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中文名称 英文名称 CAS号 化学式 结构式图片
—— 7-[[4-(dimethylamino)phenyl]methyl]-2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H31N5O2
7-[[4-(dimethylamino)phenyl]methyl]-2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-chloro-N-[(1S,2S)-2-methylcyclohexyl]-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide —— C22H29ClN2O3
7-chloro-N-[(1S,2S)-2-methylcyclohexyl]-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide
—— 7-[2-[(3S)-3-methylpiperidin-1-yl]-2-oxoethyl]-8-oxo-9-propan-2-yl-2-thiophen-2-ylpurine-6-carboxamide —— C21H26N6O3S
7-[2-[(3S)-3-methylpiperidin-1-yl]-2-oxoethyl]-8-oxo-9-propan-2-yl-2-thiophen-2-ylpurine-6-carboxamide
—— 7-cyclohexyl-2-[(2R)-1-[(2S)-2-phenylpropanoyl]piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C27H36N4O2
7-cyclohexyl-2-[(2R)-1-[(2S)-2-phenylpropanoyl]piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-acetyl-2-[(2S)-1-[(2R)-2-phenylpropanoyl]piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H28N4O3
7-acetyl-2-[(2S)-1-[(2R)-2-phenylpropanoyl]piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-Chloro-4'-(3,3-dimethylpiperidine-1-carbonyl)spiro[3,4-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-5-one —— C22H29ClN2O3
7-Chloro-4'-(3,3-dimethylpiperidine-1-carbonyl)spiro[3,4-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-5-one
—— 7-(cyclopropanecarbonyl)-2-[(2R)-1-[(2S)-2-phenylpropanoyl]piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C25H30N4O3
7-(cyclopropanecarbonyl)-2-[(2R)-1-[(2S)-2-phenylpropanoyl]piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[1-[(1S,2R)-2-methylcyclopropanecarbonyl]piperidin-4-yl]-6H-1,6-naphthyridin-5-one —— C18H21N3O2
7-[1-[(1S,2R)-2-methylcyclopropanecarbonyl]piperidin-4-yl]-6H-1,6-naphthyridin-5-one
—— 7-methylsulfonyl-2-[(2S)-1-[(2S)-2-phenylpropanoyl]piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H28N4O4S
7-methylsulfonyl-2-[(2S)-1-[(2S)-2-phenylpropanoyl]piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(cyclopropanecarbonyl)-2-[(3S)-1-[(2R)-2-phenylpropanoyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H28N4O3
7-(cyclopropanecarbonyl)-2-[(3S)-1-[(2R)-2-phenylpropanoyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-methoxy-1'-[(3S)-1-[(2R)-1-methoxypropan-2-yl]-5-oxopyrrolidine-3-carbonyl]spiro[3H-chromene-2,4'-piperidine]-4-one —— C23H30N2O6
7-methoxy-1'-[(3S)-1-[(2R)-1-methoxypropan-2-yl]-5-oxopyrrolidine-3-carbonyl]spiro[3H-chromene-2,4'-piperidine]-4-one
—— 7-cyclopentyl-2-[(2S)-1-[(3S)-3-pyrazol-1-ylbutanoyl]piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H34N6O2
7-cyclopentyl-2-[(2S)-1-[(3S)-3-pyrazol-1-ylbutanoyl]piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-methoxy-1'-[(3R)-3-(1,2,4-triazol-1-yl)butanoyl]spiro[3H-chromene-2,4'-piperidine]-4-one —— C20H24N4O4
7-methoxy-1'-[(3R)-3-(1,2,4-triazol-1-yl)butanoyl]spiro[3H-chromene-2,4'-piperidine]-4-one
—— 7-[[(3S)-oxolan-3-yl]methyl]-2-propan-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C16H25N3O2
7-[[(3S)-oxolan-3-yl]methyl]-2-propan-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-(2,2-dimethylpropanoyl)-2-propan-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C16H25N3O2
7-(2,2-dimethylpropanoyl)-2-propan-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-methylsulfonyl-2-propan-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C12H19N3O3S
7-methylsulfonyl-2-propan-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-[(2-fluorophenyl)methyl]-2-propan-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C18H22FN3O
7-[(2-fluorophenyl)methyl]-2-propan-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-[(3S)-1-(3-propan-2-yl-1,2-oxazole-5-carbonyl)pyrrolidin-3-yl]-6H-1,6-naphthyridin-5-one —— C19H20N4O3
7-[(3S)-1-(3-propan-2-yl-1,2-oxazole-5-carbonyl)pyrrolidin-3-yl]-6H-1,6-naphthyridin-5-one
—— 7-[(3-methoxy-4-propan-2-yloxyphenyl)methyl]-2-morpholin-4-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C23H32N4O4
7-[(3-methoxy-4-propan-2-yloxyphenyl)methyl]-2-morpholin-4-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-Propan-2-yl-2-[1-(pyridine-4-carbonyl)piperidin-4-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C21H27N5O2
7-Propan-2-yl-2-[1-(pyridine-4-carbonyl)piperidin-4-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-chloro-N-[(2S)-3-methylbutan-2-yl]-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide —— C20H27ClN2O3
7-chloro-N-[(2S)-3-methylbutan-2-yl]-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide
—— 7-propan-2-yl-2-[(2R)-1-(4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H32N4O2S
7-propan-2-yl-2-[(2R)-1-(4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(4-methoxy-3-propan-2-yloxyphenyl)methyl]-2-morpholin-4-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C23H32N4O4
7-[(4-methoxy-3-propan-2-yloxyphenyl)methyl]-2-morpholin-4-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-(cyclohexylmethyl)-2-[(2R)-1-(2-thiophen-3-ylacetyl)pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H32N4O2S
7-(cyclohexylmethyl)-2-[(2R)-1-(2-thiophen-3-ylacetyl)pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-acetyl-2-[(2R)-1-[(4-propan-2-yloxyphenyl)methyl]pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H30N4O3
7-acetyl-2-[(2R)-1-[(4-propan-2-yloxyphenyl)methyl]pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-cyclohexyl-2-[(3R)-1-(pyrazine-2-carbonyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H28N6O2
7-cyclohexyl-2-[(3R)-1-(pyrazine-2-carbonyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-cyclopentyl-2-[(2R)-1-(4-imidazol-1-ylbutanoyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H34N6O2
7-cyclopentyl-2-[(2R)-1-(4-imidazol-1-ylbutanoyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(2,3-difluorophenyl)methyl]-2-pyridin-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C20H18F2N4O
7-[(2,3-difluorophenyl)methyl]-2-pyridin-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-[(6-Chloro-1,3-benzodioxol-5-yl)methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C20H17ClN4O3
7-[(6-Chloro-1,3-benzodioxol-5-yl)methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-cyclopentyl-2-[(2S)-1-(pyridine-2-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H29N5O2
7-cyclopentyl-2-[(2S)-1-(pyridine-2-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-cyclopentyl-2-[(2S)-1-(2-thiophen-3-ylacetyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H30N4O2S
7-cyclopentyl-2-[(2S)-1-(2-thiophen-3-ylacetyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[[(2R)-oxolan-2-yl]methyl]-2-pyrazin-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C17H21N5O2
7-[[(2R)-oxolan-2-yl]methyl]-2-pyrazin-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-[(4-fluorophenyl)methyl]-2-pyridin-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C20H19FN4O
7-[(4-fluorophenyl)methyl]-2-pyridin-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-[(2-Morpholin-4-ylpyrimidin-5-yl)methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C21H23N7O2
7-[(2-Morpholin-4-ylpyrimidin-5-yl)methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-cyclohexyl-2-[(3R)-1-(3-pyrazol-1-ylpropanoyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H32N6O2
7-cyclohexyl-2-[(3R)-1-(3-pyrazol-1-ylpropanoyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(cyclohexylmethyl)-2-[(2R)-1-(pyridine-2-carbonyl)pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H31N5O2
7-(cyclohexylmethyl)-2-[(2R)-1-(pyridine-2-carbonyl)pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-Chloro-3-[[4-hydroxy-1-(2-pyridin-2-ylacetyl)piperidin-4-yl]methyl]quinazolin-4-one —— C21H21ClN4O3
7-Chloro-3-[[4-hydroxy-1-(2-pyridin-2-ylacetyl)piperidin-4-yl]methyl]quinazolin-4-one
—— 7-(cyclopropanecarbonyl)-2-[(3R)-1-[2-(1H-indol-3-yl)acetyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C25H27N5O3
7-(cyclopropanecarbonyl)-2-[(3R)-1-[2-(1H-indol-3-yl)acetyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(2-Oxo-2-pyrrolidin-1-ylethyl)-5-phenyl-4,5,7,9,13-pentazatricyclo[7.4.0.02,6]trideca-1(13),2(6),3-trien-8-one —— C20H22N6O2
7-(2-Oxo-2-pyrrolidin-1-ylethyl)-5-phenyl-4,5,7,9,13-pentazatricyclo[7.4.0.02,6]trideca-1(13),2(6),3-trien-8-one
—— 7-[(2R)-1-(benzenesulfonyl)pyrrolidin-2-yl]-[1,2,4]triazolo[1,5-a]pyrimidine —— C15H15N5O2S
7-[(2R)-1-(benzenesulfonyl)pyrrolidin-2-yl]-[1,2,4]triazolo[1,5-a]pyrimidine
—— 7-(cyclopropanecarbonyl)-2-[(2R)-1-(3-phenylpropanoyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C25H30N4O3
7-(cyclopropanecarbonyl)-2-[(2R)-1-(3-phenylpropanoyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[[1-(2-Chlorophenyl)pyrrol-2-yl]methyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H20ClN5O
7-[[1-(2-Chlorophenyl)pyrrol-2-yl]methyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(3R)-1-(3-phenylpropanoyl)pyrrolidin-3-yl]-6H-1,6-naphthyridin-5-one —— C21H21N3O2
7-[(3R)-1-(3-phenylpropanoyl)pyrrolidin-3-yl]-6H-1,6-naphthyridin-5-one
—— 7-(cyclopropanecarbonyl)-2-[(2S)-1-(2-phenylacetyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H28N4O3
7-(cyclopropanecarbonyl)-2-[(2S)-1-(2-phenylacetyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(cyclopropanecarbonyl)-2-[(3S)-1-(3-phenylpropanoyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H28N4O3
7-(cyclopropanecarbonyl)-2-[(3S)-1-(3-phenylpropanoyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(cyclopropanecarbonyl)-2-[(2R)-1-(2-phenylacetyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H28N4O3
7-(cyclopropanecarbonyl)-2-[(2R)-1-(2-phenylacetyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-cyclopentyl-2-[(2S)-1-[(E)-3-phenylprop-2-enoyl]piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C26H32N4O2
7-cyclopentyl-2-[(2S)-1-[(E)-3-phenylprop-2-enoyl]piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(cyclohexylmethyl)-2-[(2R)-1-(3-phenylpropanoyl)pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C27H36N4O2
7-(cyclohexylmethyl)-2-[(2R)-1-(3-phenylpropanoyl)pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(3S)-1-(3-phenylpropanoyl)pyrrolidin-3-yl]-6H-1,6-naphthyridin-5-one —— C21H21N3O2
7-[(3S)-1-(3-phenylpropanoyl)pyrrolidin-3-yl]-6H-1,6-naphthyridin-5-one
—— 7-(cyclopropanecarbonyl)-2-[(3R)-1-(2-phenylacetyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H26N4O3
7-(cyclopropanecarbonyl)-2-[(3R)-1-(2-phenylacetyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one