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—— 7-[(R)-(1-benzyltetrazol-5-yl)-[4-(furan-2-ylmethyl)piperazin-1-yl]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C28H27N7O4
7-[(R)-(1-benzyltetrazol-5-yl)-[4-(furan-2-ylmethyl)piperazin-1-yl]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— 7-[(R)-(1-tert-butyltetrazol-5-yl)-[4-(4-fluorophenyl)piperazin-1-yl]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C26H28FN7O3
7-[(R)-(1-tert-butyltetrazol-5-yl)-[4-(4-fluorophenyl)piperazin-1-yl]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— 7-[(R)-(1-tert-butyltetrazol-5-yl)-[4-(4-methoxyphenyl)piperazin-1-yl]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C27H31N7O4
7-[(R)-(1-tert-butyltetrazol-5-yl)-[4-(4-methoxyphenyl)piperazin-1-yl]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— 7-[(R)-(1-tert-butyltetrazol-5-yl)-morpholin-4-ylmethyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C20H24N6O4
7-[(R)-(1-tert-butyltetrazol-5-yl)-morpholin-4-ylmethyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— 7-[(S)-(4-hydroxyphenyl)-[(4-methylpyridin-1-ium-2-yl)amino]methyl]-2-methylquinolin-8-olate —— C23H21N3O2
7-[(S)-(4-hydroxyphenyl)-[(4-methylpyridin-1-ium-2-yl)amino]methyl]-2-methylquinolin-8-olate
—— (7S)-7-(4-tert-butylphenyl)-2-butylsulfanyl-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H35N5OS
(7S)-7-(4-tert-butylphenyl)-2-butylsulfanyl-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-(2,3-dimethylphenyl)-5-methyl-2-propylsulfanyl-7-thiophen-2-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C22H25N5OS2
(7R)-N-(2,3-dimethylphenyl)-5-methyl-2-propylsulfanyl-7-thiophen-2-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-(2,3-dimethylphenyl)-5-methyl-7-naphthalen-1-yl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C24H22N6O
(7R)-N-(2,3-dimethylphenyl)-5-methyl-7-naphthalen-1-yl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(3-bromo-4,5-dimethoxyphenyl)-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C22H22BrN5O3
(7R)-7-(3-bromo-4,5-dimethoxyphenyl)-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-(2,3-dimethylphenyl)-7-(3-fluorophenyl)-5-methyl-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C24H26FN5OS
(7R)-N-(2,3-dimethylphenyl)-7-(3-fluorophenyl)-5-methyl-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-5-methyl-N-(3-methylphenyl)-7-(3-methylthiophen-2-yl)-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C22H25N5OS2
(7R)-5-methyl-N-(3-methylphenyl)-7-(3-methylthiophen-2-yl)-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(2-ethoxyphenyl)-2-ethylsulfanyl-5-methyl-7-thiophen-2-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C21H23N5O2S2
(7S)-N-(2-ethoxyphenyl)-2-ethylsulfanyl-5-methyl-7-thiophen-2-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-[4-[2-(diethylamino)-2-oxoethoxy]-3-methoxyphenyl]-5-methyl-N-(3-methylphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C26H31N7O4
(7S)-7-[4-[2-(diethylamino)-2-oxoethoxy]-3-methoxyphenyl]-5-methyl-N-(3-methylphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(2-ethoxyphenyl)-2-ethylsulfanyl-5-methyl-7-naphthalen-1-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H27N5O2S
(7S)-N-(2-ethoxyphenyl)-2-ethylsulfanyl-5-methyl-7-naphthalen-1-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-(2,3-dimethylphenyl)-7-(3-fluorophenyl)-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C20H19FN6O
(7R)-N-(2,3-dimethylphenyl)-7-(3-fluorophenyl)-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(4-butoxy-3-methoxyphenyl)-N-(2,3-dimethylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C26H31N5O3
(7R)-7-(4-butoxy-3-methoxyphenyl)-N-(2,3-dimethylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-[4-[(2-chlorophenyl)methoxy]phenyl]-N-(2,3-dimethylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H26ClN5O2
(7R)-7-[4-[(2-chlorophenyl)methoxy]phenyl]-N-(2,3-dimethylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(3-fluorophenyl)-5-methyl-N-(3-methylphenyl)-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H24FN5OS
(7R)-7-(3-fluorophenyl)-5-methyl-N-(3-methylphenyl)-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(3-bromo-4,5-dimethoxyphenyl)-N-(2,3-dimethylphenyl)-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C22H23BrN6O3
(7R)-7-(3-bromo-4,5-dimethoxyphenyl)-N-(2,3-dimethylphenyl)-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-(2-ethoxyphenyl)-7-[3-methoxy-4-[(3-methylphenyl)methoxy]phenyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C30H31N5O4
(7R)-N-(2-ethoxyphenyl)-7-[3-methoxy-4-[(3-methylphenyl)methoxy]phenyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(2,3-dimethylphenyl)-7-(3-fluorophenyl)-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C20H19FN6O
(7S)-N-(2,3-dimethylphenyl)-7-(3-fluorophenyl)-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(3-methoxy-4-propoxyphenyl)-5-methyl-N-(3-methylphenyl)-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H33N5O3S
(7S)-7-(3-methoxy-4-propoxyphenyl)-5-methyl-N-(3-methylphenyl)-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(4-tert-butylphenyl)-N-(2,3-dimethylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C25H29N5O
(7R)-7-(4-tert-butylphenyl)-N-(2,3-dimethylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-ethylsulfanyl-5-methyl-N-(3-methylphenyl)-7-naphthalen-1-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C26H25N5OS
(7R)-2-ethylsulfanyl-5-methyl-N-(3-methylphenyl)-7-naphthalen-1-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-butylsulfanyl-N-(2-ethoxyphenyl)-7-(4-ethylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H33N5O2S
(7S)-2-butylsulfanyl-N-(2-ethoxyphenyl)-7-(4-ethylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-[3-methoxy-4-(3-methylbutoxy)phenyl]-5-methyl-N-(3-methylphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C25H30N6O3
(7S)-7-[3-methoxy-4-(3-methylbutoxy)phenyl]-5-methyl-N-(3-methylphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(4-tert-butylphenyl)-N-(2,3-dimethylphenyl)-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C24H28N6O
(7R)-7-(4-tert-butylphenyl)-N-(2,3-dimethylphenyl)-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-butylsulfanyl-N-(2-ethoxyphenyl)-7-(3-fluorophenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C25H28FN5O2S
(7S)-2-butylsulfanyl-N-(2-ethoxyphenyl)-7-(3-fluorophenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(5-bromofuran-2-yl)-2-butylsulfanyl-N-(2,3-dimethylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H26BrN5O2S
(7S)-7-(5-bromofuran-2-yl)-2-butylsulfanyl-N-(2,3-dimethylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-(2-ethoxyphenyl)-2-ethylsulfanyl-5-methyl-7-naphthalen-1-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H27N5O2S
(7R)-N-(2-ethoxyphenyl)-2-ethylsulfanyl-5-methyl-7-naphthalen-1-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-(2,3-dimethylphenyl)-5-methyl-7-(3-methylthiophen-2-yl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C19H20N6OS
(7R)-N-(2,3-dimethylphenyl)-5-methyl-7-(3-methylthiophen-2-yl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-ethylsulfanyl-7-[3-methoxy-4-(3-methylbutoxy)phenyl]-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H35N5O3S
(7R)-2-ethylsulfanyl-7-[3-methoxy-4-(3-methylbutoxy)phenyl]-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-5-methyl-N-(3-methylphenyl)-7-thiophen-2-yl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C17H16N6OS
(7R)-5-methyl-N-(3-methylphenyl)-7-thiophen-2-yl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-(2,3-dimethylphenyl)-7-(3-ethoxyphenyl)-5-methyl-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C26H31N5O2S
(7R)-N-(2,3-dimethylphenyl)-7-(3-ethoxyphenyl)-5-methyl-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(4-tert-butylphenyl)-N-(2,3-dimethylphenyl)-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C24H28N6O
(7S)-7-(4-tert-butylphenyl)-N-(2,3-dimethylphenyl)-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(3-bromo-5-methoxy-4-propoxyphenyl)-N-(2,3-dimethylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C25H28BrN5O3
(7S)-7-(3-bromo-5-methoxy-4-propoxyphenyl)-N-(2,3-dimethylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(3-methoxy-4-propan-2-yloxyphenyl)-5-methyl-N-(3-methylphenyl)-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H33N5O3S
(7R)-7-(3-methoxy-4-propan-2-yloxyphenyl)-5-methyl-N-(3-methylphenyl)-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(3,4-dichlorophenyl)-5-methyl-N-(3-methylphenyl)-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H23Cl2N5OS
(7S)-7-(3,4-dichlorophenyl)-5-methyl-N-(3-methylphenyl)-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(4-butoxyphenyl)-5-methyl-N-(3-methylphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C23H26N6O2
(7R)-7-(4-butoxyphenyl)-5-methyl-N-(3-methylphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(4-bromophenyl)-N-(2,3-dimethylphenyl)-5-methyl-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C24H26BrN5OS
(7S)-7-(4-bromophenyl)-N-(2,3-dimethylphenyl)-5-methyl-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(3-bromo-4-ethoxy-5-methoxyphenyl)-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H24BrN5O3
(7R)-7-(3-bromo-4-ethoxy-5-methoxyphenyl)-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(2,4-dimethoxyphenyl)-N-(2-ethoxyphenyl)-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C25H29N5O4S
(7S)-7-(2,4-dimethoxyphenyl)-N-(2-ethoxyphenyl)-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(3-bromo-4-ethoxy-5-methoxyphenyl)-5-methyl-N-(3-methylphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C22H23BrN6O3
(7R)-7-(3-bromo-4-ethoxy-5-methoxyphenyl)-5-methyl-N-(3-methylphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-(2-ethoxyphenyl)-7-(4-ethoxyphenyl)-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C25H29N5O3S
(7R)-N-(2-ethoxyphenyl)-7-(4-ethoxyphenyl)-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(4-butoxyphenyl)-N-(2-ethoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C25H29N5O3
(7S)-7-(4-butoxyphenyl)-N-(2-ethoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-(2,3-dimethylphenyl)-5-methyl-7-[(E)-2-phenylethenyl]-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C26H29N5OS
(7R)-N-(2,3-dimethylphenyl)-5-methyl-7-[(E)-2-phenylethenyl]-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(2-ethoxyphenyl)-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C22H23N5O2
(7S)-7-(2-ethoxyphenyl)-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-5-methyl-N-(3-methylphenyl)-7-thiophen-2-yl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C17H16N6OS
(7S)-5-methyl-N-(3-methylphenyl)-7-thiophen-2-yl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-(2,3-dimethylphenyl)-7-(4-ethylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H25N5O
(7R)-N-(2,3-dimethylphenyl)-7-(4-ethylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(2,3-dimethylphenyl)-5-methyl-7-(4-propoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C24H27N5O2
(7S)-N-(2,3-dimethylphenyl)-5-methyl-7-(4-propoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide