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—— (7S)-N-(1-ethylpyrazol-3-yl)-2,5-dimethyl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide —— C14H20N6O
(7S)-N-(1-ethylpyrazol-3-yl)-2,5-dimethyl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide
—— (7R)-N-[2-(4-fluorophenyl)ethyl]-2-methyl-5-[(E)-2-methyl-3-phenylprop-2-enyl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide —— C26H29FN4O
(7R)-N-[2-(4-fluorophenyl)ethyl]-2-methyl-5-[(E)-2-methyl-3-phenylprop-2-enyl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide
—— 7-Hydroxy-8-[[4-(2-hydroxyethyl)piperazine-1,4-diium-1-yl]methyl]-4-methylchromen-2-one —— C17H24N2O4+2
7-Hydroxy-8-[[4-(2-hydroxyethyl)piperazine-1,4-diium-1-yl]methyl]-4-methylchromen-2-one
—— (7R)-N-(1-ethylpyrazol-3-yl)-2,5-dimethyl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide —— C14H20N6O
(7R)-N-(1-ethylpyrazol-3-yl)-2,5-dimethyl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide
—— (7S)-N-[(4-methoxyphenyl)methyl]-2-methyl-5-[(4-propan-2-yloxyphenyl)methyl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide —— C26H32N4O3
(7S)-N-[(4-methoxyphenyl)methyl]-2-methyl-5-[(4-propan-2-yloxyphenyl)methyl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide
—— (7S)-5-[2-(2-fluorophenyl)acetyl]-2-methyl-N-(pyridin-2-ylmethyl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide —— C22H22FN5O2
(7S)-5-[2-(2-fluorophenyl)acetyl]-2-methyl-N-(pyridin-2-ylmethyl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide
—— (7R)-5-[4-(4-fluorophenyl)butanoyl]-2-methyl-N-(pyridin-2-ylmethyl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide —— C24H26FN5O2
(7R)-5-[4-(4-fluorophenyl)butanoyl]-2-methyl-N-(pyridin-2-ylmethyl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide
—— (7S)-N-[(2-fluorophenyl)methyl]-2-methyl-5-[2-(methylamino)pyridine-4-carbonyl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide —— C22H23FN6O2
(7S)-N-[(2-fluorophenyl)methyl]-2-methyl-5-[2-(methylamino)pyridine-4-carbonyl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide
—— (7S)-2-methyl-N-propyl-4,5,6,7-tetrahydropyrazolo[4,3-c]pyridine-7-carboxamide —— C11H18N4O
(7S)-2-methyl-N-propyl-4,5,6,7-tetrahydropyrazolo[4,3-c]pyridine-7-carboxamide
—— (7R)-N-[2-(5-fluoro-1H-indol-3-yl)ethyl]-5-[(4-fluorophenyl)methyl]-2-methyl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide —— C25H25F2N5O
(7R)-N-[2-(5-fluoro-1H-indol-3-yl)ethyl]-5-[(4-fluorophenyl)methyl]-2-methyl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide
—— (7R)-5-[2-(4-fluorophenoxy)acetyl]-N-[(2-fluorophenyl)methyl]-2-methyl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide —— C23H22F2N4O3
(7R)-5-[2-(4-fluorophenoxy)acetyl]-N-[(2-fluorophenyl)methyl]-2-methyl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide
—— (7R)-5-[2-(1H-indol-3-yl)acetyl]-2-methyl-N-(pyridin-2-ylmethyl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide —— C24H24N6O2
(7R)-5-[2-(1H-indol-3-yl)acetyl]-2-methyl-N-(pyridin-2-ylmethyl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide
—— (7S)-N-(2-fluorophenyl)-2-methyl-5-(pyridine-4-carbonyl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide —— C20H18FN5O2
(7S)-N-(2-fluorophenyl)-2-methyl-5-(pyridine-4-carbonyl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide
—— (7S)-5-(4-fluorobenzoyl)-N-[(4-methoxyphenyl)methyl]-2-methyl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide —— C23H23FN4O3
(7S)-5-(4-fluorobenzoyl)-N-[(4-methoxyphenyl)methyl]-2-methyl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide
—— (7R)-N-[2-(4-fluorophenyl)ethyl]-5-(2-methoxyacetyl)-2-methyl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide —— C19H23FN4O3
(7R)-N-[2-(4-fluorophenyl)ethyl]-5-(2-methoxyacetyl)-2-methyl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide
—— (7R)-5-[3-(4-fluorophenyl)propanoyl]-2-methyl-N-(pyridin-2-ylmethyl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide —— C23H24FN5O2
(7R)-5-[3-(4-fluorophenyl)propanoyl]-2-methyl-N-(pyridin-2-ylmethyl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide
—— (7S)-N-[2-(4-fluorophenyl)ethyl]-5-(2-methoxyacetyl)-2-methyl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide —— C19H23FN4O3
(7S)-N-[2-(4-fluorophenyl)ethyl]-5-(2-methoxyacetyl)-2-methyl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide
—— (7R)-2-methyl-5-(2-phenylacetyl)-N-(pyridin-2-ylmethyl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide —— C22H23N5O2
(7R)-2-methyl-5-(2-phenylacetyl)-N-(pyridin-2-ylmethyl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide
—— (7S)-N-(2-methoxyphenyl)-2-methyl-5-(2-phenoxyacetyl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide —— C23H24N4O4
(7S)-N-(2-methoxyphenyl)-2-methyl-5-(2-phenoxyacetyl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide
—— (7R)-5-[3-(4-methoxyphenyl)propanoyl]-2-methyl-N-(pyridin-2-ylmethyl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide —— C24H27N5O3
(7R)-5-[3-(4-methoxyphenyl)propanoyl]-2-methyl-N-(pyridin-2-ylmethyl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide
—— (7R)-2-methyl-5-(3-phenylpropanoyl)-N-(pyridin-2-ylmethyl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide —— C23H25N5O2
(7R)-2-methyl-5-(3-phenylpropanoyl)-N-(pyridin-2-ylmethyl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide
—— (7R)-5-[2-(4-fluorophenyl)acetyl]-N-[2-(4-fluorophenyl)ethyl]-2-methyl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide —— C24H24F2N4O2
(7R)-5-[2-(4-fluorophenyl)acetyl]-N-[2-(4-fluorophenyl)ethyl]-2-methyl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide
—— (7R)-5-[2-(azepan-1-yl)acetyl]-2-methyl-N-(pyridin-2-ylmethyl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide —— C22H30N6O2
(7R)-5-[2-(azepan-1-yl)acetyl]-2-methyl-N-(pyridin-2-ylmethyl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide
—— (7R)-N-(2-methoxyphenyl)-2-methyl-5-(2-pyridin-2-ylacetyl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide —— C22H23N5O3
(7R)-N-(2-methoxyphenyl)-2-methyl-5-(2-pyridin-2-ylacetyl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide
—— (7S)-N-[(4-methoxyphenyl)methyl]-2-methyl-5-(pyridine-4-carbonyl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide —— C22H23N5O3
(7S)-N-[(4-methoxyphenyl)methyl]-2-methyl-5-(pyridine-4-carbonyl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide
—— (7S)-5-(4-fluorophenyl)sulfonyl-N-(2-methoxyphenyl)-2-methyl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide —— C21H21FN4O4S
(7S)-5-(4-fluorophenyl)sulfonyl-N-(2-methoxyphenyl)-2-methyl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide
—— [(7R)-2-methyl-5-(pyridine-3-carbonyl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-7-yl]-morpholin-4-ylmethanone —— C18H21N5O3
[(7R)-2-methyl-5-(pyridine-3-carbonyl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-7-yl]-morpholin-4-ylmethanone
—— (7R)-5-benzyl-N-[2-(5-fluoro-1H-indol-3-yl)ethyl]-2-methyl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide —— C25H26FN5O
(7R)-5-benzyl-N-[2-(5-fluoro-1H-indol-3-yl)ethyl]-2-methyl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide
—— (7S)-N-[2-(5-fluoro-1H-indol-3-yl)ethyl]-2-methyl-5-(pyridin-2-ylmethyl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide —— C24H25FN6O
(7S)-N-[2-(5-fluoro-1H-indol-3-yl)ethyl]-2-methyl-5-(pyridin-2-ylmethyl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide
—— (7-chloro-4-methoxyquinolin-3-yl)-[(3R)-3-(2H-pyrazolo[3,4-b]pyrazin-3-yl)piperidin-1-yl]methanone —— C21H19ClN6O2
(7-chloro-4-methoxyquinolin-3-yl)-[(3R)-3-(2H-pyrazolo[3,4-b]pyrazin-3-yl)piperidin-1-yl]methanone
—— 7-methoxy-1'-[(3S)-1-(2-methoxyethyl)-5-oxopyrrolidine-3-carbonyl]spiro[3H-chromene-2,4'-piperidine]-4-one —— C22H28N2O6
7-methoxy-1'-[(3S)-1-(2-methoxyethyl)-5-oxopyrrolidine-3-carbonyl]spiro[3H-chromene-2,4'-piperidine]-4-one
—— 7-[[2-methoxy-5-(methoxymethyl)phenyl]methyl]-2-pyrazin-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C22H25N5O3
7-[[2-methoxy-5-(methoxymethyl)phenyl]methyl]-2-pyrazin-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-[1-[5-(methoxymethyl)furan-2-carbonyl]piperidin-4-yl]-6H-1,6-naphthyridin-5-one —— C20H21N3O4
7-[1-[5-(methoxymethyl)furan-2-carbonyl]piperidin-4-yl]-6H-1,6-naphthyridin-5-one
—— 7-[[5-(methoxymethyl)furan-2-yl]methyl]-2-pyridin-4-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C20H22N4O3
7-[[5-(methoxymethyl)furan-2-yl]methyl]-2-pyridin-4-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-[[2-Methoxy-5-(methoxymethyl)phenyl]methyl]-2-pyrazin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C21H23N5O3
7-[[2-Methoxy-5-(methoxymethyl)phenyl]methyl]-2-pyrazin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[[4-methoxy-3-(2-methoxyethoxy)phenyl]methyl]-2-pyridin-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C24H28N4O4
7-[[4-methoxy-3-(2-methoxyethoxy)phenyl]methyl]-2-pyridin-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-[[4-Methoxy-3-(2-methoxyethoxy)phenyl]methyl]-2-pyrazin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H25N5O4
7-[[4-Methoxy-3-(2-methoxyethoxy)phenyl]methyl]-2-pyrazin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[[4-methoxy-3-(2-methoxyethoxy)phenyl]methyl]-2-morpholin-4-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C23H32N4O5
7-[[4-methoxy-3-(2-methoxyethoxy)phenyl]methyl]-2-morpholin-4-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— (7E)-4,6-bis(4-chlorophenyl)-7-(naphthalene-2-carbonyl)-5-naphthalen-2-yl-3-phenyl-3,4,5,6-tetrahydro-1H-azocin-2-one —— C46H33Cl2NO2
(7E)-4,6-bis(4-chlorophenyl)-7-(naphthalene-2-carbonyl)-5-naphthalen-2-yl-3-phenyl-3,4,5,6-tetrahydro-1H-azocin-2-one
—— (7-chloro-4-methoxyquinolin-3-yl)-[(3S)-3-(2H-pyrazolo[3,4-b]pyrazin-3-yl)piperidin-1-yl]methanone —— C21H19ClN6O2
(7-chloro-4-methoxyquinolin-3-yl)-[(3S)-3-(2H-pyrazolo[3,4-b]pyrazin-3-yl)piperidin-1-yl]methanone
—— 7-[[3-(2-Methoxyethoxy)phenyl]methyl]-2-pyrazin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C21H23N5O3
7-[[3-(2-Methoxyethoxy)phenyl]methyl]-2-pyrazin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(2-methoxyphenyl)methyl]-2-[(3S)-1-(3-methoxypropanoyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H30N4O4
7-[(2-methoxyphenyl)methyl]-2-[(3S)-1-(3-methoxypropanoyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-methoxy-1'-[(3R)-1-(2-methoxyethyl)-5-oxopyrrolidine-3-carbonyl]spiro[3H-chromene-2,4'-piperidine]-4-one —— C22H28N2O6
7-methoxy-1'-[(3R)-1-(2-methoxyethyl)-5-oxopyrrolidine-3-carbonyl]spiro[3H-chromene-2,4'-piperidine]-4-one
—— 7-(cyclopropanecarbonyl)-2-[(3R)-1-(3-methoxypropanoyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C19H26N4O4
7-(cyclopropanecarbonyl)-2-[(3R)-1-(3-methoxypropanoyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(cyclopropanecarbonyl)-2-[(3S)-1-(3-methoxypropanoyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C19H26N4O4
7-(cyclopropanecarbonyl)-2-[(3S)-1-(3-methoxypropanoyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(2-fluorobenzoyl)-2-[(3S)-1-(3-methoxypropanoyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H25FN4O4
7-(2-fluorobenzoyl)-2-[(3S)-1-(3-methoxypropanoyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(1-methyl-3,4-dihydro-2H-quinolin-6-yl)methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H25N5O
7-[(1-methyl-3,4-dihydro-2H-quinolin-6-yl)methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-cyclopentyl-2-[(2S)-1-[3-(dimethylamino)benzoyl]piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C26H35N5O2
7-cyclopentyl-2-[(2S)-1-[3-(dimethylamino)benzoyl]piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[1-(cyclobutanecarbonyl)piperidin-4-yl]-2-(dimethylamino)-6H-pyrido[4,3-d]pyrimidin-5-one —— C19H25N5O2
7-[1-(cyclobutanecarbonyl)piperidin-4-yl]-2-(dimethylamino)-6H-pyrido[4,3-d]pyrimidin-5-one
—— 7-[(4-Methoxy-2,3-dimethylphenyl)methyl]-2-pyrazin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C21H23N5O2
7-[(4-Methoxy-2,3-dimethylphenyl)methyl]-2-pyrazin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one