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—— (7R)-5-methyl-7-(3-methylphenyl)-3-N-(4-methylphenyl)-6-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide —— C29H27N5O2
(7R)-5-methyl-7-(3-methylphenyl)-3-N-(4-methylphenyl)-6-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide
—— (7R)-7-(2-methoxyphenyl)-5-methyl-3-N-(4-methylphenyl)-6-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide —— C29H27N5O3
(7R)-7-(2-methoxyphenyl)-5-methyl-3-N-(4-methylphenyl)-6-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide
—— 7'-[1-(1,3-dimethyl-2,4,6-trioxo-1,3-diazinan-5-ylidene)ethylamino]-1,3-dimethylspiro[1,3-diazinane-5,4'-2,3,3a,5-tetrahydro-1H-pyrrolo[1,2-a]quinoline]-2,4,6-trione —— C25H28N6O6
7'-[1-(1,3-dimethyl-2,4,6-trioxo-1,3-diazinan-5-ylidene)ethylamino]-1,3-dimethylspiro[1,3-diazinane-5,4'-2,3,3a,5-tetrahydro-1H-pyrrolo[1,2-a]quinoline]-2,4,6-trione
—— (7S)-7-(4-chlorophenyl)-14-methyl-17-thia-2,8,14-triazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene —— C20H20ClN3S
(7S)-7-(4-chlorophenyl)-14-methyl-17-thia-2,8,14-triazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene
—— 7-methyl-4-[[4-[(5R)-5-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carbonyl]piperazin-1-yl]methyl]chromen-2-one —— C24H28N4O3
7-methyl-4-[[4-[(5R)-5-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carbonyl]piperazin-1-yl]methyl]chromen-2-one
—— (7R)-7-(4-methoxyphenyl)-11,13-dimethyl-2,8,14-triazatricyclo[8.4.0.02,6]tetradeca-1(10),3,5,11,13-pentaene —— C20H21N3O
(7R)-7-(4-methoxyphenyl)-11,13-dimethyl-2,8,14-triazatricyclo[8.4.0.02,6]tetradeca-1(10),3,5,11,13-pentaene
—— (7S)-7-thiophen-2-yl-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene —— C18H18N2S2
(7S)-7-thiophen-2-yl-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene
—— (7R)-7-methyl-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene —— C15H18N2S
(7R)-7-methyl-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene
—— (7R)-7-(3-methoxyphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene —— C21H22N2OS
(7R)-7-(3-methoxyphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene
—— (7R)-7-(4-methylphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene —— C21H22N2S
(7R)-7-(4-methylphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene
—— (7R)-N-cyclohexyl-9-oxo-8-[[(2S)-oxolan-2-yl]methyl]-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-7-carboxamide —— C26H33N3O3S
(7R)-N-cyclohexyl-9-oxo-8-[[(2S)-oxolan-2-yl]methyl]-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-7-carboxamide
—— (7S)-7-(4-methylphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene —— C21H22N2S
(7S)-7-(4-methylphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene
—— (7R)-7-(4-chlorophenyl)-14-methyl-17-thia-2,8,14-triazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene —— C20H20ClN3S
(7R)-7-(4-chlorophenyl)-14-methyl-17-thia-2,8,14-triazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene
—— (7S)-N-cyclohexyl-9-oxo-8-[[(2R)-oxolan-2-yl]methyl]-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-7-carboxamide —— C26H33N3O3S
(7S)-N-cyclohexyl-9-oxo-8-[[(2R)-oxolan-2-yl]methyl]-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-7-carboxamide
—— 7-chloro-5-[(3R)-3-methylpiperidin-1-yl]-3-[3-(trifluoromethyl)phenyl]triazolo[1,5-a]quinazoline —— C22H19ClF3N5
7-chloro-5-[(3R)-3-methylpiperidin-1-yl]-3-[3-(trifluoromethyl)phenyl]triazolo[1,5-a]quinazoline
—— 7-chloro-5-[(3S)-3-methylpiperidin-1-yl]-3-[3-(trifluoromethyl)phenyl]triazolo[1,5-a]quinazoline —— C22H19ClF3N5
7-chloro-5-[(3S)-3-methylpiperidin-1-yl]-3-[3-(trifluoromethyl)phenyl]triazolo[1,5-a]quinazoline
—— (7R)-3-[4-(3-nitrophenyl)-1,3-thiazol-2-yl]-7-phenyl-1,6,7,8-tetrahydroquinoline-2,5-dione —— C24H17N3O4S
(7R)-3-[4-(3-nitrophenyl)-1,3-thiazol-2-yl]-7-phenyl-1,6,7,8-tetrahydroquinoline-2,5-dione
—— (7S)-7-(4-methoxyphenyl)-3-[4-(3-nitrophenyl)-1,3-thiazol-2-yl]-1,6,7,8-tetrahydroquinoline-2,5-dione —— C25H19N3O5S
(7S)-7-(4-methoxyphenyl)-3-[4-(3-nitrophenyl)-1,3-thiazol-2-yl]-1,6,7,8-tetrahydroquinoline-2,5-dione
—— (7R)-3-[4-(3-fluoro-4-methoxyphenyl)-1,3-thiazol-2-yl]-7-(furan-2-yl)-1,6,7,8-tetrahydroquinoline-2,5-dione —— C23H17FN2O4S
(7R)-3-[4-(3-fluoro-4-methoxyphenyl)-1,3-thiazol-2-yl]-7-(furan-2-yl)-1,6,7,8-tetrahydroquinoline-2,5-dione
—— (7S)-7-(3,4-dimethoxyphenyl)-3-[4-(4-ethoxyphenyl)-1,3-thiazol-2-yl]-1,6,7,8-tetrahydroquinoline-2,5-dione —— C28H26N2O5S
(7S)-7-(3,4-dimethoxyphenyl)-3-[4-(4-ethoxyphenyl)-1,3-thiazol-2-yl]-1,6,7,8-tetrahydroquinoline-2,5-dione
—— (7R)-3-[4-(4-butylphenyl)-1,3-thiazol-2-yl]-7-(4-methoxyphenyl)-1,6,7,8-tetrahydroquinoline-2,5-dione —— C29H28N2O3S
(7R)-3-[4-(4-butylphenyl)-1,3-thiazol-2-yl]-7-(4-methoxyphenyl)-1,6,7,8-tetrahydroquinoline-2,5-dione
—— (7S)-3-[4-(4-chlorophenyl)-5-methyl-1,3-thiazol-2-yl]-7-(furan-2-yl)-1,6,7,8-tetrahydroquinoline-2,5-dione —— C23H17ClN2O3S
(7S)-3-[4-(4-chlorophenyl)-5-methyl-1,3-thiazol-2-yl]-7-(furan-2-yl)-1,6,7,8-tetrahydroquinoline-2,5-dione
—— (7S)-1-[5-(3,4-dimethylphenyl)-1,3-thiazol-2-yl]-2,5-dioxo-7-phenyl-7,8-dihydro-6H-quinoline-3-carbonitrile —— C27H21N3O2S
(7S)-1-[5-(3,4-dimethylphenyl)-1,3-thiazol-2-yl]-2,5-dioxo-7-phenyl-7,8-dihydro-6H-quinoline-3-carbonitrile
—— (7S)-3-[4-(3-nitrophenyl)-1,3-thiazol-2-yl]-7-phenyl-1,6,7,8-tetrahydroquinoline-2,5-dione —— C24H17N3O4S
(7S)-3-[4-(3-nitrophenyl)-1,3-thiazol-2-yl]-7-phenyl-1,6,7,8-tetrahydroquinoline-2,5-dione
—— 7,9,9-trimethyl-9a-[(E)-2-(naphthalen-1-yl)ethenyl]-9,9a-dihydro-1H-imidazo[1,2-a]indol-2(3H)-one —— C25H24N2O
7,9,9-trimethyl-9a-[(E)-2-(naphthalen-1-yl)ethenyl]-9,9a-dihydro-1H-imidazo[1,2-a]indol-2(3H)-one
—— (7R)-7-(4-methoxyphenyl)-3-[4-(3-nitrophenyl)-1,3-thiazol-2-yl]-1,6,7,8-tetrahydroquinoline-2,5-dione —— C25H19N3O5S
(7R)-7-(4-methoxyphenyl)-3-[4-(3-nitrophenyl)-1,3-thiazol-2-yl]-1,6,7,8-tetrahydroquinoline-2,5-dione
—— 7,9,9-trimethyl-9a-[(E)-2-(thiophen-2-yl)ethenyl]-9,9a-dihydro-1H-imidazo[1,2-a]indol-2(3H)-one —— C19H20N2OS
7,9,9-trimethyl-9a-[(E)-2-(thiophen-2-yl)ethenyl]-9,9a-dihydro-1H-imidazo[1,2-a]indol-2(3H)-one
—— (7R)-2-benzylsulfanyl-7-(2-chlorophenyl)-N-(2-methoxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H24ClN5O2S
(7R)-2-benzylsulfanyl-7-(2-chlorophenyl)-N-(2-methoxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(4-methoxyphenyl)-3-[4-(4-phenoxyphenyl)-1,3-thiazol-2-yl]-1,6,7,8-tetrahydroquinoline-2,5-dione —— C31H24N2O4S
(7R)-7-(4-methoxyphenyl)-3-[4-(4-phenoxyphenyl)-1,3-thiazol-2-yl]-1,6,7,8-tetrahydroquinoline-2,5-dione
—— 7-Chloro-1-hydroxy-3-(2-oxopropoxy)xanthen-9-one —— C16H11ClO5
7-Chloro-1-hydroxy-3-(2-oxopropoxy)xanthen-9-one
—— 7-chloro-1-hydroxy-3-[(3-oxobutan-2-yl)oxy]-9H-xanthen-9-one —— C17H13ClO5
7-chloro-1-hydroxy-3-[(3-oxobutan-2-yl)oxy]-9H-xanthen-9-one
—— (7S)-7-(3,4-dimethoxyphenyl)-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C17H21N5O3S
(7S)-7-(3,4-dimethoxyphenyl)-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-ethylsulfanyl-5-methyl-7-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C15H17N5OS
(7S)-2-ethylsulfanyl-5-methyl-7-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-ethylsulfanyl-5-methyl-7-pyridin-2-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C14H16N6OS
(7S)-2-ethylsulfanyl-5-methyl-7-pyridin-2-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(1,3-benzodioxol-5-yl)-2-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxylic acid —— C19H14N4O4
(7R)-7-(1,3-benzodioxol-5-yl)-2-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxylic acid
—— 7,8-dihydroxy-4-methyl-3-[2-oxo-2-(4-phenylpiperazin-1-yl)ethyl]-2H-chromen-2-one —— C22H22N2O5
7,8-dihydroxy-4-methyl-3-[2-oxo-2-(4-phenylpiperazin-1-yl)ethyl]-2H-chromen-2-one
—— 7,9,9-trimethyl-9a-[(E)-2-(3-nitrophenyl)ethenyl]-9,9a-dihydro-1H-imidazo[1,2-a]indol-2(3H)-one —— C21H21N3O3
7,9,9-trimethyl-9a-[(E)-2-(3-nitrophenyl)ethenyl]-9,9a-dihydro-1H-imidazo[1,2-a]indol-2(3H)-one
—— 7-[(3R,5R)-3,5-dimethylpiperidine-1-carbonyl]-3-[(2-methoxyphenyl)methyl]-2-sulfanylidene-1H-quinazolin-4-one —— C24H27N3O3S
7-[(3R,5R)-3,5-dimethylpiperidine-1-carbonyl]-3-[(2-methoxyphenyl)methyl]-2-sulfanylidene-1H-quinazolin-4-one
—— 7-[2-[(2R)-2-methylpiperidin-1-yl]ethyl]-6-sulfanylidene-5H-[1,3]dioxolo[4,5-g]quinazolin-8-one —— C17H21N3O3S
7-[2-[(2R)-2-methylpiperidin-1-yl]ethyl]-6-sulfanylidene-5H-[1,3]dioxolo[4,5-g]quinazolin-8-one
—— 7,9,9-trimethyl-9a-[(E)-2-(2-nitrophenyl)ethenyl]-9,9a-dihydro-1H-imidazo[1,2-a]indol-2(3H)-one —— C21H21N3O3
7,9,9-trimethyl-9a-[(E)-2-(2-nitrophenyl)ethenyl]-9,9a-dihydro-1H-imidazo[1,2-a]indol-2(3H)-one
—— 7-chloro-3-[[(2S)-1-ethylpyrrolidin-2-yl]methyl]-2-sulfanylidene-1H-quinazolin-4-one —— C15H18ClN3OS
7-chloro-3-[[(2S)-1-ethylpyrrolidin-2-yl]methyl]-2-sulfanylidene-1H-quinazolin-4-one
—— 7-(4-ethylpiperazine-1-carbonyl)-3-[[(2R)-oxolan-2-yl]methyl]-2-sulfanylidene-1H-quinazolin-4-one —— C20H26N4O3S
7-(4-ethylpiperazine-1-carbonyl)-3-[[(2R)-oxolan-2-yl]methyl]-2-sulfanylidene-1H-quinazolin-4-one
—— 7-[4-(1,3-benzodioxol-5-ylmethyl)piperazine-1-carbonyl]-3-[[(2S)-oxolan-2-yl]methyl]-2-sulfanylidene-1H-quinazolin-4-one —— C26H28N4O5S
7-[4-(1,3-benzodioxol-5-ylmethyl)piperazine-1-carbonyl]-3-[[(2S)-oxolan-2-yl]methyl]-2-sulfanylidene-1H-quinazolin-4-one
—— 7-(4-chlorophenyl)-5-[2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl]sulfanyl-1,3-dimethylpyrimido[4,5-d]pyrimidine-2,4-dione —— C22H24ClN5O4S
7-(4-chlorophenyl)-5-[2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl]sulfanyl-1,3-dimethylpyrimido[4,5-d]pyrimidine-2,4-dione
—— (7S)-7-(4-fluorophenyl)-N-(4-methoxyphenyl)-5-methyl-2-methylsulfanyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C21H20FN5O2S
(7S)-7-(4-fluorophenyl)-N-(4-methoxyphenyl)-5-methyl-2-methylsulfanyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(4-ethoxyphenyl)-N-(4-methoxyphenyl)-5-methyl-2-methylsulfanyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H25N5O3S
(7R)-7-(4-ethoxyphenyl)-N-(4-methoxyphenyl)-5-methyl-2-methylsulfanyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(3-chlorophenyl)-5-methyl-3-N,6-N-diphenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide —— C27H22ClN5O2
(7R)-7-(3-chlorophenyl)-5-methyl-3-N,6-N-diphenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide
—— (7R)-6-N,7-bis(2-methoxyphenyl)-5-methyl-3-N-(4-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide —— C30H29N5O4
(7R)-6-N,7-bis(2-methoxyphenyl)-5-methyl-3-N-(4-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide
—— 7-[(3R)-3-methylpiperidin-1-yl]sulfonyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one —— C15H20N2O3S2
7-[(3R)-3-methylpiperidin-1-yl]sulfonyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one
—— (7S)-7-(2,3-dimethoxyphenyl)-N-(4-methoxyphenyl)-5-methyl-2-methylsulfanyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H25N5O4S
(7S)-7-(2,3-dimethoxyphenyl)-N-(4-methoxyphenyl)-5-methyl-2-methylsulfanyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide