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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-(1,2,4-triazol-1-ylmethyl)-5-[(1S)-1-[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]ethyl]sulfanyl-1,3,4-oxadiazole —— C16H12F3N7O2S
2-(1,2,4-triazol-1-ylmethyl)-5-[(1S)-1-[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]ethyl]sulfanyl-1,3,4-oxadiazole
—— (2R)-N-[4-(4-fluorophenyl)-1,3-thiazol-2-yl]-2-(5-phenyltetrazol-2-yl)propanamide —— C19H15FN6OS
(2R)-N-[4-(4-fluorophenyl)-1,3-thiazol-2-yl]-2-(5-phenyltetrazol-2-yl)propanamide
—— 5-[(1R)-1-[[4-(3-methoxypropyl)-1,2,4-triazol-3-yl]sulfanyl]ethyl]-3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazole —— C17H18F3N5O2S
5-[(1R)-1-[[4-(3-methoxypropyl)-1,2,4-triazol-3-yl]sulfanyl]ethyl]-3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazole
—— N-[[(2S)-4-(2-methylpropyl)morpholin-2-yl]methyl]-1-phenylpyrazolo[3,4-d]pyrimidin-4-amine —— C20H26N6O
N-[[(2S)-4-(2-methylpropyl)morpholin-2-yl]methyl]-1-phenylpyrazolo[3,4-d]pyrimidin-4-amine
—— 1-(4-methylphenyl)-5-[(E)-piperidin-1-ylmethylideneamino]pyrazole-4-carbonitrile —— C17H19N5
1-(4-methylphenyl)-5-[(E)-piperidin-1-ylmethylideneamino]pyrazole-4-carbonitrile
—— 3-(4-methoxyphenyl)-5-[[(2R)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)pyrrolidin-1-yl]methyl]-1,2,4-oxadiazole —— C21H26N6O2
3-(4-methoxyphenyl)-5-[[(2R)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)pyrrolidin-1-yl]methyl]-1,2,4-oxadiazole
—— 2-[[ethyl-[(1S)-1-[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]ethyl]amino]methyl]-1H-quinazolin-4-one —— C22H20F3N5O2
2-[[ethyl-[(1S)-1-[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]ethyl]amino]methyl]-1H-quinazolin-4-one
—— (1S)-1-(furan-2-yl)-N,N-dimethyl-N'-(1-phenylpyrazolo[3,4-d]pyrimidin-4-yl)ethane-1,2-diamine —— C19H20N6O
(1S)-1-(furan-2-yl)-N,N-dimethyl-N'-(1-phenylpyrazolo[3,4-d]pyrimidin-4-yl)ethane-1,2-diamine
—— 5-{[(4-methyl-1-piperazinyl)methylene]amino}-1-phenyl-1H-pyrazole-4-carbonitrile —— C16H18N6
5-{[(4-methyl-1-piperazinyl)methylene]amino}-1-phenyl-1H-pyrazole-4-carbonitrile
—— 2-(1,2,4-triazol-1-ylmethyl)-5-[(1R)-1-[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]ethyl]sulfanyl-1,3,4-oxadiazole —— C16H12F3N7O2S
2-(1,2,4-triazol-1-ylmethyl)-5-[(1R)-1-[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]ethyl]sulfanyl-1,3,4-oxadiazole
—— 5-[(1S)-1-[[4-(3-methoxypropyl)-1,2,4-triazol-3-yl]sulfanyl]ethyl]-3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazole —— C17H18F3N5O2S
5-[(1S)-1-[[4-(3-methoxypropyl)-1,2,4-triazol-3-yl]sulfanyl]ethyl]-3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazole
—— (2Z,4Z)-N-[3-methyl-4-(tetrazol-1-yl)phenyl]hexa-2,4-dienamide —— C14H15N5O
(2Z,4Z)-N-[3-methyl-4-(tetrazol-1-yl)phenyl]hexa-2,4-dienamide
—— N-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-3-[(2S)-2-methyl-3,4-dihydro-2H-quinolin-1-yl]propanamide —— C24H28N4O2
N-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-3-[(2S)-2-methyl-3,4-dihydro-2H-quinolin-1-yl]propanamide
—— (Z)-N-[[1-(difluoromethyl)imidazol-2-yl]methyl]-N-methyl-3-(1-methylpyrazol-4-yl)prop-2-enamide —— C13H15F2N5O
(Z)-N-[[1-(difluoromethyl)imidazol-2-yl]methyl]-N-methyl-3-(1-methylpyrazol-4-yl)prop-2-enamide
—— 1-(4-methylphenyl)-5-[(4-morpholinylmethylene)amino]-1H-pyrazole-4-carbonitrile —— C16H17N5O
1-(4-methylphenyl)-5-[(4-morpholinylmethylene)amino]-1H-pyrazole-4-carbonitrile
—— 3-(4-methoxyphenyl)-5-[[(2S)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)pyrrolidin-1-yl]methyl]-1,2,4-oxadiazole —— C21H26N6O2
3-(4-methoxyphenyl)-5-[[(2S)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)pyrrolidin-1-yl]methyl]-1,2,4-oxadiazole
—— N-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-3-[(2R)-2-methyl-3,4-dihydro-2H-quinolin-1-yl]propanamide —— C24H28N4O2
N-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-3-[(2R)-2-methyl-3,4-dihydro-2H-quinolin-1-yl]propanamide
—— 5-{[(E)-azepan-1-ylmethylidene]amino}-1-(4-methylphenyl)-1H-pyrazole-4-carbonitrile —— C18H21N5
5-{[(E)-azepan-1-ylmethylidene]amino}-1-(4-methylphenyl)-1H-pyrazole-4-carbonitrile
—— (Z)-N-cyclopropyl-N-(furan-2-ylmethyl)-3-(1-methylpyrazol-4-yl)prop-2-enamide —— C15H17N3O2
(Z)-N-cyclopropyl-N-(furan-2-ylmethyl)-3-(1-methylpyrazol-4-yl)prop-2-enamide
—— 1-methyl-5-[(1-pyrrolidinylmethylene)amino]-1H-pyrazole-4-carbonitrile —— C10H13N5
1-methyl-5-[(1-pyrrolidinylmethylene)amino]-1H-pyrazole-4-carbonitrile
—— (Z)-1-[(2R)-2-ethylmorpholin-4-yl]-3-(1-phenylpyrazol-4-yl)prop-2-en-1-one —— C18H21N3O2
(Z)-1-[(2R)-2-ethylmorpholin-4-yl]-3-(1-phenylpyrazol-4-yl)prop-2-en-1-one
—— (Z)-1-[(2S)-2-ethylmorpholin-4-yl]-3-(1-phenylpyrazol-4-yl)prop-2-en-1-one —— C18H21N3O2
(Z)-1-[(2S)-2-ethylmorpholin-4-yl]-3-(1-phenylpyrazol-4-yl)prop-2-en-1-one
—— 3-methyl-6-propan-2-yl-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide —— C21H22N6O2
3-methyl-6-propan-2-yl-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
—— (Z)-N-[(1S)-1-[5-methyl-1-[3-(trifluoromethyl)phenyl]pyrazol-4-yl]ethyl]-3-pyridin-3-ylprop-2-enamide —— C21H19F3N4O
(Z)-N-[(1S)-1-[5-methyl-1-[3-(trifluoromethyl)phenyl]pyrazol-4-yl]ethyl]-3-pyridin-3-ylprop-2-enamide
—— 3-methyl-6-propan-2-yl-N-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide —— C21H22N6O2
3-methyl-6-propan-2-yl-N-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
—— (2E,4Z)-N-[3-methyl-4-(tetrazol-1-yl)phenyl]hexa-2,4-dienamide —— C14H15N5O
(2E,4Z)-N-[3-methyl-4-(tetrazol-1-yl)phenyl]hexa-2,4-dienamide
—— (Z)-N-[[1-(difluoromethyl)imidazol-2-yl]methyl]-N-methyl-3-(2-methyl-1,3-thiazol-4-yl)prop-2-enamide —— C13H14F2N4OS
(Z)-N-[[1-(difluoromethyl)imidazol-2-yl]methyl]-N-methyl-3-(2-methyl-1,3-thiazol-4-yl)prop-2-enamide
—— (Z)-N-[(1R)-1-[5-methyl-1-[3-(trifluoromethyl)phenyl]pyrazol-4-yl]ethyl]-3-pyridin-3-ylprop-2-enamide —— C21H19F3N4O
(Z)-N-[(1R)-1-[5-methyl-1-[3-(trifluoromethyl)phenyl]pyrazol-4-yl]ethyl]-3-pyridin-3-ylprop-2-enamide
—— (2Z,4E)-N-[3-methyl-4-(tetrazol-1-yl)phenyl]hexa-2,4-dienamide —— C14H15N5O
(2Z,4E)-N-[3-methyl-4-(tetrazol-1-yl)phenyl]hexa-2,4-dienamide
—— (5E)-3-[[5-(4-chlorophenyl)-1,2,4-oxadiazol-3-yl]methyl]-5-(thiophen-2-ylmethylidene)-1,3-thiazolidine-2,4-dione —— C17H10ClN3O3S2
(5E)-3-[[5-(4-chlorophenyl)-1,2,4-oxadiazol-3-yl]methyl]-5-(thiophen-2-ylmethylidene)-1,3-thiazolidine-2,4-dione
—— 1,5-dimethyl-4-[(Z)-(3-oxo-1H-inden-2-ylidene)methyl]-2-phenylpyrazol-3-one —— C21H18N2O2
1,5-dimethyl-4-[(Z)-(3-oxo-1H-inden-2-ylidene)methyl]-2-phenylpyrazol-3-one
—— 2-(4-fluorophenyl)-4-[[(Z)-3-phenylprop-2-enyl]sulfonylmethyl]-1,3-oxazole —— C19H16FNO3S
2-(4-fluorophenyl)-4-[[(Z)-3-phenylprop-2-enyl]sulfonylmethyl]-1,3-oxazole
—— (Z)-2-cyano-N-(2,4-dichlorophenyl)-3-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)prop-2-enamide —— C21H16Cl2N4O2
(Z)-2-cyano-N-(2,4-dichlorophenyl)-3-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)prop-2-enamide
—— 4-[(2R)-2-hydroxy-3-(7-methyl-2,3-dihydro-1,4-benzoxazin-4-yl)propyl]-3-phenyl-1,2,4-oxadiazol-5-one —— C20H21N3O4
4-[(2R)-2-hydroxy-3-(7-methyl-2,3-dihydro-1,4-benzoxazin-4-yl)propyl]-3-phenyl-1,2,4-oxadiazol-5-one
—— 4-[(Z)-(6-methoxy-1-oxo-3,4-dihydronaphthalen-2-ylidene)methyl]-1,5-dimethyl-2-phenylpyrazol-3-one —— C23H22N2O3
4-[(Z)-(6-methoxy-1-oxo-3,4-dihydronaphthalen-2-ylidene)methyl]-1,5-dimethyl-2-phenylpyrazol-3-one
—— 1,5-dimethyl-4-[(Z)-3-oxo-3-[3-(2-oxopyrrolidin-1-yl)phenyl]prop-1-enyl]-2-phenylpyrazol-3-one —— C24H23N3O3
1,5-dimethyl-4-[(Z)-3-oxo-3-[3-(2-oxopyrrolidin-1-yl)phenyl]prop-1-enyl]-2-phenylpyrazol-3-one
—— propan-2-yl (Z)-2-cyano-3-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)prop-2-enoate —— C18H19N3O3
propan-2-yl (Z)-2-cyano-3-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)prop-2-enoate
—— 4-[(2S)-2-hydroxy-3-(7-methyl-2,3-dihydro-1,4-benzoxazin-4-yl)propyl]-3-phenyl-1,2,4-oxadiazol-5-one —— C20H21N3O4
4-[(2S)-2-hydroxy-3-(7-methyl-2,3-dihydro-1,4-benzoxazin-4-yl)propyl]-3-phenyl-1,2,4-oxadiazol-5-one
—— N-[3-[[(Z)-3-(1-phenylpyrazol-4-yl)prop-2-enoyl]amino]phenyl]cyclopropanecarboxamide —— C22H20N4O2
N-[3-[[(Z)-3-(1-phenylpyrazol-4-yl)prop-2-enoyl]amino]phenyl]cyclopropanecarboxamide
—— (Z)-3-[3-(4-fluorophenyl)-1-phenylpyrazol-4-yl]-N-[4-[2-(methylamino)-2-oxoethyl]phenyl]prop-2-enamide —— C27H23FN4O2
(Z)-3-[3-(4-fluorophenyl)-1-phenylpyrazol-4-yl]-N-[4-[2-(methylamino)-2-oxoethyl]phenyl]prop-2-enamide
—— 4-[[(2-tert-butyl-1,3-thiazol-5-yl)methylamino]methyl]-N-[(1S)-1-phenylethyl]oxan-4-amine —— C22H33N3OS
4-[[(2-tert-butyl-1,3-thiazol-5-yl)methylamino]methyl]-N-[(1S)-1-phenylethyl]oxan-4-amine
—— 3-[3-phenyl-4-[[[1-[[(1R)-1-phenylethyl]amino]cyclopentyl]methylamino]methyl]pyrazol-1-yl]propanenitrile —— C27H33N5
3-[3-phenyl-4-[[[1-[[(1R)-1-phenylethyl]amino]cyclopentyl]methylamino]methyl]pyrazol-1-yl]propanenitrile
—— 3-[3-phenyl-4-[[[1-[[(1S)-1-phenylethyl]amino]cyclopentyl]methylamino]methyl]pyrazol-1-yl]propanenitrile —— C27H33N5
3-[3-phenyl-4-[[[1-[[(1S)-1-phenylethyl]amino]cyclopentyl]methylamino]methyl]pyrazol-1-yl]propanenitrile
—— 2-[2-[(2S,3S)-2,3-dimethylthiomorpholin-4-yl]ethyl]-[1,2,4]triazolo[4,3-a]pyridin-3-one —— C14H20N4OS
2-[2-[(2S,3S)-2,3-dimethylthiomorpholin-4-yl]ethyl]-[1,2,4]triazolo[4,3-a]pyridin-3-one
—— 4-N-(5-methyl-1,2-oxazol-3-yl)-1-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]piperidine-1,4-dicarboxamide —— C21H25N7O3
4-N-(5-methyl-1,2-oxazol-3-yl)-1-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]piperidine-1,4-dicarboxamide
—— (2S)-N-[5-tert-butyl-2-(2,4-dimethylphenyl)pyrazol-3-yl]-2-(1,2,4-triazol-1-yl)propanamide —— C20H26N6O
(2S)-N-[5-tert-butyl-2-(2,4-dimethylphenyl)pyrazol-3-yl]-2-(1,2,4-triazol-1-yl)propanamide
—— 2-[2-[(2S,3R)-2,3-dimethylthiomorpholin-4-yl]ethyl]-[1,2,4]triazolo[4,3-a]pyridin-3-one —— C14H20N4OS
2-[2-[(2S,3R)-2,3-dimethylthiomorpholin-4-yl]ethyl]-[1,2,4]triazolo[4,3-a]pyridin-3-one
—— 4-[[(2-tert-butyl-1,3-thiazol-5-yl)methylamino]methyl]-N-[(1R)-1-phenylethyl]oxan-4-amine —— C22H33N3OS
4-[[(2-tert-butyl-1,3-thiazol-5-yl)methylamino]methyl]-N-[(1R)-1-phenylethyl]oxan-4-amine
—— 1-[2-pyrazol-1-yl-5-(trifluoromethyl)phenyl]-3-[(6S)-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-yl]urea —— C17H16F3N7O
1-[2-pyrazol-1-yl-5-(trifluoromethyl)phenyl]-3-[(6S)-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-yl]urea
—— [1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]-[(2R)-2-methyl-1,1-dioxo-1,4-thiazinan-4-yl]methanone —— C17H20FN3O3S
[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]-[(2R)-2-methyl-1,1-dioxo-1,4-thiazinan-4-yl]methanone