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—— (7S)-7-(5-bromo-2-propoxyphenyl)-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C22H22BrN5O2
(7S)-7-(5-bromo-2-propoxyphenyl)-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-[3-ethoxy-4-[(4-methylphenyl)methoxy]phenyl]-5-methyl-N-phenyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C28H28N6O3
(7R)-7-[3-ethoxy-4-[(4-methylphenyl)methoxy]phenyl]-5-methyl-N-phenyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-5-methyl-N-(2-methylphenyl)-7-[2-[(2-methylphenyl)methoxy]phenyl]-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H27N5O2
(7S)-5-methyl-N-(2-methylphenyl)-7-[2-[(2-methylphenyl)methoxy]phenyl]-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-5-methyl-7-[4-(3-methylbutoxy)phenyl]-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C24H27N5O2
(7R)-5-methyl-7-[4-(3-methylbutoxy)phenyl]-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— 7-[(R)-(1-benzyltetrazol-5-yl)-(4-cyclohexylpiperazin-1-yl)methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C29H33N7O3
7-[(R)-(1-benzyltetrazol-5-yl)-(4-cyclohexylpiperazin-1-yl)methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— (7S)-7-[5-bromo-2-[(2-chlorophenyl)methoxy]phenyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C20H17BrClN5O2
(7S)-7-[5-bromo-2-[(2-chlorophenyl)methoxy]phenyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— 7-[(S)-[1-[(4-fluorophenyl)methyl]tetrazol-5-yl]-(4-methylpiperazin-1-yl)methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C24H24FN7O3
7-[(S)-[1-[(4-fluorophenyl)methyl]tetrazol-5-yl]-(4-methylpiperazin-1-yl)methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— 7-[(R)-[1-[(4-fluorophenyl)methyl]tetrazol-5-yl]-(4-hydroxypiperidin-1-yl)methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C24H23FN6O4
7-[(R)-[1-[(4-fluorophenyl)methyl]tetrazol-5-yl]-(4-hydroxypiperidin-1-yl)methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— (7R)-7-[3-ethoxy-4-[(3-methylphenyl)methoxy]phenyl]-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C22H24N6O3
(7R)-7-[3-ethoxy-4-[(3-methylphenyl)methoxy]phenyl]-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-5-methyl-N-phenyl-7-(3-propan-2-yloxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C22H23N5O2
(7S)-5-methyl-N-phenyl-7-(3-propan-2-yloxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— 7-[(R)-[4-(4-methoxyphenyl)piperazin-1-yl]-[1-(2-methylbutan-2-yl)tetrazol-5-yl]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C28H33N7O4
7-[(R)-[4-(4-methoxyphenyl)piperazin-1-yl]-[1-(2-methylbutan-2-yl)tetrazol-5-yl]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— 7-[(R)-[4-(4-fluorophenyl)-3,6-dihydro-2H-pyridin-1-yl]-[1-(2-methylbutan-2-yl)tetrazol-5-yl]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C28H29FN6O3
7-[(R)-[4-(4-fluorophenyl)-3,6-dihydro-2H-pyridin-1-yl]-[1-(2-methylbutan-2-yl)tetrazol-5-yl]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— (7S)-7-[4-[(2-chloro-6-fluorophenyl)methoxy]-3-methoxyphenyl]-5-methyl-N-phenyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C26H22ClFN6O3
(7S)-7-[4-[(2-chloro-6-fluorophenyl)methoxy]-3-methoxyphenyl]-5-methyl-N-phenyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— 7-[(R)-2,3-dihydroindol-1-yl-[1-[(4-methoxyphenyl)methyl]tetrazol-5-yl]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C28H24N6O4
7-[(R)-2,3-dihydroindol-1-yl-[1-[(4-methoxyphenyl)methyl]tetrazol-5-yl]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— 7-[(R)-2,3-dihydroindol-1-yl-[1-(2-methylbutan-2-yl)tetrazol-5-yl]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C25H26N6O3
7-[(R)-2,3-dihydroindol-1-yl-[1-(2-methylbutan-2-yl)tetrazol-5-yl]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— (7S)-7-[3-ethoxy-4-[(2-fluorophenyl)methoxy]phenyl]-5-methyl-N-(2-methylphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C28H27FN6O3
(7S)-7-[3-ethoxy-4-[(2-fluorophenyl)methoxy]phenyl]-5-methyl-N-(2-methylphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(4-butoxy-3-ethoxyphenyl)-5-methyl-N-(2-methylphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C25H30N6O3
(7S)-7-(4-butoxy-3-ethoxyphenyl)-5-methyl-N-(2-methylphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-[3-ethoxy-4-[(4-methylphenyl)methoxy]phenyl]-5-methyl-N-(2-methylphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C29H30N6O3
(7R)-7-[3-ethoxy-4-[(4-methylphenyl)methoxy]phenyl]-5-methyl-N-(2-methylphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-[4-[(2-fluorophenyl)methoxy]phenyl]-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C19H17FN6O2
(7S)-7-[4-[(2-fluorophenyl)methoxy]phenyl]-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-[3-ethoxy-4-[(4-methylphenyl)methoxy]phenyl]-N-(2-methoxyphenyl)-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C29H30N6O4
(7S)-7-[3-ethoxy-4-[(4-methylphenyl)methoxy]phenyl]-N-(2-methoxyphenyl)-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-[4-[(3-chlorophenyl)methoxy]phenyl]-5-methyl-N-phenyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C25H21ClN6O2
(7R)-7-[4-[(3-chlorophenyl)methoxy]phenyl]-5-methyl-N-phenyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-[3-bromo-4-[(2-fluorophenyl)methoxy]-5-methoxyphenyl]-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C20H18BrFN6O3
(7S)-7-[3-bromo-4-[(2-fluorophenyl)methoxy]-5-methoxyphenyl]-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— 7-[(R)-[4-(2,3-dimethylphenyl)piperazin-1-yl]-[1-(2-methylbutan-2-yl)tetrazol-5-yl]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C29H35N7O3
7-[(R)-[4-(2,3-dimethylphenyl)piperazin-1-yl]-[1-(2-methylbutan-2-yl)tetrazol-5-yl]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— 7-[(S)-[1-[(4-methoxyphenyl)methyl]tetrazol-5-yl]-(4-methylpiperidin-1-yl)methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C26H28N6O4
7-[(S)-[1-[(4-methoxyphenyl)methyl]tetrazol-5-yl]-(4-methylpiperidin-1-yl)methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— 7-[(R)-[4-(4-hydroxyphenyl)piperazin-1-yl]-[1-(2-methylbutan-2-yl)tetrazol-5-yl]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C27H31N7O4
7-[(R)-[4-(4-hydroxyphenyl)piperazin-1-yl]-[1-(2-methylbutan-2-yl)tetrazol-5-yl]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— 7-[(R)-[1-[(4-methoxyphenyl)methyl]tetrazol-5-yl]-piperidin-1-ylmethyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C25H26N6O4
7-[(R)-[1-[(4-methoxyphenyl)methyl]tetrazol-5-yl]-piperidin-1-ylmethyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— (7R)-5-methyl-N-(2-methylphenyl)-7-[4-(2-phenylethoxy)phenyl]-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C27H26N6O2
(7R)-5-methyl-N-(2-methylphenyl)-7-[4-(2-phenylethoxy)phenyl]-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— 7-[(R)-[4-(2,5-dimethylphenyl)piperazin-1-yl]-[1-(2-methylbutan-2-yl)tetrazol-5-yl]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C29H35N7O3
7-[(R)-[4-(2,5-dimethylphenyl)piperazin-1-yl]-[1-(2-methylbutan-2-yl)tetrazol-5-yl]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— 7-[(S)-[1-[(4-fluorophenyl)methyl]tetrazol-5-yl]-(4-propylpiperazin-1-yl)methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C26H28FN7O3
7-[(S)-[1-[(4-fluorophenyl)methyl]tetrazol-5-yl]-(4-propylpiperazin-1-yl)methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— (7R)-7-[3-bromo-5-ethoxy-4-[(3-methylphenyl)methoxy]phenyl]-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C22H23BrN6O3
(7R)-7-[3-bromo-5-ethoxy-4-[(3-methylphenyl)methoxy]phenyl]-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— 7-[(R)-[1-[(4-methoxyphenyl)methyl]tetrazol-5-yl]-pyrrolidin-1-ylmethyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C24H24N6O4
7-[(R)-[1-[(4-methoxyphenyl)methyl]tetrazol-5-yl]-pyrrolidin-1-ylmethyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— (7S)-7-[3-methoxy-4-(3-methylbutoxy)phenyl]-5-methyl-N-(2-methylphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C25H30N6O3
(7S)-7-[3-methoxy-4-(3-methylbutoxy)phenyl]-5-methyl-N-(2-methylphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— 7-methoxy-3-[(R)-[1-(2-methylbutan-2-yl)tetrazol-5-yl]-[(3R)-3-methylpiperidin-1-yl]methyl]-1H-quinolin-2-one —— C23H32N6O2
7-methoxy-3-[(R)-[1-(2-methylbutan-2-yl)tetrazol-5-yl]-[(3R)-3-methylpiperidin-1-yl]methyl]-1H-quinolin-2-one
—— (7R)-7-(4-hexoxy-3-methoxyphenyl)-5-methyl-N-(2-methylphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C26H32N6O3
(7R)-7-(4-hexoxy-3-methoxyphenyl)-5-methyl-N-(2-methylphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-[3-ethoxy-4-[(3-methylphenyl)methoxy]phenyl]-5-methyl-N-phenyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C28H28N6O3
(7R)-7-[3-ethoxy-4-[(3-methylphenyl)methoxy]phenyl]-5-methyl-N-phenyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(4-hexoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C19H25N5O2
(7S)-7-(4-hexoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-[4-[(2-chlorophenyl)methoxy]-3-ethoxyphenyl]-5-methyl-N-phenyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C27H25ClN6O3
(7R)-7-[4-[(2-chlorophenyl)methoxy]-3-ethoxyphenyl]-5-methyl-N-phenyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-5-methyl-N-phenyl-7-(3-propan-2-yloxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C22H23N5O2
(7R)-5-methyl-N-phenyl-7-(3-propan-2-yloxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(2-methoxyphenyl)-5-methyl-7-[4-(2-phenylethoxy)phenyl]-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C27H26N6O3
(7S)-N-(2-methoxyphenyl)-5-methyl-7-[4-(2-phenylethoxy)phenyl]-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-[4-[(2-chlorophenyl)methoxy]-3-methoxyphenyl]-5-methyl-N-(2-methylphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C27H25ClN6O3
(7R)-7-[4-[(2-chlorophenyl)methoxy]-3-methoxyphenyl]-5-methyl-N-(2-methylphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-[4-[(2-fluorophenyl)methoxy]-3-methoxyphenyl]-5-methyl-N-(2-methylphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C27H25FN6O3
(7S)-7-[4-[(2-fluorophenyl)methoxy]-3-methoxyphenyl]-5-methyl-N-(2-methylphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— 7-[(R)-(4-benzylpiperidin-1-yl)-[1-(2-methylbutan-2-yl)tetrazol-5-yl]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C29H34N6O3
7-[(R)-(4-benzylpiperidin-1-yl)-[1-(2-methylbutan-2-yl)tetrazol-5-yl]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— (7S)-7-[4-[(3-bromophenyl)methoxy]-3-methoxyphenyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C21H20BrN5O3
(7S)-7-[4-[(3-bromophenyl)methoxy]-3-methoxyphenyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-[4-[(4-tert-butylphenyl)methoxy]phenyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C24H27N5O2
(7S)-7-[4-[(4-tert-butylphenyl)methoxy]phenyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-[3-methoxy-4-(2-morpholin-4-yl-2-oxoethoxy)phenyl]-5-methyl-N-phenyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C25H27N7O5
(7R)-7-[3-methoxy-4-(2-morpholin-4-yl-2-oxoethoxy)phenyl]-5-methyl-N-phenyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-(2,4-dimethylphenyl)-7-[4-[(2-fluorophenyl)methoxy]-3-methoxyphenyl]-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C28H27FN6O3
(7R)-N-(2,4-dimethylphenyl)-7-[4-[(2-fluorophenyl)methoxy]-3-methoxyphenyl]-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(4-butoxy-3-ethoxyphenyl)-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C18H24N6O3
(7R)-7-(4-butoxy-3-ethoxyphenyl)-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(4-hexoxyphenyl)-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C18H24N6O2
(7R)-7-(4-hexoxyphenyl)-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-(2-methoxyphenyl)-5-methyl-7-(4-propan-2-yloxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H25N5O3
(7R)-N-(2-methoxyphenyl)-5-methyl-7-(4-propan-2-yloxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(2-methoxyphenyl)-5-methyl-7-(4-propan-2-yloxyphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C22H24N6O3
(7S)-N-(2-methoxyphenyl)-5-methyl-7-(4-propan-2-yloxyphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide