzofuran-2-yl)-[4-[(2S)-2-hydroxybutyl]piperazin-1-yl]methanone
—— 5-chloro-N-[(1R)-2-methyl-1-(3-methyl-1,2,4-oxadiazol-5-yl)propyl]thiophene-2-sulfonamide —— C11H14ClN3O3S2
5-chloro-N-[(1R)-2-methyl-1-(3-methyl-1,2,4-oxadiazol-5-yl)propyl]thiophene-2-sulfonamide
—— 5-fluoro-2-[[[(2S)-1-pyrazol-1-ylpropan-2-yl]amino]methyl]benzonitrile —— C14H15FN4
5-fluoro-2-[[[(2S)-1-pyrazol-1-ylpropan-2-yl]amino]methyl]benzonitrile
—— (5S)-2-[(2R)-3-[(4-chlorophenyl)methoxy]-2-hydroxypropyl]-7-thia-2-azaspiro[4.4]nonane-1,3-dione —— C17H20ClNO4S
(5S)-2-[(2R)-3-[(4-chlorophenyl)methoxy]-2-hydroxypropyl]-7-thia-2-azaspiro[4.4]nonane-1,3-dione
—— 5-[2-[4-[(2R)-2-hydroxybutyl]piperazin-1-yl]-2-oxoethyl]-1-methylpyrazolo[3,4-d]pyrimidin-4-one —— C16H24N6O3
5-[2-[4-[(2R)-2-hydroxybutyl]piperazin-1-yl]-2-oxoethyl]-1-methylpyrazolo[3,4-d]pyrimidin-4-one
—— 5-bromo-2-chloro-N-[(3S,4R)-1,1-dioxo-4-pyrrolidin-1-ylthiolan-3-yl]pyridine-3-carboxamide —— C14H17BrClN3O3S
5-bromo-2-chloro-N-[(3S,4R)-1,1-dioxo-4-pyrrolidin-1-ylthiolan-3-yl]pyridine-3-carboxamide
—— 5-[[(2R)-2-(pyrazol-1-ylmethyl)piperidin-1-yl]methyl]-3-pyridin-2-yl-1,2,4-oxadiazole —— C17H20N6O
5-[[(2R)-2-(pyrazol-1-ylmethyl)piperidin-1-yl]methyl]-3-pyridin-2-yl-1,2,4-oxadiazole
—— 5-bromo-2-chloro-N-[(3S,4S)-1,1-dioxo-4-pyrrolidin-1-ylthiolan-3-yl]pyridine-3-carboxamide —— C14H17BrClN3O3S
5-bromo-2-chloro-N-[(3S,4S)-1,1-dioxo-4-pyrrolidin-1-ylthiolan-3-yl]pyridine-3-carboxamide
—— 5-[[(2R)-2-naphthalen-1-ylpyrrolidin-1-yl]methyl]-3-thiophen-2-yl-1,2,4-oxadiazole —— C21H19N3OS
5-[[(2R)-2-naphthalen-1-ylpyrrolidin-1-yl]methyl]-3-thiophen-2-yl-1,2,4-oxadiazole
—— 5-bromo-2-chloro-N-[(3R,4S)-1,1-dioxo-4-pyrrolidin-1-ylthiolan-3-yl]pyridine-3-carboxamide —— C14H17BrClN3O3S
5-bromo-2-chloro-N-[(3R,4S)-1,1-dioxo-4-pyrrolidin-1-ylthiolan-3-yl]pyridine-3-carboxamide
—— (5Z)-5-[(3-ethoxy-2-propoxyphenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C15H17NO3S2
(5Z)-5-[(3-ethoxy-2-propoxyphenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one