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—— 7-[[(2S)-2-methyl-2,3-dihydroindol-1-yl]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C16H15N3OS
7-[[(2S)-2-methyl-2,3-dihydroindol-1-yl]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— (7R)-7-(2-chlorophenyl)-5-methyl-N-pyridin-2-yl-4,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C17H14ClN7O
(7R)-7-(2-chlorophenyl)-5-methyl-N-pyridin-2-yl-4,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-5-methyl-2-(3-methylphenyl)-7-pyridin-3-yl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C19H18N6O
(7R)-5-methyl-2-(3-methylphenyl)-7-pyridin-3-yl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(4-fluorophenyl)-5-methyl-N-pyridin-2-yl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C18H15FN6O
(7R)-7-(4-fluorophenyl)-5-methyl-N-pyridin-2-yl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— [7,8-dimethyl-2-(1-methylpyrazol-4-yl)quinolin-4-yl]-[(2R)-2-ethylpiperidin-1-yl]methanone —— C23H28N4O
[7,8-dimethyl-2-(1-methylpyrazol-4-yl)quinolin-4-yl]-[(2R)-2-ethylpiperidin-1-yl]methanone
—— [7-methyl-2-(2-propan-2-ylpyrimidin-5-yl)quinolin-4-yl]-[(2S)-2-methylpyrrolidin-1-yl]methanone —— C23H26N4O
[7-methyl-2-(2-propan-2-ylpyrimidin-5-yl)quinolin-4-yl]-[(2S)-2-methylpyrrolidin-1-yl]methanone
—— [7-methyl-2-(1-methylpyrazol-4-yl)quinolin-4-yl]-[(2S)-2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]methanone —— C22H21N5OS
[7-methyl-2-(1-methylpyrazol-4-yl)quinolin-4-yl]-[(2S)-2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]methanone
—— 7,8-dimethyl-N-[(1S)-1-(2-methyl-1,2,4-triazol-3-yl)propyl]-2-pyrimidin-5-ylquinoline-4-carboxamide —— C22H23N7O
7,8-dimethyl-N-[(1S)-1-(2-methyl-1,2,4-triazol-3-yl)propyl]-2-pyrimidin-5-ylquinoline-4-carboxamide
—— [7,8-dimethyl-2-(1-methylpyrazol-4-yl)quinolin-4-yl]-[(2S)-2-ethylpiperidin-1-yl]methanone —— C23H28N4O
[7,8-dimethyl-2-(1-methylpyrazol-4-yl)quinolin-4-yl]-[(2S)-2-ethylpiperidin-1-yl]methanone
—— (7-fluoro-2-pyrimidin-5-ylquinolin-4-yl)-[(2R)-2-(pyridin-3-ylmethyl)pyrrolidin-1-yl]methanone —— C24H20FN5O
(7-fluoro-2-pyrimidin-5-ylquinolin-4-yl)-[(2R)-2-(pyridin-3-ylmethyl)pyrrolidin-1-yl]methanone
—— (7-methyl-2-pyrimidin-5-ylquinolin-4-yl)-[(2R)-2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]methanone —— C22H19N5OS
(7-methyl-2-pyrimidin-5-ylquinolin-4-yl)-[(2R)-2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]methanone
—— [7-methyl-2-(2-propan-2-ylpyrimidin-5-yl)quinolin-4-yl]-[(2R)-2-methylpyrrolidin-1-yl]methanone —— C23H26N4O
[7-methyl-2-(2-propan-2-ylpyrimidin-5-yl)quinolin-4-yl]-[(2R)-2-methylpyrrolidin-1-yl]methanone
—— [7,8-dimethyl-2-(1-methylpyrazol-4-yl)quinolin-4-yl]-[(3S)-3-methylpiperidin-1-yl]methanone —— C22H26N4O
[7,8-dimethyl-2-(1-methylpyrazol-4-yl)quinolin-4-yl]-[(3S)-3-methylpiperidin-1-yl]methanone
—— [7,8-dimethyl-2-(1-methylpyrazol-4-yl)quinolin-4-yl]-[(3S)-3-propylpyrrolidin-1-yl]methanone —— C23H28N4O
[7,8-dimethyl-2-(1-methylpyrazol-4-yl)quinolin-4-yl]-[(3S)-3-propylpyrrolidin-1-yl]methanone
—— (7-methyl-2-pyrimidin-5-ylquinolin-4-yl)-[(2S)-2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]methanone —— C22H19N5OS
(7-methyl-2-pyrimidin-5-ylquinolin-4-yl)-[(2S)-2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]methanone
—— [7,8-dimethyl-2-(1-methylpyrazol-4-yl)quinolin-4-yl]-[(3R)-3-methylpiperidin-1-yl]methanone —— C22H26N4O
[7,8-dimethyl-2-(1-methylpyrazol-4-yl)quinolin-4-yl]-[(3R)-3-methylpiperidin-1-yl]methanone
—— (7-fluoro-2-pyrimidin-5-ylquinolin-4-yl)-[(2S)-2-(pyridin-3-ylmethyl)pyrrolidin-1-yl]methanone —— C24H20FN5O
(7-fluoro-2-pyrimidin-5-ylquinolin-4-yl)-[(2S)-2-(pyridin-3-ylmethyl)pyrrolidin-1-yl]methanone
—— 7,8-dimethyl-N-[(1R)-1-(2-methyl-1,2,4-triazol-3-yl)propyl]-2-pyrimidin-5-ylquinoline-4-carboxamide —— C22H23N7O
7,8-dimethyl-N-[(1R)-1-(2-methyl-1,2,4-triazol-3-yl)propyl]-2-pyrimidin-5-ylquinoline-4-carboxamide
—— (7-fluoro-2-pyrimidin-5-ylquinolin-4-yl)-[(2R)-2-(3-methyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methanone —— C21H17FN6O2
(7-fluoro-2-pyrimidin-5-ylquinolin-4-yl)-[(2R)-2-(3-methyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methanone
—— [7-methyl-2-(1-methylpyrazol-4-yl)quinolin-4-yl]-[(2S)-2-methylpiperidin-1-yl]methanone —— C21H24N4O
[7-methyl-2-(1-methylpyrazol-4-yl)quinolin-4-yl]-[(2S)-2-methylpiperidin-1-yl]methanone
—— [7-methyl-2-(1-propan-2-ylpyrazol-4-yl)quinolin-4-yl]-[(2R)-2-methylpyrrolidin-1-yl]methanone —— C22H26N4O
[7-methyl-2-(1-propan-2-ylpyrazol-4-yl)quinolin-4-yl]-[(2R)-2-methylpyrrolidin-1-yl]methanone
—— 7-[(1R)-1-(2,4-dichlorophenoxy)ethyl]-2-methylpyrazolo[1,5-a]pyrimidine —— C15H13Cl2N3O
7-[(1R)-1-(2,4-dichlorophenoxy)ethyl]-2-methylpyrazolo[1,5-a]pyrimidine
—— [7-fluoro-2-(1-methylpyrazol-4-yl)quinolin-4-yl]-[(2R)-2-(3-methyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methanone —— C21H19FN6O2
[7-fluoro-2-(1-methylpyrazol-4-yl)quinolin-4-yl]-[(2R)-2-(3-methyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methanone
—— (7-fluoro-2-pyrimidin-5-ylquinolin-4-yl)-[(2S)-2-(3-methyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methanone —— C21H17FN6O2
(7-fluoro-2-pyrimidin-5-ylquinolin-4-yl)-[(2S)-2-(3-methyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methanone
—— [7,8-dimethyl-2-(1-propylpyrazol-4-yl)quinolin-4-yl]-[(2S)-2-methylpyrrolidin-1-yl]methanone —— C23H28N4O
[7,8-dimethyl-2-(1-propylpyrazol-4-yl)quinolin-4-yl]-[(2S)-2-methylpyrrolidin-1-yl]methanone
—— [7-methyl-2-(1-propan-2-ylpyrazol-4-yl)quinolin-4-yl]-[(2S)-2-methylpyrrolidin-1-yl]methanone —— C22H26N4O
[7-methyl-2-(1-propan-2-ylpyrazol-4-yl)quinolin-4-yl]-[(2S)-2-methylpyrrolidin-1-yl]methanone
—— [7,8-dimethyl-2-(1-propylpyrazol-4-yl)quinolin-4-yl]-[(2R)-2-methylpyrrolidin-1-yl]methanone —— C23H28N4O
[7,8-dimethyl-2-(1-propylpyrazol-4-yl)quinolin-4-yl]-[(2R)-2-methylpyrrolidin-1-yl]methanone
—— 7-[(1S)-1-(2,4-dichlorophenoxy)ethyl]-2-methylpyrazolo[1,5-a]pyrimidine —— C15H13Cl2N3O
7-[(1S)-1-(2,4-dichlorophenoxy)ethyl]-2-methylpyrazolo[1,5-a]pyrimidine
—— [7-fluoro-2-(1-methylpyrazol-4-yl)quinolin-4-yl]-[(2S)-2-(3-methyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methanone —— C21H19FN6O2
[7-fluoro-2-(1-methylpyrazol-4-yl)quinolin-4-yl]-[(2S)-2-(3-methyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methanone
—— [7-methyl-2-(1-methylpyrazol-4-yl)quinolin-4-yl]-[(2R)-2-methylpiperidin-1-yl]methanone —— C21H24N4O
[7-methyl-2-(1-methylpyrazol-4-yl)quinolin-4-yl]-[(2R)-2-methylpiperidin-1-yl]methanone
—— [7,8-dimethyl-2-(1-propan-2-ylpyrazol-4-yl)quinolin-4-yl]-[(2S)-2-methylpyrrolidin-1-yl]methanone —— C23H28N4O
[7,8-dimethyl-2-(1-propan-2-ylpyrazol-4-yl)quinolin-4-yl]-[(2S)-2-methylpyrrolidin-1-yl]methanone
—— [7-methyl-2-(1-methylpyrazol-4-yl)quinolin-4-yl]-[(2R)-2-(pyridin-3-ylmethyl)pyrrolidin-1-yl]methanone —— C25H25N5O
[7-methyl-2-(1-methylpyrazol-4-yl)quinolin-4-yl]-[(2R)-2-(pyridin-3-ylmethyl)pyrrolidin-1-yl]methanone
—— [7,8-dimethyl-2-(2-methylpyrimidin-5-yl)quinolin-4-yl]-[(3R)-3-methylpiperidin-1-yl]methanone —— C23H26N4O
[7,8-dimethyl-2-(2-methylpyrimidin-5-yl)quinolin-4-yl]-[(3R)-3-methylpiperidin-1-yl]methanone
—— [7-methyl-2-(1-methylpyrazol-4-yl)quinolin-4-yl]-[(2S)-2-(pyridin-3-ylmethyl)pyrrolidin-1-yl]methanone —— C25H25N5O
[7-methyl-2-(1-methylpyrazol-4-yl)quinolin-4-yl]-[(2S)-2-(pyridin-3-ylmethyl)pyrrolidin-1-yl]methanone
—— 7-chloro-N-[2-[[(3S)-oxolan-3-yl]methyl]pyrazol-3-yl]-1,3-benzodioxole-5-carboxamide —— C16H16ClN3O4
7-chloro-N-[2-[[(3S)-oxolan-3-yl]methyl]pyrazol-3-yl]-1,3-benzodioxole-5-carboxamide
—— 7-[4-[(2S)-1-methoxypropan-2-yl]piperidin-1-yl]-2,5-dimethyl-[1,3]oxazolo[5,4-d]pyrimidine —— C16H24N4O2
7-[4-[(2S)-1-methoxypropan-2-yl]piperidin-1-yl]-2,5-dimethyl-[1,3]oxazolo[5,4-d]pyrimidine
—— 7-[4-[(2R)-1-methoxypropan-2-yl]piperidin-1-yl]-2,5-dimethyl-[1,3]oxazolo[5,4-d]pyrimidine —— C16H24N4O2
7-[4-[(2R)-1-methoxypropan-2-yl]piperidin-1-yl]-2,5-dimethyl-[1,3]oxazolo[5,4-d]pyrimidine
—— (7,8-dimethyl-2-pyrimidin-5-ylquinolin-4-yl)-[(2S)-2-methylpiperidin-1-yl]methanone —— C22H24N4O
(7,8-dimethyl-2-pyrimidin-5-ylquinolin-4-yl)-[(2S)-2-methylpiperidin-1-yl]methanone
—— (7,8-dimethyl-2-pyrimidin-5-ylquinolin-4-yl)-[(2S)-2-methylpyrrolidin-1-yl]methanone —— C21H22N4O
(7,8-dimethyl-2-pyrimidin-5-ylquinolin-4-yl)-[(2S)-2-methylpyrrolidin-1-yl]methanone
—— 7-[4-[(2R)-2-(butanoylamino)-3-ethoxy-1,1,1-trifluoro-3-oxopropan-2-yl]piperazin-1-yl]-1-ethyl-6-fluoro-4-oxoquinoline-3-carboxylic acid —— C25H30F4N4O6
7-[4-[(2R)-2-(butanoylamino)-3-ethoxy-1,1,1-trifluoro-3-oxopropan-2-yl]piperazin-1-yl]-1-ethyl-6-fluoro-4-oxoquinoline-3-carboxylic acid
—— [7-methyl-2-(1-methylpyrazol-4-yl)quinolin-4-yl]-[(2S)-2-(3-methyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methanone —— C22H22N6O2
[7-methyl-2-(1-methylpyrazol-4-yl)quinolin-4-yl]-[(2S)-2-(3-methyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methanone
—— 7-[(3R)-3-benzylmorpholin-4-yl]-2,5-dimethyl-[1,3]oxazolo[5,4-d]pyrimidine —— C18H20N4O2
7-[(3R)-3-benzylmorpholin-4-yl]-2,5-dimethyl-[1,3]oxazolo[5,4-d]pyrimidine
—— 7-[(3S)-3-benzylmorpholin-4-yl]-2,5-dimethyl-[1,3]oxazolo[5,4-d]pyrimidine —— C18H20N4O2
7-[(3S)-3-benzylmorpholin-4-yl]-2,5-dimethyl-[1,3]oxazolo[5,4-d]pyrimidine
—— 7-[(2S)-2-(3,4-dimethylphenyl)pyrrolidin-1-yl]-5-propyl-[1,2,4]triazolo[1,5-a]pyrimidine —— C20H25N5
7-[(2S)-2-(3,4-dimethylphenyl)pyrrolidin-1-yl]-5-propyl-[1,2,4]triazolo[1,5-a]pyrimidine
—— [7,8-dimethyl-2-(2-propan-2-ylpyrimidin-5-yl)quinolin-4-yl]-[(2S)-2-methylpyrrolidin-1-yl]methanone —— C24H28N4O
[7,8-dimethyl-2-(2-propan-2-ylpyrimidin-5-yl)quinolin-4-yl]-[(2S)-2-methylpyrrolidin-1-yl]methanone
—— [7,8-dimethyl-2-(1-methylpyrazol-4-yl)quinolin-4-yl]-[(2S)-2-methylpyrrolidin-1-yl]methanone —— C21H24N4O
[7,8-dimethyl-2-(1-methylpyrazol-4-yl)quinolin-4-yl]-[(2S)-2-methylpyrrolidin-1-yl]methanone
—— [7,8-dimethyl-2-(2-propan-2-ylpyrimidin-5-yl)quinolin-4-yl]-[(2R)-2-methylpyrrolidin-1-yl]methanone —— C24H28N4O
[7,8-dimethyl-2-(2-propan-2-ylpyrimidin-5-yl)quinolin-4-yl]-[(2R)-2-methylpyrrolidin-1-yl]methanone
—— (7,8-dimethyl-2-pyrimidin-5-ylquinolin-4-yl)-[(2R)-2-methylpiperidin-1-yl]methanone —— C22H24N4O
(7,8-dimethyl-2-pyrimidin-5-ylquinolin-4-yl)-[(2R)-2-methylpiperidin-1-yl]methanone
—— (7,8-dimethyl-2-pyrimidin-5-ylquinolin-4-yl)-[(2R)-2-methylpyrrolidin-1-yl]methanone —— C21H22N4O
(7,8-dimethyl-2-pyrimidin-5-ylquinolin-4-yl)-[(2R)-2-methylpyrrolidin-1-yl]methanone
—— 7-[4-[(2S)-2-(butanoylamino)-3-ethoxy-1,1,1-trifluoro-3-oxopropan-2-yl]piperazin-1-yl]-1-ethyl-6-fluoro-4-oxoquinoline-3-carboxylic acid —— C25H30F4N4O6
7-[4-[(2S)-2-(butanoylamino)-3-ethoxy-1,1,1-trifluoro-3-oxopropan-2-yl]piperazin-1-yl]-1-ethyl-6-fluoro-4-oxoquinoline-3-carboxylic acid