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—— 7-[(2-methoxyphenyl)methyl]-4-methyl-2-[(3S)-1-methylsulfonylpiperidin-3-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C21H26N4O4S
7-[(2-methoxyphenyl)methyl]-4-methyl-2-[(3S)-1-methylsulfonylpiperidin-3-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(3R)-1-benzylpiperidin-3-yl]-1,3-dimethyl-5-(trifluoromethyl)pyrido[2,3-d]pyrimidine-2,4-dione —— C22H23F3N4O2
7-[(3R)-1-benzylpiperidin-3-yl]-1,3-dimethyl-5-(trifluoromethyl)pyrido[2,3-d]pyrimidine-2,4-dione
—— 7-[(3R)-1-(cyclopropylmethyl)piperidin-3-yl]-2-phenylpyrido[2,3-d]pyrimidin-4-amine —— C22H25N5
7-[(3R)-1-(cyclopropylmethyl)piperidin-3-yl]-2-phenylpyrido[2,3-d]pyrimidin-4-amine
—— 7-benzyl-2-[(3R)-1-(2,4-dimethyl-1,3-oxazole-5-carbonyl)piperidin-3-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C25H27N5O3
7-benzyl-2-[(3R)-1-(2,4-dimethyl-1,3-oxazole-5-carbonyl)piperidin-3-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(3S)-1-[(4-chlorophenyl)methyl]piperidin-3-yl]-5-(trifluoromethyl)pyrido[2,3-d]pyrimidin-4-amine —— C20H19ClF3N5
7-[(3S)-1-[(4-chlorophenyl)methyl]piperidin-3-yl]-5-(trifluoromethyl)pyrido[2,3-d]pyrimidin-4-amine
—— 7-[(4-methoxyphenyl)methyl]-4-methyl-2-[(3S)-1-(oxan-4-yl)piperidin-3-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C25H32N4O3
7-[(4-methoxyphenyl)methyl]-4-methyl-2-[(3S)-1-(oxan-4-yl)piperidin-3-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(3S)-1-(1H-indol-5-ylmethyl)piperidin-3-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione —— C23H25N5O2
7-[(3S)-1-(1H-indol-5-ylmethyl)piperidin-3-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione
—— 7-[(2R)-1-(2-cyclopentylacetyl)pyrrolidin-2-yl]-1,3-dimethyl-5-(trifluoromethyl)pyrido[2,3-d]pyrimidine-2,4-dione —— C21H25F3N4O3
7-[(2R)-1-(2-cyclopentylacetyl)pyrrolidin-2-yl]-1,3-dimethyl-5-(trifluoromethyl)pyrido[2,3-d]pyrimidine-2,4-dione
—— 7-benzyl-4-methyl-2-[(3S)-1-(1-methylpyrazole-4-carbonyl)piperidin-3-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C24H26N6O2
7-benzyl-4-methyl-2-[(3S)-1-(1-methylpyrazole-4-carbonyl)piperidin-3-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[2-(4-fluorophenyl)ethyl]-4-methyl-2-[(2R)-1-(2-methylpyrazole-3-carbonyl)pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C24H25FN6O2
7-[2-(4-fluorophenyl)ethyl]-4-methyl-2-[(2R)-1-(2-methylpyrazole-3-carbonyl)pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[1-[(4-Fluorophenyl)methyl]piperidin-4-yl]-1-(2-methoxyethyl)-3-methylpyrido[2,3-d]pyrimidine-2,4-dione —— C23H27FN4O3
7-[1-[(4-Fluorophenyl)methyl]piperidin-4-yl]-1-(2-methoxyethyl)-3-methylpyrido[2,3-d]pyrimidine-2,4-dione
—— 7-[(4-methoxyphenyl)methyl]-4-methyl-2-[(3R)-1-(3-methylbutanoyl)piperidin-3-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C25H32N4O3
7-[(4-methoxyphenyl)methyl]-4-methyl-2-[(3R)-1-(3-methylbutanoyl)piperidin-3-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(3-methoxyphenyl)methyl]-4-methyl-2-[(3R)-1-(3-methylbutanoyl)piperidin-3-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C25H32N4O3
7-[(3-methoxyphenyl)methyl]-4-methyl-2-[(3R)-1-(3-methylbutanoyl)piperidin-3-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(3-fluorophenyl)methyl]-4-methyl-2-[(3R)-1-(2-pyrazol-1-ylacetyl)piperidin-3-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C24H25FN6O2
7-[(3-fluorophenyl)methyl]-4-methyl-2-[(3R)-1-(2-pyrazol-1-ylacetyl)piperidin-3-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-benzyl-2-[(3S)-1-(1-ethylpyrazole-3-carbonyl)piperidin-3-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C25H28N6O2
7-benzyl-2-[(3S)-1-(1-ethylpyrazole-3-carbonyl)piperidin-3-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(3S)-1-[2-(1H-indol-3-yl)acetyl]piperidin-3-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione —— C24H25N5O3
7-[(3S)-1-[2-(1H-indol-3-yl)acetyl]piperidin-3-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione
—— 7-[(2-methoxyphenyl)methyl]-4-methyl-2-[(2S)-1-(1-methylpyrazole-4-carbonyl)pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C24H26N6O3
7-[(2-methoxyphenyl)methyl]-4-methyl-2-[(2S)-1-(1-methylpyrazole-4-carbonyl)pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(3S)-1-[2-(4-fluorophenyl)acetyl]piperidin-3-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione —— C22H23FN4O3
7-[(3S)-1-[2-(4-fluorophenyl)acetyl]piperidin-3-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione
—— 7-[(4-methoxyphenyl)methyl]-4-methyl-2-[(2R)-1-(2-methylpyrazole-3-carbonyl)pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C24H26N6O3
7-[(4-methoxyphenyl)methyl]-4-methyl-2-[(2R)-1-(2-methylpyrazole-3-carbonyl)pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(2R)-1-(cyclopentanecarbonyl)pyrrolidin-2-yl]-1,3-dimethyl-5-(trifluoromethyl)pyrido[2,3-d]pyrimidine-2,4-dione —— C20H23F3N4O3
7-[(2R)-1-(cyclopentanecarbonyl)pyrrolidin-2-yl]-1,3-dimethyl-5-(trifluoromethyl)pyrido[2,3-d]pyrimidine-2,4-dione
—— 7-[(3R)-1-[(4-fluorophenyl)methyl]piperidin-3-yl]-1-(2-methoxyethyl)-3-methylpyrido[2,3-d]pyrimidine-2,4-dione —— C23H27FN4O3
7-[(3R)-1-[(4-fluorophenyl)methyl]piperidin-3-yl]-1-(2-methoxyethyl)-3-methylpyrido[2,3-d]pyrimidine-2,4-dione
—— 7-[(3-fluorophenyl)methyl]-4-methyl-2-[(3S)-1-(1-methylpyrazole-4-carbonyl)piperidin-3-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C24H25FN6O2
7-[(3-fluorophenyl)methyl]-4-methyl-2-[(3S)-1-(1-methylpyrazole-4-carbonyl)piperidin-3-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(3S)-1-[2-(4-methoxyphenyl)acetyl]piperidin-3-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione —— C23H26N4O4
7-[(3S)-1-[2-(4-methoxyphenyl)acetyl]piperidin-3-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione
—— 7-[(3R)-1-(3-methoxypropanoyl)piperidin-3-yl]-1,3-dimethyl-5-(trifluoromethyl)pyrido[2,3-d]pyrimidine-2,4-dione —— C19H23F3N4O4
7-[(3R)-1-(3-methoxypropanoyl)piperidin-3-yl]-1,3-dimethyl-5-(trifluoromethyl)pyrido[2,3-d]pyrimidine-2,4-dione
—— 7-[(3S)-1-benzylpiperidin-3-yl]-5-(trifluoromethyl)pyrido[2,3-d]pyrimidin-4-amine —— C20H20F3N5
7-[(3S)-1-benzylpiperidin-3-yl]-5-(trifluoromethyl)pyrido[2,3-d]pyrimidin-4-amine
—— 7-(cyclohexylmethyl)-2-[(2S)-1-(2-methoxyacetyl)piperidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C22H32N4O3
7-(cyclohexylmethyl)-2-[(2S)-1-(2-methoxyacetyl)piperidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(4-methoxyphenyl)methyl]-4-methyl-2-[(2S)-1-(pyridine-2-carbonyl)pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C25H25N5O3
7-[(4-methoxyphenyl)methyl]-4-methyl-2-[(2S)-1-(pyridine-2-carbonyl)pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(3-methoxyphenyl)methyl]-4-methyl-2-[(2S)-1-(2-methylpropanoyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C24H30N4O3
7-[(3-methoxyphenyl)methyl]-4-methyl-2-[(2S)-1-(2-methylpropanoyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(3-methoxyphenyl)methyl]-4-methyl-2-[(2R)-1-(5-methyl-1H-pyrazole-4-carbonyl)pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C24H26N6O3
7-[(3-methoxyphenyl)methyl]-4-methyl-2-[(2R)-1-(5-methyl-1H-pyrazole-4-carbonyl)pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[2-(4-fluorophenyl)ethyl]-4-methyl-2-[(2S)-1-propanoylpyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C22H25FN4O2
7-[2-(4-fluorophenyl)ethyl]-4-methyl-2-[(2S)-1-propanoylpyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-benzyl-2-[(2S)-1-(2,2-dimethylpropanoyl)pyrrolidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C23H28N4O2
7-benzyl-2-[(2S)-1-(2,2-dimethylpropanoyl)pyrrolidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(4-fluorophenyl)methyl]-4-methyl-2-[(2S)-1-(5-methylpyrazine-2-carbonyl)pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C24H23FN6O2
7-[(4-fluorophenyl)methyl]-4-methyl-2-[(2S)-1-(5-methylpyrazine-2-carbonyl)pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-(cyclohexylmethyl)-4-methyl-2-[(2R)-1-(2-oxo-2-pyrrolidin-1-ylethyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C25H37N5O2
7-(cyclohexylmethyl)-4-methyl-2-[(2R)-1-(2-oxo-2-pyrrolidin-1-ylethyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-(cyclopropylmethyl)-4-methyl-2-[(2S)-1-(3-methyl-1-benzofuran-2-carbonyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C26H28N4O3
7-(cyclopropylmethyl)-4-methyl-2-[(2S)-1-(3-methyl-1-benzofuran-2-carbonyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-(cyclohexylmethyl)-4-methyl-2-[(2S)-1-(thiadiazole-4-carbonyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C22H28N6O2S
7-(cyclohexylmethyl)-4-methyl-2-[(2S)-1-(thiadiazole-4-carbonyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(3-methoxyphenyl)methyl]-4-methyl-2-[(2R)-1-(2-methylpropanoyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C24H30N4O3
7-[(3-methoxyphenyl)methyl]-4-methyl-2-[(2R)-1-(2-methylpropanoyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(4-methoxyphenyl)methyl]-4-methyl-2-[(2R)-1-(2-methylpropanoyl)pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C23H28N4O3
7-[(4-methoxyphenyl)methyl]-4-methyl-2-[(2R)-1-(2-methylpropanoyl)pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(4-fluorophenyl)methyl]-4-methyl-2-[(2S)-1-(5-methyl-1H-pyrazole-4-carbonyl)pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C23H23FN6O2
7-[(4-fluorophenyl)methyl]-4-methyl-2-[(2S)-1-(5-methyl-1H-pyrazole-4-carbonyl)pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[2-(4-fluorophenyl)ethyl]-4-methyl-2-[(2R)-1-(3-methylbutanoyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C25H31FN4O2
7-[2-(4-fluorophenyl)ethyl]-4-methyl-2-[(2R)-1-(3-methylbutanoyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-benzyl-4-methyl-2-[(2R)-1-[2-(2-oxopyrrolidin-1-yl)acetyl]piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C25H29N5O3
7-benzyl-4-methyl-2-[(2R)-1-[2-(2-oxopyrrolidin-1-yl)acetyl]piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(2-methoxyphenyl)methyl]-4-methyl-2-[(2S)-1-(3-methylbutanoyl)pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C24H30N4O3
7-[(2-methoxyphenyl)methyl]-4-methyl-2-[(2S)-1-(3-methylbutanoyl)pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(4-methoxyphenyl)methyl]-4-methyl-2-[(2R)-1-propanoylpyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C22H26N4O3
7-[(4-methoxyphenyl)methyl]-4-methyl-2-[(2R)-1-propanoylpyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[2-(2-fluorophenyl)ethyl]-4-methyl-2-[(2R)-1-(5-methyl-1H-pyrazole-4-carbonyl)pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C24H25FN6O2
7-[2-(2-fluorophenyl)ethyl]-4-methyl-2-[(2R)-1-(5-methyl-1H-pyrazole-4-carbonyl)pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-(cyclohexylmethyl)-4-methyl-2-[(2R)-1-(pyridine-2-carbonyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C25H31N5O2
7-(cyclohexylmethyl)-4-methyl-2-[(2R)-1-(pyridine-2-carbonyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-(cyclopropylmethyl)-2-[(2R)-1-(4-fluorophenyl)sulfonylpiperidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C22H25FN4O3S
7-(cyclopropylmethyl)-2-[(2R)-1-(4-fluorophenyl)sulfonylpiperidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-(cyclopropylmethyl)-4-methyl-2-[(2R)-1-(5-methylpyrazine-2-carbonyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C22H26N6O2
7-(cyclopropylmethyl)-4-methyl-2-[(2R)-1-(5-methylpyrazine-2-carbonyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-(cyclopropylmethyl)-2-[(2R)-1-[2-(4-fluorophenoxy)acetyl]piperidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C24H27FN4O3
7-(cyclopropylmethyl)-2-[(2R)-1-[2-(4-fluorophenoxy)acetyl]piperidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-(cyclohexylmethyl)-4-methyl-2-[(2R)-1-(thiadiazole-4-carbonyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C22H28N6O2S
7-(cyclohexylmethyl)-4-methyl-2-[(2R)-1-(thiadiazole-4-carbonyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-(cyclopropylmethyl)-4-methyl-2-[(2S)-1-[4-(2-oxopyrrolidin-1-yl)butanoyl]piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C24H33N5O3
7-(cyclopropylmethyl)-4-methyl-2-[(2S)-1-[4-(2-oxopyrrolidin-1-yl)butanoyl]piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-(cyclopropylmethyl)-2-[(2S)-1-[2-(4-fluorophenyl)acetyl]piperidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C24H27FN4O2
7-(cyclopropylmethyl)-2-[(2S)-1-[2-(4-fluorophenyl)acetyl]piperidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one