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—— (7S)-2-benzylsulfanyl-7-(3-chlorophenyl)-5-methyl-N-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C26H22ClN5OS
(7S)-2-benzylsulfanyl-7-(3-chlorophenyl)-5-methyl-N-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-benzylsulfanyl-7-(4-chlorophenyl)-N-(2,4-dimethylphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H26ClN5OS
(7R)-2-benzylsulfanyl-7-(4-chlorophenyl)-N-(2,4-dimethylphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(4-chlorophenyl)-5-methyl-N-(2-methylphenyl)-2-[(3-methylphenyl)methylsulfanyl]-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H26ClN5OS
(7R)-7-(4-chlorophenyl)-5-methyl-N-(2-methylphenyl)-2-[(3-methylphenyl)methylsulfanyl]-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-5-methyl-2-[2-(4-methylphenyl)-2-oxoethyl]sulfanyl-N-phenyl-7-pyridin-3-yl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H24N6O2S
(7R)-5-methyl-2-[2-(4-methylphenyl)-2-oxoethyl]sulfanyl-N-phenyl-7-pyridin-3-yl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-[(4-chlorophenyl)methylsulfanyl]-N-(2,4-dimethylphenyl)-5-methyl-7-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H26ClN5OS
(7S)-2-[(4-chlorophenyl)methylsulfanyl]-N-(2,4-dimethylphenyl)-5-methyl-7-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-benzylsulfanyl-7-(4-chlorophenyl)-5-methyl-N-(2-methylphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H24ClN5OS
(7S)-2-benzylsulfanyl-7-(4-chlorophenyl)-5-methyl-N-(2-methylphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-benzylsulfanyl-N-(2,4-dimethylphenyl)-5-methyl-7-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H27N5OS
(7R)-2-benzylsulfanyl-N-(2,4-dimethylphenyl)-5-methyl-7-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-benzylsulfanyl-7-(4-chlorophenyl)-5-methyl-N-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C26H22ClN5OS
(7S)-2-benzylsulfanyl-7-(4-chlorophenyl)-5-methyl-N-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(4-fluorophenyl)-N-(2-methoxyphenyl)-5-methyl-2-[(3-methylphenyl)methylsulfanyl]-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H26FN5O2S
(7R)-7-(4-fluorophenyl)-N-(2-methoxyphenyl)-5-methyl-2-[(3-methylphenyl)methylsulfanyl]-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-ethylsulfanyl-5-methyl-N-(2-methylphenyl)-7-(4-methylsulfanylphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H25N5OS2
(7R)-2-ethylsulfanyl-5-methyl-N-(2-methylphenyl)-7-(4-methylsulfanylphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(4-ethylanilino)-6-(furan-2-ylmethyl)-7H-pyrrolo[3,4-b]pyridin-5-one —— C20H19N3O2
(7R)-7-(4-ethylanilino)-6-(furan-2-ylmethyl)-7H-pyrrolo[3,4-b]pyridin-5-one
—— (7S)-7-(3-chlorophenyl)-2-[(2,5-dimethylphenyl)methylsulfanyl]-5-methyl-N-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H26ClN5OS
(7S)-7-(3-chlorophenyl)-2-[(2,5-dimethylphenyl)methylsulfanyl]-5-methyl-N-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-5-methyl-2-[2-(4-methylphenyl)-2-oxoethyl]sulfanyl-N,7-diphenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H25N5O2S
(7R)-5-methyl-2-[2-(4-methylphenyl)-2-oxoethyl]sulfanyl-N,7-diphenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-benzylsulfanyl-7-(2,5-dimethoxyphenyl)-5-methyl-N-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H27N5O3S
(7R)-2-benzylsulfanyl-7-(2,5-dimethoxyphenyl)-5-methyl-N-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-benzylsulfanyl-7-(3-chlorophenyl)-N-(2-methoxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H24ClN5O2S
(7R)-2-benzylsulfanyl-7-(3-chlorophenyl)-N-(2-methoxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(2-methoxyphenyl)-2-[(3-methoxyphenyl)methylsulfanyl]-5-methyl-7-(4-methylphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C29H29N5O3S
(7S)-N-(2-methoxyphenyl)-2-[(3-methoxyphenyl)methylsulfanyl]-5-methyl-7-(4-methylphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-ethylsulfanyl-7-(4-hydroxy-3-methoxyphenyl)-N-(2-methoxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H25N5O4S
(7S)-2-ethylsulfanyl-7-(4-hydroxy-3-methoxyphenyl)-N-(2-methoxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-[(2,5-dimethylphenyl)methylsulfanyl]-5-methyl-7-(4-methylphenyl)-N-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C29H29N5OS
(7S)-2-[(2,5-dimethylphenyl)methylsulfanyl]-5-methyl-7-(4-methylphenyl)-N-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(2-methoxyphenyl)-5-methyl-2-[2-(4-methylphenyl)-2-oxoethyl]sulfanyl-7-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C29H27N5O3S
(7S)-N-(2-methoxyphenyl)-5-methyl-2-[2-(4-methylphenyl)-2-oxoethyl]sulfanyl-7-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(4-ethylphenyl)-2-[(3-methoxyphenyl)methylsulfanyl]-5-methyl-N-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C29H29N5O2S
(7R)-7-(4-ethylphenyl)-2-[(3-methoxyphenyl)methylsulfanyl]-5-methyl-N-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(4-chloro-2-methoxy-5-methylanilino)-6-phenyl-7H-pyrrolo[3,4-b]pyridin-5-one —— C21H18ClN3O2
(7R)-7-(4-chloro-2-methoxy-5-methylanilino)-6-phenyl-7H-pyrrolo[3,4-b]pyridin-5-one
—— (7S)-7-(4-methoxyphenyl)-5-methyl-N-(2-methylphenyl)-2-[(3-methylphenyl)methylsulfanyl]-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C29H29N5O2S
(7S)-7-(4-methoxyphenyl)-5-methyl-N-(2-methylphenyl)-2-[(3-methylphenyl)methylsulfanyl]-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-benzylsulfanyl-N-(2,4-dimethylphenyl)-5-methyl-7-(4-methylphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C29H29N5OS
(7S)-2-benzylsulfanyl-N-(2,4-dimethylphenyl)-5-methyl-7-(4-methylphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-ethylsulfanyl-5-methyl-N-(2-methylphenyl)-7-(4-methylsulfanylphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H25N5OS2
(7S)-2-ethylsulfanyl-5-methyl-N-(2-methylphenyl)-7-(4-methylsulfanylphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-ethylsulfanyl-7-(2-fluorophenyl)-N-(2-methoxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C22H22FN5O2S
(7R)-2-ethylsulfanyl-7-(2-fluorophenyl)-N-(2-methoxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-benzylsulfanyl-N-(2-methoxyphenyl)-5-methyl-7-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H25N5O2S
(7S)-2-benzylsulfanyl-N-(2-methoxyphenyl)-5-methyl-7-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(4-methoxyphenyl)-2-[(3-methoxyphenyl)methylsulfanyl]-5-methyl-N-(2-methylphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C29H29N5O3S
(7S)-7-(4-methoxyphenyl)-2-[(3-methoxyphenyl)methylsulfanyl]-5-methyl-N-(2-methylphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-benzylsulfanyl-7-(3-chlorophenyl)-N-(2-methoxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H24ClN5O2S
(7S)-2-benzylsulfanyl-7-(3-chlorophenyl)-N-(2-methoxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-benzylsulfanyl-7-(2,5-dimethoxyphenyl)-5-methyl-N-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H27N5O3S
(7S)-2-benzylsulfanyl-7-(2,5-dimethoxyphenyl)-5-methyl-N-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(2,4-dimethylphenyl)-2-[(2,5-dimethylphenyl)methylsulfanyl]-5-methyl-7-(4-methylphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C31H33N5OS
(7S)-N-(2,4-dimethylphenyl)-2-[(2,5-dimethylphenyl)methylsulfanyl]-5-methyl-7-(4-methylphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-(2-methoxyphenyl)-7-(4-methoxyphenyl)-5-methyl-2-[(3-methylphenyl)methylsulfanyl]-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C29H29N5O3S
(7R)-N-(2-methoxyphenyl)-7-(4-methoxyphenyl)-5-methyl-2-[(3-methylphenyl)methylsulfanyl]-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-[(2-chloro-6-fluorophenyl)methylsulfanyl]-5-methyl-N,7-diphenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C26H21ClFN5OS
(7R)-2-[(2-chloro-6-fluorophenyl)methylsulfanyl]-5-methyl-N,7-diphenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-5-methyl-N-(2-methylphenyl)-7-(4-methylphenyl)-2-[(3-methylphenyl)methylsulfanyl]-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C29H29N5OS
(7R)-5-methyl-N-(2-methylphenyl)-7-(4-methylphenyl)-2-[(3-methylphenyl)methylsulfanyl]-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(2-fluorophenyl)-5-methyl-2-[2-(4-methylphenyl)-2-oxoethyl]sulfanyl-N-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H24FN5O2S
(7R)-7-(2-fluorophenyl)-5-methyl-2-[2-(4-methylphenyl)-2-oxoethyl]sulfanyl-N-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(4-acetylanilino)-6-[(4-methoxyphenyl)methyl]-7H-pyrrolo[3,4-b]pyridin-5-one —— C23H21N3O3
(7S)-7-(4-acetylanilino)-6-[(4-methoxyphenyl)methyl]-7H-pyrrolo[3,4-b]pyridin-5-one
—— (7S)-2-benzylsulfanyl-5-methyl-7-(4-methylphenyl)-N-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H25N5OS
(7S)-2-benzylsulfanyl-5-methyl-7-(4-methylphenyl)-N-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(2-fluorophenyl)-2-[(3-methoxyphenyl)methylsulfanyl]-5-methyl-N-(2-methylphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H26FN5O2S
(7S)-7-(2-fluorophenyl)-2-[(3-methoxyphenyl)methylsulfanyl]-5-methyl-N-(2-methylphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(3-chlorophenyl)-2-ethylsulfanyl-N-(2-methoxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C22H22ClN5O2S
(7R)-7-(3-chlorophenyl)-2-ethylsulfanyl-N-(2-methoxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-6-(furan-2-ylmethyl)-7-(2-methoxyanilino)-7H-pyrrolo[3,4-b]pyridin-5-one —— C19H17N3O3
(7R)-6-(furan-2-ylmethyl)-7-(2-methoxyanilino)-7H-pyrrolo[3,4-b]pyridin-5-one
—— (7R)-6-benzyl-7-(4-fluoroanilino)-7H-pyrrolo[3,4-b]pyridin-5-one —— C20H16FN3O
(7R)-6-benzyl-7-(4-fluoroanilino)-7H-pyrrolo[3,4-b]pyridin-5-one
—— (7R)-7-(2-chloroanilino)-6-(thiophen-2-ylmethyl)-7H-pyrrolo[3,4-b]pyridin-5-one —— C18H14ClN3OS
(7R)-7-(2-chloroanilino)-6-(thiophen-2-ylmethyl)-7H-pyrrolo[3,4-b]pyridin-5-one
—— (7S)-7-(3,4-difluoroanilino)-6-phenyl-7H-pyrrolo[3,4-b]pyridin-5-one —— C19H13F2N3O
(7S)-7-(3,4-difluoroanilino)-6-phenyl-7H-pyrrolo[3,4-b]pyridin-5-one
—— (7R)-6-benzyl-7-(4-methoxyanilino)-7H-pyrrolo[3,4-b]pyridin-5-one —— C21H19N3O2
(7R)-6-benzyl-7-(4-methoxyanilino)-7H-pyrrolo[3,4-b]pyridin-5-one
—— (7S)-2-[(3-methoxyphenyl)methylsulfanyl]-5-methyl-7-(2-methylphenyl)-N-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H27N5O2S
(7S)-2-[(3-methoxyphenyl)methylsulfanyl]-5-methyl-7-(2-methylphenyl)-N-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(4-chloro-2-methoxy-5-methylanilino)-6-phenyl-7H-pyrrolo[3,4-b]pyridin-5-one —— C21H18ClN3O2
(7S)-7-(4-chloro-2-methoxy-5-methylanilino)-6-phenyl-7H-pyrrolo[3,4-b]pyridin-5-one
—— (7S)-7-methyl-3-(2-morpholin-4-yl-2-oxoethyl)-6,7,8,9-tetrahydropyrimido[4,5-b]quinolin-4-one —— C18H22N4O3
(7S)-7-methyl-3-(2-morpholin-4-yl-2-oxoethyl)-6,7,8,9-tetrahydropyrimido[4,5-b]quinolin-4-one
—— (7R)-3-[[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl]-7-methyl-6,7,8,9-tetrahydropyrimido[4,5-b]quinolin-4-one —— C25H26N4O4
(7R)-3-[[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl]-7-methyl-6,7,8,9-tetrahydropyrimido[4,5-b]quinolin-4-one
—— (7R)-7-methyl-3-(2-morpholin-4-yl-2-oxoethyl)-6,7,8,9-tetrahydropyrimido[4,5-b]quinolin-4-one —— C18H22N4O3
(7R)-7-methyl-3-(2-morpholin-4-yl-2-oxoethyl)-6,7,8,9-tetrahydropyrimido[4,5-b]quinolin-4-one
—— (7S)-7-methyl-3-[(4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl]-6,7,8,9-tetrahydropyrimido[4,5-b]quinolin-4-one —— C21H19N5O2
(7S)-7-methyl-3-[(4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl]-6,7,8,9-tetrahydropyrimido[4,5-b]quinolin-4-one
—— (7R)-3-[(2-chlorophenyl)methyl]-7-methyl-6,7,8,9-tetrahydropyrimido[4,5-b]quinolin-4-one —— C19H18ClN3O
(7R)-3-[(2-chlorophenyl)methyl]-7-methyl-6,7,8,9-tetrahydropyrimido[4,5-b]quinolin-4-one