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—— (7S)-2-ethylsulfanyl-5-methyl-7-[4-(3-methylbutoxy)phenyl]-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C26H31N5O2S
(7S)-2-ethylsulfanyl-5-methyl-7-[4-(3-methylbutoxy)phenyl]-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(3-ethoxyphenyl)-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C17H21N5O2S
(7R)-7-(3-ethoxyphenyl)-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(3-chlorophenyl)-2-ethylsulfanyl-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C21H20ClN5OS
(7S)-7-(3-chlorophenyl)-2-ethylsulfanyl-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— 7-[2-[(4aS,9bR)-2,8-dimethyl-3,4,4a,9b-tetrahydro-1H-pyrido[4,3-b]indol-5-yl]-2-oxoethyl]-1,3-dimethylpurine-2,6-dione —— C22H26N6O3
7-[2-[(4aS,9bR)-2,8-dimethyl-3,4,4a,9b-tetrahydro-1H-pyrido[4,3-b]indol-5-yl]-2-oxoethyl]-1,3-dimethylpurine-2,6-dione
—— (7S)-7-[3-[(4-chlorophenyl)methoxy]phenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C22H22ClN5O2S
(7S)-7-[3-[(4-chlorophenyl)methoxy]phenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-ethylsulfanyl-7-(2-methoxyphenyl)-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C22H23N5O2S
(7S)-2-ethylsulfanyl-7-(2-methoxyphenyl)-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(3-bromo-4,5-diethoxyphenyl)-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C19H24BrN5O3S
(7R)-7-(3-bromo-4,5-diethoxyphenyl)-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-[3-ethoxy-4-[(2-fluorophenyl)methoxy]phenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C24H26FN5O3S
(7R)-7-[3-ethoxy-4-[(2-fluorophenyl)methoxy]phenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-[3-ethoxy-4-[(4-methylphenyl)methoxy]phenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C25H29N5O3S
(7R)-7-[3-ethoxy-4-[(4-methylphenyl)methoxy]phenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-[4-[(2-chloro-6-fluorophenyl)methoxy]-3-methoxyphenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H23ClFN5O3S
(7S)-7-[4-[(2-chloro-6-fluorophenyl)methoxy]-3-methoxyphenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-ethylsulfanyl-5-methyl-7-(4-pentoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C20H27N5O2S
(7S)-2-ethylsulfanyl-5-methyl-7-(4-pentoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-ethylsulfanyl-5-methyl-7-(4-propan-2-yloxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C18H23N5O2S
(7S)-2-ethylsulfanyl-5-methyl-7-(4-propan-2-yloxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-ethylsulfanyl-5-methyl-7-(3-methylthiophen-2-yl)-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C20H21N5OS2
(7R)-2-ethylsulfanyl-5-methyl-7-(3-methylthiophen-2-yl)-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-ethylsulfanyl-7-[3-methoxy-4-(3-methylbutoxy)phenyl]-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H33N5O3S
(7S)-2-ethylsulfanyl-7-[3-methoxy-4-(3-methylbutoxy)phenyl]-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-[3-[(2,4-dichlorophenyl)methoxy]phenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C22H21Cl2N5O2S
(7R)-7-[3-[(2,4-dichlorophenyl)methoxy]phenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-[5-bromo-2-[(2-methylphenyl)methoxy]phenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H24BrN5O2S
(7R)-7-[5-bromo-2-[(2-methylphenyl)methoxy]phenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-ethylsulfanyl-5-methyl-7-[4-(2-phenylethoxy)phenyl]-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H25N5O2S
(7S)-2-ethylsulfanyl-5-methyl-7-[4-(2-phenylethoxy)phenyl]-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-ethylsulfanyl-7-(3-methoxy-4-propan-2-yloxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C19H25N5O3S
(7R)-2-ethylsulfanyl-7-(3-methoxy-4-propan-2-yloxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-ethylsulfanyl-7-(4-hexoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C21H29N5O2S
(7S)-2-ethylsulfanyl-7-(4-hexoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-[4-[(4-tert-butylphenyl)methoxy]-3-methoxyphenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H33N5O3S
(7R)-7-[4-[(4-tert-butylphenyl)methoxy]-3-methoxyphenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(3-bromo-5-ethoxy-4-methoxyphenyl)-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C18H22BrN5O3S
(7S)-7-(3-bromo-5-ethoxy-4-methoxyphenyl)-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-[4-[(2,6-dichlorophenyl)methoxy]phenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C22H21Cl2N5O2S
(7S)-7-[4-[(2,6-dichlorophenyl)methoxy]phenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(3-bromo-5-ethoxy-4-methoxyphenyl)-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C18H22BrN5O3S
(7R)-7-(3-bromo-5-ethoxy-4-methoxyphenyl)-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-[4-[(2-chloro-6-fluorophenyl)methoxy]-3-methoxyphenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H23ClFN5O3S
(7R)-7-[4-[(2-chloro-6-fluorophenyl)methoxy]-3-methoxyphenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-[2-[(4-tert-butylphenyl)methoxy]phenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C26H31N5O2S
(7S)-7-[2-[(4-tert-butylphenyl)methoxy]phenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-ethylsulfanyl-5-methyl-N-phenyl-7-(3-propoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C24H27N5O2S
(7S)-2-ethylsulfanyl-5-methyl-N-phenyl-7-(3-propoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(3-chlorophenyl)-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C15H16ClN5OS
(7R)-7-(3-chlorophenyl)-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-[2-[(4-chlorophenyl)methoxy]phenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C22H22ClN5O2S
(7S)-7-[2-[(4-chlorophenyl)methoxy]phenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(4-butoxyphenyl)-2-ethylsulfanyl-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C25H29N5O2S
(7S)-7-(4-butoxyphenyl)-2-ethylsulfanyl-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(3-ethoxyphenyl)-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C17H21N5O2S
(7S)-7-(3-ethoxyphenyl)-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-[2-[(2,4-dichlorophenyl)methoxy]phenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C22H21Cl2N5O2S
(7R)-7-[2-[(2,4-dichlorophenyl)methoxy]phenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(3-chlorophenyl)-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C15H16ClN5OS
(7S)-7-(3-chlorophenyl)-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-butylsulfanyl-5-methyl-7-[2-[(4-methylphenyl)methoxy]phenyl]-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C25H29N5O2S
(7S)-2-butylsulfanyl-5-methyl-7-[2-[(4-methylphenyl)methoxy]phenyl]-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-butylsulfanyl-7-(3-ethoxyphenyl)-N-(2-methoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C26H31N5O3S
(7R)-2-butylsulfanyl-7-(3-ethoxyphenyl)-N-(2-methoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-butylsulfanyl-7-[3-methoxy-4-(3-methylbutoxy)phenyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H33N5O3S
(7R)-2-butylsulfanyl-7-[3-methoxy-4-(3-methylbutoxy)phenyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-[3-[(2-chlorophenyl)methoxy]phenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C22H22ClN5O2S
(7R)-7-[3-[(2-chlorophenyl)methoxy]phenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-ethylsulfanyl-7-(3-methoxy-4-pentoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C21H29N5O3S
(7S)-2-ethylsulfanyl-7-(3-methoxy-4-pentoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(3-chloro-4,5-dimethoxyphenyl)-N-(2-methoxyphenyl)-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C21H21ClN6O4
(7S)-7-(3-chloro-4,5-dimethoxyphenyl)-N-(2-methoxyphenyl)-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-butylsulfanyl-5-methyl-N-phenyl-7-(4-phenylmethoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C30H31N5O2S
(7R)-2-butylsulfanyl-5-methyl-N-phenyl-7-(4-phenylmethoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-butylsulfanyl-5-methyl-N-phenyl-7-(2-propoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C26H31N5O2S
(7R)-2-butylsulfanyl-5-methyl-N-phenyl-7-(2-propoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-butylsulfanyl-7-[3-[(2-chlorophenyl)methoxy]phenyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C24H26ClN5O2S
(7R)-2-butylsulfanyl-7-[3-[(2-chlorophenyl)methoxy]phenyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-[4-(dimethylamino)phenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C17H22N6OS
(7S)-7-[4-(dimethylamino)phenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-[2-[(4-tert-butylphenyl)methoxy]phenyl]-2-butylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H35N5O2S
(7R)-7-[2-[(4-tert-butylphenyl)methoxy]phenyl]-2-butylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-[3-ethoxy-4-[(2-fluorophenyl)methoxy]phenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C24H26FN5O3S
(7S)-7-[3-ethoxy-4-[(2-fluorophenyl)methoxy]phenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-butylsulfanyl-7-(4-ethoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C19H25N5O2S
(7R)-2-butylsulfanyl-7-(4-ethoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-butylsulfanyl-7-[4-[(3-chlorophenyl)methoxy]phenyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C24H26ClN5O2S
(7S)-2-butylsulfanyl-7-[4-[(3-chlorophenyl)methoxy]phenyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-butylsulfanyl-7-(4-ethoxy-3-methoxyphenyl)-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C26H31N5O3S
(7S)-2-butylsulfanyl-7-(4-ethoxy-3-methoxyphenyl)-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(3-bromo-5-ethoxy-4-methoxyphenyl)-2-butylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C20H26BrN5O3S
(7S)-7-(3-bromo-5-ethoxy-4-methoxyphenyl)-2-butylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-butylsulfanyl-7-[4-[(2,6-dichlorophenyl)methoxy]phenyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C24H25Cl2N5O2S
(7S)-2-butylsulfanyl-7-[4-[(2,6-dichlorophenyl)methoxy]phenyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-butylsulfanyl-7-[4-(dimethylamino)phenyl]-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C25H30N6OS
(7S)-2-butylsulfanyl-7-[4-(dimethylamino)phenyl]-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide