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中文名称 英文名称 CAS号 化学式 结构式图片
—— 7-cyclohexyl-2-[(2S)-1-(2-fluorobenzoyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C25H31FN4O2
7-cyclohexyl-2-[(2S)-1-(2-fluorobenzoyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(2-Fluorophenyl)methyl]-2-pyrazin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C18H16FN5O
7-[(2-Fluorophenyl)methyl]-2-pyrazin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(2-fluorobenzoyl)-2-[(3S)-1-(pyridin-2-ylmethyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H24FN5O2
7-(2-fluorobenzoyl)-2-[(3S)-1-(pyridin-2-ylmethyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(pyridin-4-ylmethyl)-2-[(2S)-1-(thiophene-2-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H25N5O2S
7-(pyridin-4-ylmethyl)-2-[(2S)-1-(thiophene-2-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(2-fluorobenzoyl)-2-[(3S)-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H24FN5O2
7-(2-fluorobenzoyl)-2-[(3S)-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(2-fluorobenzoyl)-2-[(3S)-1-(pyrazine-2-carbonyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H21FN6O3
7-(2-fluorobenzoyl)-2-[(3S)-1-(pyrazine-2-carbonyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(pyridine-4-carbonyl)-2-[(2R)-1-(thiophen-2-ylmethyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H25N5O2S
7-(pyridine-4-carbonyl)-2-[(2R)-1-(thiophen-2-ylmethyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(6-Fluoroquinolin-2-yl)methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H18FN5O
7-[(6-Fluoroquinolin-2-yl)methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-chloro-N-(cyclopropylmethyl)-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide —— C19H23ClN2O3
7-chloro-N-(cyclopropylmethyl)-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide
—— 7-(2-fluorobenzoyl)-2-[(3R)-1-(pyridin-2-ylmethyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H24FN5O2
7-(2-fluorobenzoyl)-2-[(3R)-1-(pyridin-2-ylmethyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(2-fluorobenzoyl)-2-[(3R)-1-(pyrazine-2-carbonyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H21FN6O3
7-(2-fluorobenzoyl)-2-[(3R)-1-(pyrazine-2-carbonyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-Chloro-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxylic acid —— C15H16ClNO4
7-Chloro-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxylic acid
—— 7-(thiophene-2-carbonyl)-2-[(2S)-1-(thiophene-2-carbonyl)pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C21H20N4O3S2
7-(thiophene-2-carbonyl)-2-[(2S)-1-(thiophene-2-carbonyl)pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(cyclohexylmethyl)-2-[(2R)-1-(pyridine-3-carbonyl)pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H31N5O2
7-(cyclohexylmethyl)-2-[(2R)-1-(pyridine-3-carbonyl)pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(3S)-1-(pyrazine-2-carbonyl)piperidin-3-yl]-2-(trifluoromethyl)-6H-1,6-naphthyridin-5-one —— C19H16F3N5O2
7-[(3S)-1-(pyrazine-2-carbonyl)piperidin-3-yl]-2-(trifluoromethyl)-6H-1,6-naphthyridin-5-one
—— 7-[[4-(2-Oxo-2-pyrrolidin-1-ylethoxy)phenyl]methyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C25H27N5O3
7-[[4-(2-Oxo-2-pyrrolidin-1-ylethoxy)phenyl]methyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-cyclohexyl-2-[(2R)-1-(thiophene-2-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H30N4O2S
7-cyclohexyl-2-[(2R)-1-(thiophene-2-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[[(3S)-oxolan-3-yl]methyl]-4-pyridin-3-yloxy-2-pyrrolidin-1-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidine —— C21H27N5O2
7-[[(3S)-oxolan-3-yl]methyl]-4-pyridin-3-yloxy-2-pyrrolidin-1-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidine
—— 7-[[(1R)-cyclohex-3-en-1-yl]methyl]-2-pyridin-3-yl-1,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C19H22N4O
7-[[(1R)-cyclohex-3-en-1-yl]methyl]-2-pyridin-3-yl-1,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(cyclobutanecarbonyl)-2-[(3R)-1-(thiophen-2-ylmethyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C21H26N4O2S
7-(cyclobutanecarbonyl)-2-[(3R)-1-(thiophen-2-ylmethyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-cyclohexyl-2-[(2S)-1-(2-thiophen-2-ylacetyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H32N4O2S
7-cyclohexyl-2-[(2S)-1-(2-thiophen-2-ylacetyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— [7-Chloro-1-(2-pyrrolidin-1-ylethyl)pyrrolo[2,3-c]pyridin-3-yl]-(4-fluorophenyl)methanone —— C20H19ClFN3O
[7-Chloro-1-(2-pyrrolidin-1-ylethyl)pyrrolo[2,3-c]pyridin-3-yl]-(4-fluorophenyl)methanone
—— 7-(pyridine-4-carbonyl)-2-[(2R)-1-(pyridine-3-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H24N6O3
7-(pyridine-4-carbonyl)-2-[(2R)-1-(pyridine-3-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(3S)-1-(pyridine-4-carbonyl)piperidin-3-yl]-2-(trifluoromethyl)-6H-1,6-naphthyridin-5-one —— C20H17F3N4O2
7-[(3S)-1-(pyridine-4-carbonyl)piperidin-3-yl]-2-(trifluoromethyl)-6H-1,6-naphthyridin-5-one
—— 7-[(4-Fluorophenyl)methyl]-2-pyrazin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C18H16FN5O
7-[(4-Fluorophenyl)methyl]-2-pyrazin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(cyclobutanecarbonyl)-2-[(3R)-1-[(2,3-difluorophenyl)methyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H26F2N4O2
7-(cyclobutanecarbonyl)-2-[(3R)-1-[(2,3-difluorophenyl)methyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(3-fluorophenyl)methyl]-2-pyrazin-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C19H18FN5O
7-[(3-fluorophenyl)methyl]-2-pyrazin-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-[(4-methoxyphenyl)methyl]-2-[(3R)-1-(1-methylpyrazole-4-carbonyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H28N6O3
7-[(4-methoxyphenyl)methyl]-2-[(3R)-1-(1-methylpyrazole-4-carbonyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(3S)-1-(2-methylpyrazole-3-carbonyl)pyrrolidin-3-yl]-6H-1,6-naphthyridin-5-one —— C17H17N5O2
7-[(3S)-1-(2-methylpyrazole-3-carbonyl)pyrrolidin-3-yl]-6H-1,6-naphthyridin-5-one
—— 7-[(2-methylpyrimidin-5-yl)methyl]-2-pyrazin-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C18H19N7O
7-[(2-methylpyrimidin-5-yl)methyl]-2-pyrazin-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-[[3-(2-methoxyethoxy)phenyl]methyl]-2-methyl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C19H25N3O3
7-[[3-(2-methoxyethoxy)phenyl]methyl]-2-methyl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-benzyl-2-methyl-N-[[(2S)-oxolan-2-yl]methyl]-N-(pyridin-2-ylmethyl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-amine —— C26H31N5O
7-benzyl-2-methyl-N-[[(2S)-oxolan-2-yl]methyl]-N-(pyridin-2-ylmethyl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-amine
—— 7-[2-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)acetyl]-2-methyl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C20H23N3O4
7-[2-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)acetyl]-2-methyl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-[(3-fluorophenyl)methyl]-2-methyl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C16H18FN3O
7-[(3-fluorophenyl)methyl]-2-methyl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-[(3-methoxyphenyl)methyl]-2-methyl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C17H21N3O2
7-[(3-methoxyphenyl)methyl]-2-methyl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-2-methyl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C20H25N3O2
7-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-2-methyl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-benzyl-4-(6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl)-2-methyl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidine —— C20H23N7
7-benzyl-4-(6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl)-2-methyl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidine
—— 7-[(4-methoxynaphthalen-1-yl)methyl]-2-methyl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C21H23N3O2
7-[(4-methoxynaphthalen-1-yl)methyl]-2-methyl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-[(3,4-dimethoxyphenyl)methyl]-2-methyl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C18H23N3O3
7-[(3,4-dimethoxyphenyl)methyl]-2-methyl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-methoxy-1'-(3-methyl-4-oxophthalazine-1-carbonyl)spiro[3H-chromene-2,4'-piperidine]-4-one —— C24H23N3O5
7-methoxy-1'-(3-methyl-4-oxophthalazine-1-carbonyl)spiro[3H-chromene-2,4'-piperidine]-4-one
—— 7-benzyl-N-[(3R)-1,1-dioxothiolan-3-yl]-N,2-dimethyl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-amine —— C20H26N4O2S
7-benzyl-N-[(3R)-1,1-dioxothiolan-3-yl]-N,2-dimethyl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-amine
—— 7-[(3R)-1-(3-fluoro-4-methoxyphenyl)sulfonylpiperidin-3-yl]-5-methylimidazo[5,1-b][1,3]thiazole —— C18H20FN3O3S2
7-[(3R)-1-(3-fluoro-4-methoxyphenyl)sulfonylpiperidin-3-yl]-5-methylimidazo[5,1-b][1,3]thiazole
—— 7-[(3R)-1-[2-(4-methylpyrazol-1-yl)acetyl]pyrrolidin-3-yl]-6H-1,6-naphthyridin-5-one —— C18H19N5O2
7-[(3R)-1-[2-(4-methylpyrazol-1-yl)acetyl]pyrrolidin-3-yl]-6H-1,6-naphthyridin-5-one
—— 7-[1-[(2,4-Dimethoxyphenyl)methyl]piperidin-4-yl]-3,5-dimethylimidazo[5,1-b][1,3]thiazole —— C21H27N3O2S
7-[1-[(2,4-Dimethoxyphenyl)methyl]piperidin-4-yl]-3,5-dimethylimidazo[5,1-b][1,3]thiazole
—— 7-[(3R)-1-(4-fluorophenyl)sulfonylpiperidin-3-yl]-3,5-dimethylimidazo[5,1-b][1,3]thiazole —— C18H20FN3O2S2
7-[(3R)-1-(4-fluorophenyl)sulfonylpiperidin-3-yl]-3,5-dimethylimidazo[5,1-b][1,3]thiazole
—— 7-[(4-Methoxyphenyl)methyl]-2-(5-methylpyrazin-2-yl)-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C20H21N5O2
7-[(4-Methoxyphenyl)methyl]-2-(5-methylpyrazin-2-yl)-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(3-Fluorophenyl)methyl]-2-(5-methylpyrazin-2-yl)-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C19H18FN5O
7-[(3-Fluorophenyl)methyl]-2-(5-methylpyrazin-2-yl)-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(4-Fluorophenyl)methyl]-2-(5-methylpyrazin-2-yl)-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C19H18FN5O
7-[(4-Fluorophenyl)methyl]-2-(5-methylpyrazin-2-yl)-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(3R)-1-[(2S)-2-methyl-3-(3-methylpyrazol-1-yl)propanoyl]pyrrolidin-3-yl]-6H-1,6-naphthyridin-5-one —— C20H23N5O2
7-[(3R)-1-[(2S)-2-methyl-3-(3-methylpyrazol-1-yl)propanoyl]pyrrolidin-3-yl]-6H-1,6-naphthyridin-5-one
—— 7-acetyl-2-[(2S)-1-(5-methylpyrazine-2-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C20H24N6O3
7-acetyl-2-[(2S)-1-(5-methylpyrazine-2-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one