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—— 7-[(S)-[1-[(4-methoxyphenyl)methyl]tetrazol-5-yl]-(4-methylpiperazin-1-yl)methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C25H27N7O4
7-[(S)-[1-[(4-methoxyphenyl)methyl]tetrazol-5-yl]-(4-methylpiperazin-1-yl)methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— (7R)-N-(2-methoxyphenyl)-7-(4-methoxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C21H21N5O3
(7R)-N-(2-methoxyphenyl)-7-(4-methoxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-[4-[(3,4-dichlorophenyl)methoxy]-3-ethoxyphenyl]-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C21H20Cl2N6O3
(7S)-7-[4-[(3,4-dichlorophenyl)methoxy]-3-ethoxyphenyl]-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-[4-[(4-tert-butylphenyl)methoxy]phenyl]-5-methyl-N-(2-methylphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C30H32N6O2
(7R)-7-[4-[(4-tert-butylphenyl)methoxy]phenyl]-5-methyl-N-(2-methylphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(2,4-dimethylphenyl)-5-methyl-7-[3-[(2-methylphenyl)methoxy]phenyl]-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C29H29N5O2
(7S)-N-(2,4-dimethylphenyl)-5-methyl-7-[3-[(2-methylphenyl)methoxy]phenyl]-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(5-bromo-2-butoxyphenyl)-5-methyl-N-(2-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C24H26BrN5O2
(7R)-7-(5-bromo-2-butoxyphenyl)-5-methyl-N-(2-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-[3-bromo-5-methoxy-4-[(3-methylphenyl)methoxy]phenyl]-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C21H21BrN6O3
(7S)-7-[3-bromo-5-methoxy-4-[(3-methylphenyl)methoxy]phenyl]-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-[3-methoxy-4-(2-morpholin-4-yl-2-oxoethoxy)phenyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C20H24N6O5
(7S)-7-[3-methoxy-4-(2-morpholin-4-yl-2-oxoethoxy)phenyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-[4-[(3-chlorophenyl)methoxy]-3-methoxyphenyl]-5-methyl-N-phenyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C26H23ClN6O3
(7S)-7-[4-[(3-chlorophenyl)methoxy]-3-methoxyphenyl]-5-methyl-N-phenyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(2,4-dimethylphenyl)-7-[4-[(2-fluorophenyl)methoxy]phenyl]-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C27H25FN6O2
(7S)-N-(2,4-dimethylphenyl)-7-[4-[(2-fluorophenyl)methoxy]phenyl]-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(2,4-dimethylphenyl)-7-(3-hydroxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C21H21N5O2
(7S)-N-(2,4-dimethylphenyl)-7-(3-hydroxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-[4-[(3-chlorophenyl)methoxy]-3-methoxyphenyl]-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C20H19ClN6O3
(7S)-7-[4-[(3-chlorophenyl)methoxy]-3-methoxyphenyl]-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-[4-[(3-chlorophenyl)methoxy]phenyl]-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C19H17ClN6O2
(7S)-7-[4-[(3-chlorophenyl)methoxy]phenyl]-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(2,4-dimethylphenyl)-5-methyl-7-[4-[(4-methylphenyl)methoxy]phenyl]-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C28H28N6O2
(7S)-N-(2,4-dimethylphenyl)-5-methyl-7-[4-[(4-methylphenyl)methoxy]phenyl]-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-5-methyl-N-(2-methylphenyl)-7-(3-propan-2-yloxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H25N5O2
(7R)-5-methyl-N-(2-methylphenyl)-7-(3-propan-2-yloxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(2,4-dimethylphenyl)-5-methyl-7-(3-propan-2-yloxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C24H27N5O2
(7S)-N-(2,4-dimethylphenyl)-5-methyl-7-(3-propan-2-yloxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-(2,4-dimethylphenyl)-7-(3-ethoxy-4-phenylmethoxyphenyl)-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C29H30N6O3
(7R)-N-(2,4-dimethylphenyl)-7-(3-ethoxy-4-phenylmethoxyphenyl)-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-[5-bromo-2-[(2,4-dichlorophenyl)methoxy]phenyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C20H16BrCl2N5O2
(7R)-7-[5-bromo-2-[(2,4-dichlorophenyl)methoxy]phenyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-[5-bromo-2-[(2,4-dichlorophenyl)methoxy]phenyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C20H16BrCl2N5O2
(7S)-7-[5-bromo-2-[(2,4-dichlorophenyl)methoxy]phenyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(5-bromo-2-butoxyphenyl)-5-methyl-N-(2-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C24H26BrN5O2
(7S)-7-(5-bromo-2-butoxyphenyl)-5-methyl-N-(2-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— 7-[(R)-(1-benzyltetrazol-5-yl)-(2,3-dihydroindol-1-yl)methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C27H22N6O3
7-[(R)-(1-benzyltetrazol-5-yl)-(2,3-dihydroindol-1-yl)methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— 7-[(R)-[1-[(4-fluorophenyl)methyl]tetrazol-5-yl]-morpholin-4-ylmethyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C23H21FN6O4
7-[(R)-[1-[(4-fluorophenyl)methyl]tetrazol-5-yl]-morpholin-4-ylmethyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— (7S)-7-[4-[(3,4-dichlorophenyl)methoxy]-3-methoxyphenyl]-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C20H18Cl2N6O3
(7S)-7-[4-[(3,4-dichlorophenyl)methoxy]-3-methoxyphenyl]-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— 7-[(S)-(4-ethylpiperazin-1-yl)-[1-[(4-methoxyphenyl)methyl]tetrazol-5-yl]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C26H29N7O4
7-[(S)-(4-ethylpiperazin-1-yl)-[1-[(4-methoxyphenyl)methyl]tetrazol-5-yl]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— 7-[(R)-[1-(2-methylbutan-2-yl)tetrazol-5-yl]-(4-methylpiperidin-1-yl)methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C23H30N6O3
7-[(R)-[1-(2-methylbutan-2-yl)tetrazol-5-yl]-(4-methylpiperidin-1-yl)methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— (7S)-7-[5-bromo-2-[(4-chlorophenyl)methoxy]phenyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C20H17BrClN5O2
(7S)-7-[5-bromo-2-[(4-chlorophenyl)methoxy]phenyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(4-hexoxyphenyl)-5-methyl-N-(2-methylphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C25H30N6O2
(7R)-7-(4-hexoxyphenyl)-5-methyl-N-(2-methylphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-[4-[(2-fluorophenyl)methoxy]phenyl]-N-(2-methoxyphenyl)-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C26H23FN6O3
(7S)-7-[4-[(2-fluorophenyl)methoxy]phenyl]-N-(2-methoxyphenyl)-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— 7-[(R)-[1-(2-methylbutan-2-yl)tetrazol-5-yl]-piperidin-1-ylmethyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C22H28N6O3
7-[(R)-[1-(2-methylbutan-2-yl)tetrazol-5-yl]-piperidin-1-ylmethyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— (7S)-7-[4-[(2-chloro-6-fluorophenyl)methoxy]phenyl]-N-(2,4-dimethylphenyl)-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C27H24ClFN6O2
(7S)-7-[4-[(2-chloro-6-fluorophenyl)methoxy]phenyl]-N-(2,4-dimethylphenyl)-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— 7-[(R)-(4-ethylpiperazin-1-yl)-[1-(2-methylbutan-2-yl)tetrazol-5-yl]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C23H31N7O3
7-[(R)-(4-ethylpiperazin-1-yl)-[1-(2-methylbutan-2-yl)tetrazol-5-yl]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— 7-[(R)-(4-benzylpiperazin-1-yl)-[1-(2-methylbutan-2-yl)tetrazol-5-yl]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C28H33N7O3
7-[(R)-(4-benzylpiperazin-1-yl)-[1-(2-methylbutan-2-yl)tetrazol-5-yl]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— 7-[(S)-(1-benzyltetrazol-5-yl)-(4-ethylpiperazin-1-yl)methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C25H27N7O3
7-[(S)-(1-benzyltetrazol-5-yl)-(4-ethylpiperazin-1-yl)methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— 7-[(R)-[1-(2-methylbutan-2-yl)tetrazol-5-yl]-(4-methylpiperazin-1-yl)methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C22H29N7O3
7-[(R)-[1-(2-methylbutan-2-yl)tetrazol-5-yl]-(4-methylpiperazin-1-yl)methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— (7R)-7-[4-[(2,4-dichlorophenyl)methoxy]phenyl]-5-methyl-N-phenyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C25H20Cl2N6O2
(7R)-7-[4-[(2,4-dichlorophenyl)methoxy]phenyl]-5-methyl-N-phenyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— 7-[(S)-(1-benzyltetrazol-5-yl)-(4-propylpiperazin-1-yl)methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C26H29N7O3
7-[(S)-(1-benzyltetrazol-5-yl)-(4-propylpiperazin-1-yl)methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— 7-[(R)-[4-(2-methoxyphenyl)piperazin-1-yl]-[1-(2-methylbutan-2-yl)tetrazol-5-yl]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C28H33N7O4
7-[(R)-[4-(2-methoxyphenyl)piperazin-1-yl]-[1-(2-methylbutan-2-yl)tetrazol-5-yl]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— (7R)-7-[3-ethoxy-4-[(3-methylphenyl)methoxy]phenyl]-5-methyl-N-(2-methylphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C29H30N6O3
(7R)-7-[3-ethoxy-4-[(3-methylphenyl)methoxy]phenyl]-5-methyl-N-(2-methylphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— 7-[(R)-(4-hydroxypiperidin-1-yl)-[1-[(4-methoxyphenyl)methyl]tetrazol-5-yl]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C25H26N6O5
7-[(R)-(4-hydroxypiperidin-1-yl)-[1-[(4-methoxyphenyl)methyl]tetrazol-5-yl]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— 7-[(R)-[1-[(4-fluorophenyl)methyl]tetrazol-5-yl]-piperidin-1-ylmethyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C24H23FN6O3
7-[(R)-[1-[(4-fluorophenyl)methyl]tetrazol-5-yl]-piperidin-1-ylmethyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— (7R)-5-methyl-7-(4-pentoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C18H23N5O2
(7R)-5-methyl-7-(4-pentoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— 7-[(R)-[4-(4-fluorophenyl)piperazin-1-yl]-[1-(2-methylbutan-2-yl)tetrazol-5-yl]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C27H30FN7O3
7-[(R)-[4-(4-fluorophenyl)piperazin-1-yl]-[1-(2-methylbutan-2-yl)tetrazol-5-yl]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— 7-[(R)-[1-(2-methylbutan-2-yl)tetrazol-5-yl]-(4-phenylpiperazin-1-yl)methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C27H31N7O3
7-[(R)-[1-(2-methylbutan-2-yl)tetrazol-5-yl]-(4-phenylpiperazin-1-yl)methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— 7-[(R)-azepan-1-yl-[1-[(4-methoxyphenyl)methyl]tetrazol-5-yl]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C26H28N6O4
7-[(R)-azepan-1-yl-[1-[(4-methoxyphenyl)methyl]tetrazol-5-yl]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— (7R)-N-(2-methoxyphenyl)-5-methyl-7-[3-[(2-methylphenyl)methoxy]phenyl]-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H27N5O3
(7R)-N-(2-methoxyphenyl)-5-methyl-7-[3-[(2-methylphenyl)methoxy]phenyl]-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-[4-[(2-fluorophenyl)methoxy]phenyl]-N-(2-methoxyphenyl)-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C26H23FN6O3
(7R)-7-[4-[(2-fluorophenyl)methoxy]phenyl]-N-(2-methoxyphenyl)-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-(2-methoxyphenyl)-5-methyl-7-[4-(2-morpholin-4-yl-2-oxoethoxy)phenyl]-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C26H28N6O5
(7R)-N-(2-methoxyphenyl)-5-methyl-7-[4-(2-morpholin-4-yl-2-oxoethoxy)phenyl]-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— 7-[(R)-(1-benzyltetrazol-5-yl)-(4-hydroxypiperidin-1-yl)methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C24H24N6O4
7-[(R)-(1-benzyltetrazol-5-yl)-(4-hydroxypiperidin-1-yl)methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— (7R)-7-[5-bromo-2-[(4-tert-butylphenyl)methoxy]phenyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C24H26BrN5O2
(7R)-7-[5-bromo-2-[(4-tert-butylphenyl)methoxy]phenyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— 7-[(R)-(1-benzyltetrazol-5-yl)-morpholin-4-ylmethyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C23H22N6O4
7-[(R)-(1-benzyltetrazol-5-yl)-morpholin-4-ylmethyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one